NCT03346837

Brief Summary

Assess the effects of itraconazole and rifampin on the pharmacokinetics, safety, and tolerability of BMS-986205.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
53

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Nov 2017

Shorter than P25 for phase_1

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

November 6, 2017

Completed
11 days until next milestone

First Posted

Study publicly available on registry

November 17, 2017

Completed
5 days until next milestone

Study Start

First participant enrolled

November 22, 2017

Completed
28 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 20, 2017

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 20, 2017

Completed
Last Updated

February 28, 2018

Status Verified

February 1, 2018

Enrollment Period

28 days

First QC Date

November 6, 2017

Last Update Submit

February 26, 2018

Conditions

Outcome Measures

Primary Outcomes (3)

  • Maximum observed plasma concentration (Cmax)

    Measured by plasma concentration

    Up to 25 days

  • AUC from time zero to time of last quantifiable concentration (AUC(0-T))

    Measured by plasma concentration

    Up to 25 days

  • AUC from time zero extrapolated to infinite time (AUC(INF))

    Measured by plasma concentration

    Up to 25 days

Secondary Outcomes (5)

  • Incidence of Adverse Events (AEs)

    Up to 25 days

  • Incidence of Serious Adverse Events (SAEs)

    Up to 76 days

  • Number of participants with electrocardiogram abnormalities

    Up to 25 days

  • Number of participants with physical examination findings abnormalities

    Up to 25 days

  • Number of participants with clinical laboratory abnormalities

    Up to 25 days

Study Arms (4)

Inhibition (Cohort 1)

EXPERIMENTAL

Single oral dose BMS-986205

Drug: BMS-986205

Inhibition (Cohort 2)

EXPERIMENTAL

Daily oral itraconazole doses for 24 days; single oral dose BMS-986205 on day 4

Drug: BMS-986205Drug: Itraconazole

Induction (Cohort 3)

EXPERIMENTAL

Single oral dose BMS-986205

Drug: BMS-986205

Induction (Cohort 4)

EXPERIMENTAL

Daily oral rifampin doses for21 days; single oral dose BMS-986205 on day 8

Drug: BMS-986205Drug: Rifampin

Interventions

BMS-986205

Induction (Cohort 3)Induction (Cohort 4)Inhibition (Cohort 1)Inhibition (Cohort 2)

Oral solution

Inhibition (Cohort 2)

Tablet

Induction (Cohort 4)

Eligibility Criteria

Age18 Years - 50 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Body mass index 18.0 to 32.0 kg/m2, inclusive
  • Must have normal renal function demonstrated by GFR, calculated by Chronic Kidney Disease Epidemiology Collaboration formula
  • Women must not be of childbearing potential (cannot become pregnant)

You may not qualify if:

  • Any significant acute or chronic medical illness
  • History of glucose-6-phosphodiesterase (G6PD) deficiency
  • Personal or family history of cytochrome b5 reductase deficiency

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

PPD

Austin, Texas, 78744, United States

Location

Related Links

MeSH Terms

Interventions

linrodostatItraconazoleRifampin

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPiperazinesRifamycinsHeterocyclic Compounds, 4 or More RingsHeterocyclic Compounds, Fused-RingLactams, MacrocyclicMacrocyclic CompoundsPolycyclic Compounds

Study Officials

  • Bristol-Myers Squibb

    Briston-Myers Squibb

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
OTHER
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 6, 2017

First Posted

November 17, 2017

Study Start

November 22, 2017

Primary Completion

December 20, 2017

Study Completion

December 20, 2017

Last Updated

February 28, 2018

Record last verified: 2018-02

Locations