NCT01704495

Brief Summary

The purpose is to Evaluate the Efficacy, Safety, and Tolerability of 3 Different Doses of AZD5069 Twice Daily as Add-on Treatment to Medium to High Dose Inhaled Corticosteroids (ICS) and Long-acting β2 Agonists (LABA), in Patients with Uncontrolled Persistent Asthma

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
1,147

participants targeted

Target at P75+ for phase_2 asthma

Timeline
Completed

Started Nov 2012

Typical duration for phase_2 asthma

Geographic Reach
13 countries

96 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 9, 2012

Completed
2 days until next milestone

First Posted

Study publicly available on registry

October 11, 2012

Completed
21 days until next milestone

Study Start

First participant enrolled

November 1, 2012

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 1, 2014

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2014

Completed
1.6 years until next milestone

Results Posted

Study results publicly available

March 1, 2016

Completed
Last Updated

March 1, 2016

Status Verified

February 1, 2016

Enrollment Period

1.7 years

First QC Date

October 9, 2012

Results QC Date

June 30, 2015

Last Update Submit

February 1, 2016

Conditions

Keywords

Uncontrolled Asthma,Exacerbation,Safety

Outcome Measures

Primary Outcomes (1)

  • Rate of Severe Asthma Exacerbations During 6 Months

    From start of treatment up to 6 months

Secondary Outcomes (41)

  • Rate of Asthma-specific Hospital Admission/Intensive Care Unit Admissions During 6 Months

    From start of treatment up to 6 months

  • Total Number of Days of Asthma-specific Hospital Admission/Intensive Care Unit Admissions

    From start of treatment up to 6 months

  • Total Number of Days on Oral Cortecosteroids, Due to a Worsening of Asthma Symptoms

    From start of treatment up to 6 months

  • Change From Baseline to 2 Weeks Measurement of Pre-bronchodilator FEV1

    Baseline (Day 0) and 2 weeks after Day 0

  • Change From Baseline to 1 Month Measurement of Pre-bronchodilator FEV1

    Baseline (Day 0) and 1 month after Day 0

  • +36 more secondary outcomes

Study Arms (4)

AZD5069 5 mg

EXPERIMENTAL

AZD5069 oral capsules self-administered twice daily

Drug: AZD5069

AZD5069 15 mg

EXPERIMENTAL

AZD5069 oral capsules self-administered twice daily

Drug: AZD5069

AZD5069 45 mg

EXPERIMENTAL

AZD5069 oral capsules self-administered twice daily

Drug: AZD5069

Placebo

PLACEBO COMPARATOR

Placebo oral capsules self-administered twice daily

Drug: Placebo

Interventions

AZD5069 oral capsules self-administered twice daily.

AZD5069 15 mgAZD5069 45 mgAZD5069 5 mg

Placebo oral capsules self-administered twice daily.

Placebo

Eligibility Criteria

Age18 Years - 150 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Men and women aged 18 years and above. Females of childbearing potential must use a highly effective contraceptive method plus a condom by their male partner.
  • Diagnosis of asthma for at least 12 months (GINA 2011)
  • Uncontrolled persistent asthma, despite treatment with medium to high dose ICS and LABA, and with a history of exacerbations during the last year
  • Morning prebronchodilator FEV1 of ≥30% and ≤85% predicted normal at enrolment
  • Daily use of medium or high dose ICS (≥fluticasone 500 µg or the equivalent daily)

You may not qualify if:

  • Any clinically significant disease or disorder (including any chronic lower respiratory disease other than asthma) that may put the patient at risk or influence study results
  • Patients with recurrent, latent, or chronic infections
  • Active tuberculosis or latent tuberculosis without completion of an appropriate course of treatment or prophylactic treatment
  • Significant lower respiratory tract infection not resolved within 30 days prior to enrolment
  • Current smoker or smoking history of more than 20 pack years

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (96)

Research Site

Gotse Delchev, Bulgaria

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Kozloduy, Bulgaria

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Petrich, Bulgaria

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Pleven, Bulgaria

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Razgrad, Bulgaria

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Rousse, Bulgaria

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Sofia, Bulgaria

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Vidin, Bulgaria

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Mount Pearl, Newfoundland and Labrador, Canada

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Hamilton, Ontario, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Québec, Quebec, Canada

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Saint Romuald, Quebec, Canada

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Brno, Czechia

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Jindřichův Hradec, Czechia

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Karlovy Vary, Czechia

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Kutná Hora, Czechia

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Mělník, Czechia

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Prague, Czechia

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Strakonice, Czechia

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Tábor, Czechia

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Berlin, Germany

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Großhansdorf, Germany

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Hamburg, Germany

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Hanover, Germany

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München, Germany

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Aszód, Hungary

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Baja, Hungary

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Balassagyarmat, Hungary

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Budapest, Hungary

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Cegléd, Hungary

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Gyula, Hungary

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Komárom, Hungary

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Makó, Hungary

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Monor, Hungary

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Nyíregyháza, Hungary

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Pécs, Hungary

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Százhalombatta, Hungary

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Szeged, Hungary

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Szombathely, Hungary

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Guadalajara, Mexico

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México, Mexico

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Monterrey, Mexico

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Bialystok, Poland

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Gdansk, Poland

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Giżycko, Poland

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Krakow, Poland

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Lodz, Poland

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Lublin, Poland

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Poznan, Poland

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Proszowice, Poland

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Skierniewice, Poland

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Tarnów, Poland

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Wroclaw, Poland

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Żnin, Poland

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Brasov, Romania

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Bucharest, Romania

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Constanța, Romania

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Deva, Romania

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Iași, Romania

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Izhevsk, Russia

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Kazan', Russia

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Moscow, Russia

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Saint Petersburg, Russia

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Vladikavkaz, Russia

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Yaroslavl, Russia

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Yekaterinburg, Russia

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Bardejov, Slovakia

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Bratislava, Slovakia

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Komárno, Slovakia

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Košice, Slovakia

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Levice, Slovakia

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Poprad, Slovakia

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Spišská Nová Ves, Slovakia

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Šurany, Slovakia

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Topoľčany, Slovakia

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Trenčín, Slovakia

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Zvolen, Slovakia

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Cape Town, South Africa

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Durban, South Africa

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eManzimtoti, South Africa

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eMkhomazi, South Africa

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Pretoria, South Africa

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Donetsk, Ukraine

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Ivano-Frankivsk, Ukraine

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Kharkiv, Ukraine

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Kyiv, Ukraine

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Vinnytsia, Ukraine

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Zaporizhzhya, Ukraine

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Zaporizhzhzya, Ukraine

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Zaporozye, Ukraine

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Birmingham, United Kingdom

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Dundee, United Kingdom

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Liverpool, United Kingdom

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London, United Kingdom

Location

Related Publications (1)

  • O'Byrne PM, Metev H, Puu M, Richter K, Keen C, Uddin M, Larsson B, Cullberg M, Nair P. Efficacy and safety of a CXCR2 antagonist, AZD5069, in patients with uncontrolled persistent asthma: a randomised, double-blind, placebo-controlled trial. Lancet Respir Med. 2016 Oct;4(10):797-806. doi: 10.1016/S2213-2600(16)30227-2. Epub 2016 Aug 27.

MeSH Terms

Conditions

Asthma

Interventions

N-(2-(2,3-difluoro-6-benzylthio)-6-(3,4-dihydroxybutan-2-yloxy)pyrimidin-4-yl)azetidine-1-sulfonamide

Condition Hierarchy (Ancestors)

Bronchial DiseasesRespiratory Tract DiseasesLung Diseases, ObstructiveLung DiseasesRespiratory HypersensitivityHypersensitivity, ImmediateHypersensitivityImmune System Diseases

Results Point of Contact

Title
Medical Science Director Bengt Larsson
Organization
AstraZeneca

Study Officials

  • Bengt Larsson, MEDICAL SCIENCE DIRECTOR

    AZ Mondal R&D, Sweden

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
GT60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 9, 2012

First Posted

October 11, 2012

Study Start

November 1, 2012

Primary Completion

August 1, 2014

Study Completion

August 1, 2014

Last Updated

March 1, 2016

Results First Posted

March 1, 2016

Record last verified: 2016-02

Locations