NCT01098539

Brief Summary

This randomized, double-blind, active-controlled study evaluates the efficacy and safety of a weekly dose of albiglutide as compared with sitagliptin. Subjects who are renally impaired with a historical diagnosis of type 2 diabetes mellitus and whose glycemia is inadequately controlled on their current regimen of diet and exercise or their antidiabetic therapy of metformin, thiazolidinedione, sulfonylurea, or any combination of these oral antidiabetic medications will be recruited into the study.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
507

participants targeted

Target at P50-P75 for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started May 2010

Longer than P75 for phase_3 diabetes-mellitus-type-2

Geographic Reach
15 countries

218 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

April 1, 2010

Completed
1 day until next milestone

First Posted

Study publicly available on registry

April 2, 2010

Completed
29 days until next milestone

Study Start

First participant enrolled

May 1, 2010

Completed
2.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 1, 2012

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

November 1, 2012

Completed
1.5 years until next milestone

Results Posted

Study results publicly available

May 16, 2014

Completed
Last Updated

February 28, 2017

Status Verified

January 1, 2017

Enrollment Period

2.5 years

First QC Date

April 1, 2010

Results QC Date

April 17, 2014

Last Update Submit

January 16, 2017

Conditions

Keywords

sitagliptinalbiglutiderenal impairment

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Glycosylated Hemoglobin (HbA1c) at Week 26

    HbA1c is a form of hemoglobin that is measured primarily to identify the average plasma glucose concentration over a 2- to 3-month period. The Baseline HbA1c value is defined as the last non-missing value before the start of treatment. Change from Baseline in HbA1c was calculated as the value at Week 26 minus the value at Baseline. The analysis was performed using an Analysis of Covariance (ANCOVA) model with treatment group, region, history of prior myocardial infarction (yes versus no), and age category (\<65 years versus \>=65 years) as factors and Baseline HbA1c as a continuous covariate. The last observation carried forward (LOCF) method was used to impute missing data, in which the last non-missing post-Baseline on-treatment measurement was used to impute the missing measurement. If a participant had missing observation(s) immediately after Baseline, the Baseline observation was not carried forward and was left as missing.

    Baseline; Week 26

Secondary Outcomes (15)

  • Mean Change From Baseline in HbA1c at Weeks 4, 8, 12, 16, and 20: LOCF

    Baseline; Weeks 4, 8, 12, 16, and 20

  • Mean Change From Baseline in HbA1c at Weeks 4, 8, 12, 16, 20, 26, 36, 48, and Week 52: Observed Cases

    Baseline; Weeks 4, 8, 12, 16, 20, 26, 36, 48, and 52

  • Change From Baseline in Fasting Plasma Glucose (FPG) at Week 26

    Baseline; Week 26

  • Mean Change From Baseline in FPG at Weeks 4, 8, 12, 16, 20, and 26: LOCF

    Baseline; Weeks 4, 8, 12, 16, 20, and 26

  • Mean Change From Baseline in Fasting Plasma Glucose (FPG) at Weeks 1, 2, 3, 4, 8, 12, 16, 20, 26, 36, 48, and Week 52: OC

    Baseline; Weeks 1, 2, 3, 4, 8, 12, 16, 20, 26, 36, 48, Week 52

  • +10 more secondary outcomes

Study Arms (2)

albiglutide

ACTIVE COMPARATOR

albiglutide weekly subcutaneous injection + sitagliptin matching placebo

Biological: albiglutide

sitagliptin

ACTIVE COMPARATOR

albiglutide matching placebo + sitagliptin

Drug: sitagliptin

Interventions

albiglutideBIOLOGICAL

albiglutide weekly subcutaneous injection + sitagliptin matching placebo

albiglutide

albiglutide matching placebo + sitagliptin (25mg, 50mg or 100mg depending on level of renal impairment)

sitagliptin

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Renally impaired with a historical diagnosis of type 2 diabetes mellitus and is experiencing inadequate glycemic control on their current regime of diet and exercise or their antidiabetic therapy of metformin, TZD, SU, or any combination of these oral antidiabetic medications
  • BMI \>/=20 kg/m2 and \</=45 kg/m2
  • Fasting C-peptide \>/=0.8 ng/mL (\>/=0.26 nmol/L)
  • HbA1c between 7.0% and 10.0%, inclusive.

You may not qualify if:

  • History of cancer
  • History of treated diabetic gastroparesis
  • Current biliary disease or history of pancreatitis
  • History of significant gastrointestinal surgery
  • Recent clinically significant cardiovascular and/or cerebrovascular disease
  • History of human immunodeficiency virus infection
  • Abnormal liver function or acute symptomatic infection with hepatitis B or hepatitis C
  • Female subject is pregnant (confirmed by laboratory testing), lactating, or \<6 weeks postpartum
  • Known allergy to any GLP 1 analogue, sitagliptin, other study medications' excipients, excipients of albiglutide, or Baker's yeast
  • Receipt of any investigational drug or sitagliptin within the 30 days or 5 half lives, whichever is longer, before Screening or a history of receipt of an investigational antidiabetic drug within the 3 months before randomization or receipt of albiglutide in previous studies

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (218)

GSK Investigational Site

Birmingham, Alabama, 35294, United States

Location

GSK Investigational Site

Gulf Shores, Alabama, 36542, United States

Location

GSK Investigational Site

Huntsville, Alabama, 35801, United States

Location

GSK Investigational Site

Toney, Alabama, 35773, United States

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GSK Investigational Site

Phoenix, Arizona, 85028, United States

Location

GSK Investigational Site

Fresno, California, 93720, United States

Location

GSK Investigational Site

Huntington Beach, California, 92648, United States

Location

GSK Investigational Site

Los Angeles, California, 90017, United States

Location

GSK Investigational Site

Los Angeles, California, 90022, United States

Location

GSK Investigational Site

Los Angeles, California, 90073, United States

Location

GSK Investigational Site

Los Gatos, California, 95032, United States

Location

GSK Investigational Site

Orange, California, 92868, United States

Location

GSK Investigational Site

San Diego, California, 92120, United States

Location

GSK Investigational Site

San Diego, California, 92161, United States

Location

GSK Investigational Site

San Dimas, California, 91773, United States

Location

GSK Investigational Site

Tarzana, California, 91356, United States

Location

GSK Investigational Site

West Hills, California, 91307, United States

Location

GSK Investigational Site

Whittier, California, 90602, United States

Location

GSK Investigational Site

Whittier, California, 90603, United States

Location

GSK Investigational Site

Doral, Florida, 33172, United States

Location

GSK Investigational Site

Hollywood, Florida, 33021, United States

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GSK Investigational Site

Jacksonville, Florida, 32205, United States

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GSK Investigational Site

Miami, Florida, 33136, United States

Location

GSK Investigational Site

Miami Beach, Florida, 33141, United States

Location

GSK Investigational Site

New Port Richey, Florida, 34653, United States

Location

GSK Investigational Site

Pembroke Pines, Florida, 33028, United States

Location

GSK Investigational Site

Plantation, Florida, 33322, United States

Location

GSK Investigational Site

Tampa, Florida, 33613, United States

Location

GSK Investigational Site

Winter Park, Florida, 32789, United States

Location

GSK Investigational Site

Winter Park, Florida, 32792, United States

Location

GSK Investigational Site

Atlanta, Georgia, 30312, United States

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GSK Investigational Site

Atlanta, Georgia, 30342, United States

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GSK Investigational Site

Augusta, Georgia, 30909, United States

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GSK Investigational Site

Blue Ridge, Georgia, 30513, United States

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GSK Investigational Site

Decatur, Georgia, 30032, United States

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GSK Investigational Site

Roswell, Georgia, 30076, United States

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GSK Investigational Site

Stone Mountain, Georgia, 30088, United States

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GSK Investigational Site

Valparaiso, Indiana, 46383, United States

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GSK Investigational Site

Des Moines, Iowa, 50314, United States

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GSK Investigational Site

Mission, Kansas, 66202, United States

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GSK Investigational Site

Lexington, Kentucky, 40504, United States

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GSK Investigational Site

Paducah, Kentucky, 42003, United States

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GSK Investigational Site

Alexandria, Louisiana, 71301, United States

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GSK Investigational Site

Bangor, Maine, 04401, United States

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GSK Investigational Site

Hyattsville, Maryland, 20782, United States

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GSK Investigational Site

Springfield, Massachusetts, 01107, United States

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GSK Investigational Site

Dearborn, Michigan, 48124, United States

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GSK Investigational Site

Detroit, Michigan, 48235, United States

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GSK Investigational Site

Flint, Michigan, 48504, United States

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GSK Investigational Site

Saint Clair Shores, Michigan, 48081, United States

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GSK Investigational Site

Taylor, Michigan, 48180, United States

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GSK Investigational Site

Kansas City, Missouri, 64111, United States

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GSK Investigational Site

Kansas City, Missouri, 64128, United States

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GSK Investigational Site

Springfield, Missouri, 65807, United States

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GSK Investigational Site

Omaha, Nebraska, 68131, United States

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GSK Investigational Site

Las Vegas, Nevada, 89102, United States

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GSK Investigational Site

Las Vegas, Nevada, 89103, United States

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GSK Investigational Site

North Massapequa, New York, 11758, United States

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GSK Investigational Site

Staten Island, New York, 10301, United States

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GSK Investigational Site

Asheville, North Carolina, 28801, United States

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GSK Investigational Site

Hurst, North Carolina, 76054, United States

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GSK Investigational Site

Shelby, North Carolina, 28150, United States

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GSK Investigational Site

Tabor City, North Carolina, 28463, United States

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GSK Investigational Site

Wilmington, North Carolina, 28401, United States

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GSK Investigational Site

Winston-Salem, North Carolina, 27103, United States

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GSK Investigational Site

Cincinnati, Ohio, 45219, United States

Location

GSK Investigational Site

Cleveland, Ohio, 44195, United States

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GSK Investigational Site

Gallipolis, Ohio, 45631, United States

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GSK Investigational Site

Oklahoma City, Oklahoma, 73103, United States

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GSK Investigational Site

Medford, Oregon, 97501, United States

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GSK Investigational Site

Altoona, Pennsylvania, 16602, United States

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GSK Investigational Site

Downington, Pennsylvania, 19335, United States

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GSK Investigational Site

Philadelphia, Pennsylvania, 19146, United States

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GSK Investigational Site

Charleston, South Carolina, 29412, United States

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GSK Investigational Site

Columbia, South Carolina, 29204, United States

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GSK Investigational Site

Greer, South Carolina, 29651, United States

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GSK Investigational Site

North Myrtle Beach, South Carolina, 29582, United States

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GSK Investigational Site

Taylors, South Carolina, 29687, United States

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GSK Investigational Site

Bristol, Tennessee, 37620, United States

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GSK Investigational Site

Franklin, Tennessee, 37067, United States

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GSK Investigational Site

Knoxville, Tennessee, 37923, United States

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GSK Investigational Site

Tullahoma, Tennessee, 37398, United States

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GSK Investigational Site

Arlington, Texas, 76011, United States

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GSK Investigational Site

Arlington, Texas, 76014, United States

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GSK Investigational Site

Austin, Texas, 78751, United States

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GSK Investigational Site

Austin, Texas, 78758, United States

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GSK Investigational Site

Dallas, Texas, 75224, United States

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GSK Investigational Site

Dallas, Texas, 75231, United States

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GSK Investigational Site

Dallas, Texas, 75251, United States

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GSK Investigational Site

Deer Park, Texas, 77536, United States

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GSK Investigational Site

Fort Worth, Texas, 76104, United States

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GSK Investigational Site

Grapevine, Texas, 76051, United States

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GSK Investigational Site

Houston, Texas, 77027, United States

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GSK Investigational Site

Houston, Texas, 77030, United States

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GSK Investigational Site

Houston, Texas, 77036, United States

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GSK Investigational Site

Houston, Texas, 77070, United States

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GSK Investigational Site

Houston, Texas, 77074, United States

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GSK Investigational Site

Houston, Texas, 77081, United States

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GSK Investigational Site

Houston, Texas, 77088, United States

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GSK Investigational Site

Houston, Texas, 77099, United States

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GSK Investigational Site

Humble, Texas, 77338, United States

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GSK Investigational Site

Hurst, Texas, 76054, United States

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GSK Investigational Site

Irving, Texas, 75039, United States

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GSK Investigational Site

Midland, Texas, 79707, United States

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GSK Investigational Site

North Richland Hills, Texas, 76180, United States

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GSK Investigational Site

Pearland, Texas, 77584, United States

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GSK Investigational Site

Plano, Texas, 75075, United States

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GSK Investigational Site

Richardson, Texas, 75080, United States

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GSK Investigational Site

San Antonio, Texas, 78215, United States

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GSK Investigational Site

San Antonio, Texas, 78217, United States

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GSK Investigational Site

San Antonio, Texas, 78258, United States

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GSK Investigational Site

Schertz, Texas, 78154, United States

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GSK Investigational Site

Sugarland, Texas, 77479, United States

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GSK Investigational Site

Tomball, Texas, 77375, United States

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GSK Investigational Site

Bountiful, Utah, 84010, United States

Location

GSK Investigational Site

South Burlington, Vermont, 05403, United States

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GSK Investigational Site

Burke, Virginia, 22015, United States

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GSK Investigational Site

Manassas, Virginia, 20110, United States

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GSK Investigational Site

Norfolk, Virginia, 23510, United States

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GSK Investigational Site

Salem, Virginia, 24153, United States

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GSK Investigational Site

Tacoma, Washington, 98405, United States

Location

GSK Investigational Site

Garran, Australian Capital Territory, 2606, Australia

Location

GSK Investigational Site

Camperdown, New South Wales, 2050, Australia

Location

GSK Investigational Site

Auchenflower, Queensland, 4066, Australia

Location

GSK Investigational Site

Caboolture, Queensland, 4510, Australia

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GSK Investigational Site

Herston, Queensland, 4029, Australia

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GSK Investigational Site

Kippa-Ring, Queensland, 4021, Australia

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GSK Investigational Site

Box Hill, Victoria, 3128, Australia

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GSK Investigational Site

Clayton, Victoria, 3168, Australia

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GSK Investigational Site

Heidelberg, Victoria, 3081, Australia

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GSK Investigational Site

Melbourne, Victoria, 3135, Australia

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GSK Investigational Site

Parkville, Victoria, 3050, Australia

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GSK Investigational Site

Fremantle, Western Australia, 6160, Australia

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GSK Investigational Site

Porto Alegre, Rio Grande do Sul, 90035-170, Brazil

Location

GSK Investigational Site

São Paulo, São Paulo, 05302-001, Brazil

Location

GSK Investigational Site

Brasília, 71625-009, Brazil

Location

GSK Investigational Site

Mogi das Cruzes, 08780 - 090, Brazil

Location

GSK Investigational Site

Barrangquilla, Colombia

Location

GSK Investigational Site

Bogotá, 110221, Colombia

Location

GSK Investigational Site

Floridablanca-Santander, Colombia

Location

GSK Investigational Site

Bad Nauheim, Hesse, 61231, Germany

Location

GSK Investigational Site

Bad Lauterberg im Harz, Lower Saxony, 37431, Germany

Location

GSK Investigational Site

Mainz, Rhineland-Palatinate, 55116, Germany

Location

GSK Investigational Site

Dresden, Saxony, 01307, Germany

Location

GSK Investigational Site

Berlin, State of Berlin, 10115, Germany

Location

GSK Investigational Site

Ahmedabad, 380015, India

Location

GSK Investigational Site

Bangalore, 560 010, India

Location

GSK Investigational Site

Bangalore, 560 054, India

Location

GSK Investigational Site

Bangalore, 560043, India

Location

GSK Investigational Site

Bangalore, 560052, India

Location

GSK Investigational Site

Bangalore, 560078, India

Location

GSK Investigational Site

Belagavi, 590001, India

Location

GSK Investigational Site

Belagavi, 590010, India

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GSK Investigational Site

Chennai, 600013, India

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GSK Investigational Site

Lucknow, 226005, India

Location

GSK Investigational Site

Manipal, 576104, India

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GSK Investigational Site

Mumbai, 400 008, India

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GSK Investigational Site

Nashik, 422013, India

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GSK Investigational Site

Ashkelon, 78278, Israel

Location

GSK Investigational Site

Beersheba, 84101, Israel

Location

GSK Investigational Site

Haifa, 31096, Israel

Location

GSK Investigational Site

Haifa, 35251, Israel

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GSK Investigational Site

Holon, 58100, Israel

Location

GSK Investigational Site

Kfar Saba, 44281, Israel

Location

GSK Investigational Site

Safed, 13110, Israel

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GSK Investigational Site

Arequipa, Arequipa, 54, Peru

Location

GSK Investigational Site

Ica, Ica, 11, Peru

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GSK Investigational Site

Lima, Lima Province, 01, Peru

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GSK Investigational Site

Lima, Lima Province, 17, Peru

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GSK Investigational Site

Callao, Lima, Callao 2, Peru

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GSK Investigational Site

Piura, Piura, Peru

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GSK Investigational Site

Lima, Lima 1, Peru

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GSK Investigational Site

Trujillo, Peru

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GSK Investigational Site

Cebu City, 6000, Philippines

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GSK Investigational Site

Iloilo City, 5000, Philippines

Location

GSK Investigational Site

Makati City, 1218, Philippines

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GSK Investigational Site

Pasay, 1300, Philippines

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GSK Investigational Site

Tagbilaran City, 6300, Philippines

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GSK Investigational Site

Nizhny Novgorod, 603126, Russia

Location

GSK Investigational Site

Saratov, 410030, Russia

Location

GSK Investigational Site

St'Petersburg, 194156, Russia

Location

GSK Investigational Site

Yaroslavl, 150062, Russia

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GSK Investigational Site

Port Elizabeth, Eastern Cape, 6014, South Africa

Location

GSK Investigational Site

Johannesburg, Gauteng, 2013, South Africa

Location

GSK Investigational Site

Johannesburg, Gauteng, 2193, South Africa

Location

GSK Investigational Site

Lenasia, Gauteng, 1827, South Africa

Location

GSK Investigational Site

Pretoria, Gauteng, 0084, South Africa

Location

GSK Investigational Site

Durban, KwaZulu-Natal, 4092, South Africa

Location

GSK Investigational Site

Phoenix, KwaZulu-Natal, 4068, South Africa

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GSK Investigational Site

Houghton Estate, 2198, South Africa

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GSK Investigational Site

Pretoria, 0002, South Africa

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GSK Investigational Site

Somerset West, 07129, South Africa

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GSK Investigational Site

Tygerberg, 7505, South Africa

Location

GSK Investigational Site

Seongnam-si, 463712, South Korea

Location

GSK Investigational Site

Seoul, 135-720, South Korea

Location

GSK Investigational Site

Seoul, 136-705, South Korea

Location

GSK Investigational Site

Seoul, 137-701, South Korea

Location

GSK Investigational Site

Seoul, 139-872, South Korea

Location

GSK Investigational Site

Suwon, Kyonggi-do, 443-721, South Korea

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GSK Investigational Site

A Coruña, 15006, Spain

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GSK Investigational Site

Alicante, 03114, Spain

Location

GSK Investigational Site

Málaga, 29010, Spain

Location

GSK Investigational Site

Palma de Mallorca, 07014, Spain

Location

GSK Investigational Site

Santiago de Compostela, 15706, Spain

Location

GSK Investigational Site

Seville, 41003, Spain

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GSK Investigational Site

Torrevieja (Alicante), 03186, Spain

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GSK Investigational Site

Kaohsiung City, 833, Taiwan

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GSK Investigational Site

Taichung, 404, Taiwan

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GSK Investigational Site

Tainan, 71044, Taiwan

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GSK Investigational Site

Coventry, West Midlands, CV2 2DX, United Kingdom

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GSK Investigational Site

Birmingham, B9 5SS, United Kingdom

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GSK Investigational Site

Hertfordshire, United Kingdom

Location

GSK Investigational Site

Hull, HU3 2RW, United Kingdom

Location

GSK Investigational Site

Liverpool, L9 7AL, United Kingdom

Location

GSK Investigational Site

Livingston, EH54 6PP, United Kingdom

Location

GSK Investigational Site

London, SE1 9NH, United Kingdom

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GSK Investigational Site

Plymouth, PL6 8BX, United Kingdom

Location

GSK Investigational Site

Swansea, SA6 6NL, United Kingdom

Location

Related Publications (2)

  • Natale P, Green SC, Tunnicliffe DJ, Pellegrino G, Toyama T, Strippoli GF. Glucagon-like peptide 1 (GLP-1) receptor agonists for people with chronic kidney disease and diabetes. Cochrane Database Syst Rev. 2025 Feb 18;2(2):CD015849. doi: 10.1002/14651858.CD015849.pub2.

  • Young MA, Wald JA, Matthews JE, Scott R, Hodge RJ, Zhi H, Reinhardt RR. Clinical pharmacology of albiglutide, a GLP-1 receptor agonist. Postgrad Med. 2014 Nov;126(7):84-97. doi: 10.3810/pgm.2014.11.2836.

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Renal Insufficiency

Interventions

rGLP-1 proteinSitagliptin Phosphate

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesKidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

TriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrazines

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 1, 2010

First Posted

April 2, 2010

Study Start

May 1, 2010

Primary Completion

November 1, 2012

Study Completion

November 1, 2012

Last Updated

February 28, 2017

Results First Posted

May 16, 2014

Record last verified: 2017-01

Data Sharing

IPD Sharing
Will share

Patient-level data for this study will be made available through www.clinicalstudydatarequest.com following the timelines and process described on this site.

Available IPD Datasets

Study Protocol (114130)Access
Informed Consent Form (114130)Access
Dataset Specification (114130)Access
Annotated Case Report Form (114130)Access
Clinical Study Report (114130)Access
Statistical Analysis Plan (114130)Access
Individual Participant Data Set (114130)Access

Locations