NCT00528879

Brief Summary

The purpose of this clinical research study is to learn whether dapagliflozin can help reduce blood sugar levels in participants with Type 2 diabetes that is not well controlled on metformin alone. The safety of this treatment will also be studied.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
915

participants targeted

Target at P75+ for phase_3 type-2-diabetes

Timeline
Completed

Started Sep 2007

Typical duration for phase_3 type-2-diabetes

Geographic Reach
5 countries

75 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2007

Completed
10 days until next milestone

First Submitted

Initial submission to the registry

September 11, 2007

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 12, 2007

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 1, 2008

Completed
1.5 years until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2010

Completed
4 years until next milestone

Results Posted

Study results publicly available

May 2, 2014

Completed
Last Updated

October 20, 2015

Status Verified

September 1, 2015

Enrollment Period

1.2 years

First QC Date

September 11, 2007

Results QC Date

February 6, 2014

Last Update Submit

September 30, 2015

Conditions

Keywords

Diabetes Mellitus, Type 2Diabetes MellitusEndocrine System DiseasesGlucose Metabolism DisordersMetabolic DiseasesMetforminHypoglycemic AgentsPharmacologic ActionsPhysiological Effects of Drugs

Outcome Measures

Primary Outcomes (1)

  • Adjusted Mean Change From Baseline in Hemoglobin A1C (HbA1c) at Week 24 (Last Observation Carried Forward [LOCF])

    HbA1c was measured as percent of hemoglobin by a central laboratory. Data after rescue medication was excluded from this analysis. Baseline was defined as the last assessment prior to the start date and time of the first dose of the double-blind study medication. In cases where time of the first dose or time of the assessment was not available, baseline was defined as the last assessment on or prior to the date of the first dose of the double-blind study medication. HbA1c measurements were obtained during the qualification and lead-in periods and on Day 1 and Weeks 4, 8, 12, 16, 20, and 24 in the double-blind period.

    From Baseline to Week 24

Secondary Outcomes (8)

  • Adjusted Mean Change From Baseline in Fasting Plasma Glucose at Week 24 (Last Observation Carried Forward [LOCF])

    From Baseline to Week 24

  • Adjusted Mean Change From Baseline in Total Body Weight at Week 24 (Last Observation Carried Forward [LOCF])

    From Baseline to Week 24

  • Percentage of Participants Achieving a Therapeutic Glycemic Response (Hemoglobin A1c [HbA1C]) <7.0% at Week 24 (Last Observation Carried Forward [LOCF])

    From Baseline to Week 24

  • Adjusted Mean Change From Baseline in Hemoglobin A1c (HbA1c) in Participants With Baseline HbA1c ≥9.0% at Week 24 (Last Observation Carried Forward [LOCF])

    From Baseline to Week 24

  • Adjusted Mean Change From Baseline in Total Body Weight at Week 24 in Participants With Baseline Body Mass Index (BMI) ≥27 kg/m^2 (Last Observation Carried Forward [LOCF])

    From Baseline to Week 24

  • +3 more secondary outcomes

Other Outcomes (6)

  • Number of Participants With Adverse Events (AEs), Hypoglycemia Events, Related AEs, Death as Outcome, Serious AEs (SAEs), Related SAEs, SAEs Leading to Discontinuation, AEs Leading to Discontinuation, and Hypoglycemia Events Leading to Discontinuation

    From Baseline to end of Long-term Period (Week 102)

  • Number of Participants With Laboratory Test Results Meeting the Criteria for Laboratory Abnormality

    Day 1 to Week 102

  • Number of Participants With Changes in Baseline in Electrocardiogram Findings at Week 102 (Last Observation Carried Forward [LOCF])

    Baseline to Week 102

  • +3 more other outcomes

Study Arms (4)

Placebo + Metformin

PLACEBO COMPARATOR

Participants received dapagliflozin-matching placebo once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Drug: PlaceboDrug: Metformin

Dapagliflozin, 2.5 mg + Metformin

EXPERIMENTAL

Participants received dapagliflozin, 2.5 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Drug: DapagliflozinDrug: Metformin

Dapagliflozin, 5 mg + Metformin

EXPERIMENTAL

Participants received dapagliflozin, 5 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Drug: DapagliflozinDrug: Metformin

Dapagliflozin, 10 mg + Metformin

EXPERIMENTAL

Participants received dapagliflozin, 10 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Drug: DapagliflozinDrug: PlaceboDrug: Metformin

Interventions

Tablets administered orally as a 2.5-, 5-, or 10-mg dose once daily for up to 102 weeks

Also known as: BMS-512148
Dapagliflozin, 10 mg + MetforminDapagliflozin, 2.5 mg + MetforminDapagliflozin, 5 mg + Metformin

Dapagliflozin-matching placebo administered as tablets orally once daily for up to 102 weeks

Dapagliflozin, 10 mg + MetforminPlacebo + Metformin

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Dapagliflozin, 10 mg + MetforminDapagliflozin, 2.5 mg + MetforminDapagliflozin, 5 mg + MetforminPlacebo + Metformin

Eligibility Criteria

Age18 Years - 77 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Males and females, 18 to 77 years old, with type 2 diabetes and inadequate glycemic control
  • Participants who have been receiving metformin at a total daily dose ≥1500 mg per day for at least 8 weeks
  • C-peptide ≥1.0 ng/mL
  • Body mass index ≤45.0 kg/m\^2
  • Serum creatinine level \<1.50 mg/dL for men or \<1.40 mg/dL for women.

You may not qualify if:

  • Aspartate aminotransferase and/or alanine aminotransferase level \>3.0 times the upper limit of normal
  • Serum total bilirubin level \>2 mg/dL
  • Creatinine kinase level \>3 times upper limit of normal
  • Symptoms of severely uncontrolled diabetes
  • Serum creatinine level ≥1.50 mg/dL for men or ≥1.40 mg/dL for women
  • Currently unstable or serious cardiovascular, renal, hepatic, hematologic, oncologic, endocrine, psychiatric, or rheumatic diseases

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (75)

Clinical Research Advantage / Desert Clinical Res, Llc

Tempe, Arizona, 85282, United States

Location

Medical Group Of Encino

Encino, California, 91436, United States

Location

Valley Research

Fresno, California, 93720, United States

Location

Randall Shue, D.O.

Los Angeles, California, 90023, United States

Location

Diabetes Medical Center Of California

Northridge, California, 91325, United States

Location

Ritchken & First M.D.'S

San Diego, California, 92117, United States

Location

Encompass Clinical Research

Spring Valley, California, 91978, United States

Location

Raikhel, Marina

Torrance, California, 90505, United States

Location

Express Care Clinical Res

Colorado Springs, Colorado, 80909, United States

Location

Denver Internal Medicine

Denver, Colorado, 80209, United States

Location

New West Physicians

Golden, Colorado, 80401, United States

Location

Central Florida Clinical Trials, Inc.

Altamonte Springs, Florida, 32701, United States

Location

Family Care Associates Of Nw Florida

Chipley, Florida, 32428, United States

Location

Health Partners Research Foundation

Minneapolis, Minnesota, 56440, United States

Location

Woodlake Research

Chesterfield, Missouri, 63017, United States

Location

Nevada Alliance Against Diabetes

Las Vegas, Nevada, 89101, United States

Location

Diabetes & Endocrinology Consultants, Pc

Morehead City, North Carolina, 28557, United States

Location

Newark Physician Associates

Newark, Ohio, 43055, United States

Location

Integris Family Care S. Penn

Oklahoma City, Oklahoma, 73159, United States

Location

Cumberland Valley Endocrinology Center, Llc

Carlisle, Pennsylvania, 17013, United States

Location

Banksville Medical Pc

Pittsburgh, Pennsylvania, 15216, United States

Location

Palmetto Clinical Research

Summerville, South Carolina, 29485, United States

Location

Southeastern Research Assoc

Taylors, South Carolina, 29687, United States

Location

Texas Center For Drug Development, P.A.

Houston, Texas, 77081, United States

Location

Diabetes & Glandular Disease Research Associates, Inc.

San Antonio, Texas, 78229, United States

Location

S.A.M. Clinical Research Center

San Antonio, Texas, 78229, United States

Location

Optimum Clinical Research

Salt Lake City, Utah, 84102, United States

Location

Office Of Dr. Gray

Spokane, Washington, 99216, United States

Location

Local Institution

Buenos Aires, Buenos Aires, 1431, Argentina

Location

Local Institution

Capital Federal, Buenos Aires, 1034, Argentina

Location

Local Institution

Capital Federal, Buenos Aires, 1429, Argentina

Location

Local Institution

Capital Federal, Buenos Aires, C1056ABJ, Argentina

Location

Local Institution

Capital Federal, Buenos Aires, C1425AGC, Argentina

Location

Local Institution

Ciudad Auton., Buenos Aires, C1505CWB, Argentina

Location

Local Institution

Ciudad Auton, Buenos Aires, C1408INH, Argentina

Location

Local Institution

Mar del Plata, Buenos Aires, 7600, Argentina

Location

Local Institution

Zárate, Buenos Aires, 2800, Argentina

Location

Local Institution

Córdoba, Córdoba Province, 5000, Argentina

Location

Local Institution

Villa Carlos Paz, Córdoba Province, 5152, Argentina

Location

Local Institution

Fortaleza, Ceará, 60021, Brazil

Location

Local Institution

Itajubá, Minas Gerais, 37502, Brazil

Location

Local Institution

Belém, Pará, 66073, Brazil

Location

Local Institution

Rio de Janeiro, Rio de Janeiro, 20211, Brazil

Location

Local Institution

Caxias do Sul, Rio Grande do Sul, 95070, Brazil

Location

Local Institution

Porto Alegre, Rio Grande do Sul, 90020090, Brazil

Location

Local Institution

Porto Alegre, Rio Grande do Sul, 90035, Brazil

Location

Local Institution

Marília, São Paulo, 17519, Brazil

Location

Local Institution

Calgary, Alberta, T2R 0X7, Canada

Location

Local Institution

Kelowna, British Columbia, V1Y 2H4, Canada

Location

Local Institution

Winnipeg, Manitoba, R3E 3P4, Canada

Location

Local Institution

Bathurst, New Brunswick, E2A 4X7, Canada

Location

Local Institution

Mount Pearl, Newfoundland and Labrador, A1N 1W7, Canada

Location

Local Institution

St. John's, Newfoundland and Labrador, A1E 2E2, Canada

Location

Local Institution

Sarnia, Ontario, N7T 4X3, Canada

Location

Local Institution

Thornhill, Ontario, L4J 8L7, Canada

Location

Local Institution

Toronto, Ontario, M4R 2G4, Canada

Location

Local Institution

Toronto, Ontario, M9W 4L6, Canada

Location

Local Institution

Charlottetown, Prince Edward Island, C1A 5Y9, Canada

Location

Local Institution

Drummondville, Quebec, J2B 7T1, Canada

Location

Local Institution

Granby, Quebec, J2G 8Z9, Canada

Location

Local Institution

L'Ancienne-Lorette, Quebec, G2E 2X1, Canada

Location

Local Institution

Mirabel, Quebec, J7J 2K8, Canada

Location

Local Institution

Saint-Léonard, Quebec, H1S 3A9, Canada

Location

Local Institution

Saskatoon, Saskatchewan, S7K 3H3, Canada

Location

Local Institution

Saskatoon, Saskatchewan, S7K 7H9, Canada

Location

Local Institution

Durango, Durango, 64710, Mexico

Location

Local Institution

Guadalajara, Jalisco, 44650, Mexico

Location

Local Institution

Guadalajara, Jalisco, 44670, Mexico

Location

Local Institution

Df, Mexico City, 11800, Mexico

Location

Local Institution

Guadalajara, Mexico City, 44670, Mexico

Location

Local Institution

Zapopan, Mexico City, 45150, Mexico

Location

Local Institution

Monterrey, Nuevo León, 64460, Mexico

Location

Local Institution

Monterrey, Nuevo León, 64710, Mexico

Location

Local Institution

Monterrrey, Nuevo León, 64700, Mexico

Location

Local Institution

Tampico, Tamaulipas, 89109, Mexico

Location

Related Publications (7)

  • Natale P, Tunnicliffe DJ, Toyama T, Palmer SC, Saglimbene VM, Ruospo M, Gargano L, Stallone G, Gesualdo L, Strippoli GF. Sodium-glucose co-transporter protein 2 (SGLT2) inhibitors for people with chronic kidney disease and diabetes. Cochrane Database Syst Rev. 2024 May 21;5(5):CD015588. doi: 10.1002/14651858.CD015588.pub2.

  • Shah M, Stolbov L, Yakovleva T, Tang W, Sokolov V, Penland RC, Boulton D, Parkinson J. A model-based approach to investigating the relationship between glucose-insulin dynamics and dapagliflozin treatment effect in patients with type 2 diabetes. Diabetes Obes Metab. 2021 Apr;23(4):991-1000. doi: 10.1111/dom.14305. Epub 2021 Jan 25.

  • Bailey CJ, Del Prato S, Wei C, Reyner D, Saraiva G. Durability of glycaemic control with dapagliflozin, an SGLT2 inhibitor, compared with saxagliptin, a DPP4 inhibitor, in patients with inadequately controlled type 2 diabetes. Diabetes Obes Metab. 2019 Nov;21(11):2564-2569. doi: 10.1111/dom.13841. Epub 2019 Aug 26.

  • Mellander A, Billger M, Johnsson E, Traff AK, Yoshida S, Johnsson K. Hypersensitivity Events, Including Potentially Hypersensitivity-Related Skin Events, with Dapagliflozin in Patients with Type 2 Diabetes Mellitus: A Pooled Analysis. Clin Drug Investig. 2016 Nov;36(11):925-933. doi: 10.1007/s40261-016-0438-3.

  • Kohan DE, Fioretto P, Johnsson K, Parikh S, Ptaszynska A, Ying L. The effect of dapagliflozin on renal function in patients with type 2 diabetes. J Nephrol. 2016 Jun;29(3):391-400. doi: 10.1007/s40620-016-0261-1. Epub 2016 Feb 19.

  • Bailey CJ, Gross JL, Hennicken D, Iqbal N, Mansfield TA, List JF. Dapagliflozin add-on to metformin in type 2 diabetes inadequately controlled with metformin: a randomized, double-blind, placebo-controlled 102-week trial. BMC Med. 2013 Feb 20;11:43. doi: 10.1186/1741-7015-11-43.

  • Bailey CJ, Gross JL, Pieters A, Bastien A, List JF. Effect of dapagliflozin in patients with type 2 diabetes who have inadequate glycaemic control with metformin: a randomised, double-blind, placebo-controlled trial. Lancet. 2010 Jun 26;375(9733):2223-33. doi: 10.1016/S0140-6736(10)60407-2.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Diabetes MellitusEndocrine System DiseasesGlucose Metabolism DisordersMetabolic Diseases

Interventions

dapagliflozinMetformin

Condition Hierarchy (Ancestors)

Nutritional and Metabolic Diseases

Intervention Hierarchy (Ancestors)

BiguanidesGuanidinesAmidinesOrganic Chemicals

Results Point of Contact

Title
Bristol-Myers Squibb Study Director
Organization
Bristol-Myers Squibb

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

September 11, 2007

First Posted

September 12, 2007

Study Start

September 1, 2007

Primary Completion

November 1, 2008

Study Completion

May 1, 2010

Last Updated

October 20, 2015

Results First Posted

May 2, 2014

Record last verified: 2015-09

Locations