NCT01231620

Brief Summary

The purpose of this study is to test the safety and efficacy of zanamivir given intravenously and how well it works at two different doses in hospitalized adolescents and adults with flu. Zanamivir will be compared with oseltamivir, which is used for treating flu.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
626

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Jan 2011

Typical duration for phase_3

Geographic Reach
28 countries

170 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 28, 2010

Completed
4 days until next milestone

First Posted

Study publicly available on registry

November 1, 2010

Completed
3 months until next milestone

Study Start

First participant enrolled

January 15, 2011

Completed
4.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 18, 2015

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 18, 2015

Completed
2.7 years until next milestone

Results Posted

Study results publicly available

November 20, 2017

Completed
Last Updated

October 15, 2018

Status Verified

March 1, 2018

Enrollment Period

4.2 years

First QC Date

October 28, 2010

Results QC Date

April 11, 2017

Last Update Submit

September 14, 2018

Conditions

Keywords

Seasonal InfluenzaPandemicOrthomyxoviridae InfectionsInfluenzaInfluenza A Virus, H1N1 SubtypeEnzyme InhibitorsInfluenza, seasonalRespiratory Tract DiseasesZanamivirPharmacologic ActionsAntiviral AgentsAnti-Infective AgentsH1N1Neuraminidase inhibitorInfluenza B virus

Outcome Measures

Primary Outcomes (1)

  • Time to Clinical Response (TTCR) in Participants With Confirmed Influenza

    Clinical response is defined as the resolution of at least 4 of the 5 vital signs (temperature, oxygen saturation, respiratory status, heart rate, systolic blood pressure) within the respective resolution criteria, maintained for at least 24 hours, or hospital discharge, whichever occurred first. This analysis was performed for Influenza positive population, for those with symptom onset less than or equal to (\<=) 4 days, and for those on mechanical (mech) ventilation or in intensive care unit (ICU). 99 days is censored time for the participants who did not achieve TTCR.

    Up to 42 days

Secondary Outcomes (31)

  • Percentage of Participants With Respiratory Improvement

    Up to 42 days

  • Number of Participants With All Cause and Attributable Mortality at Day 14, at Day 28, and at the End of Study Visit

    On or before Day 14, Day 28, End of Study Visit (assessed up to 42 days)

  • Change From Baseline in the Katz Activities of Daily Living (ADL) Score and Each ADL Activity Score

    Baseline (Day 1) and up to 42 days

  • Median Time to Return to Pre-morbid Functional Status as Measured by the Katz ADL Score and Each ADL Activity Score

    Up to 42 days

  • Number of Participants Who Returned to Their Pre-morbid Functional Status as Assessed Per the Katz ADL Score and Each ADL Activity Score at the End of the Study

    Up to 42 days

  • +26 more secondary outcomes

Study Arms (3)

Intravenous (IV) Zanamivir 300mg Twice Daily

EXPERIMENTAL

300mg of IV zanamivir infusion twice daily plus oral oseltamivir placebo twice daily

Drug: ZanamivirDrug: Placebo to match oseltamivir

Intravenous (IV) Zanamivir 600mg Twice Daily

EXPERIMENTAL

600mg of IV zanamivir infusion twice daily plus oral oseltamivir placebo twice daily

Drug: ZanamivirDrug: Placebo to match oseltamivir

Oral Oseltamivir 75mg Twice Daily

ACTIVE COMPARATOR

75mg oral oseltamivir twice daily plus intravenous placebo zanamivir twice daily

Drug: Placebo to match zanamivirDrug: Oseltamivir

Interventions

Zanamivir aqueous solution, 10 mg/mL, will be provided as a single use, sterile clear, colorless preparation in 20 mL clear glass vials.

Also known as: Relenza
Intravenous (IV) Zanamivir 300mg Twice DailyIntravenous (IV) Zanamivir 600mg Twice Daily

Placebo to match IV zanamivir will be provided as a normal saline solution of a matched volume.

Oral Oseltamivir 75mg Twice Daily

Oseltamivir will be provided as over-encapsulated 75 mg capsules.

Also known as: Tamiflu
Oral Oseltamivir 75mg Twice Daily

Placebo to match oral oseltamivir will be provided as capsules with a common excipient of appropriate quality.

Intravenous (IV) Zanamivir 300mg Twice DailyIntravenous (IV) Zanamivir 600mg Twice Daily

Eligibility Criteria

Age16 Years+
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17), Adult (18-64), Older Adult (65+)

You may qualify if:

  • Male or female aged 16 years; a female is eligible to enter and participate in the study if she is:
  • of non-childbearing potential (i.e., physiologically incapable of becoming pregnant, including any female who is post- menopausal); or,
  • of child-bearing potential, has a negative pregnancy test at Baseline, and agrees to use protocol specified methods of birth control while on study.
  • Vital signs criteria defined as 3 or more of the following at Baseline:
  • Presence of fever \[oral temperature of 38°C or equivalent\] at Baseline. However, this requirement is waived if the subject has a history of fever within in the 24 hours prior to Baseline; or, if the subject reported symptoms of feverishness at some time during the 48 hours prior to Baseline.
  • AND at least 2 out of the following 4:
  • Oxygen saturation \<95% on room air by trans-cutaneous method or need for any supplemental oxygenation or ventilatory support, or increase in oxygen supplementation requirement of ≥2 litres for subjects with chronic oxygen dependency. For those subjects with a history of chronic hypoxia (without supplemental oxygen), an oxygen saturation of at least 3% below the patient's historical baseline oxygen saturation will satisfy this criterion.
  • Respiration rate \>24 breaths per minute. For those subjects who require ventilatory support or oxygen supplementation, this requirement is waived.
  • Heart rate \>100 beats per minute.
  • Systolic blood pressure \<90 mmHg.
  • Onset of influenza symptoms within 6 days prior to study enrolment. Symptoms may include cough, dyspnea, sore throat, feverishness, myalgias, headache, nasal symptoms (rhinorrhea, congestion), fatigue, diarrhea, anorexia, nausea and vomiting.
  • Clinical symptoms of influenza with positive influenza diagnostic test result or strong suspicion of influenza illness based on clinical symptoms and local surveillance information.
  • Subjects willing and able to give written informed consent to participate in the study and to adhere to the procedures stated in the protocol, or legally acceptable representative willing and able to give written informed consent on behalf of the subject for minors, unconscious adults and those incapable of consenting themselves due to their medical condition, or included as permitted by local regulatory authorities, IRB/IECs or local laws.
  • Severity of any medical illness that, in the Investigator's judgement, justifies hospitalization of the subject for treatment and supportive care

You may not qualify if:

  • Subjects who have taken more than a total of 3 days (6 doses) of approved anti-influenza therapy in the period from onset of symptoms and prior to enrolment.
  • Subjects who, in the opinion of the investigator, are not likely to survive beyond 48 hours from Baseline.
  • Subjects who are considered to require concurrent therapy with another influenza antiviral medication.
  • Subjects who are known or suspected to be hypersensitive to any component of the study medications.
  • Subjects with creatinine clearance ≤10 mL/min who are not being treated with continuous renal replacement therapy (CRRT).
  • Subjects who require Extra Corporeal Membrane Oxygenation (ECMO) at Baseline
  • Subjects who require routine/intermittent hemodialysis or continuous peritoneal dialysis (due to inability to provide appropriate dosing schedule for oseltamivir) at Baseline. CRRT modalities are allowed.
  • Liver toxicity criteria based on local laboratory results obtained within 24 hours of Baseline:
  • ALT or AST 3xULN and bilirubin 2xULN
  • ALT 5xULN
  • Underlying chronic liver disease with evidence of severe liver impairment.
  • History of severe cardiac disease or clinically significant arrhythmia (either on ECG or by history) which, in the opinion of the Investigator, will interfere with the safety of the individual subject.
  • Females who are pregnant or are breastfeeding.
  • Treatment with investigational parenteral anti-influenza drugs (IV peramivir, IV zanamivir or IV oseltamivir) in the 4 weeks prior to Baseline.
  • French and Korean subjects: the French or Korean subject has participated in any study using an investigational drug during the previous 30 days.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (170)

GSK Investigational Site

Birmingham, Alabama, 35249, United States

Location

GSK Investigational Site

Phoenix, Arizona, 85023, United States

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GSK Investigational Site

Chula Vista, California, 91911, United States

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GSK Investigational Site

Escondido, California, 92025, United States

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GSK Investigational Site

Fullerton, California, 92835, United States

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GSK Investigational Site

La Jolla, California, 92037, United States

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GSK Investigational Site

La Mesa, California, 91942, United States

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GSK Investigational Site

Oceanside, California, 92056, United States

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GSK Investigational Site

Aurora, Colorado, 80045, United States

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GSK Investigational Site

Stamford, Connecticut, 06902, United States

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GSK Investigational Site

Orlando, Florida, 32806, United States

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GSK Investigational Site

Sarasota, Florida, 34239, United States

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GSK Investigational Site

Sunrise, Florida, 33323, United States

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GSK Investigational Site

Atlanta, Georgia, 30342, United States

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GSK Investigational Site

Augusta, Georgia, 30912, United States

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GSK Investigational Site

Idaho Falls, Idaho, 83404, United States

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GSK Investigational Site

Chicago, Illinois, 60611, United States

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GSK Investigational Site

Oak Park, Illinois, 60302, United States

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GSK Investigational Site

Peoria, Illinois, 61637, United States

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GSK Investigational Site

Council Bluffs, Iowa, 51503, United States

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GSK Investigational Site

Topeka, Kansas, 66604, United States

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GSK Investigational Site

Louisville, Kentucky, 40241, United States

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GSK Investigational Site

Boston, Massachusetts, 02115, United States

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GSK Investigational Site

Royal Oak, Michigan, 48073, United States

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GSK Investigational Site

Troy, Michigan, 48085, United States

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GSK Investigational Site

St Louis, Missouri, 63110-1093, United States

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GSK Investigational Site

Missoula, Montana, 59802, United States

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GSK Investigational Site

Las Vegas, Nevada, 89109, United States

Location

GSK Investigational Site

Valhalla, New York, 10595, United States

Location

GSK Investigational Site

Asheville, North Carolina, 28801, United States

Location

GSK Investigational Site

Chapel Hill, North Carolina, 27599-7215, United States

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GSK Investigational Site

Bismarck, North Dakota, 58504, United States

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GSK Investigational Site

Cleveland, Ohio, 44195, United States

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GSK Investigational Site

Columbus, Ohio, 43215, United States

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GSK Investigational Site

Toledo, Ohio, 43608, United States

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GSK Investigational Site

Bethlehem, Pennsylvania, 18105, United States

Location

GSK Investigational Site

Philadelphia, Pennsylvania, 19107, United States

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GSK Investigational Site

Houston, Texas, 77030, United States

Location

GSK Investigational Site

Roanoke, Virginia, 24013, United States

Location

GSK Investigational Site

Marshfield, Wisconsin, 54449, United States

Location

GSK Investigational Site

Westmead, New South Wales, 2145, Australia

Location

GSK Investigational Site

Herston, Queensland, 4029, Australia

Location

GSK Investigational Site

Adelaide, South Australia, 5000, Australia

Location

GSK Investigational Site

Bedford Park, South Australia, 5043, Australia

Location

GSK Investigational Site

Clayton, Victoria, 3168, Australia

Location

GSK Investigational Site

Heidelberg, Victoria, 3084, Australia

Location

GSK Investigational Site

Melbourne, Victoria, 3004, Australia

Location

GSK Investigational Site

Melbourne, Victoria, 3050, Australia

Location

GSK Investigational Site

Perth, Western Australia, 6000, Australia

Location

GSK Investigational Site

Brussels, 1070, Belgium

Location

GSK Investigational Site

Brussels, 1090, Belgium

Location

GSK Investigational Site

Leuven, 3000, Belgium

Location

GSK Investigational Site

Liège, 4000, Belgium

Location

GSK Investigational Site

Rio de Janeiro, 21040-900, Brazil

Location

GSK Investigational Site

SĂ£o Paulo, 01308-050, Brazil

Location

GSK Investigational Site

Calgary, Alberta, T1Y 6J4, Canada

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GSK Investigational Site

Calgary, Alberta, T2N 2T9, Canada

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GSK Investigational Site

Halifax, Nova Scotia, B3H 3A7, Canada

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GSK Investigational Site

Hamilton, Ontario, L8N 4A6, Canada

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GSK Investigational Site

Toronto, Ontario, M5G 2C4, Canada

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GSK Investigational Site

Chicoutimi, Quebec, G7H 5H6, Canada

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GSK Investigational Site

Montreal, Quebec, H1T 2M4, Canada

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GSK Investigational Site

Montreal, Quebec, H2W1T8, Canada

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GSK Investigational Site

Trois-Rivières, Quebec, G8Z 3R9, Canada

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GSK Investigational Site

Haikou, Hainan, 570311, China

Location

GSK Investigational Site

Changsha, Hunan, 410005, China

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GSK Investigational Site

Nanchang, Jiangxi, 330006, China

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GSK Investigational Site

Changchun, Jilin, 130041, China

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GSK Investigational Site

Xi'an, Shaanxi, 710032, China

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GSK Investigational Site

Hangzhou, Zhejiang, 310003, China

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GSK Investigational Site

Beijing, 100015, China

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GSK Investigational Site

Beijing, 100044, China

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GSK Investigational Site

Chengdu, 610041, China

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GSK Investigational Site

Chongqing, 400016, China

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GSK Investigational Site

Guangzhou, 510120, China

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GSK Investigational Site

Hangzhou, 310016, China

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GSK Investigational Site

Shanghai, 200025, China

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GSK Investigational Site

Tianjin, 300052, China

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GSK Investigational Site

BogotĂ¡, Colombia

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GSK Investigational Site

Brno, 625 00, Czechia

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GSK Investigational Site

Brno-Bohunice, 625 00, Czechia

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GSK Investigational Site

Hradec KrĂ¡lovĂ©, 500 05, Czechia

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GSK Investigational Site

Prague, 180 01, Czechia

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GSK Investigational Site

Aarhus N, 8200, Denmark

Location

GSK Investigational Site

Hvidovre, DK-2650, Denmark

Location

GSK Investigational Site

Odense C, 5000, Denmark

Location

GSK Investigational Site

Dijon, 21079, France

Location

GSK Investigational Site

Limoges, 87042, France

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GSK Investigational Site

Nîmes, 30029, France

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GSK Investigational Site

Orléans, 45067, France

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GSK Investigational Site

Poitiers, 86021, France

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GSK Investigational Site

Tours, 37044, France

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GSK Investigational Site

Ulm, Baden-Wurttemberg, 89081, Germany

Location

GSK Investigational Site

Erlangen, Bavaria, 91054, Germany

Location

GSK Investigational Site

Regensburg, Bavaria, 93053, Germany

Location

GSK Investigational Site

Hanover, Lower Saxony, 30625, Germany

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GSK Investigational Site

Homburg, Saarland, 66421, Germany

Location

GSK Investigational Site

ChaĂ¯dĂ¡ri, 12462, Greece

Location

GSK Investigational Site

Goudi, Athens, 11527, Greece

Location

GSK Investigational Site

Kwun Tong, Hong Kong

Location

GSK Investigational Site

Shatin, Hong Kong

Location

GSK Investigational Site

Tuenmen, Hong Kong

Location

GSK Investigational Site

Debrecen, 4031, Hungary

Location

GSK Investigational Site

KaposvĂ¡r, 7400, Hungary

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GSK Investigational Site

Miskolc, 3529, Hungary

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GSK Investigational Site

SzĂ©kesfehĂ©rvĂ¡r, 8000, Hungary

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GSK Investigational Site

Szombathely, 9700, Hungary

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GSK Investigational Site

Bangalore, 560010, India

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GSK Investigational Site

Civil Lines, 141001, India

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GSK Investigational Site

Lucknow, 226003, India

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GSK Investigational Site

Lucknow, 226005, India

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GSK Investigational Site

Pune, 411004, India

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GSK Investigational Site

Pune, 411018, India

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GSK Investigational Site

Trivandrum, 695029, India

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GSK Investigational Site

Guadalajara, Jalisco, 44280, Mexico

Location

GSK Investigational Site

San NicolĂ¡s de los Garza, Nuevo LeĂ³n, 66480, Mexico

Location

GSK Investigational Site

CuautitlĂ¡n, Estado de MĂ©xico, State of Mexico, 54800, Mexico

Location

GSK Investigational Site

Aguascalientes, 20230, Mexico

Location

GSK Investigational Site

Chihuahua City, 31238, Mexico

Location

GSK Investigational Site

Nijmegen, 6500 HB, Netherlands

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GSK Investigational Site

Auckland, 1001, New Zealand

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GSK Investigational Site

Auckland, 1701, New Zealand

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GSK Investigational Site

Auckland, New Zealand

Location

GSK Investigational Site

Christchurch, 8001, New Zealand

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GSK Investigational Site

Hamilton, 3204, New Zealand

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GSK Investigational Site

Hastings, 4120, New Zealand

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GSK Investigational Site

Newtown, New Zealand

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GSK Investigational Site

Bergen, 5053, Norway

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GSK Investigational Site

Trondheim, 7030, Norway

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GSK Investigational Site

ChorzĂ³w, 41-500, Poland

Location

GSK Investigational Site

Dębica, 39-200, Poland

Location

GSK Investigational Site

Trzebnica, 55-100, Poland

Location

GSK Investigational Site

Warsaw, 01-201, Poland

Location

GSK Investigational Site

Barnaul, 656024, Russia

Location

GSK Investigational Site

Barnaul, 656038, Russia

Location

GSK Investigational Site

Saint Petersburg, 191167, Russia

Location

GSK Investigational Site

Saint Petersburg, 197022, Russia

Location

GSK Investigational Site

Smolensk, 214006, Russia

Location

GSK Investigational Site

Bratislava, 833 05, Slovakia

Location

GSK Investigational Site

Martin, 036 59, Slovakia

Location

GSK Investigational Site

Middelburg, Mpumalanga, 1055, South Africa

Location

GSK Investigational Site

Bellville, 7530, South Africa

Location

GSK Investigational Site

Die Wilgers, 0041, South Africa

Location

GSK Investigational Site

Les Marais, 0084, South Africa

Location

GSK Investigational Site

Panorama, 7500, South Africa

Location

GSK Investigational Site

Worcester, 6850, South Africa

Location

GSK Investigational Site

Guro Gu, 152703, South Korea

Location

GSK Investigational Site

Gyeonggi-do, 442-723, South Korea

Location

GSK Investigational Site

Kangwon-do, 220-701, South Korea

Location

GSK Investigational Site

Seoul, 150-030, South Korea

Location

GSK Investigational Site

Seoul, 150-950, South Korea

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GSK Investigational Site

Alicante, 03010, Spain

Location

GSK Investigational Site

Badalona, 08916, Spain

Location

GSK Investigational Site

Barcelona, 08003, Spain

Location

GSK Investigational Site

Granada, 18012, Spain

Location

GSK Investigational Site

Granada, 18014, Spain

Location

GSK Investigational Site

L'Hospitalet de Llobregat, 08907, Spain

Location

GSK Investigational Site

Madrid, 28007, Spain

Location

GSK Investigational Site

Madrid, 28040, Spain

Location

GSK Investigational Site

Madrid, 28046, Spain

Location

GSK Investigational Site

Murcia, 30003, Spain

Location

GSK Investigational Site

Oviedo, 33006, Spain

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GSK Investigational Site

Pama de Mallorca, 07010, Spain

Location

GSK Investigational Site

Taipei, 112, Taiwan

Location

GSK Investigational Site

Bangkok, 10400, Thailand

Location

GSK Investigational Site

Bangkok, 10700, Thailand

Location

GSK Investigational Site

Bristol, BS2 8HW, United Kingdom

Location

GSK Investigational Site

Cardiff, CF14 4XW, United Kingdom

Location

GSK Investigational Site

Liverpool, L7 8XP, United Kingdom

Location

GSK Investigational Site

Manchester, M13 9WL, United Kingdom

Location

Related Publications (2)

  • van Duijnhoven W, Van Dromme I, Haesendonckx S, Witek J, Leopold L. The Hospital Recovery Scale: A clinically useful endpoint in patients hospitalized with influenza. Contemp Clin Trials. 2022 Dec;123:106952. doi: 10.1016/j.cct.2022.106952. Epub 2022 Oct 3.

  • Marty FM, Vidal-Puigserver J, Clark C, Gupta SK, Merino E, Garot D, Chapman MJ, Jacobs F, Rodriguez-Noriega E, Husa P, Shortino D, Watson HA, Yates PJ, Peppercorn AF. Intravenous zanamivir or oral oseltamivir for hospitalised patients with influenza: an international, randomised, double-blind, double-dummy, phase 3 trial. Lancet Respir Med. 2017 Feb;5(2):135-146. doi: 10.1016/S2213-2600(16)30435-0. Epub 2017 Jan 14.

Related Links

MeSH Terms

Conditions

Influenza, HumanOrthomyxoviridae InfectionsRespiratory Tract Diseases

Interventions

ZanamivirOseltamivir

Condition Hierarchy (Ancestors)

Respiratory Tract InfectionsInfectionsRNA Virus InfectionsVirus Diseases

Intervention Hierarchy (Ancestors)

GuanidinesAmidinesOrganic ChemicalsSialic AcidsNeuraminic AcidsSugar AcidsAcids, AcyclicCarboxylic AcidsHydroxy AcidsPyransHeterocyclic Compounds, 1-RingHeterocyclic CompoundsAmino SugarsCarbohydratesAcetamidesAmidesCyclohexenesCyclohexanesCycloparaffinsHydrocarbons, AlicyclicHydrocarbons, CyclicHydrocarbons

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 28, 2010

First Posted

November 1, 2010

Study Start

January 15, 2011

Primary Completion

March 18, 2015

Study Completion

March 18, 2015

Last Updated

October 15, 2018

Results First Posted

November 20, 2017

Record last verified: 2018-03

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Annotated Case Report Form (114373)Access
Statistical Analysis Plan (114373)Access
Clinical Study Report (114373)Access
Individual Participant Data Set (114373)Access
Dataset Specification (114373)Access
Informed Consent Form (114373)Access
Study Protocol (114373)Access

Locations