NCT06034743

Brief Summary

This is a Phase III, multicentre, randomised, double-blinded, placebo-controlled, parallel group study to evaluate the safety, tolerability and effect of 1 or 2 mg baxdrostat versus placebo, administered once daily (QD) orally, on the reduction of systolic blood pressure in approximately 720 participants aged ≥ 18 years with hypertension, despite a stable regimen of 2 antihypertensive agents at baseline, one of which is a diuretic (uncontrolled hypertension); or ≥ 3 antihypertensive agents at baseline, one of which is a diuretic (treatment-resistant hypertension).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
796

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Nov 2023

Geographic Reach
28 countries

260 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 6, 2023

Completed
7 days until next milestone

First Posted

Study publicly available on registry

September 13, 2023

Completed
2 months until next milestone

Study Start

First participant enrolled

November 22, 2023

Completed
1.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 21, 2025

Completed
5 months until next milestone

Study Completion

Last participant's last visit for all outcomes

October 10, 2025

Completed
Last Updated

November 10, 2025

Status Verified

November 1, 2025

Enrollment Period

1.5 years

First QC Date

September 6, 2023

Last Update Submit

November 6, 2025

Conditions

Keywords

HypertensionUncontrolled hypertensionResistant hypertensionBlood pressureBaxdrostatCIN-107AldosteroneAldosterone synthase

Outcome Measures

Primary Outcomes (2)

  • Change from baseline in seated systolic blood pressure for 2 mg baxdrostat

    To assess the effect of 2 mg baxdrostat versus placebo on seated systolic blood pressure at Week 12

    At Week 12

  • Change from baseline in seated systolic blood pressure for 1 mg baxdrostat

    To assess the effect of 1 mg baxdrostat versus placebo on seated systolic blood pressure at Week 12

    At Week 12

Secondary Outcomes (7)

  • Change from randomised withdrawal baseline (Week 24) in seated systolic blood pressure (SBP) for 2 mg baxdrostat

    At Week 32

  • Change from baseline in seated SBP for 2 mg baxdrostat

    At Week 12

  • Change from baseline in seated diastolic blood pressure (DBP) for 2 mg baxdrostat

    At Week 12

  • Achieving seated SBP < 130 mmHg for 2 mg baxdrostat

    At Week 12

  • Change from baseline in seated SBP for 1 mg baxdrostat

    At Week 12

  • +2 more secondary outcomes

Other Outcomes (1)

  • Number of participants with adverse events (AEs)

    Up to Week 54

Study Arms (3)

2 mg baxdrostat

EXPERIMENTAL

2 mg baxdrostat administered orally, once daily (QD).

Drug: Baxdrostat

1 mg baxdrostat

EXPERIMENTAL

1 mg baxdrostat administered orally, once daily (QD).

Drug: Baxdrostat

Placebo

PLACEBO COMPARATOR

Placebo administered orally, once daily (QD).

Drug: Placebo

Interventions

Baxdrostat tablet administered orally, once daily (QD). Unit dose strengths: * 1 mg per tablet for 1 mg baxdrostat Arm; * 2 mg per tablet for 2 mg baxdrostat Arm.

Also known as: CIN-107
1 mg baxdrostat2 mg baxdrostat

Placebo tablet matching baxdrostat, administered orally, once daily (QD).

Placebo

Eligibility Criteria

Age18 Years - 130 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male or female participants must be ≥ 18 years old
  • Mean sitting systolic blood pressure on automated office blood pressure measurement ≥ 140 mmHg and \< 170 mmHg at Screening
  • Fulfil at least 1 of the following 2 criteria:
  • uHTN subpopulation: have a stable regimen of 2 antihypertensive medications, from different therapeutic classes (at least one must be a diuretic), at maximum tolerated dose in the judgement of the Investigator
  • rHTN subpopulation: have a stable regimen of ≥ 3 antihypertensive medications, from different therapeutic classes (at least one must be a diuretic), at maximum tolerated dose in the judgement of the Investigator
  • Estimated glomerular filtration rate ≥ 45 mL/min/1.73m2 at Screening
  • Serum potassium (K+) level ≥ 3.5 and \< 5.0 mmol/L at Screening
  • Randomisation Criterion:
  • Sitting systolic blood pressure on attended automated office blood pressure measurement of ≥ 135 mmHg at the Baseline Visit

You may not qualify if:

  • Mean sitting systolic blood pressure on attended automated office blood pressure measurement ≥ 170 mmHg
  • Mean seated diastolic blood pressure on attended automated office blood pressure measurement ≥ 110 mmHg
  • Serum sodium level \< 135 mmol/L at Screening
  • Has the following known secondary causes of hypertension: renal artery stenosis, uncontrolled or untreated hyperthyroidism, uncontrolled or untreated hypothyroidism, pheochromocytoma, Cushing's syndrome, aortic coarctation
  • New York Heart Association functional heart failure class IV at Screening
  • Persistent atrial fibrillation

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (263)

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Saraland, Alabama, 36571, United States

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Scottsdale, Arizona, 85054, United States

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Sun City West, Arizona, 85375, United States

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Surprise, Arizona, 85374, United States

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Little Rock, Arkansas, 72211, United States

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Fresno, California, 93720, United States

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Lincoln, California, 95648, United States

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Orange, California, 92868, United States

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Rancho Cucamonga, California, 91730, United States

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Stanford, California, 94304, United States

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New Haven, Connecticut, 06510, United States

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Clearwater, Florida, 33765, United States

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Jacksonville, Florida, 32204, United States

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Port Orange, Florida, 32127, United States

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Atlanta, Georgia, 30344, United States

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Decatur, Georgia, 30033, United States

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Springfield, Illinois, 62702, United States

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Munster, Indiana, 46321, United States

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Lexington, Kentucky, 40503, United States

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Detroit, Michigan, 48202, United States

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Rochester, Minnesota, 55905, United States

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Olive Branch, Mississippi, 38654, United States

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Kansas City, Missouri, 64111, United States

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Kansas City, Missouri, 64128, United States

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Kansas City, Missouri, 64151, United States

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Rosedale, New York, 11422, United States

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The Bronx, New York, 10455, United States

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Chapel Hill, North Carolina, 27599, United States

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New Bern, North Carolina, 28562, United States

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Toledo, Ohio, 43614, United States

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Grants Pass, Oregon, 97527, United States

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Bethlehem, Pennsylvania, 18017, United States

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Langhorne, Pennsylvania, 19047, United States

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East Providence, Rhode Island, 02914, United States

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Memphis, Tennessee, 38105, United States

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Brownsville, Texas, 78526, United States

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Corpus Christi, Texas, 78404, United States

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Houston, Texas, 77054, United States

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Sugar Land, Texas, 77479, United States

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Manassas, Virginia, 20110, United States

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Suffolk, Virginia, 23435, United States

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Madison, Wisconsin, 53792, United States

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Milwaukee, Wisconsin, 53295, United States

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CABA, C1119ACN, Argentina

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CABA, C1425AGC, Argentina

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Ciudad de Buenos Aires, AR-CP 1221, Argentina

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Córdoba, 5000, Argentina

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Córdoba, X5003DCP, Argentina

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Mar del Plata, B7600, Argentina

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Mendoza, M5500, Argentina

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Rosario, S2000PBJ, Argentina

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San Miguel de Tucumán, 4000, Argentina

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San Nicolás, B2900DMH, Argentina

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San Vicente, 5006, Argentina

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Clayton, 3168, Australia

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Darlinghurst, 2010, Australia

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Epping, 3076, Australia

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Geelong, 3220, Australia

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Liverpool, 2170, Australia

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New Lambton Heights, 2305, Australia

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Perth, 6000, Australia

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Wollongong, 2500, Australia

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Woolloongabba, 4102, Australia

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Braunau am Inn, 5280, Austria

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Sankt Pölten, 3100, Austria

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Vienna, 1090, Austria

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Ghent, 9000, Belgium

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Liège, 4000, Belgium

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Mons, 7000, Belgium

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Pleven, 5800, Bulgaria

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Sofia, 1527, Bulgaria

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Sofia, 1618, Bulgaria

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Sofia, 1680, Bulgaria

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Sofia, 1709, Bulgaria

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Edmonton, Alberta, T6G 2C8, Canada

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North Vancouver, British Columbia, V7M 2H4, Canada

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Cambridge, Ontario, N1R 6V6, Canada

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Markham, Ontario, L3S 0A2, Canada

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Newmarket, Ontario, L3Y 2P6, Canada

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Ottawa, Ontario, K1H 7W9, Canada

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Scarborough Village, Ontario, M1B 4Z8, Canada

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Toronto, Ontario, M6G 1M2, Canada

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Waterloo, Ontario, N2T 0C1, Canada

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Chicoutimi, Quebec, G7H 7K9, Canada

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Saint-Jean-sur-Richelieu, Quebec, J3A 1J2, Canada

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Benešov, 256 01, Czechia

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Brandýs nad Labem, 250 01, Czechia

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Broumov, 55001, Czechia

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Louny, 440 01, Czechia

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Ostrava, 708 52, Czechia

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Příbram, 261 01, Czechia

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Uherské Hradiště, 68601, Czechia

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Aarhus, 8200, Denmark

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Herning, 7400, Denmark

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Holbæk, 4300, Denmark

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Bobigny, 93000, France

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Bordeaux, 33076, France

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Paris, 75013, France

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Paris, 75015, France

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Saint-Priest-en-Jarez, 42270, France

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Toulon, 83100, France

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Toulouse, 31059, France

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Tours, 37044, France

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Bad Homburg, 61348, Germany

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Bad Oeynhausen, 32545, Germany

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Berlin, 12203, Germany

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Berlin, 13347, Germany

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Dortmund, 44137, Germany

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Düsseldorf, 40225, Germany

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Elsterwerda, 04910, Germany

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Erlangen, 91054, Germany

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Essen, 45355, Germany

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Frankfurt, 60590, Germany

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Frankfurt, 60596, Germany

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Hanover, 30449, Germany

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Hanover, 30625, Germany

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Homburg, 66424, Germany

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Kaiserslautern, 67655, Germany

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Leipzig, 04103, Germany

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Mannheim, 68167, Germany

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Wermsdorf, 04779, Germany

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Balatonfüred, 8230, Hungary

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Budapest, 1115, Hungary

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Kalocsa, 6300, Hungary

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Kaposvár, 7400, Hungary

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Nyíregyháza, 4400, Hungary

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Pécs, 7623, Hungary

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Delhi, 110029, India

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Delhi, 110060, India

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Guntur, 522001, India

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Kanpur, 208002, India

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Kolkata, 700014, India

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Kolkata, 700020, India

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Mysuru, 570004, India

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Mysuru, 570015, India

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New Delhi, 110002, India

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New Delhi, 110017, India

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Surat, 395001, India

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Ashdod, 7747629, Israel

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Haifa, 3109601, Israel

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Petah Tikva, 49100, Israel

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Ramat Gan, 52621, Israel

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Rehovot, 76100, Israel

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Acquaviva delle Fonti, 70021, Italy

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Bologna, 40138, Italy

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Brescia, 25123, Italy

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Milan, 20122, Italy

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Milan, 20138, Italy

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Milan, 20149, Italy

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Pisa, 56126, Italy

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Roma, 00189, Italy

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Torino, 10126, Italy

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Udine, 33100, Italy

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Adachi-ku, 121-0815, Japan

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Chūōku, 103-0027, Japan

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Chūōku, 260-0804, Japan

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Kanazawa, 920-8530, Japan

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Koga-shi, 306-0232, Japan

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Kyoto, 607-8062, Japan

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Nagasaki, 850-8555, Japan

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Okayama, 700-0804, Japan

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Osaka, 559-0012, Japan

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Sapporo, 003-0026, Japan

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Tsuchiura-shi, 300-0062, Japan

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Yufu-shi, 879-5593, Japan

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Kajang, 43000, Malaysia

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Kota Bharu, 15586, Malaysia

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Kuching, 93586, Malaysia

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Malacca, 75400, Malaysia

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Muar town, 84000, Malaysia

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Sarawak Miri, 98000, Malaysia

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Seri Manjung, 32040, Malaysia

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Hoogeveen, 7909 AA, Netherlands

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Nijmegen, 6525 GA, Netherlands

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Utrecht, 3508 AB, Netherlands

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Bialystok, 15-540, Poland

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Bydgoszcz, 85-095, Poland

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Chrzanów, 32-500, Poland

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Gdansk, 80-214, Poland

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Gdynia, 81-338, Poland

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Krakow, 30-688, Poland

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Lodz, 91-002, Poland

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Poznan, 61-848, Poland

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Warsaw, 02-172, Poland

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Warsaw, 02-758, Poland

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Warsaw, 04-628, Poland

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Brezno, 977 01, Slovakia

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Košice, 04022, Slovakia

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Moldava nad Bodvou, 04501, Slovakia

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Prešov, 080 01, Slovakia

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Rimavská Sobota, 979 01, Slovakia

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Svidník, 08901, Slovakia

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Cape Town, 7500, South Africa

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Centurion, 0157, South Africa

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Claremont, 7708, South Africa

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Durban, 4001, South Africa

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Kwadwesi, 6201, South Africa

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Somerset West, 7130, South Africa

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Worcester, 6850, South Africa

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Bucheon-si, 420-717, South Korea

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Busan, 49241, South Korea

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Daejeon, 35015, South Korea

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Incheon, 21565, South Korea

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Seoul, 02841, South Korea

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Seoul, 03080, South Korea

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Seoul, 03722, South Korea

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Seoul, 04763, South Korea

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Seoul, 05505, South Korea

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Seoul, 07441, South Korea

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Seoul, 07804, South Korea

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Seoul, 08308, South Korea

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Barcelona, 08003, Spain

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Barcelona, 08036, Spain

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Ferrol, 15405, Spain

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Granada, 18014, Spain

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Madrid, 28040, Spain

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Madrid, 28041, Spain

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Majadahonda, 28222, Spain

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Seville, 41004, Spain

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Terrassa (Barcelona), 08221, Spain

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Gothenburg, 413 45, Sweden

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Uppsala, 75185, Sweden

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Kaohsiung City, 80756, Taiwan

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Kaohsiung City, 81362, Taiwan

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Taichung, 40201, Taiwan

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Taichung, 40447, Taiwan

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Taichung, 433004, Taiwan

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Taipei, 10002, Taiwan

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Taipei, 110, Taiwan

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Taipei, 11217, Taiwan

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Yung Kang City, 71044, Taiwan

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Bangkok, 10330, Thailand

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Bangkok, 10400, Thailand

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Bangkok, 10700, Thailand

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Chiang Mai, 50200, Thailand

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Hat Yai, 90110, Thailand

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Khon Kaen, 40002, Thailand

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Pathum Thani, 12120, Thailand

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Adana, 01060, Turkey (Türkiye)

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Ankara, 06530, Turkey (Türkiye)

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Bursa, 16059, Turkey (Türkiye)

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Dinar, 03400, Turkey (Türkiye)

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Istanbul, 34862, Turkey (Türkiye)

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Izmir, Turkey (Türkiye)

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Kütahya, 43100, Turkey (Türkiye)

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Odunpazari, 26080, Turkey (Türkiye)

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Bollington, SK10 5JH, United Kingdom

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Bristol, BS34 6BQ, United Kingdom

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Chesterfield, S40 4AA, United Kingdom

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Dundee, DD1 9SY, United Kingdom

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Glasgow, G51 4TF, United Kingdom

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Harrow, HA3 7LT, United Kingdom

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Hownslow, TW3 3LN, United Kingdom

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London, EC1M 6BQ, United Kingdom

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London, W6 7HY, United Kingdom

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Prescot, L35 5DR, United Kingdom

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Weston-super-Mare, BS24 7PR, United Kingdom

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Yate, BS37 4AX, United Kingdom

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Da Nang, 550000, Vietnam

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Hanoi, 100000, Vietnam

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Ho Chi Minh City, 700000, Vietnam

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Ho Chi Minh City, 70000, Vietnam

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Hochiminh City, 700000, Vietnam

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Related Publications (1)

  • Flack JM, Azizi M, Brown JM, Dwyer JP, Fronczek J, Jones ESW, Olsson DS, Perl S, Shibata H, Wang JG, Wilderang U, Wittes J, Williams B; BaxHTN Investigators. Efficacy and Safety of Baxdrostat in Uncontrolled and Resistant Hypertension. N Engl J Med. 2025 Oct 9;393(14):1363-1374. doi: 10.1056/NEJMoa2507109. Epub 2025 Aug 30.

MeSH Terms

Conditions

Hypertension

Condition Hierarchy (Ancestors)

Vascular DiseasesCardiovascular Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 6, 2023

First Posted

September 13, 2023

Study Start

November 22, 2023

Primary Completion

May 21, 2025

Study Completion

October 10, 2025

Last Updated

November 10, 2025

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data from AstraZeneca group of companies sponsored clinical trials via the request portal Vivli.org. All requests will be evaluated as per the AZ disclosure commitment: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure. "Yes", indicates that AZ are accepting requests for IPD, but this does not mean all requests will be approved.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
AstraZeneca will meet or exceed data availability as per the commitments made to the EFPIA/PhRMA Data-Sharing Principles. For details of our timelines, please refer to our disclosure commitment at: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
Access Criteria
When a request has been approved AstraZeneca will provide access to the anonymized individual patient-level data via secure research environment Vivli.org. A Signed Data Usage Agreement (non-negotiable contract for data accessors) must be in place before accessing requested information.
More information

Locations