NCT07669584

Brief Summary

The test medication Gel PKB171 is a vaginal gel that has not yet been licensed by the regulatory authorities. However, the active substance pentoxifylline has been available as tablets for decades and is used to increase peripheral blood flow in patients with circulation problems. Additionally, pentoxifylline is used to treat sperm samples in artificial insemination and test tube fertilisation to increase the mobility of sperm. A phase I clinical trial, 30 women were treated with Gel PKB171 for up to three times. Gel PKB171 was generally well tolerated and the most common side effects were local reactions like vaginal discharge and itching. A phase II clinical trial, investigate the efficacy and safety of two concentrations of PKB171 versus placebo in couples with asthenozoospermia who wish to conceive. A total of 72 couples were planned to be included in the study. Finally, 28 couples were enrolled, and 11 couples were randomised. Within this trial, two concentrations of pentoxifylline gel were compared (5 mL of gel PKB171 containing 150 mg (3%) of pentoxifiylline, and 5 mL of gel PKB171 containing and 200 mg (4%) of pentoxifylline. Both doses were tolerated well and revealed no safety concerns as assessed by AEs, local Gel PKB171 tolerability, laboratory parameters, vital signs, gynaecologic and physical examination, or transvaginal ultrasound findings. This study was prematurely discontinued due to low numbers of eligible subjects and high recruitment failure rates, despite several protocol amendments. PKB171 gel was well tolerated and revealed no safety concerns as assessed by AEDTs, local IMP tolerability, analytical parameters, vital signs, physical and gynecological examination, or transvaginal ultrasound findings. The aim of this clinical trial is to assess the safety and efficacy of the gel PKB171 compared to a placebo gel in couples with mild male factor infertility, unable to conceive in the last 6 and 24 months. Additionally, the safety and local tolerability of Gel PKB171 will be further investigated.

Trial Health

77
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
732

participants targeted

Target at P75+ for phase_2

Timeline
15mo left

Started Oct 2025

Geographic Reach
1 country

12 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress38%
Oct 2025Oct 2027

Study Start

First participant enrolled

October 28, 2025

Completed
4 months until next milestone

First Submitted

Initial submission to the registry

February 25, 2026

Completed
4 months until next milestone

First Posted

Study publicly available on registry

June 25, 2026

Completed
1.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 28, 2027

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

October 28, 2027

Last Updated

June 25, 2026

Status Verified

June 1, 2026

Enrollment Period

2 years

First QC Date

February 25, 2026

Last Update Submit

June 22, 2026

Conditions

Keywords

asthenozoospermiapentoxifylinemale infertility

Outcome Measures

Primary Outcomes (1)

  • To assess the efficacy up to three treaament cycles with Gel PKB171 compared with placebo in couples with mild male factor fertility

    Heartbeat by the 6th-8th weeks of gestation by ecography

    6-8 weeks

Secondary Outcomes (6)

  • To assess the efficacy of PKB171 gel compared to placebo on biochemical pregnancy rate

    6-8 months

  • To assess the efficacy of PKB171 gel compared to placebo on ongoing pregnancy rate

    12 months

  • To assess the efficacy of PKB171 gel compared to placebo on live birth rate.

    9 months

  • To assess the pregnancy loss rate after PKB171 gel treatment compared to placebo on-viable intrauterine pregnancy up to 20 weeks

    9 months

  • To compare the obstetrics characteristics of pregnancies achieved after PKB171 gel compared to placebo,

    10 months

  • +1 more secondary outcomes

Study Arms (2)

Gel PKB171 200 mg (equivalent to 4% pentoxiphylline)

EXPERIMENTAL

Intravaginal application of Gel PKB171 4% with a single-use applicator (syringe). The content fo the applicator (5g) was inserted will be inserted as deep as possible into the vagina, and the female will be rested for at least 45 minutes in bed

Drug: Intravaginal gel

Gel PKB171 placebo

PLACEBO COMPARATOR

Intravaginal application of Gel PKB171 4% with a single-use applicator (syringe). The content fo the applicator (5g) was inserted will be inserted as deep as possible into the vagina, and the female will be rested for at least 45 minutes in bed

Drug: Vaginal Gel with Applicator

Interventions

Intravaginal application of gel PKB171 with a single-use applicator (syringe)

Also known as: PKB171 200 mg
Gel PKB171 200 mg (equivalent to 4% pentoxiphylline)

Intravaginal application of gel PKB171 with a single-use applicator (syringe)

Also known as: PKB171 placebo
Gel PKB171 placebo

Eligibility Criteria

Age18 Years - 38 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64)

You may qualify if:

  • Written informed consent form signed before any study test or procedure.
  • Unable to conceive for more than 6 months and less than 24 months, despite regular and adequate unprotected sexual intercourse.
  • Willing and able to comply with the protocol.
  • Female subjects with the following criteria:
  • Age ≥ 18 and ≤ 38 years.
  • Regular spontaneous menstrual cycles with a 25- to 35-day length (intercycle variation less than 5 days) within the last six cycles before the first visit.
  • Normal uterine cavity shown on transvaginal sonography.
  • Normal ovarian reserve, demonstrated by AMH ≥ 1 ng/ml at day 2-5 of the cycle.
  • Antral follicle count (sum of both ovaries) ≥ 6
  • Male subjects with the following criteria:
  • Age ≥ 18 and ≤ 50 years.
  • Spermiogram with semen volume ≥ 1mL, concentration \> 11 M/mL, \< 42% total mobility and normal forms ≥ 2%

You may not qualify if:

  • Subjects eligible for this study, both women and men, must not meet any of the following criteria:
  • Body mass Index (BMI) \< 18 and ≥ 32 kg/m².
  • Any sexual intercourse with another partner (other than corresponding trial subject) within 12 weeks entry in the study and during it.
  • Active hepatitis B, C, HIV, genital herpes, Chlamydia, Gonorrhea or Syphilis infection.
  • History of malignant disease (cancer). Previous or planned chemotherapy or radiotherapy.
  • History of cerebral or retinal hemorrhage, acute myocardial infarction.
  • In females: Prohibited concomitant intravaginal products or procedures.
  • Hypersensitivity or intolerance to pentoxifylline, xanthine derivatives or any of the excipients of the IMP.
  • Employees of the investigator or trial center, with direct involvement in the proposed trial or other studies under the direction of that investigator or trial center, as well as family members of the employees or the principal investigator.
  • People committed to an institution by virtue of an order issued either by the judicial or other authorities.
  • Reasonable expectation that the subject will not be able to satisfactorily complete the study:
  • History of current psychiatric illness that would interfere with the subject's ability to comply with protocol requirements or give informed consent.
  • History of alcohol or drug abuse that would interfere with the subject's ability to comply with protocol requirements.
  • Receipt of any investigational drug within three months of screening visit.
  • Previous enrolment in this trial.
  • +25 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (12)

Clinica Universidad de Navarra

Pamplona, Navarre, 31008, Spain

RECRUITING

Hospital del Mar

Barcelona, 08003, Spain

RECRUITING

Clinica Fertty

Barcelona, 08010, Spain

NOT YET RECRUITING

Clinica Sagrada Familia

Barcelona, 08022, Spain

RECRUITING

Assir Dreta-Cap Pare Claret

Barcelona, 08037, Spain

NOT YET RECRUITING

Assir Dreta-Cap Roger de Flor

Barcelona, 08037, Spain

NOT YET RECRUITING

Hospital de la Santa Creu i Sant Pau

Barcelona, 08041, Spain

NOT YET RECRUITING

HM Gabinete Médico Velázquez

Madrid, 28001, Spain

NOT YET RECRUITING

Hospital Universitario San Rafael

Madrid, 28016, Spain

RECRUITING

Clinica Universidad de Navarra

Madrid, 28027, Spain

RECRUITING

Hospital Universitario L Paz

Madrid, 28046, Spain

NOT YET RECRUITING

Hospital Universitario Nuestra Señora de Valme

Seville, 41014, Spain

RECRUITING

MeSH Terms

Conditions

AsthenozoospermiaInfertility, Male

Interventions

Vaginal Creams, Foams, and Jellies

Condition Hierarchy (Ancestors)

Genital Diseases, MaleGenital DiseasesUrogenital DiseasesInfertilityMale Urogenital Diseases

Intervention Hierarchy (Ancestors)

Dosage FormsPharmaceutical PreparationsFeminine Hygiene ProductsEquipment and Supplies

Study Officials

  • Cristina Trilla Solà, MD, PhD

    Coordinator Investigator

    STUDY CHAIR

Central Study Contacts

Elena Vernet Arias, MD, PhD

CONTACT

Miquel Raurell, MD

CONTACT

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Model Details: The couple will be randomized to Gel PKB171 200 mg or placebo (randomization ratio 1:1).
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

February 25, 2026

First Posted

June 25, 2026

Study Start

October 28, 2025

Primary Completion (Estimated)

October 28, 2027

Study Completion (Estimated)

October 28, 2027

Last Updated

June 25, 2026

Record last verified: 2026-06

Data Sharing

IPD Sharing
Will not share

Locations