NCT04135833

Brief Summary

This is a phase I study to assess the effect of itraconazole and rifampicin on the pharmacokinetic parameters of BPI-7711 in Chinese healthy volunteers.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
31

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started Dec 2019

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 21, 2019

Completed
2 days until next milestone

First Posted

Study publicly available on registry

October 23, 2019

Completed
2 months until next milestone

Study Start

First participant enrolled

December 12, 2019

Completed
7 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 22, 2020

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

July 22, 2020

Completed
Last Updated

April 22, 2021

Status Verified

April 1, 2021

Enrollment Period

7 months

First QC Date

October 21, 2019

Last Update Submit

April 21, 2021

Conditions

Outcome Measures

Primary Outcomes (2)

  • Cmax

    Pharmacokinetics of BPI-7711 by assessment of maximum plasma concentration

    Blood samples collected on Day 1 and Day 20 (arm 1)/Day 25 (arm 2) at pre-dose, 1, 2, 3, 4, 5, 6, 8, 10, 12, 24, 48, 72, 96, 120, 144, 168 and 336 hours post BPI-7711 dose

  • AUC(0-last)

    Pharmacokinetics of BPI-7711 by assessment of area under the plasma concentration time curve from zero to last assessed timepoint

    Blood samples collected on Day 1 and Day 20 (arm 1)/Day 25 (arm 2) at pre-dose, 1, 2, 3, 4, 5, 6, 8, 10, 12, 24, 48, 72, 96, 120, 144, 168 and 336 hours post BPI-7711 dose

Study Arms (2)

Itraconazole and BPI-7711

EXPERIMENTAL

BPI-7711 alone followed by BPI-7711 +Itraconazole, followed by Itraconazole alone.

Drug: BPI-7711Drug: Itraconazole

Rifampicin and BPI-7711

EXPERIMENTAL

BPI-7711 alone followed by BPI-7711 +Rifampicin, followed by Rifampicin alone.

Drug: BPI-7711Drug: Rifampicin

Interventions

BPI-7711 60 mg

Also known as: BPI-7711 capsule
Itraconazole and BPI-7711

Itraconazole 200 mg

Also known as: Itraconazole capsule
Itraconazole and BPI-7711

Rifampicin 600 mg

Also known as: Rifampicin capsule
Rifampicin and BPI-7711

Eligibility Criteria

Age18 Years - 45 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Male, aged from 18 to 45 years
  • BMI from 18.5 to 28.0 kg/m2
  • Medical history, vital signs, physical examination and lab tests are normal or abnormal without clinical significance

You may not qualify if:

  • Subjects with clinical significant diseases
  • Subjects with allergic disease history
  • Subjects with gastrointestinal disease history that can affect study drug absorption
  • Subjects with drug abuse history

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Shanghai Xuhui Central Hospital

Shanghai, 200000, China

Location

MeSH Terms

Interventions

rezivertinibItraconazoleRifampin

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPiperazinesRifamycinsHeterocyclic Compounds, 4 or More RingsHeterocyclic Compounds, Fused-RingLactams, MacrocyclicMacrocyclic CompoundsPolycyclic Compounds

Study Officials

  • Jingying Jia

    Shanghai Xuhui Central Hospital

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
OTHER
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 21, 2019

First Posted

October 23, 2019

Study Start

December 12, 2019

Primary Completion

July 22, 2020

Study Completion

July 22, 2020

Last Updated

April 22, 2021

Record last verified: 2021-04

Data Sharing

IPD Sharing
Will not share

Locations