NCT00418782

Brief Summary

CE-224535 is a new medication being developed as an analgesic and anti-inflammatory agent for the treatment of the signs and symptoms of osteoarthritis (OA). The purpose of this study is to evaluate the analgesic and anti inflammatory efficacy and safety of CE 224,535 versus placebo and naproxen treatment in patients with OA knee pain.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
212

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Jan 2007

Shorter than P25 for phase_2

Geographic Reach
1 country

46 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

January 1, 2007

Completed
3 days until next milestone

First Submitted

Initial submission to the registry

January 4, 2007

Completed
1 day until next milestone

First Posted

Study publicly available on registry

January 5, 2007

Completed
7 months until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2007

Completed
Last Updated

December 5, 2018

Status Verified

December 1, 2018

First QC Date

January 4, 2007

Last Update Submit

December 3, 2018

Conditions

Outcome Measures

Primary Outcomes (2)

  • To determine the safety, tolerability, pharmacokinetics (PK), and pharmacodynamics (PD) of oral multiple doses of CE 224,535 in subjects with OA of the knee

    ongoing

  • The primary endpoint is the change from Baseline (Day 1) to Week 2 (Day 14) in the WOMAC Pain domain score.

    Day 1-14

Secondary Outcomes (9)

  • The change from Baseline to each day (Days 1 to 6) and over the average response in Days 1 to 6 using an 11 point numeric rating scale (NRS) from 0-10 on daily pain diary;

    (Days 1 to 6)

  • Patient's Global Impression of Change (PGIC) at Week 2;

    Week 2

  • The change from Baseline to Weeks 1 and 2 in the Patient's Global Assessment of Arthritic Condition;

    Baseline to Weeks 1 and 2

  • The change from Baseline to Week 1 (Day 7) in the WOMAC Pain domain score;

    Day 7

  • The change from Baseline to Weeks 1 and 2 (Days 7 and 14) in the WOMAC Stiffness domain score;

    Days 7 and 14

  • +4 more secondary outcomes

Study Arms (3)

1

ACTIVE COMPARATOR
Drug: naproxen

2

EXPERIMENTAL
Drug: CE-224535

3

PLACEBO COMPARATOR
Drug: placebo

Interventions

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Is a healthy adult 18 to 75 years of age, inclusive, in general good health and with diagnosis of knee OA, as determined by the American College of Rheumatology (ACR) clinical/radiographic classification criteria for OA of the knee.
  • Women must be of non childbearing potential (amenorrhea for at least 1 year PLUS have a serum follicle stimulating hormone (FSH) level \>30 IU/L, bilateral oophorectomy or hysterectomy), and have a confirmed negative serum pregnancy test at the screening visit prior to randomization.

You may not qualify if:

  • History of other diseases that may involve the study joint, including inflammatory joint diseases, crystalline disease, endocrinopathies, metabolic diseases, infections, neuropathic disorders, avascular necrosis, Paget's disease, or tumors.
  • Women of childbearing potential, or who are pregnant or lactating.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (46)

Pfizer Investigational Site

Anniston, Alabama, 36207, United States

Location

Pfizer Investigational Site

Bayou La Batre, Alabama, 36509, United States

Location

Pfizer Investigational Site

Birmingham, Alabama, 35209, United States

Location

Pfizer Investigational Site

Birmingham, Alabama, 35216, United States

Location

Pfizer Investigational Site

Birmingham, Alabama, 35242, United States

Location

Pfizer Investigational Site

Hot Springs, Arkansas, 71913, United States

Location

Pfizer Investigational Site

Northridge, California, 91325, United States

Location

Pfizer Investigational Site

Sacramento, California, 95825, United States

Location

Pfizer Investigational Site

Tarzana, California, 91356, United States

Location

Pfizer Investigational Site

Denver, Colorado, 80204, United States

Location

Pfizer Investigational Site

Denver, Colorado, 80206, United States

Location

Pfizer Investigational Site

Westminster, Colorado, 80030, United States

Location

Pfizer Investigational Site

Clearwater, Florida, 33761, United States

Location

Pfizer Investigational Site

DeFuniak Springs, Florida, 32435, United States

Location

Pfizer Investigational Site

Destin, Florida, 32541, United States

Location

Pfizer Investigational Site

Pensacola, Florida, 32503, United States

Location

Pfizer Investigational Site

Chicago, Illinois, 60053, United States

Location

Pfizer Investigational Site

Gurnee, Illinois, 60031, United States

Location

Pfizer Investigational Site

Avon, Indiana, 46123, United States

Location

Pfizer Investigational Site

Indianapolis, Indiana, 46250, United States

Location

Pfizer Investigational Site

Gretna, Louisiana, 70056, United States

Location

Pfizer Investigational Site

Kenner, Louisiana, 70065, United States

Location

Pfizer Investigational Site

Metairie, Louisiana, 70002, United States

Location

Pfizer Investigational Site

Baltimore, Maryland, 21218, United States

Location

Pfizer Investigational Site

Frederick, Maryland, 21702, United States

Location

Pfizer Investigational Site

Flowood, Mississippi, 39232, United States

Location

Pfizer Investigational Site

Columbia, Missouri, 65212, United States

Location

Pfizer Investigational Site

Kansas City, Missouri, 64114, United States

Location

Pfizer Investigational Site

Missoula, Montana, 59802, United States

Location

Pfizer Investigational Site

Trenton, New Jersey, 08611, United States

Location

Pfizer Investigational Site

Beavercreek, Ohio, 45440, United States

Location

Pfizer Investigational Site

Cincinnati, Ohio, 45242, United States

Location

Pfizer Investigational Site

Kettering, Ohio, 45429, United States

Location

Pfizer Investigational Site

Ashland, Oregon, 97520, United States

Location

Pfizer Investigational Site

Eugene, Oregon, 97404, United States

Location

Pfizer Investigational Site

Duncansville, Pennsylvania, 16635, United States

Location

Pfizer Investigational Site

Summerville, South Carolina, 29485, United States

Location

Pfizer Investigational Site

Collierville, Tennessee, 38017, United States

Location

Pfizer Investigational Site

Knoxville, Tennessee, 37909-1900, United States

Location

Pfizer Investigational Site

Memphis, Tennessee, 38104, United States

Location

Pfizer Investigational Site

Bryan, Texas, 77802, United States

Location

Pfizer Investigational Site

Longview, Texas, 75605, United States

Location

Pfizer Investigational Site

San Antonio, Texas, 78213, United States

Location

Pfizer Investigational Site

San Antonio, Texas, 78229, United States

Location

Pfizer Investigational Site

Arlington, Virginia, 22205, United States

Location

Pfizer Investigational Site

Spokane, Washington, 99216, United States

Location

Related Links

MeSH Terms

Conditions

Osteoarthritis

Interventions

NaproxenCE 224,535

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic Diseases

Intervention Hierarchy (Ancestors)

Naphthaleneacetic AcidsNaphthalenesPolycyclic Aromatic HydrocarbonsHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsPolycyclic Compounds

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

January 4, 2007

First Posted

January 5, 2007

Study Start

January 1, 2007

Study Completion

August 1, 2007

Last Updated

December 5, 2018

Record last verified: 2018-12

Locations