NCT01671787

Brief Summary

This is an open-label study evaluating multiple doses of GS-7340 versus Tenofovir disoproxil fumarate (TDF).

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
51

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Mar 2012

Geographic Reach
5 countries

19 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 1, 2012

Completed
6 months until next milestone

First Submitted

Initial submission to the registry

August 21, 2012

Completed
3 days until next milestone

First Posted

Study publicly available on registry

August 24, 2012

Completed
7 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2013

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 1, 2013

Completed
Last Updated

October 23, 2018

Status Verified

May 1, 2014

Enrollment Period

1.1 years

First QC Date

August 21, 2012

Last Update Submit

October 19, 2018

Conditions

Keywords

Hepatitis BHBVGS-7340TDFTenofovir disoproxil fumarateGileadViread

Outcome Measures

Primary Outcomes (1)

  • Change in serum hepatitis B virus (HBV) DNA

    Time-weighted average change from baseline through Week 4 (DAVG4) in serum HBV DNA (log10 IU/mL) for GS-7340 8-, 25-, 40 and 120-mg.

    Up to Week 4

Secondary Outcomes (4)

  • Change in HBV DNA for tenofovir disoproxil fumarate (TDF)

    Up to Week 4

  • Change in HBV DNA of GS-7340 through 28 days of therapy

    Up to week 4

  • Pharmacokinetics (PK) of GS-7340 and/or tenofovir (TVF) following single and multiple doses of GS-7340 and TDF

    Up to week 4

  • Safety and Tolerability of Therapy

    Up to week 4

Study Arms (5)

GS-7340 8mg

EXPERIMENTAL

After Screening procedures, eligible subjects will be randomized 1:1:1:1:1 to receive either open-label GS-7340 8, 25, 40, or 120 mg (3 x 40 mg), or open-label TDF 300 mg for 28 days.

Drug: GS-7340

GS-7340 25mg

EXPERIMENTAL

After Screening procedures, eligible subjects will be randomized 1:1:1:1:1 to receive either open-label GS-7340 8, 25, 40, or 120 mg (3 x 40 mg), or open-label TDF 300 mg for 28 days.

Drug: GS-7340

GS-7340 40mg

EXPERIMENTAL

After Screening procedures, eligible subjects will be randomized 1:1:1:1:1 to receive either open-label GS-7340 8, 25, 40, or 120 mg (3 x 40 mg), or open-label TDF 300 mg for 28 days.

Drug: GS-7340

GS-7340 120mg

EXPERIMENTAL

After Screening procedures, eligible subjects will be randomized 1:1:1:1:1 to receive either open-label GS-7340 8, 25, 40, or 120 mg (3 x 40 mg), or open-label TDF 300 mg for 28 days.

Drug: GS-7340

Tenofovir disoproxil fumarate 300mg

EXPERIMENTAL

After Screening procedures, eligible subjects will be randomized 1:1:1:1:1 to receive either open-label GS-7340 8, 25, 40, or 120 mg (3 x 40 mg), or open-label TDF 300 mg for 28 days.

Drug: Tenofovir disoproxil fumarate

Interventions

Subjects are randomized to receive one of four different doses of GS-7340 over 28 days of therapy.

GS-7340 120mgGS-7340 25mgGS-7340 40mgGS-7340 8mg

Subjects will receive 300mg of Tenofovir disoproxil fumarate (TDF) over 28 days of therapy

Also known as: Viread
Tenofovir disoproxil fumarate 300mg

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Must be between 18 and 65 years of age
  • Must have Screening plasma HBV DNA ≥ 2x10\^3 IU/mL
  • Must have chronic HBV infection for at least 6 months
  • Must have estimated creatinine clearance (CLCr) ≥ 70 mL/min
  • Not pregnant or nursing
  • Women must be of non-childbearing potential OR of childbearing potential with confirmed negative pregnancy tests
  • Consistent and correct use of recommended methods of birth control for men and women

You may not qualify if:

  • Pregnant or lactating subjects
  • Receipt of anti-HBV nucleoside/nucleotide therapy. Subjects who have failed prior Interferon treatment, greater than 6 months prior to screening, are permitted to participate in the study screening
  • Known co-infection with HIV, hepatitis C virus (HCV) or hepatitis D virus (HDV)
  • Presence of autoimmune disorders
  • History of liver disease other than Hepatitis B
  • History of Gilbert's Disease
  • Any sign of decompensated liver disease
  • Known or suspected cirrhosis
  • Evidence of hepatocellular carcinoma
  • Presence or history of cardiovascular disease, cardiomyopathy, and/or cardiac conduction abnormalities
  • Electrolyte abnormalities
  • History of treatment that permanently alters the gastric condition
  • Alcohol or substance abuse
  • History of bleeding diathesis
  • Significant bone disease

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (19)

Research and Education Inc.

San Diego, California, 92105, United States

Location

University of Maryland Institute of Human Virology

Baltimore, Maryland, 21201, United States

Location

Henry Ford Health System

Detroit, Michigan, 48202, United States

Location

Baylor College of Medicine - St. Luke's Episcopal Hospital

Houston, Texas, 77030, United States

Location

Monash Medical Centre

Melborne, Victoria, 03168, Australia

Location

Alfred Hospital

Melbourne, Victoria, 3004, Australia

Location

Austin Health

Melbourne, Victoria, 3084, Australia

Location

Linear Clinical Research Ltd

Nedlands, Western Australia, 6009, Australia

Location

Downtown Infectious Diseases Clinic (University of British Columbia)

Vancouver, British Columbia, V6Z2C9, Canada

Location

The Ottawa Hospital, General Campus

Ottawa, Ontario, K1H8L6, Canada

Location

Toronto General Hospital

Toronto, Ontario, M5G 2C4, Canada

Location

Algorithme Pharma

Montreal, Quebec, H3P3P1, Canada

Location

Pro-recherche

Saint Romuald, Quebec, G6W 8H1, Canada

Location

Auckland Clinical Studies

Auckland, 1042, New Zealand

Location

University Hospitals Birmingham NHS Foundation Trust

Birmingham, B152TH, United Kingdom

Location

Grahame Hayton Unit

London, E1 1BB, United Kingdom

Location

University College London Hospital

London, NW1-2BU, United Kingdom

Location

Institute of Liver Studies, King's College Hospital

London, SE5 9RS, United Kingdom

Location

Nottingham University Hospitals NHS Trust - Queens Medical Centre

Nottingham, NG7 2UH, United Kingdom

Location

MeSH Terms

Conditions

Hepatitis B, ChronicHepatitis B

Interventions

tenofovir alafenamideTenofovir

Condition Hierarchy (Ancestors)

Blood-Borne InfectionsCommunicable DiseasesInfectionsHepadnaviridae InfectionsDNA Virus InfectionsVirus DiseasesHepatitis, Viral, HumanHepatitis, ChronicHepatitisLiver DiseasesDigestive System DiseasesChronic DiseaseDisease AttributesPathologic ProcessesPathological Conditions, Signs and Symptoms

Intervention Hierarchy (Ancestors)

OrganophosphonatesOrganophosphorus CompoundsOrganic ChemicalsAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Study Officials

  • John Flaherty, MD

    Gilead Sciences

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 21, 2012

First Posted

August 24, 2012

Study Start

March 1, 2012

Primary Completion

April 1, 2013

Study Completion

April 1, 2013

Last Updated

October 23, 2018

Record last verified: 2014-05

Data Sharing

IPD Sharing
Will share

Qualified external researchers may request IPD for this study after study completion. For more information, please visit our website at http://www.gilead.com/research/disclosure-and-transparency.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
18 months after study completion
Access Criteria
A secured external environment with username, password, and RSA code.
More information

Locations