NCT03493685

Brief Summary

To determine the long-term nephroprotective potential of treatment with sparsentan as compared to an angiotensin receptor blocker in patients with primary and genetic focal segmental glomerulosclerosis (FSGS).

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
371

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Apr 2018

Longer than P75 for phase_3

Geographic Reach
21 countries

206 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 3, 2018

Completed
7 days until next milestone

First Posted

Study publicly available on registry

April 10, 2018

Completed
7 days until next milestone

Study Start

First participant enrolled

April 17, 2018

Completed
4.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 20, 2023

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

April 30, 2024

Completed
1.9 years until next milestone

Study Completion

Last participant's last visit for all outcomes

March 19, 2026

Completed
Last Updated

April 17, 2026

Status Verified

April 1, 2026

Enrollment Period

4.9 years

First QC Date

April 3, 2018

Results QC Date

March 15, 2024

Last Update Submit

April 15, 2026

Conditions

Outcome Measures

Primary Outcomes (2)

  • Slope of Estimated Glomerular Filtration Rate (eGFR)

    The total eGFR slope over 2 years, defined as the slope of eGFR following initiation of randomized treatment (ie, Day 1 to Week 108). Estimates are calculated from a mixed-effects model with treatment, Baseline eGFR, analysis visit, treatment-by-analysis visit, randomization stratification factors as fixed effects, and intercept and slope for each participant as a random effect.

    From Day 1 to Week 108

  • Percentage of Participants Achieving FSGS Partial Remission Endpoint (FPRE)

    Percentage of participants achieving FPRE, defined as urine protein-to-creatinine ratio (UP/C) ≤1.5 grams/gram (g/g) (170 milligrams per millimoles \[mg/mmol\]) and a \>40% reduction from Baseline was analyzed using a generalized linear model to model probability of achieving FPRE. Missing responses were imputed prior to analysis using multiple imputation. A generalized linear model with appropriate link function was implemented with Baseline log (UP/C), treatment, analysis visit, treatment by analysis visit interaction, and randomization strata as fixed effects. For estimates of probability of achieving FPRE, risk difference, and odds ratio, binomial distribution with logit link was used. For relative risk, Poisson distribution with log link was used. Using Rubin's approach, estimated treatment effects are combined across all imputations to obtain overall estimates for probabilities.

    Week 36

Secondary Outcomes (2)

  • Slope of eGFR Following the Initial Acute Effect of Randomized Treatment

    From Week 6 to Week 108

  • Change From Baseline in eGFR to 4 Weeks Post-cessation of Randomized Treatment

    Baseline (Day 1) to Week 112

Study Arms (2)

sparsentan for double-blind and open-label extension

EXPERIMENTAL

Sparsentan will be administered as a single oral dose; an initial dose of 400 mg daily titrating up to a target dose of 800 mg, daily

Drug: sparsentan

Irbesartan

ACTIVE COMPARATOR

Irbesartan will be administered as a single oral dose; an initial dose of 150 mg daily titrating up to a target dose of 300 mg, daily

Drug: Irbesartan

Interventions

Double-blind period: target dose of 800 mg daily; Open-label extension: target dose based on dosage from week 114 daily

Also known as: RE-021
sparsentan for double-blind and open-label extension

target dose of 300 mg daily

Also known as: Irbesartan Tablets USP
Irbesartan

Eligibility Criteria

Age8 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17), Adult (18-64), Older Adult (65+)

You may qualify if:

  • Sites within the US and UK: The patient is male or female aged 8 to 75 years, inclusive, weighing ≥20 kg at screening
  • Sites outside the US and UK: The patient is male or female aged 18 to 75 years, inclusive, weighing ≥20 kg at screening
  • Biopsy-proven focal segmental glomerulosclerosis (FSGS) lesion(s) or documentation of a genetic mutation in a podocyte protein associated with FSGS.
  • Urine protein/creatinine (UP/C) ≥1.5 g/g (170 mg/mmol) at screening
  • eGFR ≥30 mL/min/1.73 m2 at screening.
  • Women of childbearing potential must agree to the use of one highly reliable method of contraception from 7 days prior to the first dose of study medication until 90 days after the last dose of study medication, plus one additional barrier method during sexual activity

You may not qualify if:

  • FSGS secondary to another condition
  • Positive serological tests of another primary or secondary glomerular disease not consistent with a diagnosis of primary or genetic FSGS
  • History of type 1 diabetes mellitus, uncontrolled type 2 diabetes mellitus, or nonfasting blood glucose \>180 mg/dL (10.0 mmol/L)
  • Treated with rituximab, cyclophosphamide, or abatacept within ≤3 months prior to screening; if taking other chronic immunosuppressive medications, the dosage must be stable prior to screening
  • Documented history of heart failure, coronary artery disease, or cerebrovascular disease
  • Significant liver disease
  • Positive at screening for the human immunodeficiency virus or markers indicating acute or chronic hepatitis B virus infection or hepatitis C infection
  • History of malignancy other than adequately treated basal cell or squamous cell skin cancer or cervical carcinoma within the past 2 years
  • Screening hematocrit value \<27% (0.27 L/L) or hemoglobin value \<9 g/dL (90 g/L)
  • Screening potassium value of \>5.5 mEq/L (5.5 mmol/L)
  • Extreme obesity (ie, ≥18 years of age with a body mass index (BMI) \>40, or is \<18 years of age with a BMI in the 99th percentile plus 5 units at screening, in whom there is a causal relationship between obesity and the development of FSGS
  • History of alcohol or illicit drug use disorder
  • History of serious side effect or allergic response to any angiotensin II antagonist or endothelin receptor antagonist
  • Female patient is pregnant, plans to become pregnant during the course of the study, or is breastfeeding.
  • Complete participation in the double-blind period, including the Week 112 visit.
  • +5 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (226)

Travere Investigational Site

Mesa, Arizona, 85210, United States

Location

Travere Investigational Site

Phoenix, Arizona, 85027, United States

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Travere Investigational Site

Los Angeles, California, 90048, United States

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Travere Investigational Site

Northridge, California, 91324, United States

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Travere Investigational Site

Palo Alto, California, 94304, United States

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Travere Investigational Site

San Diego, California, 92103, United States

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Travere Investigational Site

San Dimas, California, 91773, United States

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Travere Investigational Site

San Francisco, California, 94118, United States

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Travere Investigational Site

Torrance, California, 90502, United States

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Travere Investigational Site

Victorville, California, 92395, United States

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Travere Investigational Site

Denver, Colorado, 80205, United States

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Travere Investigational Site

Denver, Colorado, 80230, United States

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Travere Investigational Site

Middlebury, Connecticut, 06762, United States

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Travere Investigational Site

Wilmington, Delaware, 19803, United States

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Travere Investigational Site

Washington D.C., District of Columbia, 20010, United States

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Travere Investigational Site

Coral Springs, Florida, 33071, United States

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Fort Lauderdale, Florida, 33308, United States

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Travere Investigational Site

Gainesville, Florida, 32610, United States

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Travere Investigational Site

Miami, Florida, 33126, United States

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Travere Investigational Site

Miami, Florida, 33136, United States

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Travere Investigational Site

Miami, Florida, 33155, United States

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Travere Investigational Site

Ocala, Florida, 34471, United States

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Travere Investigational Site

Orlando, Florida, 32827, United States

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Travere Investigational Site

Port Charlotte, Florida, 33952, United States

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Travere Investigational Site

Temple Terrace, Florida, 33637, United States

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Travere Investigational Site

Winter Park, Florida, 32789, United States

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Travere Investigational Site

Lawrenceville, Georgia, 30046, United States

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Nampa, Idaho, 86387, United States

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Chicago, Illinois, 60611, United States

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Hinsdale, Illinois, 60521, United States

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Kansas City, Kansas, 66160, United States

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Wichita, Kansas, 67214, United States

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Louisville, Kentucky, 40202, United States

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Monroe, Louisiana, 71201, United States

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New Orleans, Louisiana, 70121, United States

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Shreveport, Louisiana, 71101, United States

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Boston, Massachusetts, 02111, United States

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Springfield, Massachusetts, 01107, United States

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Ann Arbor, Michigan, 48109, United States

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Detroit, Michigan, 48202, United States

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Minneapolis, Minnesota, 55404, United States

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Minneapolis, Minnesota, 55455, United States

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Rochester, Minnesota, 55902, United States

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Travere Investigational Site

Kansas City, Missouri, 64108, United States

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Travere Investigational Site

Kansas City, Missouri, 64111, United States

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Travere Investigational Site

Las Vegas, Nevada, 89129, United States

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Reno, Nevada, 89511, United States

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Hackensack, New Jersey, 07601, United States

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Fresh Meadows, New York, 11365, United States

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New Hyde Park, New York, 11040, United States

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Travere Investigational Site

New York, New York, 10016, United States

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Travere Investigational Site

New York, New York, 10029, United States

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Travere Investigational Site

New York, New York, 10032, United States

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The Bronx, New York, 10467, United States

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Chapel Hill, North Carolina, 27514, United States

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Durham, North Carolina, 27710, United States

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Raleigh, North Carolina, 27609, United States

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Winston-Salem, North Carolina, 27103, United States

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Cleveland, Ohio, 44195, United States

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Columbus, Ohio, 43210, United States

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Oklahoma City, Oklahoma, 73104, United States

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Roseburg, Oregon, 97471, United States

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Bethlehem, Pennsylvania, 18017, United States

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Camp Hill, Pennsylvania, 17011, United States

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Philadelphia, Pennsylvania, 19104, United States

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Pittsburgh, Pennsylvania, 15224, United States

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Upland, Pennsylvania, 19013, United States

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Columbia, South Carolina, 29203, United States

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Memphis, Tennessee, 38103, United States

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Corpus Christi, Texas, 78412, United States

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Dallas, Texas, 75231, United States

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Dallas, Texas, 75235, United States

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Dallas, Texas, 75246, United States

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Travere Investigational Site

El Paso, Texas, 79902, United States

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Fort Worth, Texas, 76104, United States

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Houston, Texas, 77030, United States

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Houston, Texas, 77054, United States

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Lewisville, Texas, 75057, United States

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Sherman, Texas, 75090, United States

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Salt Lake City, Utah, 84112, United States

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Salt Lake City, Utah, 84115, United States

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St. George, Utah, 84790, United States

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Hampton, Virginia, 23666, United States

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Spokane, Washington, 99204, United States

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Morgantown, West Virginia, 26506, United States

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Marshfield, Wisconsin, 54449, United States

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Wauwatosa, Wisconsin, 53226, United States

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Buenos Aires, C1280AEB, Argentina

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Córdoba, X5000JHGQ, Argentina

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Córdoba, X5016LIG, Argentina

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Santa Fe, S3000, Argentina

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Concord, New South Wales, 2139, Australia

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New Lambton Heights, New South Wales, 2305, Australia

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Saint Leonards, New South Wales, 2065, Australia

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Wollongong, New South Wales, 2522, Australia

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Birtinya, Queensland, 4575, Australia

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Woolloongabba, Queensland, 4102, Australia

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Adelaide, South Australia, 5000, Australia

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Parkville, Victoria, 3050, Australia

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Nedlands, Western Australia, 6009, Australia

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Leuven, 3000, Belgium

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Liège, 4000, Belgium

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Roeselare, 8800, Belgium

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Travere Investigational Site

Botucatu, 18618-686, Brazil

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Travere Investigational Site

Itaquera, 08270-120, Brazil

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Travere Investigational Site

Passo Fundo, 99010-080, Brazil

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Porto Alegre, 90035-903, Brazil

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Recife, 50670-901, Brazil

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Rio de Janeiro, 20551-030, Brazil

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São Paulo, 04038-002, Brazil

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Travere Investigational Site

São Paulo, 05403-000, Brazil

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Travere Investigational Site

Edmonton, Alberta, T6G 2B7, Canada

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London, Ontario, N6A 5A5, Canada

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Greenfield Park, Quebec, J4V 2H1, Canada

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Travere Investigational Site

Zagreb, 10000, Croatia

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Prague, Prague, 100 34, Czechia

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Prague, Prague, 120 00, Czechia

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Nový Jičín, 74101, Czechia

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Travere Investigational Site

Aarhus, Central Jutland, 8200, Denmark

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Kolding, Southern Denmark, 6000, Denmark

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Tallinn, 10617, Estonia

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Tartu, 50406, Estonia

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Bordeaux, 33076, France

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Clermont-Ferrand, 63003, France

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Créteil, 94000, France

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Grenoble, 38043, France

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Marseille, 13005, France

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Nice, 06001, France

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Paris, 75010, France

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Paris, 75015, France

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Paris, 75743, France

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Saint-Priest-en-Jarez, 42270, France

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Toulouse, 31059, France

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Valenciennes, 59322, France

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Düsseldorf, Westfalen, 40210, Germany

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Aachen, 52074, Germany

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Berlin, 10117, Germany

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Berlin, 12203, Germany

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Hanover, 30625, Germany

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Stuttgart, 70376, Germany

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Travere Investigational Site

Villingen-Schwenningen, 78052, Germany

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Hong Kong, Hong Kong

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Lai Chi Kok, Hong Kong

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Bari, 70124, Italy

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Bergamo, 24127, Italy

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Bologna, 40138, Italy

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Florence, 50134, Italy

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Genova, 16132, Italy

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Germaneto, 88100, Italy

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Lecco, 23900, Italy

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Milan, 20122, Italy

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Monza, 20900, Italy

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Pavia, 27100, Italy

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Roma, 168, Italy

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Verona, 37126, Italy

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Auckland, 1051, New Zealand

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Hamilton, 3204, New Zealand

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Lodz, 93-347, Poland

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Olsztyn, 10-117, Poland

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Olsztyn, 10-561, Poland

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Piotrkow Trybunalski, 97-300, Poland

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Warsaw, 00-631, Poland

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Warsaw, 04-749, Poland

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Wroclaw, 50-556, Poland

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Travere Investigational Site

Amadora, 2720-276, Portugal

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Carnaxide, 2790-134, Portugal

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Lisbon, 1050-099, Portugal

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Lisbon, 1649-035, Portugal

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Loures, 2674-514, Portugal

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Porto, 4200-319, Portugal

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Setúbal, 2910-446, Portugal

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Vila Nova de Gaia, 4434-502, Portugal

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Travere Investigational Site

Busan, 47392, South Korea

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Daejeon, 35015, South Korea

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Gyeonggi-do, 13620, South Korea

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Travere Investigational Site

Gyeonggi-do, 14068, South Korea

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Seoul, 3080, South Korea

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Seoul, 3722, South Korea

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Palma de Mallorca, Balearic Islands, 07120, Spain

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Lugo, Burela, 27880, Spain

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Sagunto, Valencia, 46520, Spain

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Badalona, 8916, Spain

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Barcelona, 08003, Spain

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Barcelona, 08025, Spain

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Barcelona, 08035, Spain

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Barcelona, 08036, Spain

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Ciudad Real, 13005, Spain

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Córdoba, 14004, Spain

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Madrid, 28040, Spain

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Madrid, 28041, Spain

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Majadahonda, 28222, Spain

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Málaga, 29010, Spain

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Santiago de Compostela, 15706, Spain

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Seville, 41009, Spain

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Seville, 41013, Spain

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Valencia, 46014, Spain

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Valencia, 46017, Spain

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Zaragoza, 50009, Spain

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Solna, SE-171 64, Sweden

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Uppsala, 75237, Sweden

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Travere Investigational Site

Uppsala, SE-751 85, Sweden

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Travere Investigational Site

Hualien City, 970, Taiwan

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Kaohsiung City, 81362, Taiwan

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New Taipei City, 235, Taiwan

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Taichung, 404, Taiwan

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Taichung, 40705, Taiwan

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Tainan, 710, Taiwan

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Taipei, 10048, Taiwan

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Taipei, 104, Taiwan

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Taipei, 110, Taiwan

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Travere Investigational Site

Taoyuan District, 333, Taiwan

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Carshalton, London, SM5 1AA, United Kingdom

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Whitechapel, London, E1 1BB, United Kingdom

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Travere Investigational Site

Fulwood, Preston, PR2 9HT, United Kingdom

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Brighton, BN2 5BE, United Kingdom

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Cambridge, CB2 0QQ, United Kingdom

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Cardiff, CF14 4XW, United Kingdom

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Leicester, LE5 4PW, United Kingdom

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London, NW3 2QG, United Kingdom

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London, SE5 9RS, United Kingdom

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Manchester, M13 9WL, United Kingdom

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Newcastle, NE7 7DN, United Kingdom

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Reading, RG1 5AN, United Kingdom

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Salford, M6 8HD, United Kingdom

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Swansea, SA6 6NL, United Kingdom

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York, YO31 8HE, United Kingdom

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Related Publications (6)

  • Yee J, Gong W, Inrig J, Rheault MN, Gruber AJ, Bedard PW, Komers R, Trachtman H. Antiproteinuric Effect of Sparsentan in Patients with Genetic-Associated FSGS Enrolled in the DUPLEX Trial. Clin J Am Soc Nephrol. 2025 Dec 23. doi: 10.2215/CJN.0000000948. Online ahead of print. No abstract available.

  • Rheault MN. Treatment Approaches for Alport Syndrome. J Am Soc Nephrol. 2026 Jan 1;37(1):172-179. doi: 10.1681/ASN.0000000897. Epub 2025 Sep 12.

  • Liu ID, Willis NS, Craig JC, Hodson EM. Interventions for idiopathic steroid-resistant nephrotic syndrome in children. Cochrane Database Syst Rev. 2025 May 8;5(5):CD003594. doi: 10.1002/14651858.CD003594.pub7.

  • Rheault MN, Alpers CE, Barratt J, Bieler S, Canetta P, Chae DW, Coppock G, Diva U, Gesualdo L, Heerspink HJL, Inrig JK, Kirsztajn GM, Kohan D, Komers R, Kooienga LA, Lieberman K, Mercer A, Noronha IL, Perkovic V, Radhakrishnan J, Rote W, Rovin B, Tesar V, Trimarchi H, Tumlin J, Wong MG, Trachtman H; DUPRO Steering Committee and DUPLEX Investigators. Sparsentan versus Irbesartan in Focal Segmental Glomerulosclerosis. N Engl J Med. 2023 Dec 28;389(26):2436-2445. doi: 10.1056/NEJMoa2308550. Epub 2023 Nov 3.

  • Obadina M, Wilson S, Derebail VK, Little J. Emerging Therapies and Advances in Sickle Cell Disease with a Focus on Renal Manifestations. Kidney360. 2023 Jul 1;4(7):997-1005. doi: 10.34067/KID.0000000000000162. Epub 2023 May 31.

  • Hodson EM, Sinha A, Cooper TE. Interventions for focal segmental glomerulosclerosis in adults. Cochrane Database Syst Rev. 2022 Feb 28;2(2):CD003233. doi: 10.1002/14651858.CD003233.pub3.

Related Links

MeSH Terms

Conditions

Glomerulosclerosis, Focal Segmental

Interventions

sparsentanIrbesartan

Condition Hierarchy (Ancestors)

GlomerulonephritisNephritisKidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

Biphenyl CompoundsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsSpiro CompoundsTetrazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPolycyclic Compounds

Results Point of Contact

Title
Travere Therapeutics Call Center
Organization
Travere Therapeutics, Inc

Study Officials

  • Radko Komers, MD, PhD

    Travere Therapeutics, Inc.

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 3, 2018

First Posted

April 10, 2018

Study Start

April 17, 2018

Primary Completion

March 20, 2023

Study Completion

March 19, 2026

Last Updated

April 17, 2026

Results First Posted

April 30, 2024

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will share

Requests for clinical trial data, including language stating its intended use, should be directed to datarequest@travere.com. If approved, the requested information will be provided to the requestor after signing a data access agreement. Requests can be made following completion of the study and full publication of the study data in a peer reviewed journal for up to 36 months following its publication. Travere reserves the right to decline or recommend modifications to a request if it does not comply with the data sharing policy or if it is determined that the request is made by a biased source.

Time Frame
Requests can be made following completion of the study and full publication of the study data in a peer reviewed journal for up to 36 months following its publication.
Access Criteria
Requires submission and approval of intended use and a data sharing agreement.

Locations