NCT00565812

Brief Summary

The objective of this 2-year study is to evaluate the safety, tolerability and disease modifying efficacy of SD 6010, an inhibitor of inducible nitric oxide synthase (iNOS), in overweight and obese subjects with knee osteoarthritis. The efficacy of SD-6010 will be evaluated by radiography using joint space narrowing in the medial tibiofemoral compartment of the study knee as the primary endpoint.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,457

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Nov 2007

Typical duration for phase_2

Geographic Reach
14 countries

183 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 1, 2007

Completed
28 days until next milestone

First Submitted

Initial submission to the registry

November 29, 2007

Completed
1 day until next milestone

First Posted

Study publicly available on registry

November 30, 2007

Completed
3.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 1, 2011

Completed
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

November 1, 2011

Completed
5.2 years until next milestone

Results Posted

Study results publicly available

December 30, 2016

Completed
Last Updated

December 30, 2016

Status Verified

November 1, 2016

Enrollment Period

3.9 years

First QC Date

November 29, 2007

Results QC Date

June 22, 2016

Last Update Submit

November 1, 2016

Conditions

Keywords

knee Osteoarthritis Disease Modifying Osteoarthritis Drug

Outcome Measures

Primary Outcomes (3)

  • Rate of Progression of Joint Space Narrowing

    Rate of progression of joint space narrowing (JSN) was defined as narrowing in joint space width (JSW) over the course of the study. It was measured radiographically in the medial tibiofemoral of knee of participants with OA. The slope reported in millimeter per year (mm/year) over a 2 year period was used to assess the rate of progression of JSN. Negative values indicating a worsening of osteoarthritis.

    Baseline up to Month 24

  • Rate of Progression of Joint Space Narrowing in Participants With Kellgren and Lawrence Grade Less Than or Equal to (<=) 2

    Rate of progression of JSN was defined as narrowing in joint space width over the course of the study. It was measured radiographically in the medial tibiofemoral of knee of participants with OA. The slope reported in mm/year over a 2 year period was used to assess the rate of progression of JSN. KLG system was a method of classifying the severity of knee OA using five grades (0 \[no severity\] to 4 \[maximum severity\], higher grade indicating worse knee function). Negative values of slope indicating a worsening of osteoarthritis.

    Baseline up to Month 24

  • Rate of Progression of Joint Space Narrowing in Participants With Kellgren and Lawrence Grade Equal to (=) 3

    Rate of progression of JSN was defined as narrowing in joint space width over the course of the study. It was measured radiographically in the medial tibiofemoral of knee of participants with OA. The slope reported in mm/year over a 2 year period was used to assess the rate of progression of JSN. KLG system was a method of classifying the severity of knee OA using five grades (0 \[no severity\] to 4 \[maximum severity\], higher grade indicating worse knee function). Negative values of slope indicating a worsening of osteoarthritis.

    Baseline up to Month 24

Secondary Outcomes (35)

  • Change From Baseline in Western Ontario and MacMaster Osteoarthritis Index (WOMAC) Composite Index Score at Month 3, 6, 12, 18 and 24

    Baseline, Month 3, 6, 12, 18, 24

  • Change From Baseline in Western Ontario and MacMaster Osteoarthritis Index Pain Subscale Score at Month 3, 6, 12, 18 and 24

    Baseline, Month 3, 6, 12, 18, 24

  • Change From Baseline in Western Ontario and MacMaster Osteoarthritis Index Pain Stiffness Subscale Score at Month 3, 6, 12, 18 and 24

    Baseline, Month 3, 6, 12, 18, 24

  • Change From Baseline in Western Ontario and MacMaster Osteoarthritis Index Physical Function Subscale Score at Month 3, 6, 12, 18 and 24

    Baseline, Month 3, 6, 12, 18, 24

  • Change From Baseline in Patient Assessment of Arthritic Pain Visual Analog Scale (VAS) Score at Month 3, 6, 12, 18 and 24

    Baseline, Month 3, 6, 12, 18, 24

  • +30 more secondary outcomes

Other Outcomes (6)

  • Number of Participants With Treatment-Emergent Adverse Events (AEs) and Serious Adverse Events (SAEs)

    Baseline up to 7-10 days after last dose of study drug (Week 111)

  • Number of Participants With Electrocardiogram (ECG) Abnormalities

    Baseline, Month 3, 6, 12, 18, 24

  • Number of Participants With Laboratory Test Abnormalities

    Baseline up to Week 111

  • +3 more other outcomes

Study Arms (3)

200 mg

ACTIVE COMPARATOR

High dose active comparator

Drug: SD-6010

50 mg

ACTIVE COMPARATOR

Low dose active comparator

Drug: SD-6010

Placebo

PLACEBO COMPARATOR

Placebo comparator to be used for control purposes

Drug: Placebo

Interventions

200 mg tablets once a day for 2 years

200 mg

Placebo tablets once a day for 2 years

Placebo

Eligibility Criteria

Age40 Years - 99 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects aged \>= 40 years with a BMI \>= 25 and \<= 40 kg/m2
  • In the past, has been diagnosed with knee OA
  • Radiographic evidence of OA in the study knee

You may not qualify if:

  • A diagnosis of any other rheumatic disease
  • Current conditions in the study knee that would confound efficacy
  • Selected, traditional clinical safety and laboratory parameters

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (183)

Brookwood Internists, P.C.

Birmingham, Alabama, 35209, United States

Location

Greystone Medical Center

Birmingham, Alabama, 35242, United States

Location

Pivotal Research Centers

Peoria, Arizona, 85381, United States

Location

Arizona Research Center

Phoenix, Arizona, 85023, United States

Location

Pivotal Research Centers

Phoenix, Arizona, 85027, United States

Location

University of Arizona

Tucson, Arizona, 85724, United States

Location

Martin Bowen Hefley Orthopedics

Little Rock, Arkansas, 72205, United States

Location

Teton Research, LLC

Little Rock, Arkansas, 72205, United States

Location

Med Center

Carmichael, California, 95608, United States

Location

College Hospital Costa Mesa

Costa Mesa, California, 92627, United States

Location

NeuroNetwork Trials

Costa Mesa, California, 92627, United States

Location

Med Investigations, Inc.

Fair Oaks, California, 95628, United States

Location

Sierra Clinical Research

Roseville, California, 95661, United States

Location

University of California Davis Health System

Sacramento, California, 95817, United States

Location

University of California Davis

Sacramento, California, 95817, United States

Location

Scripps Clinic-Clinical Research

San Diego, California, 92128, United States

Location

Plaza Medical Imaging

Santa Ana, California, 92704, United States

Location

Denver Internal Medicine Group

Denver, Colorado, 80209, United States

Location

Mountain View Clinical Research, Inc.

Denver, Colorado, 80209, United States

Location

New West Physicians Clinical Research

Golden, Colorado, 80401, United States

Location

Advanced Radiology Consultants

Fairfield, Connecticut, 06824, United States

Location

Advanced Radiology Consultants

Stamford, Connecticut, 06902, United States

Location

Stamford Therapeutics Consortium

Stamford, Connecticut, 06905, United States

Location

New England Research Associates, LLC

Trumbull, Connecticut, 06611, United States

Location

Southeastern Arthritis Center

Gainesville, Florida, 32607, United States

Location

Southeastern Imaging & Diagnostics

Gainesville, Florida, 32607, United States

Location

Southeastern Integrated Medical, PL, d/b/a Florida Medical Research Institute

Gainesville, Florida, 32607, United States

Location

Jacksonville Center for Clincal Research

Jacksonville, Florida, 32216, United States

Location

Memorial Hospital Jacksonville

Jacksonville, Florida, 32216, United States

Location

Gold Coast Research, LLC

Plantation, Florida, 33317, United States

Location

Marin E. Hale, M.D., P.A.

Plantation, Florida, 33317, United States

Location

Sabiha Khan, M.D.

Plantation, Florida, 33324, United States

Location

Kanner, Mendelson, Shteinman, LLC

West Palm Beach, Florida, 33407, United States

Location

Radiant Research

West Palm Beach, Florida, 33407, United States

Location

Rheumatology and Endocrinology Specialists of the Palm Beaches, P.A.

West Palm Beach, Florida, 33407, United States

Location

North Georgia Clinical Research

Marietta, Georgia, 30060, United States

Location

North Georgia Clinical Research

Woodstock, Georgia, 30189, United States

Location

East-West Medical Research Institute

Honolulu, Hawaii, 96814, United States

Location

Preventive Medicine

Chicago, Illinois, 60611, United States

Location

Rehabilitation Institue of Chicago

Chicago, Illinois, 60611, United States

Location

NorthShore University HealthSystem

Evanston, Illinois, 60201, United States

Location

NorthShore University HealthSystem

Glenview, Illinois, 60025, United States

Location

Clinical Investigation Specialists, Inc.

Gurnee, Illinois, 60031, United States

Location

Illinois Bone and Joint Institute, LLC

Morton Grove, Illinois, 60053, United States

Location

The Arthritis Center

Springfield, Illinois, 62704, United States

Location

NorthShore University HealthSystem

Vernon Hills, Illinois, 60061, United States

Location

Ronald Keith Stegemoller, American Health Network

Avon, Indiana, 46123, United States

Location

Floyd Memorial Hospital

New Albany, Indiana, 47150, United States

Location

Heartland Research Associates, LLC

Wichita, Kansas, 67205, United States

Location

Family Medicine East, Chartered/Radiology

Wichita, Kansas, 67207, United States

Location

Heartland Research Associates, LLC

Wichita, Kansas, 67207, United States

Location

Office of Manoj Kohli, M.D.

Lexington, Kentucky, 40517, United States

Location

L-MARC Research Center

Louisville, Kentucky, 40213, United States

Location

Commonwealth Biomedical Research, LLC

Madisonville, Kentucky, 42431, United States

Location

TFD Research, LLC

Shreveport, Louisiana, 71115, United States

Location

Rheumatology Associates

Portland, Maine, 04102, United States

Location

The Center for Rheumatology and Bone Research

Rockville, Maryland, 20850, United States

Location

The Center for Rheumatology and Bone Research

Wheaton, Maryland, 20902, United States

Location

Miray Medical Center

Brockton, Massachusetts, 02301, United States

Location

Phase III Clinical Research

Fall River, Massachusetts, 02720, United States

Location

Fall River Clinical Research

Fall River, Massachusetts, 02721, United States

Location

HCI Metromedic Walk-In

New Bedford, Massachusetts, 02740, United States

Location

MedVadis Research Corporation

Wellesley Hills, Massachusetts, 02481-2106, United States

Location

Fallon Clinic, Inc. (Drug Shipment)

Worcester, Massachusetts, 01605, United States

Location

Fallon Clinic, Inc.

Worcester, Massachusetts, 01605, United States

Location

Cadillac Clinical Research, LLC, located at Great Lakes Family Care

Cadillac, Michigan, 49601, United States

Location

Arthritis and Osteoporosis Treatment and Research Center

Flowood, Mississippi, 39232, United States

Location

Planters Clinic

Port Gibson, Mississippi, 39150, United States

Location

North Mississippi Medical Center, Inc.

Tupelo, Mississippi, 38801, United States

Location

Mercy Medical Group/Woodlake Research

Clarkson Valley, Missouri, 63011, United States

Location

Dynamic Clinical Research, Inc.

Kansas City, Missouri, 64114, United States

Location

Joan Prouty Moore, MD

Kansas City, Missouri, 64114, United States

Location

Orthopaedic and Occupational Medicine

Kansas City, Missouri, 64114, United States

Location

The Center for Pharmaceutical Research, P.C.

Kansas City, Missouri, 64114, United States

Location

Affiliated Clinical Research, Inc.

Las Vegas, Nevada, 89106, United States

Location

Office of Michael Mall, M.D.

Las Vegas, Nevada, 89109, United States

Location

Nevada Imaging Centers

Las Vegas, Nevada, 89117, United States

Location

Nevada Imaging Centers

Las Vegas, Nevada, 89118, United States

Location

Office of Danka Michaels, MD

Las Vegas, Nevada, 89128, United States

Location

Office of Stephen H. Miller, MD

Las Vegas, Nevada, 89144, United States

Location

Regional Clinical Research, Inc.

Endwell, New York, 13760, United States

Location

NYU Hospital for Joint Diseases

New York, New York, 10003, United States

Location

VirtualScopics, Inc.

Rochester, New York, 14625, United States

Location

Crouse Medical Practice, PLLC d/b/a Internist Associates of Central New York

Syracuse, New York, 13210, United States

Location

Kernodle Clinic Inc.

Burlington, North Carolina, 27215, United States

Location

Southeastern Radiology

Greensboro, North Carolina, 27407, United States

Location

PharmQuest

Greensboro, North Carolina, 27408, United States

Location

Research Institute of the Carolinas, PLLC

Mooresville, North Carolina, 28117, United States

Location

PMG Research of Salisbury

Salisbury, North Carolina, 28144, United States

Location

Piedmont Healthcare/Research

Statesville, North Carolina, 28625, United States

Location

Carolina Arthritis Associates, PA

Wilmington, North Carolina, 28401, United States

Location

PMG Research of Wilmington, LLC

Wilmington, North Carolina, 28401, United States

Location

Internal Medicine Associates

Fargo, North Dakota, 58103, United States

Location

Lillestol Research, LLC

Fargo, North Dakota, 58103, United States

Location

Advantage Diagnostics

Beachwood, Ohio, 44122, United States

Location

Rapid Medical Research, Inc.

Cleveland, Ohio, 44122, United States

Location

Columbus Clinical Research, Inc.

Columbus, Ohio, 43213, United States

Location

Optimed Research, LLC

Columbus, Ohio, 43235, United States

Location

Lake Health Lyndhurst Clinic

Lyndhurst, Ohio, 44124, United States

Location

East Penn Rheumatology Associates, PC

Bethlehem, Pennsylvania, 18015, United States

Location

Altoona Center for Clinical Research

Duncansville, Pennsylvania, 16635, United States

Location

BioImaging Technologies, Inc.

Newtown, Pennsylvania, 18940, United States

Location

Memorial Hospital of Rhode Island

Pawtucket, Rhode Island, 02860, United States

Location

Rheumatology Associates

Charleston, South Carolina, 29407, United States

Location

Radiant Research, Inc.

Greer, South Carolina, 29651, United States

Location

Parkway Medical Group

Fayetteville, Tennessee, 37334, United States

Location

Holston Medical Group

Kingsport, Tennessee, 37660, United States

Location

D. Matthew Sellers MD PC

Knoxville, Tennessee, 37920, United States

Location

Southwind Medical Specialists

Memphis, Tennessee, 38125, United States

Location

Baylor Research Institute

Dallas, Texas, 75231, United States

Location

Metroplex Clinical Research Center

Dallas, Texas, 75231, United States

Location

Radiant Research San Antonio Northeast

San Antonio, Texas, 78217, United States

Location

South Texas Radiology Imaging Center

San Antonio, Texas, 78217, United States

Location

Oakwell Clinical Research, LLC

San Antonio, Texas, 78218, United States

Location

Pivotal Research Centers

Midvale, Utah, 84047, United States

Location

National Clinical Research - Norfolk, Inc.

Norfolk, Virginia, 23502, United States

Location

National Clinical Research, Incorporated

Richmond, Virginia, 23294, United States

Location

Advanced Pain Management

Virginia Beach, Virginia, 23454, United States

Location

Tacoma Center for Arthritis Research, PS

Tacoma, Washington, 98405, United States

Location

Clinical Investigation Specialists, Inc.

Kenosha, Wisconsin, 53142, United States

Location

OMI - Organización Médica de Investigación

Buenos Aires, C1013AAR, Argentina

Location

Saint Dennis Medical Group S.A.

Buenos Aires, C1034ACO, Argentina

Location

Investigaciones Reumatológicas y Osteológicas S.R.L.

Buenos Aires, C1114AAH, Argentina

Location

Instituto Médico Especializado (IME)

Buenos Aires, C1405BCH, Argentina

Location

IMAI Research

Buenos Aires, C1425AWC, Argentina

Location

Menzies Research Institute

Hobart, Tasmania, 7000, Australia

Location

Cliniques Universitaires St Luc

Brussels, 1200, Belgium

Location

Universitair Ziekenhuis Gasthuisberg / Rheumatology

Leuven, 3000, Belgium

Location

Rheumatology Research Associates Ltd.

Edmonton, Alberta, T5M 0H4, Canada

Location

Nexus Clinic Research

St. John's, Newfoundland and Labrador, A1A 5E8, Canada

Location

The Arthritis Program Research Group Inc.

Newmarket, Ontario, L3Y 3R7, Canada

Location

Centre de Rhumatologie St-Louis

Sainte-Foy, Quebec, G1W 4R4, Canada

Location

Fakultni nemocnice u sv. Anny v Brne

Brno, 656 91, Czechia

Location

Revmacentrum MUDr. Mostera, s.r.o.

Brno-Židenice, 615 00, Czechia

Location

MEDIPONT Plus, s.r.o.

České Budějovice, 370 01, Czechia

Location

MEDIPONT, s.r.o.

České Budějovice, 370 01, Czechia

Location

ARTMEDI UPD s r.o.

Hostivice, 253 01, Czechia

Location

Nemocnice Na Frantisku s poliklinikou

Prague, 11000, Czechia

Location

Revmatologicky ustav

Prague, 128 50, Czechia

Location

Centrum pro zdravotnicke zabezpeceni sportovni reprezentace

Prague, 162 00, Czechia

Location

Ustredni vojenska nemocnice Praha

Prague, 162 00, Czechia

Location

MSI - Muskuloskeletalni institut

Prague, 169 00, Czechia

Location

DC Mediscan

Praha 11 - Chodov, 148 00, Czechia

Location

MediCentrum Praha, a.s.

Praha 11 - Chodov, 148 00, Czechia

Location

Nemocnice Atlas, a.s.

Zlín, 760 01, Czechia

Location

PV-Medical s.r.o.

Zlín, 760 01, Czechia

Location

Praxis fuer Orthopaedie, Chirotherapie und Akupunktur

Bad Hersfeld, 36251, Germany

Location

Praxis fuer Orthopaedie

Berlin, 12247, Germany

Location

Klinische Forschung Berlin-Buch

Berlin, 13125, Germany

Location

Praxis Dr. Thomas Jung

Deggingen, 73326, Germany

Location

Klinische Forschung Schwerin

Schwerin, 19055, Germany

Location

Orszagos Gerincgyogyaszati Kozpont

Budapest, 1126, Hungary

Location

Synexus Magyarorszag Kft.

Budapest, H-1036, Hungary

Location

Heves Megyei Onkormanyzat Markhot Ferenc Korhaz

Eger, 3300, Hungary

Location

Bekes Megyei Kepviselo-testulet Pandy Kalman Korhaz, Reumatologia

Gyula, 5700, Hungary

Location

Selye Janos Korhaz, Reumatologiai Szakrendelo

Komárom, 2900, Hungary

Location

MAV Korhaz es Rendelointezet

Szolnok, H-5000, Hungary

Location

Veszprem Megyei Onkormanyzat Csolnoky Ferenc Korhaz-Rendelointezet

Veszprém, H-8200, Hungary

Location

Azienda Sanitaria Genovese, Ospedale La Colletta, Dipartimento Apparato Locomotore

Arenzano, 16011, Italy

Location

Presidio Ospedaliero Augusto Murri, Reparto di Reumatologia

Jesi (Ancona), 60035, Italy

Location

Ospedale Luigi Sacco, Azienda Ospedaliera Polo Universitario Unita' Operativa di Reumatologia

Milan, 20157, Italy

Location

Clínica San Felipe

Lima, Lima Province, L-11, Peru

Location

Hospital Nacional "Edgardo Rebagliati Martins" - Essalud

Lima, Lima Province, L-11, Peru

Location

Instituto Peruano del Hueso y la Articulación SAC.

Lima, Lima Province, L-27, Peru

Location

Hospital Maria Auxiliadora

Lima, Lima Province, L-29, Peru

Location

Centro Medico Corpac

Lima, Lima Province, Lima-27, Peru

Location

Centro Empresarial - Altavista Polo 4

Santiago de Surco, Lima region, Lima 33, Peru

Location

Instituto de Ginecologia y Reproducción & Cirugia Minimamente Invasiva

Santiago de Surco, Lima region, Lima 33, Peru

Location

Hospital Nacional "Alberto Sabogal Sologuren" - Essalud

Callao, Provincia Constitucional del Callao, Callao-02, Peru

Location

NSZOZ "MEDICUS II" S.C. Irena Klimczak, Malgorzata Klimczak, Jerzy Klimczak

Cieszyn, 43-400, Poland

Location

"SYNEXUS SCM" Sp. z o.o.

Wroclaw, 50-088, Poland

Location

Katedra i Klinika Ortopedii i Traumatologii Narzadu Ruchu

Wroclaw, 50-556, Poland

Location

Russian State Medical University, Moscow Faculty, City Clinical Hospital #4

Moscow, 115093, Russia

Location

Institute of Rheumatology

Moscow, 115522, Russia

Location

City Alexandrovskaya Hospital

Saint Petersburg, 193312, Russia

Location

L.G. Sokolov Clinical Hospital #122 of Federal Medical-Biology Agency of Russia, Central Polyclinic

Saint Petersburg, 194291, Russia

Location

Research Institute of Traumatology and Orthopedy Named After R. R. Vredena

Saint Petersburg, 195427, Russia

Location

V. Interna klinika FN a LF UK

Bratislava, 826 06, Slovakia

Location

Ivan Ujvari

Bratislava, Slovakia

Location

Narodny ustav reumatickych chorob

Piešťany, 921 12, Slovakia

Location

Hospital Ntra. Sra. de La Esperanza

Santiago de Compostela, A Coruña, 15705, Spain

Location

Hospital General Universitario de Guadalajara

Guadalajara, Guadalajara, 19002, Spain

Location

Hospital Nuestra Señora de Valme

Seville, Sevilla, 41014, Spain

Location

Related Publications (1)

  • Hellio le Graverand MP, Clemmer RS, Redifer P, Brunell RM, Hayes CW, Brandt KD, Abramson SB, Manning PT, Miller CG, Vignon E. A 2-year randomised, double-blind, placebo-controlled, multicentre study of oral selective iNOS inhibitor, cindunistat (SD-6010), in patients with symptomatic osteoarthritis of the knee. Ann Rheum Dis. 2013 Feb;72(2):187-95. doi: 10.1136/annrheumdis-2012-202239. Epub 2012 Nov 10.

Related Links

MeSH Terms

Conditions

Osteoarthritis

Interventions

cindunistat

Condition Hierarchy (Ancestors)

ArthritisJoint DiseasesMusculoskeletal DiseasesRheumatic Diseases

Results Point of Contact

Title
Pfizer ClinicalTrials.gov Call Center
Organization
Pfizer, Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 29, 2007

First Posted

November 30, 2007

Study Start

November 1, 2007

Primary Completion

October 1, 2011

Study Completion

November 1, 2011

Last Updated

December 30, 2016

Results First Posted

December 30, 2016

Record last verified: 2016-11

Locations