NCT00745316

Brief Summary

The main purpose of this study is to determine the safety and tolerability of tonapofylline (BG9928) when given at different doses to patients with heart failure and renal insufficiency. This study will also explore:

  • Disease related quality-of-life
  • Exercise capacity
  • Renal function
  • Concomitant medications

Trial Health

57
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
34

participants targeted

Target at P25-P50 for phase_2

Timeline
Completed

Started Feb 2009

Shorter than P25 for phase_2

Geographic Reach
1 country

30 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 2, 2008

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 3, 2008

Completed
5 months until next milestone

Study Start

First participant enrolled

February 1, 2009

Completed
11 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

January 1, 2010

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

January 1, 2010

Completed
Last Updated

September 11, 2023

Status Verified

September 1, 2023

Enrollment Period

11 months

First QC Date

September 2, 2008

Last Update Submit

September 4, 2023

Conditions

Keywords

Heart FailureRenal InsufficiencyCongestive Heart Failure

Outcome Measures

Primary Outcomes (1)

  • To assess the safety and tolerability of BG9928 administered to subjects with heart failure and renal insufficiency.

    16 Weeks

Study Arms (6)

1

EXPERIMENTAL

oral Dose 1

Drug: Tonapofylline

2

EXPERIMENTAL

oral Dose 2

Drug: Tonapofylline

3

EXPERIMENTAL

oral Dose 3

Drug: Tonapofylline

4

EXPERIMENTAL

oral Dose 4

Drug: Tonapofylline

5

EXPERIMENTAL

oral Dose 5

Drug: Tonapofylline

6

PLACEBO COMPARATOR

Placebo - 2 capsules bid

Drug: Placebo

Interventions

Oral Tonapofylline - 2 capsules bid

Also known as: BG9928; Selective Adenosine A1 Receptor Antagonist
12345

Oral placebo - 2 capsules bid

6

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • years of age or older
  • Diagnosis of heart failure requiring hospitalization \>1 and ≤12 months prior to screening
  • NYHA Class III or IV at the time of screening
  • Renal insufficiency as defined by eGFR ≥20 and ≤70 mL/min/1.73 m2
  • Negative pregnancy test

You may not qualify if:

  • History of an allergic reaction to any xanthine-containing compound.
  • History of seizure
  • History of stroke
  • Serious systemic infection
  • Sustained systolic blood pressure \>170 or \<90 mmHg
  • Myocardial infarction within 30 days of Day 1
  • Hemodynamically destabilizing arrhythmia within 30 days of Day 1
  • Uncorrected hemodynamically significant primary valvular disease
  • Known obstructive or restrictive cardiomyopathy
  • Cardiac surgery within 60 days prior to Day 1
  • Likely to undergo cardiac transplantation, device implantation, or other cardiac surgery within next three months
  • Evidence of malignancy within 6 months prior to Day 1.
  • Participation in any other investigational study of drugs or devices within 30 days prior to Day 1.
  • Receiving aminophylline, theophylline, pentoxifylline, dyphylline or adenosine
  • Presence of any clinically significant condition that might interfere with optimal safe participation in this study

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (30)

Unknown Facility

Huntsville, Alabama, 35801, United States

Location

Unknown Facility

Mobile, Alabama, 36608, United States

Location

Unknown Facility

Scottsdale, Arizona, 85251, United States

Location

Unknown Facility

Tucson, Arizona, 85710, United States

Location

Unknown Facility

Beverly Hills, California, 90210, United States

Location

Unknown Facility

San Diego, California, 92103, United States

Location

Unknown Facility

Denver, Colorado, 80218, United States

Location

Unknown Facility

Bridgeport, Connecticut, 06606, United States

Location

Unknown Facility

Jacksonville, Florida, 32209, United States

Location

Unknown Facility

Melbourne, Florida, 32901, United States

Location

Unknown Facility

Ormond Beach, Florida, 32174, United States

Location

Unknown Facility

Chicago, Illinois, 60612, United States

Location

Unknown Facility

Maywood, Illinois, 60153, United States

Location

Unknown Facility

Indianapolis, Indiana, 46260, United States

Location

Unknown Facility

Iowa City, Iowa, 52242, United States

Location

Unknown Facility

Owensboro, Kentucky, 42303, United States

Location

Unknown Facility

Baltimore, Maryland, 21201, United States

Location

Unknown Facility

Boston, Massachusetts, 02114, United States

Location

Unknown Facility

Boston, Massachusetts, 02115, United States

Location

Unknown Facility

Minneapolis, Minnesota, 55415, United States

Location

Unknown Facility

Lincoln, Nebraska, 68506, United States

Location

Unknown Facility

The Bronx, New York, 10461, United States

Location

Unknown Facility

Cincinnati, Ohio, 45219, United States

Location

Unknown Facility

Cincinnati, Ohio, 45267, United States

Location

Unknown Facility

Oklahoma City, Oklahoma, 73120, United States

Location

Unknown Facility

Lancaster, Pennsylvania, 17602, United States

Location

Unknown Facility

Germantown, Tennessee, 38138, United States

Location

Unknown Facility

Roanoke, Virginia, 24014, United States

Location

Unknown Facility

Beloit, Wisconsin, 53511, United States

Location

Unknown Facility

Madison, Wisconsin, 53792, United States

Location

MeSH Terms

Conditions

Renal InsufficiencyHeart Failure

Interventions

BG 9928

Condition Hierarchy (Ancestors)

Kidney DiseasesUrologic DiseasesFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesMale Urogenital DiseasesHeart DiseasesCardiovascular Diseases

Study Officials

  • Medical Director

    Biogen

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 2, 2008

First Posted

September 3, 2008

Study Start

February 1, 2009

Primary Completion

January 1, 2010

Study Completion

January 1, 2010

Last Updated

September 11, 2023

Record last verified: 2023-09

Locations