NCT00477581

Brief Summary

This purpose of this study is to compare the effect of exenatide to that of sitagliptin on 2-hour postprandial glucose in subjects with type 2 diabetes mellitus.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
102

participants targeted

Target at P50-P75 for phase_4 type-2-diabetes-mellitus

Timeline
Completed

Started May 2007

Shorter than P25 for phase_4 type-2-diabetes-mellitus

Geographic Reach
1 country

19 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

May 1, 2007

Completed
20 days until next milestone

First Submitted

Initial submission to the registry

May 21, 2007

Completed
2 days until next milestone

First Posted

Study publicly available on registry

May 23, 2007

Completed
3 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

September 1, 2007

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

September 1, 2007

Completed
Last Updated

August 26, 2015

Status Verified

August 1, 2015

Enrollment Period

4 months

First QC Date

May 21, 2007

Last Update Submit

August 25, 2015

Conditions

Keywords

diabetesexenatidesitagliptinAmylinLilly

Outcome Measures

Primary Outcomes (1)

  • Effect of Exenatide on postprandial glucose

    To compare the effect of exenatide to that of sitagliptin on 2-hour postprandial glucose in subjects with type 2 diabetes mellitus

    28 days

Secondary Outcomes (1)

  • Assessment of effect of exenatide to the effect of sitagliptin the acetaminophen absorption test, and 6-point self-monitored blood glucose (SMBG) profiles

    28 days

Study Arms (2)

Sequence A

EXPERIMENTAL
Drug: exenatideDrug: sitagliptin

Sequence B

EXPERIMENTAL
Drug: exenatideDrug: sitagliptin

Interventions

subcutaneous injection (5mcg or 10mcg), twice a day

Also known as: Byetta
Sequence ASequence B

oral administration (100mg), once a day in the morning

Also known as: Januvia
Sequence ASequence B

Eligibility Criteria

Age18 Years - 70 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Treatment with metformin for at least 2 months
  • Has HbA1c 7.0% to 11.0%, inclusive, at screening
  • Body mass index (BMI)25 kg/m\^2 to 45 kg/m\^2, inclusive
  • List of medications that are not allowed or the patient has been on stable treatment for at least 2 months:
  • Hormone replacement therapy (female subjects)
  • Oral contraceptives (female subjects)
  • Antihypertensive agents
  • Lipid-lowering agents
  • Thyroid replacement therapy

You may not qualify if:

  • Has been treated with exenatide (BYETTA®) or any DPP-4 inhibitor prior to screening
  • Received any study medication or participated in any type of clinical trial within 30 days prior to screening
  • Has donated blood within 60 days of screening visit or is planning to donate blood during the study
  • Treated with any of the following medications:
  • Sulfonylurea or Thiazolidinedione within 3 months of screening;
  • Alpha-glucosidase inhibitor, meglitinide, nateglinide, or pramlintide (SYMLIN®)within 30 days of screening;
  • Insulin within 2 weeks prior to screening or insulin for longer than 1 week within 6 months of screening;
  • Drugs that directly affect gastrointestinal motility, including but not limited to, anticholinergics, macrolide antibiotics, dopamine antagonists, opioids, and Reglan®(metoclopramide);
  • Systemic corticosteroids by oral, intravenous, or intramuscular route; or potent, inhaled, or intrapulmonary (including ADVAIR®) steroids known to have a high rate of systemic absorption;

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (19)

Research Site

Los Angeles, California, United States

Location

Research Site

Spring Valley, California, United States

Location

Research Site

Miami, Florida, United States

Location

Research Site

Pembroke Pines, Florida, United States

Location

Research Site

Chicago, Illinois, United States

Location

Research Site

Indianapolis, Indiana, 46260, United States

Location

Research Site

Indianapolis, Indiana, United States

Location

Research Site

Detroit, Michigan, United States

Location

Research Site

Butte, Montana, United States

Location

Research Site

Winston-Salem, North Carolina, United States

Location

Research Site

Cincinnati, Ohio, United States

Location

Research Site

Marion, Ohio, United States

Location

Research Site

Eugene, Oregon, United States

Location

Research Site

Portland, Oregon, United States

Location

Research Site

Charleston, South Carolina, United States

Location

Research Site

Greer, South Carolina, United States

Location

Research Site

Austin, Texas, United States

Location

Research Site

Corpus Christi, Texas, United States

Location

Research Site

San Antonio, Texas, United States

Location

Related Publications (1)

  • DeFronzo RA, Okerson T, Viswanathan P, Guan X, Holcombe JH, MacConell L. Effects of exenatide versus sitagliptin on postprandial glucose, insulin and glucagon secretion, gastric emptying, and caloric intake: a randomized, cross-over study. Curr Med Res Opin. 2008 Oct;24(10):2943-52. doi: 10.1185/03007990802418851. Epub 2008 Sep 10.

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Diabetes Mellitus

Interventions

ExenatideSitagliptin Phosphate

Condition Hierarchy (Ancestors)

Glucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Intervention Hierarchy (Ancestors)

PeptidesAmino Acids, Peptides, and ProteinsVenomsComplex MixturesToxins, BiologicalBiological FactorsTriazolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPyrazines

Study Officials

  • Lisa Porter, MD

    Amylin Pharmaceuticals, LLC.

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 4
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 21, 2007

First Posted

May 23, 2007

Study Start

May 1, 2007

Primary Completion

September 1, 2007

Study Completion

September 1, 2007

Last Updated

August 26, 2015

Record last verified: 2015-08

Locations