NCT02638948

Brief Summary

The purpose of this study is to determine whether the study drug, BMS-986142, is safe and effective in treating moderate to severe rheumatoid arthritis in subjects with an inadequate response to methotrexate or methotrexate and up to 2 tumour necrosis factor (TNF) Inhibitors. Patients who qualify will be randomized to either one of 3 doses of BMS-986142 or placebo in 1:1:1 randomization for 12 weeks. Disease activity and safety will be assessed over the course of the study.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
508

participants targeted

Target at P75+ for phase_2 rheumatoid-arthritis

Timeline
Completed

Started Feb 2016

Typical duration for phase_2 rheumatoid-arthritis

Geographic Reach
17 countries

104 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

December 21, 2015

Completed
2 days until next milestone

First Posted

Study publicly available on registry

December 23, 2015

Completed
2 months until next milestone

Study Start

First participant enrolled

February 16, 2016

Completed
2.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 3, 2018

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 3, 2018

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

May 28, 2019

Completed
Last Updated

May 28, 2019

Status Verified

May 1, 2019

Enrollment Period

2.2 years

First QC Date

December 21, 2015

Results QC Date

May 1, 2019

Last Update Submit

May 2, 2019

Conditions

Outcome Measures

Primary Outcomes (2)

  • Percentage of Participants Achieving American College of Rheumatology 20% (ACR20) Response at Week 12

    ACR responses are assessed with a composite rating scale of the American College of Rheumatology that includes 7 variables: tender joint count (TJC); swollen joint count (SJC); levels of an acute phase reactant C-reactive Protein levels (CRP); participant's assessment of pain; participant's global assessment of disease activity; physician's global assessment of disease activity; participant's assessment of physical function by health assessment questionnaire disability index (HAQ-DI). ACR20 is defined as achieving at least 20% improvement in both TJC and SJC, and at least 20% improvement in at least 3 of the 5 other assessments of the ACR. Percentage of Participants achieving ACR20 = (number of participants with measure/event of interest)/(number of particpants in the analysis)\*100

    Week 12

  • Percentage of Participants Achieving American College of Rheumatology 70% (ACR70) Response at Week 12

    ACR responses are assessed with a composite rating scale of the American College of Rheumatology that includes 7 variables: TJC; SJC; levels of an acute phase reactant (CRP level); participant's assessment of pain; participant's global assessment of disease activity; physician's global assessment of disease activity; participant's assessment of physical function by HAQ--DI. ACR70 is defined as achieving at least 70% improvement in both TJC and SJC, and at least 70% improvement in at least 3 of the 5 other assessments of the ACR. Percentage of Participants achieving ACR70 = (number of participants with measure/event of interest)/(number of particpants in the analysis)\*100

    Week 12

Secondary Outcomes (18)

  • Percentage of Participants Achieving American College of Rheumatology 20% Response Over Time From Baseline to Week 12

    Baseline, Day 15, Day 29, Day 57, Day 85

  • Percentage of Participants Achieving American College of Rheumatology 50% (ACR50) Response Over Time From Baseline to Week 12

    Baseline, Day 15, Day 29, Day 57, Day 85

  • Percentage of Participants Achieving American College of Rheumatology 70% Response Over Time From Baseline to Week 12

    Baseline, Day 15, Day 29, Day 57, Day 85

  • Percentage of Participants Achieving < 2.6 Response in Disease Activity Score for 28 Joints -C-Reactive Protein (DAS28--CRP) Score at Week 12

    Week 12

  • Percentage of Participants Achieving < 2.6 Response in Disease Activity Score for 28 Joints Erythrocyte Sedimentation Rate (DAS28--ESR) Score at Week 12

    Week 12

  • +13 more secondary outcomes

Study Arms (3)

Placebo

PLACEBO COMPARATOR

Placebo + Methotrexate dose as specified

Drug: PlaceboDrug: Methotrexate

Dose Level 1

EXPERIMENTAL

BMS-986142 at dose level 1+ Methotrexate as specified

Drug: BMS-986142Drug: Methotrexate

Dose Level 2

EXPERIMENTAL

BMS-986142 at dose level 2 + Methotrexate as specified

Drug: BMS-986142Drug: Methotrexate

Interventions

BMS986142 specific dose on specific days

Dose Level 1Dose Level 2

Placebo of BMS-986142 specific dose on specific days

Placebo

Methotrexate specific dose on specific days

Dose Level 1Dose Level 2Placebo

Eligibility Criteria

Age18 Years - 120 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Male and female age 18 and above
  • Diagnosed with active rheumatoid arthritis (RA) by standard criteria at least 16 weeks before screening, have functional ACR class I-III
  • Have an inadequate response to methotrexate
  • In addition to an inadequate response to methotrexate have an inadequate response or intolerance to 1 but not more than 2 TNF inhibitors
  • Have a minimum of 6 swollen and 6 tender joints (from 66/68 joint count)
  • Have hsCRP of ≥ 0.8 mg/dL (8mg/L) \[by central laboratory values\] or an ESR ≥ 28 mm/hr
  • Willing to use effective birth control for the entire length of the study

You may not qualify if:

  • Diagnosed with juvenile Rheumatoid Arthritis
  • Have been treated with other biologic treatment than a TNF inhibitor
  • Active systemic bacterial, viral or fungal infection or evidence of prior or current Hepatitis B or C infection or HIV infection, latent bacterial, viral or fungal infections
  • Have been treated with Intramuscular or Intra-articular glucocorticosteroids within 4 weeks of randomization
  • Taking Oral steroids at dose above 10 mg/day of prednisone (or prednisone equivalents)
  • Have other autoimmune disease other than RA like lupus, multiple sclerosis
  • Have significant concurrent medical condition at the time of screening or baseline visit

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (104)

Rheumatology Associates Of North Alabama, P.C.

Huntsville, Alabama, 35801, United States

Location

St. Joseph Heritage Medical Group

Fullerton, California, 92835, United States

Location

C.V Mehta M.D Medical Corp

Hemet, California, 92543, United States

Location

HCP Clinical Research, LLC

Huntington Beach, California, 92646, United States

Location

Leon Medical Research

Miami, Florida, 33015, United States

Location

San Marcus Research Clinic, Inc.

Miami, Florida, 33015, United States

Location

Coral Research Clinic Corp

Miami, Florida, 33175, United States

Location

Precision Research Organization

Miami Lakes, Florida, 33016, United States

Location

The Arthritis Center

Palm Harbor, Florida, 34684, United States

Location

Vizae Clinical Trials Management

Pembroke Pines, Florida, 33026, United States

Location

Integral Rheumatology & Immunology Specialists

Plantation, Florida, 33324, United States

Location

North Georgia Rheumatology Group

Lawrenceville, Georgia, 30046, United States

Location

Arthritis And Diabetes Clinic

Monroe, Louisiana, 71203, United States

Location

Clinical Pharmacology Study Group

Worcester, Massachusetts, 01605, United States

Location

Aa Mrc Llc

Grand Blanc, Michigan, 48439, United States

Location

Albuquerque Center For Rheumatology

Albuquerque, New Mexico, 87102, United States

Location

Albuquerque Clinical Trials

Albuquerque, New Mexico, 87102, United States

Location

Paramount Medical Research & Consulting, Llc

Middleburg Heights, Ohio, 44130, United States

Location

East Penn Rheumatology

Bethlehem, Pennsylvania, 18015, United States

Location

Altoona Center For Clinical Research

Duncansville, Pennsylvania, 16635-8406, United States

Location

Advanced Rheumatology & Arthritis Research Center, P.C

Wexford, Pennsylvania, 15090, United States

Location

Local Institution

Wyomissing, Pennsylvania, 19610, United States

Location

West Tennessee Research Institute

Jackson, Tennessee, 38305, United States

Location

Pharma Tex Research

Amarillo, Texas, 79106, United States

Location

Tekton Research Inc

Austin, Texas, 78745, United States

Location

Southwest Rheumatology Research LLC

Mesquite, Texas, 75150, United States

Location

Local Institution

Capital Federal, Buenos Aires, 1015, Argentina

Location

Aprillus Asistencia e Investigacion

Capital Federal, Buenos Aires, Argentina

Location

Instituto De Rehabilitacion Psicofisica

Buenos Aires, 1428, Argentina

Location

Instituto Reumatologico Strusberg

Córdoba, 5000, Argentina

Location

Universitaetsklinik Fuer Innere Medizin 3

Vienna, 1090, Austria

Location

Local Institution

Goiânia, Goiás, 74110-120, Brazil

Location

Local Institution

Juiz de Fora, Minas Gerais, 36010570, Brazil

Location

Local Institution

Curitiba, Paraná, 80030-110, Brazil

Location

Local Institution

Porto Alegre, Rio Grande do Sul, 90035-903, Brazil

Location

Local Institution

Porto Alegre, Rio Grande do Sul, 90480-000, Brazil

Location

Local Institution

Santo André, São Paulo, 09190510, Brazil

Location

Local Institution

São Paulo, 04032-060, Brazil

Location

Local Institution

São Paulo, 04266-010, Brazil

Location

Aggarwal And Associates

Brampton, Ontario, L6T 0G1, Canada

Location

Dr. Anil K Gupta Med Prof Corp

Toronto, Ontario, M9V 4B4, Canada

Location

Local Institution

Corbeil-Essonnes, 91100, France

Location

Local Institution

Montpellier, 34295, France

Location

Local Institution

Orléans, 45067, France

Location

Local Institution

Strasbourg, 67098, France

Location

Asklepios Gesundheitszentrum

Elmshorn, Germany

Location

Medizinsche Universitaetsklinik Freiburg

Freiburg im Breisgau, 79106, Germany

Location

Smo.Md Gmbh

Magdeburg, 39120, Germany

Location

Local Institution

Florence, 50139, Italy

Location

Local Institution

Padua, 35128, Italy

Location

Local Institution

Nagoya, Aichi-ken, 4578511, Japan

Location

Local Institution

Fukuoka, Fukuoka, 8108563, Japan

Location

Local Institution

Kitakyushu-shi, Fukuoka, 8078555, Japan

Location

Local Institution

Sapporo, Hokkaido, 0608604, Japan

Location

Local Institution

Sapporo, Hokkaido, 0608648, Japan

Location

Local Institution

Sapporo, Hokkaido, 0630811, Japan

Location

Local Institution

Kato-shi, Hyōgo, 6731462, Japan

Location

Local Institution

Sagamihara-shi, Kanagawa, 2520392, Japan

Location

Local Institution

Kumamoto, Kumamoto, 8620976, Japan

Location

Local Institution

Sendai, Miyagi, 9808574, Japan

Location

Local Institution

Sasebo-shi, Nagasaki, 8571195, Japan

Location

Local Institution

Kawachi-Nagano, Osaka, 5868521, Japan

Location

Local Institution

Osaka, Osaka, 5458586, Japan

Location

Local Institution

Iruma-gun, Saitama, 3500495, Japan

Location

Local Institution

Kawagoe-shi, Saitama, 3508550, Japan

Location

Local Institution

Hamamatsu, Shizuoka, 4308558, Japan

Location

Local Institution

Chuo-ku, Tokyo, 1048560, Japan

Location

Local Institution

Itabashi-ku, Tokyo, 1738610, Japan

Location

Local Institution

Meguro-ku, Tokyo, 1538515, Japan

Location

Local Institution

Shinjuku-Ku, Tokyo, 1608582, Japan

Location

Local Institution

Osaki-shi, 9896183, Japan

Location

CINTRE - Centro de investigacion y tratamiento reumatologico, S.C.

Mexico City, Distrito Fededral, 11850, Mexico

Location

Consultorio Privado de Especialidad

Guadalajara, Jalisco, 42650, Mexico

Location

Clinica de Investigacion en Reumatologia y Obesidad S.C.

Guadalajara, Jalisco, 44650, Mexico

Location

Local Institution

Monterrey, Nuevo León, 64460, Mexico

Location

Local Institution

Villahermosa, Tabasco, 86190, Mexico

Location

Unidad Reumatologica Las Americas, S.C. P.

Mérida, Yucatán, 97000, Mexico

Location

Centro de Alta Especialidad en Reumatologia e Investigacion del Potosi S.C.

Distrito Federal, 03100, Mexico

Location

Maasstad Ziekenhuis Rotterdam

Rotterdam, 3079 DZ, Netherlands

Location

Nzoz Osteo-Medic S.C. A. Racewicz, J.Supronik

Bialystok, 15-351, Poland

Location

Local Institution

Bialystok, 15-879, Poland

Location

Centrum Badan Klinicznych JCI Life Science Park

Krakow, 30-348, Poland

Location

Local Institution

Lublin, 20-954, Poland

Location

Local Institution

Nadarzyn, 05-830, Poland

Location

Local Institution

Poznan, 60-218, Poland

Location

Local Institution

Warsaw, 00-465, Poland

Location

Narodowy Instytut Geriatrii, Reumatologii i Rehabilitacji

Warsaw, 02-637, Poland

Location

Local Institution

Warsaw, 02-691, Poland

Location

Local Institution

Moscow, 119049, Russia

Location

Local Institution

Moscow, 121374, Russia

Location

Local Institution

Saint Petersburg, 191124, Russia

Location

Local Institution

Saint Petersburg, 194356, Russia

Location

Local Institution

Tolyatti, 445039, Russia

Location

Local Institution

Benoni, Gauteng, 1500, South Africa

Location

Local Institution

Cape Town, Western Cape, 7500, South Africa

Location

Local Institution

George, Western Cape, 6529, South Africa

Location

Local Institution

Somerset West, Western Cape, 7129, South Africa

Location

Local Institution

Daegu, 41931, South Korea

Location

Local Institution

Seoul, 03080, South Korea

Location

Local Institution

A Coruña, 15006, Spain

Location

Fundacion Jimenez Diaz

Madrid, 28040, Spain

Location

Local Institution

Santiago Compostela, 15702, Spain

Location

Local Institution

Taichung, 402, Taiwan

Location

Local Institution

Taipei, 11031, Taiwan

Location

Related Publications (1)

  • Conaghan PG, Nowak M, Du S, Luo Y, Landis J, Pachai C, Fura A, Catlett IM, Grasela DM, Ostergaard M. Evaluation of BMS-986142, a reversible Bruton's tyrosine kinase inhibitor, for the treatment of rheumatoid arthritis: a phase 2, randomised, double-blind, dose-ranging, placebo-controlled, adaptive design study. Lancet Rheumatol. 2023 May;5(5):e263-e273. doi: 10.1016/S2665-9913(23)00089-9.

Related Links

MeSH Terms

Conditions

Arthritis, Rheumatoid

Interventions

Methotrexate

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic DiseasesConnective Tissue DiseasesSkin and Connective Tissue DiseasesAutoimmune DiseasesImmune System Diseases

Intervention Hierarchy (Ancestors)

AminopterinPterinsPteridinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Results Point of Contact

Title
Bristol-Myers Squibb Study Director
Organization
Bristol-Myers Squibb Study Director

Study Officials

  • Bristol Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

December 21, 2015

First Posted

December 23, 2015

Study Start

February 16, 2016

Primary Completion

May 3, 2018

Study Completion

May 3, 2018

Last Updated

May 28, 2019

Results First Posted

May 28, 2019

Record last verified: 2019-05

Locations