NCT00984113

Brief Summary

The purpose of the study is to determine the pharmacokinetics and safety of elinogrel and its metabolite in patients with mild, moderate, and severe renal impairment compared to healthy volunteers.

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
44

participants targeted

Target at P50-P75 for phase_1

Timeline
Completed

Started Sep 2009

Shorter than P25 for phase_1

Geographic Reach
1 country

2 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2009

Completed
15 days until next milestone

First Submitted

Initial submission to the registry

September 16, 2009

Completed
9 days until next milestone

First Posted

Study publicly available on registry

September 25, 2009

Completed
2 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 1, 2009

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

December 1, 2009

Completed
Last Updated

August 4, 2023

Status Verified

August 1, 2023

Enrollment Period

3 months

First QC Date

September 16, 2009

Last Update Submit

August 3, 2023

Conditions

Keywords

ElinogrelRenal impairmentHealthyKidney dysfunction

Outcome Measures

Primary Outcomes (1)

  • Pharmacokinetics of elinogrel and its metabolite

    The PK parameters calculated for both elinogrel and PRT060301 were: * AUC0-12h, Cmax, and Tmax on Day 1/Day 7 and T1/2, RACC \& CLR on Day 7 * For elinogrel only, CLss/F and Vss/F were also calculated

    7 days

Secondary Outcomes (2)

  • Safety assessments will include vital signs, electrocardiograms and adverse events

    9 days

  • Measures of platelet function

    7 days

Study Arms (6)

A-Patients with mild renal impairment

EXPERIMENTAL
Drug: Elinogrel

B-Healthy subjects matched to Group A

EXPERIMENTAL
Drug: Elinogrel

C-Patients with moderate renal impairment

EXPERIMENTAL
Drug: Elinogrel

D-Healthy subjects matched to Group C

EXPERIMENTAL
Drug: Elinogrel

E-Patients with severe renal impairment

EXPERIMENTAL
Drug: Elinogrel

F-Healthy subjects matched to Group E

EXPERIMENTAL
Drug: Elinogrel

Interventions

100 mg elinogrel b.i.d. with aspirin q.d. for 7 days and aspirin alone for 4 days (Dose of aspirin is 81 mg in the US and 100 mg in Germany)

Also known as: PRT060128
A-Patients with mild renal impairmentB-Healthy subjects matched to Group AC-Patients with moderate renal impairmentD-Healthy subjects matched to Group CE-Patients with severe renal impairmentF-Healthy subjects matched to Group E

Eligibility Criteria

Age18 Years - 80 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Able to understand and sign the written informed consent
  • Subjects should have either normal renal function or have stable renal disease

You may not qualify if:

  • History of heart disease
  • Unstable or clinically significant other disorders such as respiratory, hepatic, metabolic, psychiatric or gastrointestinal disorder

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (2)

DaVita Clinical Research

Minneapolis, Minnesota, 55404, United States

Location

NOCR-Knoxville

Knoxville, Tennessee, 37920, United States

Location

MeSH Terms

Conditions

Renal Insufficiency

Interventions

elinogrel

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital Diseases

Study Officials

  • Matthew W McClure, MD

    Portola Pharmaceuticals Inc.

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY

Study Record Dates

First Submitted

September 16, 2009

First Posted

September 25, 2009

Study Start

September 1, 2009

Primary Completion

December 1, 2009

Study Completion

December 1, 2009

Last Updated

August 4, 2023

Record last verified: 2023-08

Locations