NCT04595370

Brief Summary

The purpose of the study is to evaluate the efficacy and safety of AZD9977 in combination with dapagliflozin compared with dapagliflozin alone and to assess the dose-response relationship, dapagliflozin alone and 3 doses of AZD9977 combined with dapagliflozin on urinary albumin to creatinine ratio (UACR). The study will be conducted in participants with heart failure (HF) with left ventricular ejection fraction (LVEF \[below 60%\]) and chronic kidney disease (CKD) with estimated glomerular filtration rate (eGFR \[between ≥ 20 and ≤ 60 mL/min/1.73 m\^2, with at least 20% of participants with eGFR ≥ 20 to \<30 mL/min/1.73\^2 and a maximum of 35% of participants with eGFR ≥ 45 mL/min/1.73 m\^2\]).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
153

participants targeted

Target at P50-P75 for phase_2 heart-failure

Timeline
Completed

Started Jan 2021

Typical duration for phase_2 heart-failure

Geographic Reach
22 countries

156 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 14, 2020

Completed
6 days until next milestone

First Posted

Study publicly available on registry

October 20, 2020

Completed
3 months until next milestone

Study Start

First participant enrolled

January 26, 2021

Completed
2.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 22, 2023

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 22, 2023

Completed
1.2 years until next milestone

Results Posted

Study results publicly available

November 19, 2024

Completed
Last Updated

November 19, 2024

Status Verified

October 1, 2024

Enrollment Period

2.7 years

First QC Date

October 14, 2020

Results QC Date

September 20, 2024

Last Update Submit

October 28, 2024

Conditions

Keywords

Heart FailureType 2 diabetes mellitusDiabetic kidney diseaseChronic kidney diseaseMineralocorticoid receptor modulatorSodium-glucose co-transporter-2 inhibitorAZD9977DapagliflozinUrinary albumin creatinine ratio

Outcome Measures

Primary Outcomes (1)

  • Percent Change From Baseline in Urinary Albumin to Creatinine Ratio (UACR) at Week 12

    The effect of AZD9977 in combination with dapagliflozin compared with dapagliflozin alone on UACR assessed. Urine samples were collected for the analysis of UACR. UACR (milligrams per gram \[mg/g\]) was calculated as 10 x urine albumin (mg per deciliter \[mg/dL\])/urine creatinine (g/dL). Change from baseline in UACR at the end of 12 weeks of study treatment was calculated as the average of the UACR values at Week 12 and was analyzed by a mixed-effects model for repeated measures (MMRM). Due to early removal of arms (AZD9977 150 mg monotherapy and Placebo), the study objectives were revised and the MMRM analysis included the 4 remaining arms (AZD9977 15 mg + Dapagliflozin, AZD9977 50 mg + Dapagliflozin, AZD9977 150 mg + Dapagliflozin, and Dapagliflozin 10 mg). Since 2 arms were removed from the study resulting in fewer participants only descriptive statistics are shown for those two arms without formal comparison.

    Baseline (Day 1) to Week 12

Secondary Outcomes (6)

  • Percent Change From Baseline in Urinary Albumin to Creatinine Ratio (UACR) at 12 Weeks to Assess Dose-Response Relationship

    Baseline (Day 1) to Week 12

  • Number of Participants With Adverse Events (AEs)

    From baseline (Day 1) until Day 113

  • Change From Baseline in Serum Potassium (K+)

    Baseline (Day 1) and Week 12

  • Absolute Value of Serum Potassium Over Time

    Baseline (Day 1) and Week 12

  • Change From Baseline in Estimated Glomerular Filtration Rate (eGFR)

    Baseline (Day 1) and Week 12

  • +1 more secondary outcomes

Study Arms (4)

AZD9977 Dose A + dapagliflozin 10 mg

EXPERIMENTAL

Participants will receive once daily oral dose A of AZD9977 and 10 mg dapagliflozin for 12 weeks.

Drug: AZD9977Drug: Dapagliflozin

AZD9977 Dose B + dapagliflozin 10 mg

EXPERIMENTAL

Participants will receive once daily oral dose B of AZD9977 and 10 mg dapagliflozin for 12 weeks.

Drug: AZD9977Drug: Dapagliflozin

AZD9977 Dose C + dapagliflozin 10 mg

EXPERIMENTAL

Participants will receive once daily oral dose C of AZD9977 and 10 mg dapagliflozin for 12 weeks.

Drug: AZD9977Drug: Dapagliflozin

Dapagliflozin 10 mg

EXPERIMENTAL

Participants will receive once daily oral dose of dapagliflozin 10 mg alone for 12 weeks.

Drug: Dapagliflozin

Interventions

Participants will receive AZD9977 as per the arms they are randomized.

AZD9977 Dose A + dapagliflozin 10 mgAZD9977 Dose B + dapagliflozin 10 mgAZD9977 Dose C + dapagliflozin 10 mg

Participants will receive dapagliflozin as per the arms they are randomized.

AZD9977 Dose A + dapagliflozin 10 mgAZD9977 Dose B + dapagliflozin 10 mgAZD9977 Dose C + dapagliflozin 10 mgDapagliflozin 10 mg

Eligibility Criteria

Age21 Years - 130 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants are included in the study if any of the following criteria apply:
  • Documented diagnosis of stable symptomatic HF (New York Heart Association class II-III) at screening, and a medical history of typical symptoms and signs of HF in those who are currently receiving loop diuretic treatment
  • Left ventricular ejection fraction \<60% documented by the most recent echocardiogram or cardiac magnetic resonance imaging within the last 12 months prior to screening
  • Stable background treatment for HF, hypertension, diabetes mellitus or renal disease according to guidelines
  • N-terminal-pro-brain natriuretic peptide (NT proBNP) ≥300 pg/mL for participants with sinus rhythm at screening; and NT proBNP ≥600 pg/mL for participants with atrial fibrillation/flutter at screening
  • The eGFR ≥30 and ≤60 mL/min/1.73\^2 (by CKD- EPI formula) and UACR ≥30 mg/g (3 mg/mmol) and \<3000 mg/g (300 mg/mmol)
  • Body mass index less than 40 kg/m\^2
  • Serum/plasma K+ level ≥ 3.5 and \< 5.0 mmol/L within 10 days prior to randomization
  • Serum/ plasma Na+ level within normal reference values within 10 days prior to randomization
  • Systolic blood pressure should be at protocol defined range at randomization (Visit 3), with no change to antihypertensive treatments in previous 3 weeks
  • Male or female of non-childbearing potential
  • All participants must follow protocol defined contraceptives procedures

You may not qualify if:

  • Participants are excluded from the study if any of the following criteria apply:
  • Primary glomerulopathy, vasculitic renal disease, prior dialysis or unstable rapidly progressing renal disease, autosomal dominant or autosomal recessive polycystic kidney disease, lupus nephritis or anti-neutrophil cytoplasm antibody-associated vasculitis
  • Participants with currently decompensated HF requiring hospitalization for optimization of HF treatment and are not on stable HF therapy at the time of enrollment
  • HF due to cardiomyopathies
  • High output HF (e.g., due to hyperthyroidism or Paget's disease)
  • HF due to pericardial disease, congenital heart disease or clinically significant uncorrected primary cardiac valvular disease or planned cardiac valve repair/replacement
  • Participants with uncontrolled diabetes mellitus (Glycated hemoglobin \>10%)
  • Participants with Type 1 diabetes mellitus
  • Intermittent or persistent 2nd or 3rd degree atrioventricular block, sinus node dysfunction with clinically significant bradycardia or sinus pauses, not treated with a pacemaker
  • History of any life-threatening cardiac dysrhythmia or uncontrolled ventricular rate in participants with atrial fibrillation or atrial flutter
  • Acute coronary syndrome and/or elective/non-elective percutaneous cardiac interventions (within 3 months) prior to randomisation or is planned to undergo any of these procedures during the study
  • Any major cardiovascular (eg, open chest, coronary artery bypass grafting or valvular repair/replacement) or major non-cardiovascular surgery within 3 months prior to randomisation or is planned to undergo any cardiovascular surgery during the study
  • Heart transplantation or left ventricular assist device at any time or if these are planned
  • Kidney or any organ transplantation or if these are planned
  • Medical conditions associated with development of hyperkalaemia (Addison's disease )
  • +8 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (156)

Research Site

Beverly Hills, California, 90211, United States

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Fountain Valley, California, 92708, United States

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Northridge, California, 91324, United States

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South Gate, California, 90280, United States

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Hialeah, Florida, 33016, United States

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Homestead, Florida, 33032, United States

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Jacksonville, Florida, 32216, United States

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Miami, Florida, 33155, United States

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Ocala, Florida, 34474, United States

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Tampa, Florida, 33603, United States

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Augusta, Georgia, 30904, United States

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Columbus, Georgia, 31904, United States

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Baltimore, Maryland, 21287, United States

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Methuen, Massachusetts, 01844, United States

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St Louis, Missouri, 63136, United States

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The Bronx, New York, 10455, United States

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New Bern, North Carolina, 28562, United States

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Rapid City, South Dakota, 57701, United States

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Memphis, Tennessee, 38119, United States

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Houston, Texas, 77087, United States

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Houston, Texas, 77099, United States

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Kingwood, Texas, 77339, United States

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McKinney, Texas, 75069, United States

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San Antonio, Texas, 78207, United States

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Sherman, Texas, 75092, United States

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Webster, Texas, 77598, United States

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Roeselare, 8800, Belgium

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Pleven, 5800, Bulgaria

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Plovdiv, 1606, Bulgaria

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Plovdiv, 4002, Bulgaria

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Plovdiv, 4003, Bulgaria

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Sofia, 1233, Bulgaria

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Sofia, 1309, Bulgaria

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Sofia, 1431, Bulgaria

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Sofia, 1510, Bulgaria

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Sofia, 1784, Bulgaria

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Veliko Tarnovo, 5000, Bulgaria

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Peterborough, Ontario, K9J 0B2, Canada

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Toronto, Ontario, M4N 3M5, Canada

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Montreal, Quebec, H2X 0A9, Canada

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Québec, Quebec, G1R 2J6, Canada

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Pardubice, 532 03, Czechia

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Prague, 120 00, Czechia

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Prague, 158 00, Czechia

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Uherské Hradiště, 68601, Czechia

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Aarhus, 8200, Denmark

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Herlev, 2730, Denmark

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Svendborg, 5700, Denmark

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Dresden, 1307, Germany

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Frankfurt, 60313, Germany

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Jena, 07747, Germany

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Leipzig, 04103, Germany

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Balatonfüred, 8230, Hungary

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Budapest, 1036, Hungary

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Budapest, 1122, Hungary

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Debrecen, 4032, Hungary

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Miskolc, 3530, Hungary

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Orosháza, H-5900, Hungary

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Ahmedabad, 382421, India

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Chennai, 600081, India

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Kolkata, 700020, India

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Pune, 411011, India

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Roma, 00168, Italy

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Chūōku, 103-0027, Japan

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Hamada-shi, 697-8511, Japan

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Hamamatsu, 430-0929, Japan

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Hanyu-shi, 348-8505, Japan

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Itabashi-ku, 173-8610, Japan

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Kasugai-shi, 487-0016, Japan

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Kawaguchi, 333-0842, Japan

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Kishiwada-shi, 596-8522, Japan

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Kobe, 650-0047, Japan

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Kobe, 654-0155, Japan

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Matsudo-Shi, 271-0077, Japan

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Matsumoto-shi, 390-8621, Japan

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Ono, 675-1392, Japan

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Osaka, 530-0001, Japan

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Sapporo, 006-0811, Japan

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Sayama, 350-1305, Japan

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Takasago-shi, 676-0812, Japan

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Takasaki-shi, 370-0829, Japan

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Ueda-shi, 386-8610, Japan

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Yokohama, 231-8682, Japan

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Yokohama, 234-8503, Japan

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Yokohama, 236-0004, Japan

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Kaunas, 50177, Lithuania

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Klaipėda, 92231, Lithuania

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Šiauliai, LT-76231, Lithuania

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Vilnius, 08661, Lithuania

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Gdansk, 80-382, Poland

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Gdansk, 80-952, Poland

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Katowice, 40-040, Poland

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Lodz, 90-127, Poland

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Lodz, 92-213, Poland

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Lodz, 95-513, Poland

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Lublin, 20-709, Poland

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Ostrowiec Świętokrzyski, 27-400, Poland

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Oświęcim, 32-600, Poland

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Oława, 55-200, Poland

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Pabianice, 95-200, Poland

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Poznan, 60-702, Poland

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Skorzewo, 60-185, Poland

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Sopot, 81-717, Poland

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Szczecin, 71-434, Poland

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Torun, 87-100, Poland

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Warsaw, 01-192, Poland

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Kazan', 420101, Russia

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Kazan, Tatarstan, 420012, Russia

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Kemerovo, 650002, Russia

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Moscow, 111539, Russia

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Moscow, 121552, Russia

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Moscow, 125284, Russia

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Moscow, 129110, Russia

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Saint Petersburg, 195067, Russia

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Saint Petersburg, 195257, Russia

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Saint Petersburg, 197022, Russia

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Saint Petersburg, 197089, Russia

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Banská Bystrica, 974 01, Slovakia

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Brezno, 977 01, Slovakia

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Lučenec, 984 01, Slovakia

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Prešov, 080 01, Slovakia

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Svidník, 08901, Slovakia

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Trenčín, 911 01, Slovakia

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Busan, 49201, South Korea

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Gangwon-do, 26426, South Korea

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Seongnam-si, 463-707, South Korea

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Seoul, 03080, South Korea

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Seoul, 06351, South Korea

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Seoul, 06591, South Korea

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A Coruña, 15006, Spain

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Barcelona, 08003, Spain

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El Palmar, 30120, Spain

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Madrid, 28041, Spain

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Málaga, 29010, Spain

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Santiago(A Coruña), 15706, Spain

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Seville, 41009, Spain

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Valencia, 46010, Spain

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Valencia, 46026, Spain

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Gothenburg, 413 46, Sweden

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Stockholm, 14186, Sweden

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Stockholm, 18288, Sweden

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Uppsala, 75185, Sweden

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Kaohsiung City, 80756, Taiwan

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Taichung, 40201, Taiwan

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Taipei, 10449, Taiwan

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Taipei, 110, Taiwan

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Taipei, 11217, Taiwan

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Bangkok, 10400, Thailand

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Bangkok, 10700, Thailand

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Chaingmai, 50200, Thailand

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Khon Kaen, 40002, Thailand

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Adana, 01060, Turkey (Türkiye)

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Kocaeli, 41380, Turkey (Türkiye)

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Ivano-Frankivsk, 76018, Ukraine

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Kharkiv, 61039, Ukraine

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Kyiv, 02091, Ukraine

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Related Links

MeSH Terms

Conditions

Heart FailureRenal Insufficiency, ChronicDiabetes Mellitus, Type 2Diabetic Nephropathies

Interventions

AZD9977dapagliflozin

Condition Hierarchy (Ancestors)

Heart DiseasesCardiovascular DiseasesRenal InsufficiencyKidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and SymptomsDiabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesDiabetes Complications

Limitations and Caveats

Enrolment stopped early because of slow recruitment. Therefore, pre-specified sample size of 500 and planned statistical power were not achieved. Nine subjects were excluded from analysis due to site misconduct and GCP non-compliance.

Results Point of Contact

Title
Global Clinical Lead
Organization
AstraZeneca

Study Officials

  • John McMurray

    University of Glasgow, United Kingdom

    PRINCIPAL INVESTIGATOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Model Details: Participants who meet the eligibility criteria will be randomized to one of the following treatment group: 1. AZD9977 Dose A + dapagliflozin 10 mg 2. AZD9977 Dose B + dapagliflozin 10 mg 3. AZD9977 Dose C + dapagliflozin 10 mg 4. Dapagliflozin 10 mg
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 14, 2020

First Posted

October 20, 2020

Study Start

January 26, 2021

Primary Completion

September 22, 2023

Study Completion

September 22, 2023

Last Updated

November 19, 2024

Results First Posted

November 19, 2024

Record last verified: 2024-10

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data from AstraZeneca group of companies sponsored clinical trials via the request portal. All requests will be evaluated as per the AZ disclosure commitment: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure. Yes, indicates that AZ are accepting requests for IPD, but this does not mean all requests will be shared.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
AstraZeneca will meet or exceed data availability as per the commitments made to the EFPIA Pharma Data Sharing Principles. For details of our timelines, please rerefer to our disclosure commitment at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
Access Criteria
When a request has been approved AstraZeneca will provide access to the de-identified individual patient-level data in an approved sponsored tool . Signed Data Sharing Agreement (non-negotiable contract for data accessors) must be in place before accessing requested information. Additionally, all users will need to accept the terms and conditions of the SAS MSE to gain access. For additional details, please review the Disclosure Statements at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
More information

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