NCT00143611

Brief Summary

The purpose of this study is to determine the optimal dose of Resatorvid for reducing 28-day all-cause mortality in subjects with severe sepsis.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
277

participants targeted

Target at P50-P75 for phase_3 sepsis

Timeline
Completed

Started Sep 2005

Shorter than P25 for phase_3 sepsis

Geographic Reach
16 countries

142 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

August 31, 2005

Completed
1 day until next milestone

Study Start

First participant enrolled

September 1, 2005

Completed
1 day until next milestone

First Posted

Study publicly available on registry

September 2, 2005

Completed
1.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2007

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

February 1, 2007

Completed
Last Updated

February 2, 2012

Status Verified

January 1, 2012

Enrollment Period

1.4 years

First QC Date

August 31, 2005

Last Update Submit

January 31, 2012

Conditions

Keywords

Shock, SepticSepsis SyndromeRespiratory InsufficiencySIRS (Systemic Inflammatory Response Syndrome)Respiratory FailureDrug Therapy

Outcome Measures

Primary Outcomes (1)

  • 28-day All-cause Mortality.

    Day 28

Secondary Outcomes (6)

  • Change from Baseline in Organ Failure Assessment

    Day 28

  • Mean Systemic Inflammatory Response

    Day 28

  • Mean Vasopressor-free days

    Day 28

  • Mean Ventilator-free days

    Day 28

  • Mean Intensive Care Unit free days

    Day 28

  • +1 more secondary outcomes

Study Arms (3)

Resatorvid 1.2 mg/kg/day

EXPERIMENTAL
Drug: Resatorvid

Resatorvid 2.4 mg/kg/day

EXPERIMENTAL
Drug: Resatorvid

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

Resatorvid 1.2 mg/kg, injection, subcutaneously for thirty minutes; then resatorvid 0.05 mg/kg/h (1.2 mg/kg/day), injection, subcutaneously over 96 hours.

Also known as: TAK-242
Resatorvid 1.2 mg/kg/day

Resatorvid placebo-matching injection, subcutaneously for thirty minutes; then resatorvid placebo-matching injection, subcutaneously over 96 hours.

Placebo

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has clinical evidence of infection defined as the presence of a known or probable source of infection requiring the initiation of parenteral antimicrobial therapy.
  • Must meet at least 3 of the following 4 criteria for SIRS:
  • A core temperature greater than 38°C or less than 36°C.
  • A heart rate greater than 90 beats per minute.
  • A respiratory rate greater than 20 breaths/min or partial pressure of carbon dioxide in arterial blood less than 32 mm Hg or mechanical ventilation for an acute process.
  • A total white blood cell absolute count greater than 12,000 cells/mm3 or less than 4,000 cells/mm3, or a white blood cell differential count that showed greater than 10% immature (band) forms.
  • Must have sepsis with shock and/or respiratory failure.

You may not qualify if:

  • If female, the subject is pregnant, nursing and the milk is intended to be ingested by the infant, or the participant plans to become pregnant, or nurse and the milk is intended to be ingested by the infant.
  • Is receiving immunosuppressive therapy such as cyclosporine, azathioprine, or cancer-related chemotherapy.
  • Has a granulocyte count of less than 1000/mm3 except if the decreased count was believed to be due to sepsis.
  • Has documented or suspected acute myocardial infarction within the last 6 weeks prior to Pretreatment Period.
  • Has a documented history of moderate to severe chronic heart failure as defined by New York Heart Association Functional Classification III or IV.
  • Is known to be positive for human immunodeficiency virus with known CD4 count less than or equal to 50/mm3 or had known end-stage processes.
  • Has a known history of glucose-6-phosphate dehydrogenase deficiency.
  • Has a methemoglobin level greater than 5% at Pretreatment Period or had a known history of methemoglobinemia.
  • Is moribund and death was considered imminent.
  • Is classified as "Do Not Resuscitate", or "Do Not Treat", or the participant's family has not committed to aggressive management of the participant's condition.
  • Is not expected to survive for 28 days and was not likely be given life support due to a pre-existing, uncorrectable medical condition.
  • Has a known esophageal varices, chronic jaundice, cirrhosis, or chronic ascites.
  • Is in a chronic vegetative state or has a similar long-term neurological condition.
  • Has known portal hypertension or Child-Pugh hepatic impairment class C.
  • Has acute third degree burns involving more than 30% of body surface within 120 hours prior to Pretreatment Period.
  • +3 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (144)

Unknown Facility

Birmingham, Alabama, United States

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Mobile, Alabama, United States

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Phoenix, Arizona, United States

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Scottsdale, Arizona, United States

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Escondido, California, United States

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Los Angeles, California, United States

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Orange, California, United States

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Poway, California, United States

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San Diego, California, United States

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Colorado Springs, Colorado, United States

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New Haven, Connecticut, United States

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Newark, Delaware, United States

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Atlantis, Florida, United States

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Bay Pines, Florida, United States

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Jacksonville, Florida, United States

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Miami, Florida, United States

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Orlando, Florida, United States

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Sarasota, Florida, United States

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Atlanta, Georgia, United States

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Augusta, Georgia, United States

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Chicago, Illinois, United States

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Peoria, Illinois, United States

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Indianapolis, Indiana, United States

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Des Moines, Iowa, United States

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Louisville, Kentucky, United States

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Shreveport, Louisiana, United States

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Portland, Maine, United States

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Baltimore, Maryland, United States

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Springfield, Massachusetts, United States

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Kalamazoo, Michigan, United States

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Kansas City, Missouri, United States

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St Louis, Missouri, United States

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Butte, Montana, United States

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Englewood, New Jersey, United States

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Buffalo, New York, United States

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New York, New York, United States

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Rochester, New York, United States

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Greensboro, North Carolina, United States

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Winston-Salem, North Carolina, United States

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Akron, Ohio, United States

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Columbus, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Greenville, South Carolina, United States

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Nashville, Tennessee, United States

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Fort Worth, Texas, United States

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Galveston, Texas, United States

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Houston, Texas, United States

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Lubbock, Texas, United States

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Bellevue, Washington, United States

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Adelaide, Australia

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Fremantle, Australia

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Heidelberg, Australia

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Linz, Austria

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Vienna, Austria

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Aalst, Belgium

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Antwerp, Belgium

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Brussels, Belgium

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Genk, Belgium

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Ghent, Belgium

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Liège, Belgium

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Ottignies, Belgium

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Yvoir, Belgium

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Calgary, Alberta, Canada

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Vancouver, British Columbia, Canada

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Victoria, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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Halifax, Nova Scotia, Canada

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London, Ontario, Canada

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Brno, Czechia

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Havlíčkův Brod, Czechia

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Hradec Králové, Czechia

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Opava, Czechia

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Pilsen, Czechia

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Prague, Czechia

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Helsinki, Finland

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Joensuu, Finland

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Kokkola, Finland

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Kuopio, Finland

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Lappeenranta, Finland

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Oulu, Finland

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Seinäjoki, Finland

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Tampere, Finland

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Turku, Finland

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Berlin, Germany

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Dresden, Germany

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Erfurt, Germany

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Jena, Germany

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Krefeld, Germany

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Ludwigshafen, Germany

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Mannheim, Germany

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München, Germany

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Wuppertal, Germany

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Afula, Israel

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Ashkelon, Israel

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Haifa, Israel

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Holon, Israel

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Jerusalem, Israel

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Kfar Saba, Israel

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Petah Tikva, Israel

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Ẕerifin, Israel

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Lecco, Italy

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Monza, Italy

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Pavia, Italy

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Chiba, Japan

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Fukuoka, Japan

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Hiroshima, Japan

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Hokkaido, Japan

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Kumamoto, Japan

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Kyoto, Japan

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Numakunai, Japan

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Osaka, Japan

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Shizuoka, Japan

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Tokyo, Japan

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Yamaguchi, Japan

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's-Hertogenbosch, Netherlands

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Apeldoorn, Netherlands

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Groningen, Netherlands

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Leeuwarden, Netherlands

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Nijmegen, Netherlands

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Rotterdam, Netherlands

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Tilburg, Netherlands

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Auckland, New Zealand

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Christchurch, New Zealand

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Hastings, New Zealand

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Tauranga, New Zealand

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San Juan, Puerto Rico

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Barcelona, Spain

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Getafe, Spain

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Madrid, Spain

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Valladolid, Spain

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Vitoria-Gasteiz, Spain

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Gävle, Sweden

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Gothenburg, Sweden

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Karlstad, Sweden

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Kristianstad, Sweden

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Linköping, Sweden

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Lund, Sweden

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Stockholm, Sweden

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Uppsala, Sweden

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Brighton, United Kingdom

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Glasgow, United Kingdom

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Leeds, United Kingdom

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Livingston, United Kingdom

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London, United Kingdom

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Related Publications (1)

  • Rice TW, Wheeler AP, Bernard GR, Vincent JL, Angus DC, Aikawa N, Demeyer I, Sainati S, Amlot N, Cao C, Ii M, Matsuda H, Mouri K, Cohen J. A randomized, double-blind, placebo-controlled trial of TAK-242 for the treatment of severe sepsis. Crit Care Med. 2010 Aug;38(8):1685-94. doi: 10.1097/CCM.0b013e3181e7c5c9.

MeSH Terms

Conditions

SepsisShock, SepticSystemic Inflammatory Response SyndromeRespiratory Insufficiency

Interventions

ethyl 6-(N-(2-chloro-4-fluorophenyl)sulfamoyl)cyclohex-1-ene-1-carboxylate

Condition Hierarchy (Ancestors)

InfectionsInflammationPathologic ProcessesPathological Conditions, Signs and SymptomsShockRespiration DisordersRespiratory Tract Diseases

Study Officials

  • VP Clinical Science

    Takeda

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

August 31, 2005

First Posted

September 2, 2005

Study Start

September 1, 2005

Primary Completion

February 1, 2007

Study Completion

February 1, 2007

Last Updated

February 2, 2012

Record last verified: 2012-01

Locations