NCT04765657

Brief Summary

A multicenter study to evaluate safety and efficacy of inclisiran in Asian patients with ASCVD or ASCVD high risk and elevated LDL-C

Trial Health

78
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
345

participants targeted

Target at P50-P75 for phase_3

Timeline
9mo left

Started Mar 2021

Longer than P75 for phase_3

Geographic Reach
4 countries

45 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress88%
Mar 2021Dec 2026

First Submitted

Initial submission to the registry

February 5, 2021

Completed
16 days until next milestone

First Posted

Study publicly available on registry

February 21, 2021

Completed
8 days until next milestone

Study Start

First participant enrolled

March 1, 2021

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 9, 2022

Completed
4.6 years until next milestone

Study Completion

Last participant's last visit for all outcomes

December 28, 2026

Expected
Last Updated

December 30, 2025

Status Verified

December 1, 2025

Enrollment Period

1.3 years

First QC Date

February 5, 2021

Last Update Submit

December 22, 2025

Conditions

Keywords

inclisiransiRNAdyslipidemiaKJX839

Outcome Measures

Primary Outcomes (2)

  • Core: Percentage change in low- density lipoprotein cholesterol (LDL-C)

    Superiority of inclisiran compared to placebo in reducing LDL-C from baseline to Day 330

    Baseline, Day 330

  • Extension: Number of participants with Adverse Events

    Evaluation of the safety and tolerability of inclisiran, treatment emergent Adverse events and Serious Adverse Events

    Day 360 until study completion, an average of 3 years

Secondary Outcomes (10)

  • Core: Time adjusted percentage change in LDL-C

    From baseline after Day 90 and up to Day 360

  • Core: Absolute change in LDL-C

    From baseline to Day 330

  • Core: Time adjusted absolute change in LDL-C

    From baseline after Day 90 and up to Day 360

  • Core: Percentage change in PCSK9

    From baseline to Day 330

  • Core: Absolute change in PCSK9

    From baseline to Day 330

  • +5 more secondary outcomes

Study Arms (2)

inclisiran sodium 300 mg

EXPERIMENTAL

Subcutaneous injection

Drug: inclisiran sodium

Placebo

PLACEBO COMPARATOR

Subcutaneous injection

Drug: Placebo

Interventions

Subcutaneously injected on Day 1, 90 and 270 (Core Part). Subcutaneously injected on Day 360 and every 6 months thereafter until EOS visit (Extension Part)

Also known as: KJX839
inclisiran sodium 300 mg

Subcutaneously injected on Day 1, 90, and 270.

Placebo

Eligibility Criteria

Age18 Years - 100 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • At screening participants with: ASCVD (including acute coronary syndrome (ACS), stable coronary heart disease, post revascularization, ischemic cardiomyopathy, ischemic stroke, transient ischemic attack (TIA), and peripheral atherosclerosis) and Serum LDL-C ≥1.8 mmol/L (≥70 mg/dL) OR ASCVD high risk (LDL-C ≥4.9 mmol/L, diabetes, high 10-year ASCVD risk assessed by Chinese ASCVD Risk Assessment Flow Chart , or high risk per local guidelines with a target LDL-C of \<100 mg/dL) and Serum LDL-C ≥2.6 mmol/L (≥100 mg/dL)
  • Fasting triglyceride \< 400 mg/dL (\< 4.52 mmol/L) at screening.
  • Participants on statins should be receiving a maximally tolerated dose . Maximum tolerated dose is defined as the maximum dose of statin that can be taken on a regular basis without intolerable AE. Intolerance to any dose of statin must be documented as historical AEs attributed to the statin in question on the source documentation and on the Medical history page of the eCRF
  • Participants not receiving statin must have a documented evidence of intolerance to all doses of at least 2 different statins(or the corresponding local definition of complete intolerance to statins)
  • Participants following lifestyle modification should be on the therapy of LDL-C lowering (such as statin monotherapy, or statin incombination with ezetimibe) with a stable dose for ≥30 days before screening and have no planned medication or dose change during study participation.
  • Participants are willing and able to give informed consent before initiation of any study related procedures and willing to comply with all required study procedures.

You may not qualify if:

  • New York Heart Association (NYHA) class IV heart failure or last known left ventricular ejection fraction \<25%.
  • Cardiac arrhythmia with clinical significance within 3 months prior to randomization that is not controlled by medication or via ablation.
  • Major adverse cardiovascular event within 3 months prior to randomization.
  • Uncontrolled severe hypertension: systolic blood pressure ≥160 mmHg or diastolic blood pressure ≥100 mmHg prior to randomization despite antihypertensive therapy.
  • Calculated glomerular filtration rate ≤30 mL/min by estimated glomerular filtration rate (eGFR) using standardized clinical methodology.
  • Severe concomitant non-cardiovascular disease that carries the risk of reducing life expectancy to less than 2 years.
  • History of malignancy that required surgery (excluding local and wide-local excision), radiation therapy and/or systemic therapy during the three years prior to randomization.
  • Barrier method: Condom or Occlusive cap (e.g. diaphragm or cervical/vault caps).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (45)

Novartis Investigative Site

Lanzhou, Gansu, 730030, China

Location

Novartis Investigative Site

Foshan, Guangdong, 528000, China

Location

Novartis Investigative Site

Guangzhou, Guangdong, 510080, China

Location

Novartis Investigative Site

Shijiazhuang, Hebei, 050000, China

Location

Novartis Investigative Site

Baotou, Inner Mongolia, 014040, China

Location

Novartis Investigative Site

Hohhot, Inner Mongolia, 010017, China

Location

Novartis Investigative Site

Nanjing, Jiangsu, 210008, China

Location

Novartis Investigative Site

Nanjing, Jiangsu, 211166, China

Location

Novartis Investigative Site

Nantong, Jiangsu, 226000, China

Location

Novartis Investigative Site

Suzhou, Jiangsu, 215004, China

Location

Novartis Investigative Site

Xuzhou, Jiangsu, 221003, China

Location

Novartis Investigative Site

Changchun, Jilin, 130000, China

Location

Novartis Investigative Site

Changchun, Jilin, 130021, China

Location

Novartis Investigative Site

Jinan, Shandong, 250013, China

Location

Novartis Investigative Site

Zhujing, Shanghai Municipality, 201508, China

Location

Novartis Investigative Site

Taiyuan, Shanxi, 030002, China

Location

Novartis Investigative Site

Xian, Shanxi, 710061, China

Location

Novartis Investigative Site

Tianjin, Tianjin Municipality, 300121, China

Location

Novartis Investigative Site

Hangzhou, Zhejiang, 310014, China

Location

Novartis Investigative Site

Beijing, 100034, China

Location

Novartis Investigative Site

Beijing, 100039, China

Location

Novartis Investigative Site

Beijing, 100050, China

Location

Novartis Investigative Site

Beijing, 100191, China

Location

Novartis Investigative Site

Shanghai, 200032, China

Location

Novartis Investigative Site

Shanghai, 200040, China

Location

Novartis Investigative Site

Shanghai, 200080, China

Location

Novartis Investigative Site

Shanghai, 200120, China

Location

Novartis Investigative Site

Tianjin, 300052, China

Location

Novartis Investigative Site

Tianjin, 300140, China

Location

Novartis Investigative Site

Xiamen, 361004, China

Location

Novartis Investigative Site

Singapore, 119074, Singapore

Location

Novartis Investigative Site

Singapore, 169609, Singapore

Location

Novartis Investigative Site

Wŏnju, Gangwon-do, 26427, South Korea

Location

Novartis Investigative Site

Incheon, Korea, 405 760, South Korea

Location

Novartis Investigative Site

Seoul, Korea, 02841, South Korea

Location

Novartis Investigative Site

Seoul, Korea, 03080, South Korea

Location

Novartis Investigative Site

Seoul, Seoul, 06351, South Korea

Location

Novartis Investigative Site

Seoul, South Korea, 110-746, South Korea

Location

Novartis Investigative Site

Gwangju, 61469, South Korea

Location

Novartis Investigative Site

Seoul, 03722, South Korea

Location

Novartis Investigative Site

Seoul, 05505, South Korea

Location

Novartis Investigative Site

Kaohsiung City, 80756, Taiwan

Location

Novartis Investigative Site

Taipei, 10002, Taiwan

Location

Novartis Investigative Site

Taipei, 11217, Taiwan

Location

Novartis Investigative Site

Taipei, 11220, Taiwan

Location

Related Publications (1)

  • Huo Y, Lesogor A, Lee CW, Chiang CE, Mena-Madrazo J, Poh KK, Jeong MH, Maheux P, Zhang M, Wei S, Han Y, Li Y. Efficacy and Safety of Inclisiran in Asian Patients: Results From ORION-18. JACC Asia. 2023 Nov 14;4(2):123-134. doi: 10.1016/j.jacasi.2023.09.006. eCollection 2024 Feb.

MeSH Terms

Conditions

HypercholesterolemiaDyslipidemias

Condition Hierarchy (Ancestors)

HyperlipidemiasLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 5, 2021

First Posted

February 21, 2021

Study Start

March 1, 2021

Primary Completion

June 9, 2022

Study Completion (Estimated)

December 28, 2026

Last Updated

December 30, 2025

Record last verified: 2025-12

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with applicable laws and regulations. This trial data availability is according to the criteria and process described on www.clinicalstudydatarequest.com

Locations