NCT01063920

Brief Summary

LT-NS001 is a prodrug of Naproxen, which is inactive as a cox inhibitor while intact and is rapidly metabolized to Naproxen once absorbed. This trial will compare the rate of gastric ulcer by endoscopy over three months in patients with knee osteoarthritis, with patients receiving either LT-NS001 at a dose which provides comparable dose levels of Naproxen, or Naprosyn® 500mg (an approved treatment for OA).

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
534

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Feb 2010

Shorter than P25 for phase_2

Geographic Reach
1 country

65 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 29, 2010

Completed
3 days until next milestone

Study Start

First participant enrolled

February 1, 2010

Completed
4 days until next milestone

First Posted

Study publicly available on registry

February 5, 2010

Completed
9 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 1, 2010

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

November 1, 2010

Completed
Last Updated

January 24, 2011

Status Verified

January 1, 2011

Enrollment Period

9 months

First QC Date

January 29, 2010

Last Update Submit

January 20, 2011

Conditions

Keywords

LT-NS001Gastric UlcersNSAIDOsteoarthritisNaproxen

Outcome Measures

Primary Outcomes (1)

  • Gastric Ulcer by Endoscopy

    Baseline, Day 29, Day 57 and Day 85

Secondary Outcomes (2)

  • Western Ontario and McMaster Universities Osteoarthritis Index (WOMAC) score

    Screening, Baseline, Days 15, 29, 57 and 85

  • Population pharmacokinetic analysis will assess the influence of covariates on the absorption/metabolism of LT-NS001 to naproxen

    Two separate days after Day 14, at least two weeks apart

Study Arms (2)

LT-NS001

EXPERIMENTAL

LT-NS001 1200 mg b.i.d. p.o. for 12 weeks

Drug: LT-NS001

Naprosyn®

ACTIVE COMPARATOR

Naprosyn® 500 mg b.i.d for 12 weeks

Drug: Naprosyn®

Interventions

1200 mg b.i.d. p.o. for 12 weeks

LT-NS001

500 mg b.i.d. p.o. for 12 weeks

Naprosyn®

Eligibility Criteria

Age45 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Osteoarthritis of knee
  • Appropriate candidate for chronic NSAID therapy due to moderate or severe pain on most days in the 28 days before screening for study.

You may not qualify if:

  • Pregnant/Nursing women
  • History of GI bleeding, perforation or obstruction
  • A documented symptomatic GI ulcer during past 5 years
  • Presence of GI ulcer or more than 2 erosions on screening endoscopy
  • Allergy to naproxen (or naproxen intolerance), acetylsalicylic acid, or other NSAID drug

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (65)

Greystone Medical Research, LLC

Birmingham, Alabama, 35242, United States

Location

Clinical Research Associates

Huntsville, Alabama, 35801, United States

Location

Radiant Research

Chandler, Arizona, 85225, United States

Location

Dedicated Clinical Research Inc.

Surprise, Arizona, 85340, United States

Location

Radiant Research Inc.

Tucson, Arizona, 85710, United States

Location

Adobe Gastroenterology Research, LLC

Tucson, Arizona, 85712, United States

Location

Genova Clinical Research Inc.

Tucson, Arizona, 85741, United States

Location

Lynn Institute of the Ozarks

Little Rock, Arkansas, 72205, United States

Location

Orange County Clinical Trials

Anaheim, California, 92801, United States

Location

Theresa Sligh, MD

Burbank, California, 91505, United States

Location

Torrance Clinical Research

Lomeita, California, 90274, United States

Location

West Gastroenterology Associates

Los Angeles, California, 90045, United States

Location

Facey Medical Center

Mission Hills, California, 91345, United States

Location

Desert Medical Group

Palm Springs, California, 92262, United States

Location

Medical Affiliated Research Center Inc.

San Diego, California, 35801, United States

Location

Cynthia Schaeffer, MD

San Diego, California, 92114, United States

Location

Medical Associates Research Group

San Diego, California, 92123, United States

Location

Lynn Institute of the Rockies

Colorado Springs, Colorado, 80907, United States

Location

Rocky Mountain Center for Clinical Research

Wheat Ridge, Colorado, 80033, United States

Location

Eastern Clinical Research Unit

Hialeah, Florida, 33013, United States

Location

Nature Coast Clinical Research

Inverness, Florida, 33452, United States

Location

Drug Study Institute

Jupiter, Florida, 33458, United States

Location

University Clinical Research Inc.

Pembroke Pines, Florida, 33024, United States

Location

Radiant Research

Pinellas Park, Florida, 33781, United States

Location

Accord Clinical Research LLC

Port Orange, Florida, 32129, United States

Location

Miami Research Associates

South Miami, Florida, 33143, United States

Location

Palm Beach Research Center

West Palm Beach, Florida, 33409, United States

Location

Gold Coast Research LLC

Weston, Florida, 33317, United States

Location

Thomas Schnitzer, MD

Chicago, Illinois, 60611, United States

Location

Welborn Clinic

Evansville, Indiana, 47710, United States

Location

MediSphere Medical Research Center LLC

Evansville, Indiana, 47714, United States

Location

Venture Resource Group Inc.

Mission, Kansas, 66202, United States

Location

Pinnacle Medical Research

Overland Park, Kansas, 66215, United States

Location

Delta Research Partners LLC

Bastrop, Louisiana, 71201, United States

Location

SNBL Clinical Pharmacology Center

Baltimore, Maryland, 21201, United States

Location

Metropolitan Gastroenterolgy Group PC

Chevy Chase, Maryland, 20815, United States

Location

Arthritis and Osteoporosis Cener of Maryland

Frederick, Maryland, 21702, United States

Location

MidAtlantic Medical Research Centers/Bean Medical Center

Hollywood, Maryland, 20636, United States

Location

Dynamic Clinical Research

Kansas City, Missouri, 64114, United States

Location

Sundance Clinical Research

St Louis, Missouri, 63141, United States

Location

Montana Health Research Institute Inc.

Billings, Montana, 59102, United States

Location

Advanced Biomedical Research of America

Las Vegas, Nevada, 89123, United States

Location

Affiliated Clinical Research Inc.

Las Vegas, Nevada, 89144, United States

Location

Clifton-Wallington Medical Group

Clifton, New Jersey, 07013, United States

Location

Research Across America

New York, New York, 10022, United States

Location

Allergy Asthma Immunology of Rochester Research Center

Rochester, New York, 14618, United States

Location

Carolina Digestive Health Associates PA

Charlotte, North Carolina, 28075, United States

Location

Peters Medical Research LLC

High Point, North Carolina, 27262, United States

Location

Wake Research Associates

Raleigh, North Carolina, 27612, United States

Location

Radiant Research-Akron

Akron, Ohio, 44311, United States

Location

Consultants for Clinical Research

Cincinnati, Ohio, 45219, United States

Location

Health Research of Oklahoma

Oklahoma City, Oklahoma, 73103, United States

Location

Lynn Health Science Institute

Oklahoma City, Oklahoma, 73112, United States

Location

Sooner Clinical Research

Oklahoma City, Oklahoma, 73112, United States

Location

Clinical Research Associates LLC

Oklahoma City, Oklahoma, 73116, United States

Location

Keith Klatt, MD

Portland, Oregon, 97739, United States

Location

Altoona Center for Clinical Research

Duncansville, Pennsylvania, 16635, United States

Location

Corsicana Medical Research PLLC

Corsicana, Texas, 75110, United States

Location

Galenos Research

Dallas, Texas, 75251, United States

Location

Clinical Trial Network

Houston, Texas, 77074, United States

Location

Houston Endoscopy and Research Center

Houston, Texas, 77079, United States

Location

Houston Medical Research Associates

Houston, Texas, 77090, United States

Location

Quality Research Inc.

San Antonio, Texas, 78209, United States

Location

Arthritis and Osteoporosis Clinic Research Center of Central Texas

Waco, Texas, 76708, United States

Location

Physicians Research Options LLC

Draper, Utah, 84020, United States

Location

MeSH Terms

Conditions

OsteoarthritisStomach Ulcer

Interventions

Naproxen

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic DiseasesPeptic UlcerDuodenal DiseasesIntestinal DiseasesGastrointestinal DiseasesDigestive System DiseasesStomach Diseases

Intervention Hierarchy (Ancestors)

Naphthaleneacetic AcidsNaphthalenesPolycyclic Aromatic HydrocarbonsHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsPolycyclic Compounds

Study Officials

  • Jay L Goldstein, MD

    University of Illinois at Chicago, Department of Medicine

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, CARE PROVIDER
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

January 29, 2010

First Posted

February 5, 2010

Study Start

February 1, 2010

Primary Completion

November 1, 2010

Study Completion

November 1, 2010

Last Updated

January 24, 2011

Record last verified: 2011-01

Locations