NCT03373383

Brief Summary

The purpose of the study is to characterize the dose-response relationship with respect to efficacy of Padsevonil administered concomitantly with up to 3 anti-epileptic drugs (AEDs) for treatment of observable focal-onset seizures in subjects with drug-resistant epilepsy.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
411

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2018

Geographic Reach
19 countries

148 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

December 7, 2017

Completed
7 days until next milestone

First Posted

Study publicly available on registry

December 14, 2017

Completed
2 months until next milestone

Study Start

First participant enrolled

February 12, 2018

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 30, 2020

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 30, 2020

Completed
1.2 years until next milestone

Results Posted

Study results publicly available

April 9, 2021

Completed
Last Updated

December 19, 2023

Status Verified

December 1, 2023

Enrollment Period

2 years

First QC Date

December 7, 2017

Results QC Date

January 28, 2021

Last Update Submit

December 15, 2023

Conditions

Keywords

EpilepsyPadsevonil

Outcome Measures

Primary Outcomes (4)

  • Change in Log-transformed Observable Focal Onset Seizure Frequency From Baseline Over the 12 Week Maintenance Period

    During the study, participants kept diaries to record daily seizure activity. Seizure frequency refers to 28-day adjusted frequency. Seizure frequency was based on investigator assessment of participants' reports of daily seizure type and frequency. Observable focal-onset seizures refer to Type IA1, IB, and IC (ILAE Classification of Epileptic Seizures, 1981). Based on ANCOVA on change in log-transformed, 28-day adjusted seizure frequency from Baseline with treatment group as the main factor, Baseline log-transformed seizure frequency as a continuous covariate, Baseline SV2A use (yes or no) and Region (Europe, Non-Europe) as categorical factors.

    From Baseline over the 12 Week Maintenance Period

  • Percentage of Participants With Treatment-Emergent Adverse Events (TEAEs) Reported by the Subject and/or Caregiver or Observed by the Investigator During the Entire Study

    An Adverse Event is any untoward medical occurrence in a patient or clinical investigation subject administered a pharmaceutical product that does not necessarily have a causal relationship with this treatment.

    From Baseline until Safety Follow-Up (up to Week 23)

  • Percentage of Participants With Treatment-Emergent Adverse Events (TEAEs) Leading to Study Withdrawal

    An Adverse Event is any untoward medical occurrence in a patient or clinical investigation subject administered a pharmaceutical product that does not necessarily have a causal relationship with this treatment.

    From Baseline until Safety Follow-Up (up to Week 23)

  • Percentage of Participants With Treatment-Emergent Serious Adverse Events (SAEs) During the Entire Study

    A Serious Adverse Event (SAE) is any untoward medical occurrence that at any dose: * Results in death * Is life-threatening * Requires in patient hospitalization or prolongation of existing hospitalization * Is a congenital anomaly or birth defect * Is an infection that requires treatment parenteral antibiotics * Other important medical events which based on medical or scientific judgement may jeopardize the patients, or may require medical or surgical intervention to prevent any of the above.

    From Baseline until Safety Follow-Up (up to Week 23)

Secondary Outcomes (3)

  • 75 % Responder Rate Over the 12 Week Maintenance Period

    End of Maintenance Period (Week 16) following 3 Weeks of titration and 1 Week stabilization

  • 50 % Responder Rate Over the 12 Week Maintenance Period

    End of Maintenance Period (Week 16) following 3 Weeks of titration and 1 Week stabilization

  • Percent Change in Observable Focal-onset Seizure Frequency From Baseline Over the 12 Week Maintenance Period

    End of Maintenance Period (Week 16) following 3 Weeks of titration and 1 Week stabilization

Study Arms (5)

Padsevonil dosing regimen 1

EXPERIMENTAL

Subjects will be randomized to receive a combination of tablets of Padsevonil and Placebo (as appropriate) to maintain the blinding.

Drug: PadsevonilOther: Placebo

Padsevonil dosing regimen 2

EXPERIMENTAL

Subjects will be randomized to receive a combination of tablets of Padsevonil and Placebo (as appropriate) to maintain the blinding.

Drug: PadsevonilOther: Placebo

Padsevonil dosing regimen 3

EXPERIMENTAL

Subjects will be randomized to receive a combination of tablets of Padsevonil and Placebo (as appropriate) to maintain the blinding.

Drug: PadsevonilOther: Placebo

Padsevonil dosing regimen 4

EXPERIMENTAL

Subjects will be randomized to receive a combination of tablets of Padsevonil and Placebo (as appropriate) to maintain the blinding.

Drug: PadsevonilOther: Placebo

Placebo

PLACEBO COMPARATOR

Subjects randomized to the placebo group will receive a combination of several Placebo tablets to maintain the blinding.

Other: Placebo

Interventions

Padsevonil in different dosages.

Padsevonil dosing regimen 1Padsevonil dosing regimen 2Padsevonil dosing regimen 3Padsevonil dosing regimen 4
PlaceboOTHER

Placebo will be provided matching Padsevonil.

Padsevonil dosing regimen 1Padsevonil dosing regimen 2Padsevonil dosing regimen 3Padsevonil dosing regimen 4Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Diagnosis of focal epilepsy per 1989 International League Against Epilepsy (ILAE) criteria at least 3 years before study entry
  • Subject has failed to achieve seizure control with 4 tolerated and appropriately chosen prior antiepileptic drugs (AED), including past and ongoing treatment, that were individually optimized for adequate dose and duration. Prior discontinued AED treatment would need to be assessed by the Investigator considering the patient medical records and patient and/or caregiver interview. 'Prior AED' is defined as all past and ongoing AED treatments with a start date before the Screening Visit (Visit 1)
  • Average of \>= 4 spontaneous and observable focal seizures (type IA1 (i.e. focal aware), IB (i.e. focal impaired awareness), IC (i.e. focal to bilateral tonic-clonic)) per month
  • Current treatment with an individually optimized and stable dose of at least 1 and up to 3 AEDs for the 8 weeks prior to the Screening Visit with or without additional Vagus Nerve Stimulation (VNS) or other neurostimulation treatments

You may not qualify if:

  • Subject has a history of or signs of generalized or combined generalized and focal epilepsy
  • Cluster seizures which are uncountable in the previous 8 weeks before study entry and during 4 weeks prospective baseline
  • Current treatment with carbamazepine, phenytoin, primidone, phenobarbital
  • Current treatment/ use of (non-AED) prescription, nonprescription, dietary (eg, grapefruit or passion fruit), or herbal products that are potent inducers or inhibitors of the CYP3A4 or 2C19 pathway for 2 weeks (or 5 half-lives, whichever is longer) prior to the Baseline Visit
  • Subjects taking sensitive substrates of CYP2C19 for 2 weeks (or 5 half-lives, whichever is longer) prior to the Baseline Visit
  • Subject has been taking vigabatrin less than 2 years at study entry
  • Subject has been taking felbamate for less than 12 months
  • Subject taking retigabine for less than 4 years
  • Current treatment with benzodiazepines (i.e. GABA-A-ergic drugs like zolpidem, zaleplon, or zopiclone, excluding GABA-A-ergic AEDs) \<3 times per week for emergencies
  • Subject has a current medical condition that occurred within the last 12 months which, in the opinion of the investigator, could compromise his/her safety or ability to participate in this study

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (148)

Ep0091 839

Chandler, Arizona, 85226, United States

Location

Ep0091 810

Little Rock, Arkansas, 72205, United States

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Ep0091 815

La Jolla, California, 92037, United States

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Ep0091 801

San Francisco, California, 94115, United States

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Ep0091 845

Washington D.C., District of Columbia, 20037, United States

Location

Ep0091 809

Ocala, Florida, 34471, United States

Location

Ep0091 823

Orlando, Florida, 32806, United States

Location

Ep0091 825

Port Charlotte, Florida, 33952, United States

Location

Ep0091 820

Tallahassee, Florida, 32308, United States

Location

Ep0091 873

Atlanta, Georgia, 30303, United States

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Ep0091 803

Honolulu, Hawaii, 96817, United States

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Ep0091 832

Peoria, Illinois, 61637, United States

Location

Ep0091 822

Baltimore, Maryland, 21287, United States

Location

Ep0091 818

Bethesda, Maryland, 20817, United States

Location

Ep0091 817

Saint Paul, Minnesota, 55102, United States

Location

Ep0091 806

Hackensack, New Jersey, 07601, United States

Location

Ep0091 827

New York, New York, 10016-48, United States

Location

Ep0091 800

Philadelphia, Pennsylvania, 19104, United States

Location

Ep0091 802

Philadelphia, Pennsylvania, 19107, United States

Location

Ep0091 838

Cordova, Tennessee, 38018, United States

Location

Ep0091 835

Nashville, Tennessee, 37232, United States

Location

Ep0091 805

Austin, Texas, 78701, United States

Location

Ep0091 844

Austin, Texas, 78758, United States

Location

Ep0091 836

Dallas, Texas, 75231, United States

Location

Ep0091 830

Dallas, Texas, 75390-91, United States

Location

Ep0091 824

Round Rock, Texas, 78681, United States

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Ep0091 870

San Antonio, Texas, 78229, United States

Location

Ep0091 855

Box Hill, Australia

Location

Ep0091 857

Clayton, Australia

Location

Ep0091 850

Fitzroy, Australia

Location

Ep0091 859

Herston, Australia

Location

Ep0091 852

Melbourne, Australia

Location

Ep0091 853

Melbourne, Australia

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Ep0091 856

Randwick, Australia

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Westmead, Australia

Location

Ep0091 102

Bruges, Belgium

Location

Ep0091 101

Brussels, Belgium

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Ep0091 105

Ghent, Belgium

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Ep0091 100

Leuven, Belgium

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Ep0091 150

Blagoevgrad, Bulgaria

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Ep0091 151

Pleven, Bulgaria

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Ep0091 153

Pleven, Bulgaria

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Ep0091 152

Sofia, Bulgaria

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Ep0091 154

Sofia, Bulgaria

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Ep0091 155

Sofia, Bulgaria

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Ep0091 200

Greenfield Park, Canada

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Ep0091 205

London, Canada

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Ep0091 201

Montreal, Canada

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Ep0091 254

Brno, Czechia

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Ostrava-Poruba, Czechia

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Ep0091 250

Prague, Czechia

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Ep0091 251

Prague, Czechia

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Ep0091 252

Prague, Czechia

Location

Ep0091 253

Prague, Czechia

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Ep0091 307

Clermont-Ferrand, France

Location

Ep0091 309

Dijon, France

Location

Ep0091 300

Lille, France

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Ep0091 302

Montpellier, France

Location

Ep0091 305

Paris, France

Location

Ep0091 303

Rennes, France

Location

Ep0091 306

Toulouse, France

Location

Ep0091 361

Bad Neustadt an der Saale, Germany

Location

Ep0091 365

Berlin, Germany

Location

Ep0091 362

Bernau, Germany

Location

Ep0091 363

Bielefeld, Germany

Location

Ep0091 358

Bonn, Germany

Location

Ep0091 350

Frankfurt am Main, Germany

Location

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Freiburg im Breisgau, Germany

Location

Ep0091 364

Hamburg, Germany

Location

Ep0091 368

Jena, Germany

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Ep0091 366

Kork, Germany

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Ep0091 357

Leipzig, Germany

Location

Ep0091 353

Marburg, Germany

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Ep0091 354

München, Germany

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Ep0091 351

Münster, Germany

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Ep0091 356

Osnabrück, Germany

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Ep0091 367

Ravensburg, Germany

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Ep0091 301

Strausberg, Germany

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Ep0091 352

Tübingen, Germany

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Ep0091 400

Budapest, Hungary

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Ep0091 403

Budapest, Hungary

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Ep0091 402

Debrecen, Hungary

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Ep0091 462

Bologna, Italy

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Ep0091 450

Cagliari, Italy

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Ep0091 461

Foggia, Italy

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Milan, Italy

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Ep0091 459

Pavia, Italy

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Ep0091 453

Perugia, Italy

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Pozzilli, Italy

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Reggio Calabria, Italy

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Ep0091 455

Roma, Italy

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Ep0091 457

Roma, Italy

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Ep0091 460

Roma, Italy

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Ep0091 501

Asaka, Japan

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Ep0091 511

Fukuoka, Japan

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Ep0091 505

Hiroshima, Japan

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Ep0091 513

Hōfu, Japan

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Ep0091 507

Itami, Japan

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Ep0091 503

Kodaira, Japan

Location

Ep0091 514

Kyoto, Japan

Location

Ep0091 512

Nagakute, Japan

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Ep0091 510

Niigata, Japan

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Ep0091 515

Saitama, Japan

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Ep0091 509

Shizuoka, Japan

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Ep0091 703

Kaunas, Lithuania

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Ep0091 701

Vilnius, Lithuania

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Ep0091 702

Vilnius, Lithuania

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Ep0091 553

Culiacán, Mexico

Location

Ep0091 552

Mexico City, Mexico

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Ep0091 601

Gdansk, Poland

Location

Ep0091 607

Grodzisk Mazowiecki, Poland

Location

Ep0091 605

Katowice, Poland

Location

Ep0091 608

Katowice, Poland

Location

Ep0091 603

Krakow, Poland

Location

Ep0091 604

Lublin, Poland

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Ep0091 606

Nowa Sól, Poland

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Ep0091 600

Poznan, Poland

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Ep0091 609

Poznan, Poland

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Ep0091 602

Świdnik, Poland

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Ep0091 952

Santa Maria da Feira, Portugal

Location

Ep0091 004

Bardejov, Slovakia

Location

Ep0091 001

Hlohovec, Slovakia

Location

Ep0091 662

Alicante, Spain

Location

Ep0091 651

Barcelona, Spain

Location

Ep0091 652

Barcelona, Spain

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Ep0091 658

Barcelona, Spain

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Ep0091 664

Barcelona, Spain

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Ep0091 668

Bilbao, Spain

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Ep0091 666

Córdoba, Spain

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Ep0091 650

Madrid, Spain

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Ep0091 656

Madrid, Spain

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Ep0091 660

Madrid, Spain

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Ep0091 661

Madrid, Spain

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Ep0091 659

Málaga, Spain

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Ep0091 663

Seville, Spain

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Ep0091 665

Terrassa, Spain

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Ep0091 657

Valencia, Spain

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Ep0091 667

Valencia, Spain

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Ep0091 653

Valladolid, Spain

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Ep0091 904

Eskişehir, Turkey (Türkiye)

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Ep0091 900

Istanbul, Turkey (Türkiye)

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Ep0091 901

Istanbul, Turkey (Türkiye)

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Ep0091 752

Birmingham, United Kingdom

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Ep0091 751

Cardiff, United Kingdom

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Ep0091 756

Inverness, United Kingdom

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Ep0091 757

London, United Kingdom

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Ep0091 750

Manchester, United Kingdom

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Ep0091 753

Swansea, United Kingdom

Location

Related Publications (2)

  • Rademacher M, Toledo M, Van Paesschen W, Liow KK, Milanov IG, Esch ML, Wang N, MacPherson M, Byrnes WJ, Minh TDC, Webster E, Werhahn KJ. Efficacy and safety of adjunctive padsevonil in adults with drug-resistant focal epilepsy: Results from two double-blind, randomized, placebo-controlled trials. Epilepsia Open. 2022 Dec;7(4):758-770. doi: 10.1002/epi4.12656. Epub 2022 Oct 22.

  • Kramer H, Bicer C, Otoul C, Rospo C, Macpherson M, Watling M, Bani M, Sciberras D, Chanteux H. Clinical Bridging Studies and Modeling Approach for Implementation of a Patient Centric Sampling Technique in Padsevonil Clinical Development. AAPS J. 2023 Nov 16;26(1):1. doi: 10.1208/s12248-023-00866-7.

MeSH Terms

Conditions

Drug Resistant EpilepsySeizuresEpilepsy

Interventions

padsevonil

Condition Hierarchy (Ancestors)

Brain DiseasesCentral Nervous System DiseasesNervous System DiseasesNeurologic ManifestationsSigns and SymptomsPathological Conditions, Signs and Symptoms

Results Point of Contact

Title
UCB
Organization
Cares

Study Officials

  • UCB Cares

    001 844 599 2273 (UCB)

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
GT60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 7, 2017

First Posted

December 14, 2017

Study Start

February 12, 2018

Primary Completion

January 30, 2020

Study Completion

January 30, 2020

Last Updated

December 19, 2023

Results First Posted

April 9, 2021

Record last verified: 2023-12

Data Sharing

IPD Sharing
Will share

Data from this trial may be requested by qualified researchers six months after product approval in the US and/or Europe, or global development is discontinued, and 18 months after trial completion. Investigators may request access to anonymized individual patient-level data and redacted trial documents which may include: analysis-ready datasets, study protocol, annotated case report form, statistical analysis plan, dataset specifications, and clinical study report. Prior to use of the data, proposals need to be approved by an independent review panel at www.Vivli.org and a signed data sharing agreement will need to be executed. All documents are available in English only, for a prespecified time, typically 12 months, on a password protected portal. This plan may change if the risk of re-identifying trial participants is determined to be too high after the trial is completed; in this case and to protect participants, individual patient-level data would not be made available.

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
Data from this trial may be requested by qualified researchers six months after product approval in the US and/or Europe or global development is discontinued, and 18 months after trial completion.
Access Criteria
Qualified researchers may request access to anonymized IPD and redacted study documents which may include: raw datasets, analysis-ready datasets, study protocol, blank case report form, annotated case report form, statistical analysis plan, dataset specifications, and clinical study report. Prior to use of the data, proposals need to be approved by an independent review panel at www.Vivli.org and a signed data sharing agreement will need to be executed. All documents are available in English only, for a pre-specified time, typically 12 months, on a password protected portal.
More information

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