NCT05929066

Brief Summary

The purpose of this study is to evaluate the efficacy and safety of retatrutide in participants who have obesity or overweight (J1I-MC-GZBJ master protocol) including subsets of participants who have knee osteoarthritis (OA) (J1I-MC-GOA1) or who have obstructive sleep apnea (OSA) (J1I-MC-GSA1). This study will last about 89 weeks and will include up to 24 visits. Addendum (2) is optional and available to approximately 500 participants to continue treatment with retatrutide for up to an additional 24 weeks.

Trial Health

67
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Trial has exceeded expected completion date
Strong global presence with extensive site network
Enrollment
2,300

participants targeted

Target at P75+ for phase_3 obesity

Timeline
Completed

Started Jul 2023

Typical duration for phase_3 obesity

Geographic Reach
12 countries

134 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 26, 2023

Completed
7 days until next milestone

First Posted

Study publicly available on registry

July 3, 2023

Completed
7 days until next milestone

Study Start

First participant enrolled

July 10, 2023

Completed
2.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2026

Completed
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2026

Completed
Last Updated

April 18, 2025

Status Verified

April 1, 2025

Enrollment Period

2.7 years

First QC Date

June 26, 2023

Last Update Submit

April 17, 2025

Conditions

Outcome Measures

Primary Outcomes (4)

  • Percent Change From Baseline in Body Weight

    Baseline, Week 80

  • Change from Baseline in the Western Ontario and McMaster Universities Osteoarthritis Index (WOMAC) Pain Subscale Score for GOA1 Subset

    Baseline, Week 80

  • Change from Baseline in Apnea-Hypopnea Index (AHI) Events Per Hour for GSA1 Subset

    Baseline, Week 80

  • Percent Change from Baseline in Body Weight to

    Baseline, Week 104

Secondary Outcomes (14)

  • Change from Baseline in Body Mass Index (BMI)

    Baseline, Week 80

  • Change from Baseline in Waist Circumference

    Baseline, Week 80

  • Change from Baseline in Systolic Blood Pressure (SBP)

    Baseline, Week 80

  • Percent Change form Baseline in Fasting Insulin

    Baseline, Week 80

  • Change from Baseline in HbA1c

    Baseline, Week 80

  • +9 more secondary outcomes

Study Arms (5)

Retatrutide Dose 1

EXPERIMENTAL

Participants will receive retatrutide subcutaneously (SC).

Drug: Retatrutide

Retatrutide Dose 2

EXPERIMENTAL

Participants will receive retatrutide SC.

Drug: Retatrutide

Retatrutide Dose 3

EXPERIMENTAL

Participants will receive retatrutide SC.

Drug: Retatrutide

Placebo

PLACEBO COMPARATOR

Participants will receive placebo.

Drug: Placebo

Retatrutide Extension Period

EXPERIMENTAL

Participants will receive retatrutide after the placebo-controlled 80 week treatment period for an additional 24 weeks.

Drug: Retatrutide

Interventions

Administered SC

Also known as: LY3437943
Retatrutide Dose 1Retatrutide Dose 2Retatrutide Dose 3Retatrutide Extension Period

Administered SC

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have body mass index (BMI) ≥30.0 kilograms per square meter (kg/m²), or ≥27.0 kg/m² with at least one of the following:
  • hypertension
  • dyslipidemia
  • obstructive sleep apnea, or
  • cardiovascular disease
  • History of of at least one unsuccessful dietary effort to reduce body weight
  • Have index knee pain for \>12 weeks prior to screening, and presence of index knee pain for \>15 days over the previous month
  • Have knee X-ray with moderate radiographic changes (Kellgren-Lawrence Grade 2 or 3) per central reading at screening
  • Currently meets American College of Rheumatology (ACR) Criteria (clinical and radiological) for OA.
  • Previously diagnosed with OSA
  • Have AHI ≥15 on polysomnography at screening (definition of moderate-to-severe OSA)
  • For participants not on positive airway pressure (PAP) therapy: unable or unwilling to use PAP therapy and have not used PAP for at least 4 weeks prior to screening.
  • If on PAP therapy, have been on PAP therapy for at least 3 consecutive months prior to screening, and willing to temporarily stop using PAP therapy for approximately 7 days prior to each of the sleep study (PSG) visits.
  • Have completed the final treatment visit of GZBJ Week 80.

You may not qualify if:

  • Have a self-reported or documented change in body weight \>5 kg (11 pounds) within 90 days.
  • Have taken weight loss drugs, including over-the-counter medications, within 90 days prior to screening.
  • Have a prior or planned surgical treatment for obesity.
  • Have diabetes mellitus.
  • Have family or personal history of medullary thyroid carcinoma (MTC) or multiple endocrine neoplasia syndrome type 2 (MEN-2)
  • Have had pancreatitis.
  • Have had steroid joint injections within 90 days of screening.
  • Have had other joint injections and procedures within 6 months of screening.
  • Have joint disease other than osteoarthritis.
  • Use stimulants (for example, modafinil, armodafinil, solriamfetol, pitolisant, amphetamine) less than 3 months prior to screening.
  • Use hypnotics, mirtazapine, opioids, trazodone, and zonisamide less than 3 months prior to screening.
  • Use a dental appliance or other device to treat OSA other than PAP therapy.
  • Have had study intervention discontinuation.
  • Have had permanent dose reduction.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (134)

Central Phoenix Medical Clinic

Phoenix, Arizona, 85020, United States

Location

Arizona Research Center

Phoenix, Arizona, 85053, United States

Location

Medical Investigations

Little Rock, Arkansas, 72211, United States

Location

Neuro-Pain Medical Center

Fresno, California, 93710, United States

Location

Valley Research

Fresno, California, 93720, United States

Location

Artemis Institute for Clinical Research

San Diego, California, 92103, United States

Location

University of Colorado Anschutz Medical Campus

Aurora, Colorado, 80045, United States

Location

Yale University School of Medicine

New Haven, Connecticut, 06519, United States

Location

Chase Medical Research, LLC

Waterbury, Connecticut, 06708, United States

Location

Teradan Clinical Trials, LLC

Brandon, Florida, 33511, United States

Location

Suncoast Research Group

Miami, Florida, 33135, United States

Location

New Horizon Research Center

Miami, Florida, 33165, United States

Location

Clinical Neuroscience Solutions

Orlando, Florida, 32801, United States

Location

Progressive Medical Research

Port Orange, Florida, 32127, United States

Location

NeuroTrials Research Inc

Atlanta, Georgia, 30328, United States

Location

North Georgia Clinical Research

Woodstock, Georgia, 30189, United States

Location

East-West Medical Research Institute

Honolulu, Hawaii, 96814, United States

Location

Northwestern University

Chicago, Illinois, 60611, United States

Location

Central Illinois Diabetes and Clinical Research a Division of Prairie Education and Research Cooperative

Springfield, Illinois, 62711, United States

Location

Brengle Family Medicine

Indianapolis, Indiana, 46260, United States

Location

Cotton O'Neil Diabetes & Endocrinology

Topeka, Kansas, 66606, United States

Location

MedVadis Research Corporation

Waltham, Massachusetts, 02451, United States

Location

Great Lakes Research Group, Inc.

Bay City, Michigan, 48706, United States

Location

StudyMetrix Research

City of Saint Peters, Missouri, 63303, United States

Location

Clinvest Research LLC

Springfield, Missouri, 65807, United States

Location

Palm Research Center Tenaya

Las Vegas, Nevada, 89128, United States

Location

Rochester Clinical Research, LLC

Rochester, New York, 14609, United States

Location

Carteret Medical Group

Morehead City, North Carolina, 28557, United States

Location

Trial Management Associates - Wilmington - Floral Parkway

Wilmington, North Carolina, 28403, United States

Location

Lillestol Research

Fargo, North Dakota, 58104, United States

Location

Altoona Center For Clinical Research

Duncansville, Pennsylvania, 16635, United States

Location

Tribe Clinical Research, LLC

Greenville, South Carolina, 29607, United States

Location

Tribe Clinical Research - Spartanburg

Spartanburg, South Carolina, 29301, United States

Location

Vanderbilt Health One Hundred Oaks

Nashville, Tennessee, 37204, United States

Location

FutureSearch Trials of Neurology

Austin, Texas, 78731, United States

Location

Juno Research

Houston, Texas, 77040, United States

Location

Advanced Research Institute

Ogden, Utah, 84405, United States

Location

Northwest Clinical Research Center

Bellevue, Washington, 98007, United States

Location

Rainier Clinical Research Center

Renton, Washington, 98057, United States

Location

Emeritus Research

Botany, New South Wales, 2019, Australia

Location

The AIM Centre / Hunter Diabetes Centre

Merewether, New South Wales, 2291, Australia

Location

Logan Hospital

Meadowbrook, Queensland, 4131, Australia

Location

Fusion Clinical Research

Adelaide, South Australia, 5000, Australia

Location

Nightingale Research

Adelaide, South Aust, 5000, Australia

Location

Emeritus Research

Camberwell, Victoria, 3124, Australia

Location

Barwon Health

Geelong, Victoria, 3220, Australia

Location

One Clinical Research

Nedlands, Western Australia, 6009, Australia

Location

CPCLIN

São Paulo, São Paulo, 01228-200, Brazil

Location

CPQuali Pesquisa Clínica

São Paulo, 01228-000, Brazil

Location

CEPIC - Centro Paulista de Investigação Clínica

São Paulo, 04266-010, Brazil

Location

Aggarwal and Associates Limited

Brampton, Ontario, L6T 0G1, Canada

Location

Dr. Steven V. Zizzo Medicine Professional Corporation

Hamilton, Ontario, L8J 0B6, Canada

Location

Wharton Medical Clinic

Hamilton, Ontario, L8L 5G8, Canada

Location

Your Research Network

Niagara Falls, Ontario, L2H 1H5, Canada

Location

Bluewater Clinical Research Group Inc.

Sarnia, Ontario, N7T 4X3, Canada

Location

Canadian Phase Onward

Toronto, Ontario, M3J 0K2, Canada

Location

Centre de Recherche Clinique de Laval

Laval, Quebec, H7T 2P5, Canada

Location

Clinique de médecine Urbaine du Quartier Latin

Montreal, Quebec, H2L 4E9, Canada

Location

C.I.C. Mauricie inc.

Trois-Rivières, Quebec, G8T 7A1, Canada

Location

Szegedi Tudományegyetem Szent-Györgyi Albert Klinikai Központ

Szeged, Csongrád megye, 6725, Hungary

Location

Regia Med Kft

Székesfehérvár, Fejér, 8000, Hungary

Location

Medifarma 98 Kft

Nyíregyháza, Nyíregyháza, 4400, Hungary

Location

DRC Gyógyszervizsgáló Központ

Balatonfüred, Veszprém megye, 8230, Hungary

Location

Óbudai Egészségügyi Centrum

Budapest, 1036, Hungary

Location

ClinDiab Kft.

Budapest, 1089, Hungary

Location

Debreceni Egyetem Klinikai Központ

Debrecen, 4031, Hungary

Location

Debreceni Egyetem Klinikai Kozpont

Debrecen, 4032, Hungary

Location

Endolife Speciality Hospitals

Guntur, Andhra Pradesh, 522001, India

Location

Avron Hospitals

Ahmedabad, Gujarat, 380013, India

Location

Surat Institute of Digestive Sciences Hospitals

Surat, Gujarat, 395002, India

Location

Karnataka Institute of Medical Sciences

Hubli, Karnataka, 580021, India

Location

Indian Institute of Diabetes

Thiruvananthapuram, Kerala, 695031, India

Location

Jothydev's Diabetes and Research Center

Trivandrum, Kerala, 695032, India

Location

Wockhardt Hospital - Mumbai Central

Mumbai, Maharashtra, 400011, India

Location

Deenanath Mangeshkar Hospital & Research Centre

Pune, Maharashtra, 411004, India

Location

Chellaram Diabetes Institute

Pune, Maharashtra, 411021, India

Location

Lifepoint Multispeciality Hospital

Pune, Maharashtra, 411057, India

Location

All India Institute of Medical Sciences

Bhubaneswar, Odisha, 751019, India

Location

Eternal Heart Care Center and Research Institute

Jaipur, Rajasthan, 302020, India

Location

Christian Medical College Vellore

Vellore, Tamil Nadu, 632004, India

Location

ILS Hospitals

Kolkata, West Benga, 700064, India

Location

Centro de Investigacion en Artritis y Osteoporosis SC

Mexicali, Estado de Baja California, 21200, Mexico

Location

Diseno y Planeacion en Investigacion Medica

Guadalajara, Jalisco, 44130, Mexico

Location

Clinica de Investigacion en Reumatologia y Obesidad S. C.

Guadalajara, Jalisco, 44650, Mexico

Location

Private Practice - Dr. Arechavaleta Granell Maria del Rosario

Guadalajara, Jalisco, 44670, Mexico

Location

Unidad de Investigación Clínica y Atención Médica HEPA

Guadalajara, Jalisco, 44670, Mexico

Location

RM Pharma Specialists

Mexico City, Mexico City, 03100, Mexico

Location

Clinica Omega

Mexico City, Mexico City, 06700, Mexico

Location

Instituto de Diabetes, Obesidad y Nutricion

Cuernavaca, Morelos, 62250, Mexico

Location

Unidad biomedica avanzada monterrey

Monterrey, Nuevo León, 64460, Mexico

Location

Hospital Universitario Dr. Jose Eleuterio Gonzalez

Monterrey, Nuevo León, 66460, Mexico

Location

EME RED Hospitalaria

Mérida, Yucatán, 97000, Mexico

Location

Kohler and Milstein Research S.A. de C.V.

Mérida, Yucatán, 97070, Mexico

Location

Centro de Atención e Investigación Clínica

Aguascalientes, 20119, Mexico

Location

Investigacion En Salud Y Metabolismo S.C / Nutricion Clinica / Unidad de Base de Datos

Chihuahua City, 31110, Mexico

Location

Arké SMO S.A de C.V

Veracruz, 91910, Mexico

Location

Centrum Zdrowia Metabolicznego Pawel Bogdanski

Poznan, Greater Poland Voivodeship, 60-589, Poland

Location

INTERCOR

Bydgoszcz, Kuyavian-Pomeranian Voivodeship, 85-605, Poland

Location

Private Practice - Dr. Robert Witek

Tarnów, Lesser Poland Voivodeship, 33-100, Poland

Location

CenterMed Lublin NZOZ

Lublin, Lublin Voivodeship, 20-044, Poland

Location

Gabinety TERPA

Lublin, Lublin Voivodeship, 20-333, Poland

Location

MICS Centrum Medyczne Warszawa

Warsaw, Masovian Voivodeship, 00-874, Poland

Location

Uniwersytecki Szpital Kliniczny w Białymstoku

Bialystok, Podlaskie Voivodeship, 15-276, Poland

Location

Centrum Badan Klinicznych PI-House sp. z o.o.

Gdansk, Pomeranian Voivodeship, 80-546, Poland

Location

NZOZ Salvia CM

Katowice, Silesian Voivodeship, 40-772, Poland

Location

Ambulatorium Sp. z o.o.

Elblag, Warmian-Masurian Voivodeship, 82-300, Poland

Location

Centrum Kliniczno-Badawcze

Elblag, Warmian-Masurian Voivodeship, 82-300, Poland

Location

Specjalistyczna Praktyka Lekarska Diabetologia, Leczenie Cukrzycy i Otylosci

Kielce, Świętokrzyskie Voivodeship, 25-355, Poland

Location

Ponce Medical School Foundation Inc.

Ponce, 00716, Puerto Rico

Location

Diabdana

Oradea, Bihor County, 410147, Romania

Location

C.M.D.T.A. Neomed

Brasov, Brașov County, 500283, Romania

Location

Hightech Medical Services SRL-Centrul pentru Studiul Metabolismului

Bucharest, București, 011053, Romania

Location

Gama Diamed

Mangalia, Constanța County, 905500, Romania

Location

Cabinet Medical Dr.Geru

Timișoara, Timiș County, 300288, Romania

Location

SC Minimed SRL

Bacau, 600274, Romania

Location

Diamed Obesity

Galați, 800291, Romania

Location

Centrul Medical Consultmed

Iași, 700547, Romania

Location

Clinica Korall

Satu Mare, 440055, Romania

Location

Policlinica Astra Sibiu

Sibiu, 550371, Romania

Location

CHUAC-Complejo Hospitalario Universitario A Coruña

A Coruña, A Coruña [La Coruña], 15006, Spain

Location

Complejo Hospitalario Universitario de Ferrol (CHUF)- Hospital Naval

Ferrol, A Coruña [La Coruña], 15405, Spain

Location

Hospital Universitari Vall d'Hebron

Barcelona, Barcelona [Barcelona], 08035, Spain

Location

Hospital Universitario Marqués de Valdecilla

Santander, Cantabria, 39008, Spain

Location

Hospital General Universitario de Valencia

Valencia, Valenciana, Comunitat, 46014, Spain

Location

Clínica nuevas Tecnologías en Diabetes y Endocrinología (NTDE)

Seville, 41003, Spain

Location

Rowden Surgery

Chippenham, England, SN15 2SB, United Kingdom

Location

Layton Medical Centre

Blackpool, Lancashire, FY3 7EN, United Kingdom

Location

Leicester General Hospital

Leicester, Leicestershire, LE5 4PW, United Kingdom

Location

Panthera Biopartners - North London

Enfield, London, City of, EN3 4GS, United Kingdom

Location

Glasgow Royal Infirmary

Glasgow, Scotland, G31 2ER, United Kingdom

Location

Heartlands Hospital

Birmingham, B9 5SS, United Kingdom

Location

Aintree University Hospital NHS Foundation Trust

Liverpool, L9 7AL, United Kingdom

Location

St Clare Medical Centre

Penzance, TR18 3DX, United Kingdom

Location

Panthera Biopartners - Sheffield

Sheffield, S2 5FX, United Kingdom

Location

Related Links

MeSH Terms

Conditions

ObesityOverweightOsteoarthritis, KneeSleep Apnea, Obstructive

Interventions

retatrutide

Condition Hierarchy (Ancestors)

OvernutritionNutrition DisordersNutritional and Metabolic DiseasesBody WeightSigns and SymptomsPathological Conditions, Signs and SymptomsOsteoarthritisArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic DiseasesSleep Apnea SyndromesApneaRespiration DisordersRespiratory Tract DiseasesSleep Disorders, IntrinsicDyssomniasSleep Wake DisordersNervous System Diseases

Study Officials

  • Call 1-877-CTLILLY (1-877-285-4559 or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern Time (UTC/GMT - 5 hours, EST)

    Eli Lilly and Company

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 26, 2023

First Posted

July 3, 2023

Study Start

July 10, 2023

Primary Completion

April 1, 2026

Study Completion

May 1, 2026

Last Updated

April 18, 2025

Record last verified: 2025-04

Data Sharing

IPD Sharing
Will share

Anonymized individual patient level data will be provided in a secure access environment upon approval of a research proposal and a signed data sharing agreement.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
Data are available 6 months after the primary publication and approval of the indication studied in the US and European Union (EU), whichever is later. Data will be indefinitely available for requesting
Access Criteria
A research proposal must be approved by an independent review panel and researchers must sign a data sharing agreement.
More information

Locations