NCT04411641

Brief Summary

Primary Objective: To determine the efficacy of SAR442168 compared to placebo in delaying disability progression in NRSPMS Secondary Objective: To evaluate efficacy of SAR442168 compared to placebo on clinical endpoints, magnetic resonance imaging (MRI) lesions, cognitive performance, physical function, and quality of life To evaluate safety and tolerability of SAR442168 To evaluate population pharmacokinetics (PK) of SAR442168 and relevant metabolites in NRSPMS and its relationship to efficacy and safety To evaluate pharmacodynamics (PD) of SAR442168

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,131

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Sep 2020

Typical duration for phase_3

Geographic Reach
29 countries

298 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

May 28, 2020

Completed
5 days until next milestone

First Posted

Study publicly available on registry

June 2, 2020

Completed
4 months until next milestone

Study Start

First participant enrolled

September 24, 2020

Completed
3.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 29, 2024

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 29, 2024

Completed
10 months until next milestone

Results Posted

Study results publicly available

June 18, 2025

Completed
Last Updated

July 2, 2025

Status Verified

June 1, 2025

Enrollment Period

3.9 years

First QC Date

May 28, 2020

Results QC Date

June 3, 2025

Last Update Submit

July 1, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Time to Onset of 6-Month Confirmed Disability Progression (CDP) as Assessed by Expanded Disability Status Scale (EDSS)

    The EDSS is a disability scale that assesses the following 7 functional domains: visual, brainstem, pyramidal \[motor\], cerebellar \[coordination\], sensory, cerebral, and bowel/bladder. The total EDSS ranges from 0 (normal) to 10 (death due to multiple sclerosis \[MS\]) (0.5 increments from 1-10; next increase after 0 is 1). Higher scores indicated increased disability. Time to onset of 6-month CDP was defined as the time from randomization to the onset of a sustained increase from baseline in EDSS score of \>=1.0 point from the baseline EDSS score when the baseline score was \<=5.0 or of \>=0.5 points when the baseline EDSS score was \>5.0 confirmed after a minimum 6-month interval.

    Baseline (Day 1) up to approximately 47 months

Secondary Outcomes (16)

  • Time to Onset of 3-month Confirmed Disability Progression as Assessed by Expanded Disability Status Scale

    Baseline (Day 1) up to approximately 47 months

  • Mean Number of New and/or Enlarging T2-hyperintense Lesions Per Year

    Baseline (Day 1) up to approximately 47 months

  • Time to Onset of Sustained 20% Increase in the 9-hole Peg Test (HPT) for at Least 3 Months

    Baseline (Day 1) up to approximately 47 months

  • Time to Onset of Sustained 20% Increase in the Timed 25-foot Walk (T25-FW) for at Least 3 Months

    Baseline (Day 1) up to approximately 47 months

  • Time to Onset of 6-month Confirmed Disability Improvement (CDI) as Assessed by Expanded Disability Status Scale

    Baseline (Day 1) up to approximately 47 months

  • +11 more secondary outcomes

Study Arms (2)

SAR442168

EXPERIMENTAL

60 mg of oral SAR442168 once daily

Drug: Tolebrutinib

Placebo

PLACEBO COMPARATOR

Placebo tablet to match SAR442168 once daily

Drug: Placebo to match Tolebrutinib

Interventions

Pharmaceutical form: Film-coated tablet Route of administration: Oral

Also known as: SAR442168
SAR442168

Pharmaceutical form: Film-coated tablet Route of administration: Oral

Placebo

Eligibility Criteria

Age18 Years - 60 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64)

You may qualify if:

  • to 60 years of age inclusive
  • Diagnosis of nonrelapsing secondary progressive multiple sclerosis according to the 2017 McDonald criteria
  • Expanded disability status scale (EDSS) between 3.0 to 6.5 points inclusive, at screening
  • The participant must have documented evidence of disability progression observed during the 12 months before screening
  • Absence of clinical relapses for at least 24 months
  • Contraceptive use by men or women should be consistent with local regulations regarding the methods of contraception for those participating in clinical studies
  • A female participant is eligible to participate if she is not pregnant or breastfeeding, and at least one of the following conditions applies:
  • Is not a WOCBP OR
  • Is a WOCBP and agrees to use an acceptable contraceptive method

You may not qualify if:

  • The participant has conditions that would adversely affect study participation such as short life expectancy.
  • Evidence of infection with human immuodeficiency virus (HIV), transplantation, progressive multifocal leukoencephalopathy (PML), active hepatitis B or C, active or latent tuberculosis or other active infections that would adversely affect study participation.
  • Persistent chronic or active or recurring system infection, that may adversely affect participation or IMP administration in this study, as judged by the Investigator.
  • History of malignancy within 5 years prior to screening.
  • History of alcohol or drug abuse within 1 year prior to screening.
  • Hospitalized for psychiatric disease within 2 years prior to screening.
  • Clinically significant laboratory abnormalities (including evidence of liver injury) or electrocardiogram abnormalities at screening
  • Bleeding disorder, known platelet dysfunctionat any time prior to the screening visit
  • A platelet count \<150 000/μL at the screening visit
  • A history of significant bleeding event within 6 months prior to screening, according to the Investigator's judgment such as, but not limited to cerebral or gastrointestinal bleeding.
  • Lymphocyte count below the lower limit of normal at screening.
  • Recent live (attenuated) vaccine within 2 months before the first treatment visit.
  • Recent major surgery (within 4 weeks of screening) or planned major surgery during the study.
  • The participant has received medications/treatments for MS within a specified time frame.
  • Receiving potent and moderate inducers or inhibitors of cytochrome P450 3A (CYP3A) or potent inhibitors of CYP2C8 hepatic enzymes.
  • +3 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (306)

University of Alabama MS Center-Site Number:8400013

Birmingham, Alabama, 35233, United States

Location

Center for Neurology and Spine-Site Number:8400089

Phoenix, Arizona, 84018, United States

Location

Arcadia Neurology Center-Site Number:8400070

Arcadia, California, 91006, United States

Location

UC San Diego ACTRI-Site Number:8400101

La Jolla, California, 92037, United States

Location

Collaborative Neuroscience Research-Site Number:8400045

Long Beach, California, 90806, United States

Location

Multiple Sclerosis Center-Site Number:8400143

Los Angeles, California, 90033, United States

Location

University of San Francisco, Sandler Neurosciences Center-Site Number:8400137

San Francisco, California, 94158, United States

Location

Harbor UCLA-Site Number:8400088

Torrance, California, 90502, United States

Location

Regina Berkovich, MD, PhD-Site Number:8400059

West Hollywood, California, 90048, United States

Location

Mountain Neurological Research Center, Inc.-Site Number:8400128

Basalt, Colorado, 81621, United States

Location

University of Colorado-Site Number:8400012

Denver, Colorado, 80262, United States

Location

Advanced Neurosciences Research-Site Number:8400025

Fort Collins, Colorado, 80528, United States

Location

South Florida Neurology Associates-Site Number:8400029

Boca Raton, Florida, 33487, United States

Location

Neurology Associates, PA-Site Number:8400004

Maitland, Florida, 32761, United States

Location

Aqualane Clinical Research-Site Number:8400027

Naples, Florida, 34105, United States

Location

Axiom Clinical Research of Florida-Site Number:8400001

Tampa, Florida, 33609-4052, United States

Location

University of South Florida-Site Number:8400006

Tampa, Florida, 33612, United States

Location

Meridian Clinical Research-Site Number:8400003

Savannah, Georgia, 31406, United States

Location

Consultants In Neurology-Site Number:8400011

Northbrook, Illinois, 60062, United States

Location

University of Kansas Medical Center-Site Number:8400023

Kansas City, Kansas, 66160-7321, United States

Location

CHI Saint Joseph Medical Group Neurology-Site Number:8400110

Lexington, Kentucky, 40509, United States

Location

Tufts Medical Center-Site Number:8400072

Boston, Massachusetts, 02111, United States

Location

University of Massachusetts-Site Number:8400014

Worcester, Massachusetts, 01655, United States

Location

Wayne State University-Site Number:8400046

Detroit, Michigan, 48201, United States

Location

The Memorial Hospital-Site Number:8400033

Owosso, Michigan, 48867, United States

Location

Minneapolis Clinic of Neurology-Site Number:8400051

Minneapolis, Minnesota, 55422, United States

Location

Mayo Clinic-Site Number:8400111

Rochester, Minnesota, 55905, United States

Location

Missouri Baptist Medical Center-Site Number:8400019

St Louis, Missouri, 63131, United States

Location

Lou Ruvo Center for Brain Health-Site Number:8400117

Las Vegas, Nevada, 89106, United States

Location

Holy Name Hospital-Site Number:8400104

Teaneck, New Jersey, 07666, United States

Location

University of New Mexico-Site Number:8400032

Albuquerque, New Mexico, 87131, United States

Location

Icahn School of Medicine at Mount Sinai (Department of Endoc-Site Number:8400038

New York, New York, 10029-6501, United States

Location

Neurology Associates of Stony Brook-Site Number:8400042

Stony Brook, New York, 11794, United States

Location

Meridian Clinical Research, LLC-Site Number:8400005

Raleigh, North Carolina, 27607, United States

Location

Sanford Brain & Spine Center-Site Number:8400126

Fargo, North Dakota, 58103, United States

Location

University Hospitals CMC-Site Number:8400083

Cleveland, Ohio, 44106, United States

Location

Cleveland Clinic-Site Number:8400125

Cleveland, Ohio, 44195, United States

Location

Optimed Research, LTD-Site Number:8400147

Columbus, Ohio, 43235, United States

Location

Neurology Specialists-Site Number:8400002

Dayton, Ohio, 45417, United States

Location

Columbus Neuroscience-Site Number:8400010

Westerville, Ohio, 40382, United States

Location

Providence Multiple Sclerosis Center-Site Number:8400020

Portland, Oregon, 97225, United States

Location

Perelman Center for Advanced Medicine-Site Number:8400142

Philadelphia, Pennsylvania, 19104, United States

Location

Jefferson Neurology Associates-Site Number:8400016

Philadelphia, Pennsylvania, 19107, United States

Location

Premier Neurology-Site Number:8400069

Greer, South Carolina, 29650, United States

Location

Mountain View Clinical Research-Site Number:8400024

Greer, South Carolina, 29651-1817, United States

Location

Neurology Clinic, PC-Site Number:8400087

Cordova, Tennessee, 38018, United States

Location

Advanced Neuroscience Center-Site Number:8400035

Franklin, Tennessee, 37064, United States

Location

Baylor College of Medicine-Site Number:8400136

Houston, Texas, 77030, United States

Location

Neurology Center of San Antonio-Site Number:8400036

San Antonio, Texas, 78258, United States

Location

University Of Vermont College Of Medicine-Site Number:8400130

Burlington, Vermont, 05401, United States

Location

Medical College of Wisconsin-Site Number:8400028

Milwaukee, Wisconsin, 53226, United States

Location

Investigational Site Number :0320002

Capital Federal, Buenos Aires, 1012, Argentina

Location

Investigational Site Number :0320001

CABA, Buenos Aires F.D., C1061, Argentina

Location

Investigational Site Number :0320007

Buenos Aires, 1860, Argentina

Location

Investigational Site Number :0320006

Córdoba, 5000, Argentina

Location

Investigational Site Number :0320005

San Miguel de Tucumán, T4000AXL, Argentina

Location

Investigational Site Number : 0360007

St Leonards, New South Wales, 2065, Australia

Location

Investigational Site Number :0360003

Woolloongabba, Queensland, 4102, Australia

Location

Investigational Site Number :0360002

Kent Town, South Australia, Australia

Location

Investigational Site Number :0360004

Hobart, Tasmania, 7001, Australia

Location

Investigational Site Number :0360001

Fitzroy, Victoria, 3065, Australia

Location

Investigational Site Number :0360006

Heidelberg West, Victoria, 3081, Australia

Location

Investigational Site Number :0400003

Innsbruck, 6020, Austria

Location

Investigational Site Number :0400001

Linz, 4020, Austria

Location

Investigational Site Number :0400004

Linz, 4021, Austria

Location

Investigational Site Number :0400002

Vienna, 1090, Austria

Location

Investigational Site Number :1120004

Vitebsk, 210009, Belarus

Location

Investigational Site Number :1120005

Vitebsk, 210037, Belarus

Location

Investigational Site Number : 0560009

Brussels, 1070, Belgium

Location

Investigational Site Number :0560007

Brussels, 1200, Belgium

Location

Investigational Site Number :0560003

Edegem, B-2650, Belgium

Location

Investigational Site Number : 0560004

Ghent, 9000, Belgium

Location

Investigational Site Number :0560006

Leuven, 3000, Belgium

Location

Investigational Site Number :0560008

Liège, 4000, Belgium

Location

Investigational Site Number :0560002

Mons, 7000, Belgium

Location

Investigational Site Number :0560001

Overpelt, 3900, Belgium

Location

Investigational Site Number :1000002

Pleven, 5800, Bulgaria

Location

Investigational Site Number :1000005

Plovdiv, 4000, Bulgaria

Location

Investigational Site Number :1000004

Sofia, 1113, Bulgaria

Location

Investigational Site Number :1000008

Sofia, 1407, Bulgaria

Location

Investigational Site Number :1000001

Sofia, 1431, Bulgaria

Location

Investigational Site Number :1000006

Sofia, 1431, Bulgaria

Location

Investigational Site Number :1000009

Sofia, 1680, Bulgaria

Location

Investigational Site Number :1240017

Burnaby, British Columbia, V5G 2X6, Canada

Location

Investigational Site Number :1240011

Halifax, Nova Scotia, B3H 1V7, Canada

Location

Investigational Site Number :1240003

Ottawa, Ontario, K1H 8L6, Canada

Location

Investigational Site Number :1240008

Toronto, Ontario, M4N 3M5, Canada

Location

Investigational Site Number :1240006

Gatineau, Quebec, J8Y 1W2, Canada

Location

Investigational Site Number :1240005

Greenfield Park, Quebec, J4V 2J2, Canada

Location

Investigational Site Number :1240004

Montreal, Quebec, H2X 0A9, Canada

Location

Investigational Site Number :1240015

Montreal, Quebec, H3A 2B4, Canada

Location

Investigational Site Number :1240007

Sherbrooke, Quebec, J1H 5N4, Canada

Location

Investigational Site Number : 1240001

Québec, G1J 1Z4, Canada

Location

Investigational Site Number :1240021

Québec, G1W 4R4, Canada

Location

Investigational Site Number :1560006

Beijing, 100034, China

Location

Investigational Site Number :1560012

Beijing, 100053, China

Location

Investigational Site Number :1560021

Beijing, 100700, China

Location

Investigational Site Number :1560003

Beijing, 100730, China

Location

Investigational Site Number :1560009

Beijing, 100730, China

Location

Investigational Site Number :1560004

Changchun, 130021, China

Location

Investigational Site Number :1560015

Changsha, 410008, China

Location

Investigational Site Number :1560005

Chengdu, 610041, China

Location

Investigational Site Number :1560019

Chongqing, 400016, China

Location

Investigational Site Number :1560035

Fuzhou, 350005, China

Location

Investigational Site Number :1560001

Guangzhou, 510630, China

Location

Investigational Site Number :1560007

Hangzhou, 310009, China

Location

Investigational Site Number :1560014

Shijiazhuang, 050000, China

Location

Investigational Site Number :1560008

Taiyuan, 030001, China

Location

Investigational Site Number :1560017

Xi'an, 710038, China

Location

Investigational Site Number :2030002

Brno, 65691, Czechia

Location

Investigational Site Number :2030004

Hradec Králové, 50005, Czechia

Location

Investigational Site Number :2030001

Jihlava, 58633, Czechia

Location

Investigational Site Number :2030010

Ostrava - Poruba, 70852, Czechia

Location

Investigational Site Number :2030005

Prague, 12808, Czechia

Location

Investigational Site Number :2030003

Teplice, 415 29, Czechia

Location

Investigational Site Number :2080001

Esbjerg, 6700, Denmark

Location

Investigational Site Number :2080005

Holstebro, 7500, Denmark

Location

Investigational Site Number :2080004

Odense, 5000, Denmark

Location

Investigational Site Number :2460003

Helsinki, 00180, Finland

Location

Investigational Site Number :2460001

Tampere, 33520, Finland

Location

Investigational Site Number :2460002

Turku, 20520, Finland

Location

Investigational Site Number :2500011

Bron, 69500, France

Location

Investigational Site Number :2500005

Clermont-Ferrand, 63003, France

Location

Investigational Site Number :2500015

Gonesse, 95500, France

Location

Investigational Site Number :2500009

Lille, 59037, France

Location

Investigational Site Number :2500006

Montpellier, 34295, France

Location

Investigational Site Number :2500008

Nancy, 54035, France

Location

Investigational Site Number :2500010

Nantes, 44093, France

Location

Investigational Site Number :2500017

Nîmes, 30029, France

Location

Investigational Site Number :2500016

Paris, 75012, France

Location

Investigational Site Number :2500014

Paris, 75013, France

Location

Investigational Site Number :2500007

Paris, 75019, France

Location

Investigational Site Number :2500003

Rennes, 35033, France

Location

Investigational Site Number :2500001

Strasbourg, 67098, France

Location

Investigational Site Number :2500012

Toulouse, 31059, France

Location

Investigational Site Number :2760005

Bayreuth, 95445, Germany

Location

Investigational Site Number :2760009

Berlin, 10117, Germany

Location

Investigational Site Number :2760001

Dresden, 01307, Germany

Location

Investigational Site Number :2760012

Essen, 45147, Germany

Location

Investigational Site Number :2760002

Giessen, 35385, Germany

Location

Investigational Site Number :2760010

Halle, 06120, Germany

Location

Investigational Site Number :2760006

Hanover, 30625, Germany

Location

Investigational Site Number :2760008

Münster, 48149, Germany

Location

Investigational Site Number :2760004

Rostock, 18055, Germany

Location

Investigational Site Number :2760011

Ulm, 89081, Germany

Location

Investigational Site Number :3000001

Athens, 115 28, Greece

Location

Investigational Site Number :3000006

Athens, 11535, Greece

Location

Investigational Site Number :3000002

Athens, 12462, Greece

Location

Investigational Site Number :3000007

Athens, 15125, Greece

Location

Investigational Site Number :3000004

Larissa, 41110, Greece

Location

Investigational Site Number :3000003

Thessaloniki, 546 36, Greece

Location

Investigational Site Number :3000005

Thessaloniki, 57010, Greece

Location

Investigational Site Number :3480008

Budapest, 1135, Hungary

Location

Investigational Site Number :3480004

Budapest, 1145, Hungary

Location

Investigational Site Number :3480007

Budapest, 1152, Hungary

Location

Investigational Site Number :3480002

Pécs, 7623, Hungary

Location

Investigational Site Number :3480001

Szeged, 6725, Hungary

Location

Investigational Site Number :3480006

Tatabánya, 2800, Hungary

Location

Investigational Site Number :3560007

Gūrgaon, 122001, India

Location

Investigational Site Number :3560003

Gūrgaon, 122002, India

Location

Investigational Site Number :3560005

India, India

Location

Investigational Site Number :3560004

Mangaluru, 575018, India

Location

Investigational Site Number : 3560009

Nagpur, 440012, India

Location

Investigational Site Number :3560006

New Delhi, 110029, India

Location

Investigational Site Number :3560002

New Delhi, 110060, India

Location

Investigational Site Number :3760002

Ashkelon, 78278, Israel

Location

Investigational Site Number :3760003

Haifa, 31096, Israel

Location

Investigational Site Number :3760008

Jerusalem, 91120, Israel

Location

Investigational Site Number :3760004

Safed, 13100, Israel

Location

Investigational Site Number :3760001

Tel Litwinsky, 52621, Israel

Location

Investigational Site Number :3800011

Bergamo, 24127, Italy

Location

Investigational Site Number :3800007

Cagliari, 09126, Italy

Location

Investigational Site Number :3800012

Florence, 50134, Italy

Location

Investigational Site Number :3800016

Florence, 50141, Italy

Location

Investigational Site Number :3800014

Genova, 16132, Italy

Location

Investigational Site Number :3800013

L’Aquila, 67010, Italy

Location

Investigational Site Number :3800004

Milan, 20122, Italy

Location

Investigational Site Number :3800001

Milan, 20132, Italy

Location

Investigational Site Number :3800010

Milan, 20133, Italy

Location

Investigational Site Number :3800008

Pavia, 27100, Italy

Location

Investigational Site Number :3800005

Roma, 00152, Italy

Location

Investigational Site Number :3800009

Roma, 00168, Italy

Location

Investigational Site Number :3920016

Chiba, Chiba, 260-8677, Japan

Location

Investigational Site Number :3920022

Morioka, Iwate, 020-8505, Japan

Location

Investigational Site Number :3920011

Kyoto, Kyoto, 616-8255, Japan

Location

Investigational Site Number :3920020

Sendai, Miyagi, 980-8574, Japan

Location

Investigational Site Number :3920005

Niigata, Niigata, 951-8520, Japan

Location

Investigational Site Number :3920004

Moriguchi-shi, Osaka, 570-8507, Japan

Location

Investigational Site Number :3920001

Osaka, Osaka, 556-0016, Japan

Location

Investigational Site Number :3920018

Kawagoe-shi, Saitama, 350-8550, Japan

Location

Investigational Site Number :3920003

Kodaira-shi, Tokyo, 187-8551, Japan

Location

Investigational Site Number :3920010

Ōta-ku, Tokyo, 146-0065, Japan

Location

Investigational Site Number :3920009

Ube-shi, Yamaguchi, 755-8505, Japan

Location

Investigational Site Number :3920023

Sagamihara-shi, 252-0392, Japan

Location

Investigational Site Number :4400003

Kaunas, 50161, Lithuania

Location

Investigational Site Number :4400002

Klaipėda, 92288, Lithuania

Location

Investigational Site Number :4400001

Vilnius, 08661, Lithuania

Location

Investigational Site Number :5280001

Amsterdam, 1081 GN, Netherlands

Location

Investigational Site Number :5280003

Breda, 4818 CK, Netherlands

Location

Investigational Site Number :5280006

Groningen, 9728 NZ, Netherlands

Location

Investigational Site Number :5280002

Sittard-Geleen, 6162 BG, Netherlands

Location

Investigational Site Number :5780003

Bergen, 5021, Norway

Location

Investigational Site Number :5780002

Namsos, 7800, Norway

Location

Investigational Site Number :5780001

Oslo, 0450, Norway

Location

Investigational Site Number :6160008

Plewiska, Greater Poland Voivodeship, 62-064, Poland

Location

Investigational Site Number :6160003

Bydgoszcz, Kuyavian-Pomeranian Voivodeship, 85-796, Poland

Location

Investigational Site Number :6160005

Warsaw, Masovian Voivodeship, 01-211, Poland

Location

Investigational Site Number :6160006

Warsaw, Masovian Voivodeship, 01-684, Poland

Location

Investigational Site Number :6160002

Katowice, Silesian Voivodeship, 40-571, Poland

Location

Investigational Site Number :6160007

Katowice, Silesian Voivodeship, 40-684, Poland

Location

Investigational Site Number :6160004

Katowice, Silesian Voivodeship, 40-686, Poland

Location

Investigational Site Number :6160001

Lodz, 90-549, Poland

Location

Investigational Site Number :6160012

Lublin, 20-016, Poland

Location

Investigational Site Number :6160011

Zabrze, 41-800, Poland

Location

Investigational Site Number :6200001

Braga, 4710-243, Portugal

Location

Investigational Site Number :6200011

Lisbon, 1162-050, Portugal

Location

Investigational Site Number :6200007

Lisbon, 1349-019, Portugal

Location

Investigational Site Number :6200006

Lisbon, 1649-035, Portugal

Location

Investigational Site Number :6200002

Matosinhos Municipality, 4464-513, Portugal

Location

Investigational Site Number :6200010

Porto, 4099-001, Portugal

Location

Investigational Site Number :6420008

Bucharest, 022328, Romania

Location

Investigational Site Number :6420004

Campulung Muscel, 115100, Romania

Location

Investigational Site Number :6420006

Cluj-Napoca, 400012, Romania

Location

Investigational Site Number :6420003

Constanța, 900123, Romania

Location

Investigational Site Number :6420013

Oradea, 410154, Romania

Location

Investigational Site Number :6420005

Sibiu, 550052, Romania

Location

Investigational Site Number :6420001

Târgu Mureş, 540136, Romania

Location

Investigational Site Number :6420002

Timișoara, 300736, Romania

Location

Investigational Site Number :6430018

Barnaul, 656024, Russia

Location

Investigational Site Number :6430025

Kaliningrad, 236035, Russia

Location

Investigational Site Number :6430003

Kazan', 420021, Russia

Location

Investigational Site Number :6430022

Kemerovo, 650099, Russia

Location

Investigational Site Number :6430017

Kirov, 610998, Russia

Location

Investigational Site Number :6430024

Krasnoyarsk, 660029, Russia

Location

Investigational Site Number :6430020

Moscow, 117997, Russia

Location

Investigational Site Number :6430002

Moscow, 125367, Russia

Location

Investigational Site Number :6430013

Moscow, 127015, Russia

Location

Investigational Site Number :6430001

Moscow, 129110, Russia

Location

Investigational Site Number :6430008

Moscow, 129128, Russia

Location

Investigational Site Number :6430021

Nizhny Novgorod, 603137, Russia

Location

Investigational Site Number :6430006

Nizhny Novgorod, 603155, Russia

Location

Investigational Site Number :6430005

Novosibirsk, 630087, Russia

Location

Investigational Site Number :6430026

Perm, 614990, Russia

Location

Investigational Site Number :6430007

Pyatigorsk, 357538, Russia

Location

Investigational Site Number :6430016

Rostov-on-Don, 344022, Russia

Location

Investigational Site Number :6430011

Saint Petersburg, 197022, Russia

Location

Investigational Site Number :6430004

Saint Petersburg, 197110, Russia

Location

Investigational Site Number :6430009

Samara, 443095, Russia

Location

Investigational Site Number :6430019

Saransk, 430032, Russia

Location

Investigational Site Number :6430014

Smolensk, 214018, Russia

Location

Investigational Site Number :6430012

Tyumen, 625000, Russia

Location

Investigational Site Number :6430010

Ufa, 450005, Russia

Location

Investigational Site Number :6430023

Yekaterinburg, 620102, Russia

Location

Investigational Site Number :7240007

Seville, Andalusia, 41009, Spain

Location

Investigational Site Number :7240013

Barcelona, Barcelona [Barcelona], 08035, Spain

Location

Investigational Site Number :7240016

Barcelona, Barcelona [Barcelona], 08036, Spain

Location

Investigational Site Number :7240012

Donostia / San Sebastian, Basque Country, 20014, Spain

Location

Investigational Site Number :7240014

Salt, Girona [Gerona], 17190, Spain

Location

Investigational Site Number :7240017

Las Palmas de Gran Canaria, Las Palmas, 35010, Spain

Location

Investigational Site Number :7240004

Majadahonda, Madrid, 28222, Spain

Location

Investigational Site Number :7240001

Pozuelo de Alarcón, Madrid, 28223, Spain

Location

Investigational Site Number :7240008

Córdoba, 14004, Spain

Location

Investigational Site Number :7240015

Lleida, 25198, Spain

Location

Investigational Site Number :7240005

Madrid, 28007, Spain

Location

Investigational Site Number :7240002

Madrid, 28034, Spain

Location

Investigational Site Number :7240003

Madrid, 28040, Spain

Location

Investigational Site Number :7240009

Málaga, 29010, Spain

Location

Investigational Site Number :7240010

Murcia, 30120, Spain

Location

Investigational Site Number :7240011

Valencia, 46026, Spain

Location

Investigational Site Number :7920005

Eskişehir, Turkey (Türkiye)

Location

Investigational Site Number :7920010

Hatay, Turkey (Türkiye)

Location

Investigational Site Number :7920002

Istanbul, 34098, Turkey (Türkiye)

Location

Investigational Site Number :7920009

Istanbul, 34688, Turkey (Türkiye)

Location

Investigational Site Number :7920007

Istanbul, 34785, Turkey (Türkiye)

Location

Investigational Site Number :7920006

Istanbul, 34896, Turkey (Türkiye)

Location

Investigational Site Number :7920003

Istanbul, Turkey (Türkiye)

Location

Investigational Site Number :7920013

Izmir, 35100, Turkey (Türkiye)

Location

Investigational Site Number :7920001

İzmit, 41380, Turkey (Türkiye)

Location

Investigational Site Number :7920011

Kütahya, 43100, Turkey (Türkiye)

Location

Investigational Site Number :7920012

Mersin, 33070, Turkey (Türkiye)

Location

Investigational Site Number :7920008

Trabzon, 61080, Turkey (Türkiye)

Location

Investigational Site Number :8040008

Chernivtsi, 58000, Ukraine

Location

Investigational Site Number :8040016

Chernivtsi, 58023, Ukraine

Location

Investigational Site Number :8040003

Dnipro, 49005, Ukraine

Location

Investigational Site Number :8040010

Ivano-Frankivsk, 76018, Ukraine

Location

Investigational Site Number :8040007

Kharkiv, 61068, Ukraine

Location

Investigational Site Number :8040011

Kharkiv, 61103, Ukraine

Location

Investigational Site Number :8040012

Kharkiv, 61103, Ukraine

Location

Investigational Site Number :8040013

Kyiv, 03115, Ukraine

Location

Investigational Site Number :8040005

Lutsk, 43005, Ukraine

Location

Investigational Site Number :8040009

Lviv, 79010, Ukraine

Location

Investigational Site Number :8040004

Lviv, 79013, Ukraine

Location

Investigational Site Number :8040002

Odesa, 65025, Ukraine

Location

Investigational Site Number :8040006

Vinnytsia, 21050, Ukraine

Location

Investigational Site Number :8040014

Zhytomyr, 10002, Ukraine

Location

Investigational Site Number :8260003

Exeter, Devon, EX2 5DW, United Kingdom

Location

Investigational Site Number :8260008

Plymouth, Devon, PL6 8DH, United Kingdom

Location

Investigational Site Number :8260010

Swansea, Neath Port Talbot, SA6 6NL, United Kingdom

Location

Investigational Site Number :8260012

Nottingham, Nottinghamshire, NG7 2UH, United Kingdom

Location

Investigational Site Number :8260013

Oxford, Oxfordshire, OX3 9DZ, United Kingdom

Location

Investigational Site Number :8260009

Bristol, BS10 5NB, United Kingdom

Location

Investigational Site Number :8260001

Cardiff, CF4 4XY, United Kingdom

Location

Investigational Site Number :8260005

London, SW17 0RE, United Kingdom

Location

Investigational Site Number :8260018

London, W6 8RF, United Kingdom

Location

Investigational Site Number :8260014

Newcastle upon Tyne, NE1 4LP, United Kingdom

Location

Investigational Site Number :8260019

Salford, M6 8HD, United Kingdom

Location

Related Publications (1)

  • Fox RJ, Bar-Or A, Traboulsee A, Oreja-Guevara C, Giovannoni G, Vermersch P, Syed S, Li Y, Vargas WS, Turner TJ, Wallstroem E, Reich DS; HERCULES Trial Group. Tolebrutinib in Nonrelapsing Secondary Progressive Multiple Sclerosis. N Engl J Med. 2025 May 15;392(19):1883-1892. doi: 10.1056/NEJMoa2415988. Epub 2025 Apr 8.

Related Links

Results Point of Contact

Title
Trial Transparency Team
Organization
Sanofi aventis recherche & développement

Study Officials

  • Clinical Sciences & Operations

    Sanofi

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 28, 2020

First Posted

June 2, 2020

Study Start

September 24, 2020

Primary Completion

August 29, 2024

Study Completion

August 29, 2024

Last Updated

July 2, 2025

Results First Posted

June 18, 2025

Record last verified: 2025-06

Data Sharing

IPD Sharing
Will share

Qualified researchers may request access to patient level data and related study documents including the clinical study report, study protocol with any amendments, blank case report form, statistical analysis plan, and dataset specifications. Patient level data will be anonymized and study documents will be redacted to protect the privacy of trial participants. Further details on Sanofi's data sharing criteria, eligible studies, and process for requesting access can be found at: https://vivli.org

Locations