NCT00516672

Brief Summary

This is a two part phase I study in Japanese patients that will determine the safety, tolerability and pharmacokinetics of pazopanib monotherapy and of pazopanib in combination with lapatinib.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
30

participants targeted

Target at P25-P50 for phase_1

Timeline
Completed

Started Sep 2007

Longer than P75 for phase_1

Geographic Reach
1 country

2 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

August 13, 2007

Completed
2 days until next milestone

First Posted

Study publicly available on registry

August 15, 2007

Completed
26 days until next milestone

Study Start

First participant enrolled

September 10, 2007

Completed
3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 30, 2010

Completed
5.1 years until next milestone

Study Completion

Last participant's last visit for all outcomes

October 14, 2015

Completed
Last Updated

November 13, 2017

Status Verified

November 1, 2017

Enrollment Period

3 years

First QC Date

August 13, 2007

Last Update Submit

November 8, 2017

Conditions

Keywords

lapatinib,cancerpharmacokinetics,safety,pazopanib,Japanese patients,

Outcome Measures

Primary Outcomes (1)

  • Safety and tolerability

    The safety and tolerability endpoints will consist of the evaluation of adverse events (AEs), and changes in vital signs and laboratory values.

    before and after taking the study medications

Secondary Outcomes (2)

  • Pharmacokinetics

    over a 24 hour period

  • Tumor response

    9 weeks

Study Arms (1)

Arm 1

EXPERIMENTAL

Pazopanib monotherapy or in combination with lapatinib

Drug: pazopanibDrug: Lapatinib

Interventions

Pazopanib oral tablet

Arm 1

Lapatinib oral tablet

Arm 1

Eligibility Criteria

Age20 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Signed informed consent.
  • Histologically or cytologically confirmed diagnosis of advanced solid tumor.
  • Women and men with potential to have children must be willing to practice acceptable methods of birth control during the study.
  • ECOG performance status of 0 or 1.
  • Adequate bone marrow reserve and hepato-renal function.
  • Able to swallow and retain oral medication.
  • For combo part, left ventricular ejection fraction within normal range or above 50%.

You may not qualify if:

  • Prior treatment with pazopanib, and with lapatinib for combo part.
  • Clinically significant gastrointestinal abnormalities.
  • Sevier diseases or conditions other than cancer.
  • Poorly controlled hypertension.
  • Use of warfarin for therapeutic anticoagulation.
  • Use of other anti-angiogenesis agents, and other ErbB inhibitors for combo part.
  • Unresolved and/or unstable toxicities
  • Pregnant or lactating females

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (2)

GSK Investigational Site

Aichi, 466-8560, Japan

Location

GSK Investigational Site

Saitama, 350-1298, Japan

Location

Related Publications (1)

  • Inada-Inoue M, Ando Y, Kawada K, Mitsuma A, Sawaki M, Yokoyama T, Sunakawa Y, Ishida H, Araki K, Yamashita K, Mizuno K, Nagashima F, Takekura A, Nagamatsu K, Sasaki Y. Phase 1 study of pazopanib alone or combined with lapatinib in Japanese patients with solid tumors. Cancer Chemother Pharmacol. 2014 Apr;73(4):673-83. doi: 10.1007/s00280-014-2374-3. Epub 2014 Jan 24.

Related Links

MeSH Terms

Conditions

Carcinoma, Renal CellNeoplasms

Interventions

pazopanibLapatinib

Condition Hierarchy (Ancestors)

AdenocarcinomaCarcinomaNeoplasms, Glandular and EpithelialNeoplasms by Histologic TypeKidney NeoplasmsUrologic NeoplasmsUrogenital NeoplasmsNeoplasms by SiteFemale Urogenital DiseasesFemale Urogenital Diseases and Pregnancy ComplicationsUrogenital DiseasesKidney DiseasesUrologic DiseasesMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

QuinazolinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingHeterocyclic Compounds

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 13, 2007

First Posted

August 15, 2007

Study Start

September 10, 2007

Primary Completion

August 30, 2010

Study Completion

October 14, 2015

Last Updated

November 13, 2017

Record last verified: 2017-11

Locations