NCT07635563

Brief Summary

The goal of this randomized, double-blind, multi-dose crossover clinical trial is to determine the safety and efficacy of IHL-42X in subjects with obstructive sleep apnea. The primary endpoint is: Change in AHI4 at the end of each treatment period compared to baseline (each treatment period is 28 days). The study will consist of three separate four-way crossover dose-comparison studies each comparing three dose strengths of IHL-42X to placebo. The double-blind four-way crossover will be conducted according to a Williams design. Each of the crossover studies will test different doses of dronabinol in combination with a distinct, set dose of acetazolamide. In total, nine different combinations of dronabinol and acetazolamide formulated as IHL-42X will be tested in the study. The optimal dose strength will be selected based on safety and efficacy over a 4-week treatment period.

Trial Health

63
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
120

participants targeted

Target at P50-P75 for phase_2

Timeline
11mo left

Started Jun 2026

Shorter than P25 for phase_2

Geographic Reach
1 country

14 active sites

Status
not yet recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress4%
Jun 2026May 2027

Study Start

First participant enrolled

June 1, 2026

Completed
2 days until next milestone

First Submitted

Initial submission to the registry

June 3, 2026

Completed
6 days until next milestone

First Posted

Study publicly available on registry

June 9, 2026

Completed
10 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2027

Expected
1 month until next milestone

Study Completion

Last participant's last visit for all outcomes

May 1, 2027

Last Updated

June 9, 2026

Status Verified

June 1, 2026

Enrollment Period

10 months

First QC Date

June 3, 2026

Last Update Submit

June 3, 2026

Conditions

Keywords

OSAObstructive sleep apneaObstructive sleep apnoeaCPAPCannabinoidIHL-42XIncannexDronabinolTHCAceazolamideACZAHIPSGPolysomnographyPAPFOS-QFOSQPROMISPGIESSREMPhase II

Outcome Measures

Primary Outcomes (1)

  • Change in AHI4 at the end of each treatment period compared to baseline

    To assess the change in efficacy at the end of each dosing period compared with baseline.

    Each treatment period (28 days)

Secondary Outcomes (14)

  • Percent change in AHI4 at the end of each treatment period compared to baseline

    Each treatment period (28 days)

  • Change in Functional Outcomes of Sleep Questionnaire 10-items (FOSQ-10) at the end of each treatment period compared to baseline

    Each treatment period (28 days)

  • Change in Patient-reported outcome measurement information system (PROMIS)-Fatigue 7a at the end of each treatment period compared to baseline

    Each treatment period (28 days)

  • Change in Patient-reported outcome measurement information system - Sleep Related Impairment (PROMIS-SRI) 8a at the end of each treatment period compared to baseline

    Each treatment period (28 days)

  • Change in Patient Global Impression of Severity (PGI-S) the end of each treatment period compared to baseline

    Each treatment period (28 days)

  • +9 more secondary outcomes

Study Arms (10)

IHL-42X: 2.5 mg dronabinol + 125 mg acetazolamide

EXPERIMENTAL

IHL-42X (2.5 mg dronabinol + 125 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 2.5 mg dronabinol + 125 mg acetazolamide

IHL-42X: 5 mg dronabinol + 125 mg acetazolamide

EXPERIMENTAL

IHL-42X (5 mg dronabinol + 125 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 5 mg dronabinol + 125 mg acetazolamide

IHL-42X: 7.5 mg dronabinol + 125 mg acetazolamide

EXPERIMENTAL

IHL-42X (7.5 mg dronabinol + 125 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 7.5 mg dronabinol + 125 mg acetazolamide

IHL-42X: 2.5 mg dronabinol + 250 mg acetazolamide

EXPERIMENTAL

IHL-42X (2.5 mg dronabinol + 250 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 2.5 mg dronabinol + 250 mg acetazolamide

IHL-42X: 5 mg dronabinol + 250 mg acetazolamide

EXPERIMENTAL

IHL-42X (5 mg dronabinol + 250 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 5 mg dronabinol + 250 mg acetazolamide

IHL-42X: 7.5 mg dronabinol + 250 mg acetazolamide

EXPERIMENTAL

IHL-42X (7.5 mg dronabinol + 250 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 7.5 mg dronabinol + 250 mg acetazolamide

IHL-42X: 2.5 mg dronabinol + 375 mg acetazolamide

EXPERIMENTAL

IHL-42X (2.5 mg dronabinol + 375 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 2.5 mg dronabinol + 375 mg acetazolamide

IHL-42X: 5 mg dronabinol + 375 mg acetazolamide

EXPERIMENTAL

IHL-42X (5 mg dronabinol + 375 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 5 mg dronabinol + 375 mg acetazolamide

IHL-42X: 7.5 mg dronabinol + 375 mg acetazolamide

EXPERIMENTAL

IHL-42X (7.5 mg dronabinol + 375 mg acetazolamide), self-administered once daily every night approximately 1 hour prior to bed for 4 weeks.

Drug: IHL-42X: 7.5 mg dronabinol + 375 mg acetazolamide

Placebo: Negative control

PLACEBO COMPARATOR

One capsule self-administered once daily every night approximately 1 hour prior to bed for 4 weeks

Drug: Placebo: Negative control

Interventions

DReAMzz Phase 2 Placebo

Placebo: Negative control

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 3

IHL-42X: 7.5 mg dronabinol + 125 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 4

IHL-42X: 2.5 mg dronabinol + 250 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 5

IHL-42X: 5 mg dronabinol + 250 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 6

IHL-42X: 7.5 mg dronabinol + 250 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 7

IHL-42X: 2.5 mg dronabinol + 375 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 8

IHL-42X: 5 mg dronabinol + 375 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 9

IHL-42X: 7.5 mg dronabinol + 375 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 1

IHL-42X: 2.5 mg dronabinol + 125 mg acetazolamide

DReAMzz Phase 2 Investigational Product - IHL-42X Dose 2

IHL-42X: 5 mg dronabinol + 125 mg acetazolamide

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants must satisfy all the following criteria at screening unless otherwise stated:
  • Aged ≥18 and ≤65 years of age at the time of consent.
  • Two screening PSG findings confirmed on central over-read that both must meet the below criteria:
  • AHI4 ≥5
  • ≤25% central or mixed apneas out of total AHI
  • no Cheyne-Stokes respiration
  • total sleep time ≥ 4 hours in each PSG
  • \< 30 periodic leg movement disorder arousals per hour.
  • A difference in AHI4 of ≤15 between screening PSG 1 and screening PSG 2.
  • A PROMIS-SRI 8a score of \>16.
  • Intolerant or non-compliant to PAP, or has refused PAP after physician recommendation. Participants will be identified as intolerant or non-compliant to PAP devices by the following criteria (NB: OSA diagnosis must be entered in participant medical history):
  • Participants are regarded as PAP-non-compliant if they do not use PAP for ≥ 4 hours for at least 63 nights during consecutive 90-day period based on data collected from the PAP device (e.g., SD storage cards) and/or a cloud-based repository of PAP device data.
  • Participants are regarded as PAP-intolerant if they are former PAP users, i.e., a PAP device that they have not used for \>90 days, have tried PAP and not continued to use it or refusal of PAP after prior positive sleep study or prior refusal of provider recommended sleep study due to unwillingness to consider PAP.
  • NB: Participants will have the benefits and risks of PAP explained at screening, including that PAP is standard of care for OSA. Participants also have the option to withdraw from the study at any time if he/she elects to be treated with PAP or other alternative therapy such as an oral appliance or surgery.
  • Must agree not to take any form of cannabis or cannabinoid with the exception of the IP, or any other illicit or recreational drug while participating in this study.
  • +11 more criteria

You may not qualify if:

  • Participants will be excluded from the study if they satisfy any of the following criteria at screening, unless otherwise stated:
  • Body mass index (BMI) \>40 kg/m2 (men) and \>42 kg/m2 (women).
  • Diagnosed obesity hypoventilation syndrome or hypercapnia.
  • PAP-compliant, defined by use of PAP for ≥4 hours for at least 63 nights during the consecutive 90-day period.
  • Current use of custom-made oral appliances (mandibular advancement device, tongue retaining device, or mouth guard) or hypoglossal nerve stimulation devices. Devices must not be used for the duration of the study.
  • Maxillomandibular advancement, upper airway, or bariatric surgery within the last 6 months prior to first administration of the study drug; or participants who are planning surgical treatment.
  • Have commenced glucagon-like peptide-1 receptor agonist therapy within the last 6 months.
  • Use of benzodiazepines, sedative-hypnotics or stimulants (Anatomical Therapeutic Chemical \[ATC\] N06B, N05C, N05BA, N03AE, and N01AF categories) to treat insomnia, OSA, and other sleep disorders, or other disorders that require the drug to be taken prior to sleep.
  • Use of other prescription medications to treat insomnia.
  • Pierre Robin, Treacher Collins, or other craniofacial malformation syndrome, or grade ≥3 tonsillar hypertrophy.
  • Respiratory and neuromuscular diseases that could interfere with the results of the trial in the opinion of the investigator.
  • Known allergic or other severe reaction to cannabis products with previous use.
  • Known allergic reaction to sesame oil.
  • Known allergic reaction to acetazolamide.
  • Pregnant or breastfeeding.
  • +18 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (14)

Exalt Clinical Research

Chula Vista, California, 91910, United States

Location

Teradan Clinical Trials LLC

Brandon, Florida, 33511, United States

Location

CNS Healthcare - Jacksonville

Jacksonville, Florida, 32256, United States

Location

CNS Healthcare Orlando

Orlando, Florida, 32801, United States

Location

Palm Beach Research Center

West Palm Beach, Florida, 33409, United States

Location

Conquest Research/Neurotrials

Winter Park, Florida, 32789, United States

Location

Tandem Clinical Research

Marrero, Louisiana, 70072, United States

Location

Velocity Clinical Research, Rockville

Rockville, Maryland, 20854, United States

Location

CTI Clinical Research Center

Cincinnati, Ohio, 45212, United States

Location

Intrepid Research

Cincinnati, Ohio, 45245, United States

Location

Velocity Clinical Research, Anderson

Anderson, South Carolina, 29621, United States

Location

CNS Healthcare - Memphis

Memphis, Tennessee, 38119, United States

Location

FutureSearch Trials of Dallas

Dallas, Texas, 75251, United States

Location

Sleep Therapy & Research Center

San Antonio, Texas, 78229, United States

Location

MeSH Terms

Conditions

Sleep Apnea, Obstructive

Interventions

DronabinolAcetazolamide

Condition Hierarchy (Ancestors)

Sleep Apnea SyndromesApneaRespiration DisordersRespiratory Tract DiseasesSleep Disorders, IntrinsicDyssomniasSleep Wake DisordersNervous System Diseases

Intervention Hierarchy (Ancestors)

CannabinoidsTerpenesHydrocarbonsOrganic ChemicalsThiadiazolesThiazolesSulfur CompoundsAzolesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Central Study Contacts

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
CROSSOVER
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 3, 2026

First Posted

June 9, 2026

Study Start

June 1, 2026

Primary Completion (Estimated)

April 1, 2027

Study Completion (Estimated)

May 1, 2027

Last Updated

June 9, 2026

Record last verified: 2026-06

Locations