NCT03402087

Brief Summary

The purpose of this study is to investigate effects of BMS-986165 on blood levels of methotrexate given as a single dose in healthy male patients.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
30

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started Jan 2018

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 5, 2018

Completed
3 days until next milestone

Study Start

First participant enrolled

January 8, 2018

Completed
10 days until next milestone

First Posted

Study publicly available on registry

January 18, 2018

Completed
2 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 20, 2018

Completed
5 days until next milestone

Study Completion

Last participant's last visit for all outcomes

March 25, 2018

Completed
Last Updated

February 25, 2020

Status Verified

February 1, 2020

Enrollment Period

2 months

First QC Date

January 5, 2018

Last Update Submit

February 24, 2020

Conditions

Outcome Measures

Primary Outcomes (7)

  • Maximum observed plasma concentration (Cmax)

    Approximately 14 days

  • Time to attain maximum observed plasma concentration (Tmax)

    Approximately 14 days

  • Area under the plasma concentration-time curve up to time T, where T is the last point with concentrations above the lower limit of quantitation [AUC(0-T)]

    Approximately 14 days

  • Area under the plasma concentration-time curve from time 0 to infinity [AUC(INF)]

    Approximately 14 days

  • Terminal elimination rate constant (kel)

    Approximately 14 days

  • Terminal elimination half life, calculated as 0.693/kel (T-HALF)

    Approximately 14 days

  • Apparent oral clearance (CL/F)

    Approximately 14 days

Secondary Outcomes (2)

  • Incidence of adverse events (AEs)

    Approximately 19 days

  • Incidence of serious adverse events (SAEs)

    Approximately 19 days

Study Arms (1)

BMS-986165+Methotrexate+Leucovorin

EXPERIMENTAL

Three treatments administered

Drug: MethotrexateDrug: LeucovorinDrug: BMS-986165

Interventions

Specified dose on specified days

Also known as: MTX
BMS-986165+Methotrexate+Leucovorin

Specified dose on specified days

Also known as: LEU
BMS-986165+Methotrexate+Leucovorin

Specified dose on specified days

BMS-986165+Methotrexate+Leucovorin

Eligibility Criteria

Age18 Years - 50 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Body Mass Index (BMI): 18.0 - 32.0 kg/m2
  • Normal renal function at screening

You may not qualify if:

  • Any medical condition that presents a potential risk to the participant and/or that may compromise the objectives of the study, including active, or history of, liver disease
  • Any contraindication indicated in the MTX package insert
  • History or presence of chronic bacterial or viral infection
  • History or presence of an autoimmune disorder
  • Any significant acute or chronic medical illness
  • Active TB requiring treatment or documented latent TB within the previous 3 years
  • Current or recent (within 3 months of study treatment administration) gastrointestinal disease that could affect absorption

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

PRA Health Sciences

Groningen, 9728 NZ, Netherlands

Location

Related Links

MeSH Terms

Conditions

Arthritis, Psoriatic

Interventions

MethotrexateLeucovorindeucravacitinib

Condition Hierarchy (Ancestors)

SpondylarthropathiesSpondylarthritisSpondylitisSpinal DiseasesBone DiseasesMusculoskeletal DiseasesArthritisJoint DiseasesPsoriasisSkin Diseases, PapulosquamousSkin DiseasesSkin and Connective Tissue Diseases

Intervention Hierarchy (Ancestors)

AminopterinPterinsPteridinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic CompoundsFormyltetrahydrofolatesTetrahydrofolatesFolic AcidCoenzymesEnzymes and Coenzymes

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 5, 2018

First Posted

January 18, 2018

Study Start

January 8, 2018

Primary Completion

March 20, 2018

Study Completion

March 25, 2018

Last Updated

February 25, 2020

Record last verified: 2020-02

Locations