NCT01137552

Brief Summary

This is a first in human, open-label, sequential dose escalation and expansion study of AMG 780 in up to 62 subjects with advanced solid tumors. The dose escalation part of the study is aimed at evaluating the safety, tolerability, pharmacokinetics and pharmacodynamics of AMG 780. The dose expansion will consist of up to 20 subjects and the dose level of AMG 780 will be dependent upon emerging safety and PK data from the dose escalation part of the study.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
44

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Jun 2010

Longer than P75 for phase_1

Geographic Reach
1 country

3 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 22, 2010

Completed
1 month until next milestone

Study Start

First participant enrolled

June 1, 2010

Completed
3 days until next milestone

First Posted

Study publicly available on registry

June 4, 2010

Completed
3.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 1, 2013

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

April 1, 2014

Completed
Last Updated

March 4, 2015

Status Verified

February 1, 2015

Enrollment Period

3.5 years

First QC Date

April 22, 2010

Last Update Submit

March 2, 2015

Conditions

Keywords

First-In-HumanDose EscalationDose ExpansionAdvance Solid TumorsAnti-AngiopoietinAdvance MalignancyCancerOncologyOncology PatientsPhase 1Clinical TrialTumorsSolid TumorsAngiogenesis Inhibitors

Outcome Measures

Primary Outcomes (2)

  • To assess the safety and tolerability of AMG 780 in subjects with advanced solid malignancies (including adverse event rate, incidence of dose-limiting toxicities, and determination of maximum tolerated dose)

    2.5 years

  • To evaluate the pharmacokinetic (PK) parameters of AMG 780 including, but not limited to Cmax, AUC, and accumulation ratio

    2.5 years

Secondary Outcomes (4)

  • To evaluate tumor response using RECIST criteria (measured by CT/MRI)

    2.5 years

  • To evaluate changes in tumor volume (measured by volumetric CT/MRI)

    2.5 years

  • To evaluate changes in tumor vascularity and to estimate the relationship between dose/pharmacokinetics and vascular response (measured by DCE-MRI)

    2.5 years

  • To evaluate the incidence of anti-AMG 780 antibody formation

    2.5 years

Study Arms (2)

A

EXPERIMENTAL

Dose Escalation

Drug: AMG 780

B

EXPERIMENTAL

Dose Expansion

Drug: AMG 780

Interventions

AMG 780 will be administered by IV infusion every 2 weeks

AB

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Men and women ≥ 18 years old
  • Must have a pathologically documented, and definitely diagnosed, advanced solid tumor that is refractory to standard treatment, or for which no curative therapy is available, or for subjects who refuse standard therapy
  • Measurable disease by RECIST criteria
  • Must be able to undergo MRI evaluation
  • Eastern Cooperative Oncology Group (ECOG) performance status ≤ 2
  • Competent to sign and date an Institutional Review Board approved informed consent form

You may not qualify if:

  • Presence of untreated or symptomatic primary central nervous system tumors or metastases
  • Presence of leukemia or myelodysplastic syndrome
  • Subjects with head and neck cancer
  • Previous hematopoietic stem cell transplant (allogeneic)
  • Unresolved hematological toxicities \> grade 1 with the exception of grade 2 lymphopenia and non-hematological toxicities \> grade 1, excluding alopecia and grade 2 neuropathy, from prior anti-cancer therapy
  • Myocardial infarction within 1 year before study day 1, or unstable or uncontrolled disease/condition related to or affecting cardiac function
  • History of stroke, arterial or venous thrombosis, or pulmonary embolism within 1 year before study
  • Active peripheral vascular disease
  • History of bleeding diathesis
  • History of pulmonary hemorrhage or gross hemoptysis within 6 months before study
  • Known history of adrenal hemorrhage
  • Known positive test for human immunodeficiency virus infection, or active hepatitis B or hepatitis C
  • Major surgery within 1 month before study
  • Prior treatment with any agent targeting the angiopoietin-Tie2 signaling pathway
  • Concurrent antitumor treatment, except Lupron for subjects with prostate cancer and selective estrogen receptor modulators (SERMS) for subjects with breast cancer, within 4 weeks (6 weeks for nitrosoureas or mitomycin) before study day 1
  • +4 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (3)

Research Site

Los Angeles, California, 90048, United States

Location

Research Site

Durham, North Carolina, 27710, United States

Location

Research Site

Cleveland, Ohio, 44106, United States

Location

Related Publications (1)

  • Crockett SD, Barry EL, Mott LA, Snover DC, Wallace K, Baron JA. Predictors of Incident Serrated Polyps: Results from a Large Multicenter Clinical Trial. Cancer Epidemiol Biomarkers Prev. 2022 May 4;31(5):1058-1067. doi: 10.1158/1055-9965.EPI-21-1226.

Related Links

MeSH Terms

Conditions

Neoplasms

Study Officials

  • MD

    Amgen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 22, 2010

First Posted

June 4, 2010

Study Start

June 1, 2010

Primary Completion

December 1, 2013

Study Completion

April 1, 2014

Last Updated

March 4, 2015

Record last verified: 2015-02

Locations