NCT02085538

Brief Summary

Since the amount of palbociclib eliminated in urine is 6.9%, renal impairment is not expected to have much impact on palbociclib. However, the Federal Drug Administration (FDA) Guidance recommends a study in subjects with renal impairment when the drug is likely to be used in patients with impaired renal function. Palbociclib is intended for chronic use in cancer patients who may have some degree of impaired renal function.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
31

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started May 2014

Typical duration for phase_1

Geographic Reach
1 country

3 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 11, 2014

Completed
2 days until next milestone

First Posted

Study publicly available on registry

March 13, 2014

Completed
2 months until next milestone

Study Start

First participant enrolled

May 1, 2014

Completed
2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 1, 2016

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2016

Completed
Last Updated

April 30, 2018

Status Verified

April 1, 2018

Enrollment Period

2 years

First QC Date

March 11, 2014

Last Update Submit

April 26, 2018

Conditions

Keywords

renal impairmentAUCCmaxpalbociclibnormal matched subjects

Outcome Measures

Primary Outcomes (2)

  • Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUC (0 - 8)]

    AUC (0 - 8)= Area under the plasma concentration versus time curve (AUC) from time zero (pre-dose) to extrapolated infinite time (0 - 8). It is obtained from AUC (0 - t) plus AUC (t - 8).

    8 days

  • Maximum Observed Plasma Concentration (Cmax)

    8 days

Secondary Outcomes (11)

  • Area Under the Curve From Time Zero to Last Quantifiable Concentration (AUClast)

    8 days

  • Apparent Oral Clearance (CL/F)

    8 days

  • Time to Reach Maximum Observed Plasma Concentration (Tmax)

    8 days

  • Apparent Volume of Distribution (Vz/F)

    8 days

  • Plasma Decay Half-Life (t1/2)

    8 days

  • +6 more secondary outcomes

Study Arms (4)

Normal Renal Function

EXPERIMENTAL
Drug: palbociclib

Mild Renal Impairment

EXPERIMENTAL
Drug: palbociclib

Moderate Renal Impairment

EXPERIMENTAL
Drug: palbociclib

Severe Renal Impairment

EXPERIMENTAL
Drug: palbociclib

Interventions

palbociclib 125 mg oral capsule with food once

Normal Renal Function

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Personally signed and dated informed consent document.
  • Renal function calculated by the Cockcroft Gault equation: normal function (CLcr \>=90 mL/min), mild: CLcr \>=60 mL/min and \<90 mL/min, moderate: CLcr \>=30 mL/min and \<60 mL/min, severe: CLcr \<30 mL/min but not requiring hemodialysis.
  • Subjects with normal renal function matched for age, weight, gender and race to subjects in impaired renal function groups.

You may not qualify if:

  • Any condition possibly affecting drug absorption.
  • Renal allograft recipients.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (3)

Avail Clinical Research, LLC

DeLand, Florida, 32720, United States

Location

Orlando Clinical Research Center

Orlando, Florida, 32809, United States

Location

Prism Research

Saint Paul, Minnesota, 55114, United States

Location

Related Links

MeSH Terms

Conditions

Renal Insufficiency

Interventions

palbociclib

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital Diseases

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
BASIC SCIENCE
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 11, 2014

First Posted

March 13, 2014

Study Start

May 1, 2014

Primary Completion

May 1, 2016

Study Completion

May 1, 2016

Last Updated

April 30, 2018

Record last verified: 2018-04

Locations