NCT07235046

Brief Summary

The main purpose of this study is to determine the safety and efficacy of DII235 in adults with elevated lipoprotein(a).

Trial Health

80
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
200

participants targeted

Target at P75+ for phase_2

Timeline
22mo left

Started Dec 2025

Geographic Reach
4 countries

66 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress22%
Dec 2025Apr 2028

First Submitted

Initial submission to the registry

November 14, 2025

Completed
5 days until next milestone

First Posted

Study publicly available on registry

November 19, 2025

Completed
13 days until next milestone

Study Start

First participant enrolled

December 2, 2025

Completed
1.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 26, 2027

Expected
1 year until next milestone

Study Completion

Last participant's last visit for all outcomes

April 25, 2028

Last Updated

June 8, 2026

Status Verified

June 1, 2026

Enrollment Period

1.4 years

First QC Date

November 14, 2025

Last Update Submit

June 4, 2026

Conditions

Keywords

Lipoprotein(a)cardiovascular diseaseatherosclerotic cardiovascular disease (ASCVD)lipoprotein disordercardiovascularcholesterolhyperlipidemiadyslipidemiaDII235

Outcome Measures

Primary Outcomes (3)

  • Time averaged percentage change from baseline between Day 60 and Day 180

    Time averaged change from baseline in log Lp(a) measured between Day 60 and Day 180, defined as the area under the curve (AUC) between the Day 60 Visit date and the Day 180 Visit date, divided by the duration between the two visit dates.

    baseline to day 60 and day 180

  • Difference between DII235 dose 2 and placebo in time-averaged percent change from baseline in Lp(a) measured between Day 60 and Day 360

    Time averaged change from baseline in log Lp(a) measured between Day 60 and Day 360, defined as the area under the curve (AUC) between the Day 60 visit date and the Day 360 visit date, divided by the duration between the two visit dates.

    baseline to day 60 and day 360

  • Difference between DII235 dose 4 and placebo in time-averaged percent change from baseline in Lp(a) measured between Day 60 and Day 360

    Time averaged change from baseline in log Lp(a) measured between Day 60 and Day 360, defined as the area under the curve (AUC) between the Day 60 visit date and the Day 360 visit date, divided by the duration between the two visit dates.

    baseline to day 60 and day 360

Secondary Outcomes (4)

  • Difference between DII235 dose 1, dose 3 and placebo versus placebo in time-averaged percent change from baseline in Lp(a) measured between Day 60 and Day 360

    baseline to day 60 and 360

  • Difference between DII235 doses versus placebo in time-averaged percent change from baseline in Lp(a) measured between Day 240 and Day 360

    baseline to day 240 and Day 360

  • Difference between DII235 doses versus placebo with respect to the proportion of participants in achieving Lp(a) < 125 nmol/L at Day 180 and Day 360

    Day 180 and Day 360

  • Difference between DII235 doses versus placebo with respect to the proportion of participants in achieving Lp(a) < 75 nmol/L at Day 180 and Day 360

    Day 180 and Day 360

Study Arms (5)

Arm 1

PLACEBO COMPARATOR

Placebo

Drug: Saline

Arm 2

EXPERIMENTAL

DII235 dose 1

Drug: DII235

Arm 3

EXPERIMENTAL

DII235 dose 2

Drug: DII235

Arm 4

EXPERIMENTAL

DII235 dose 3

Drug: DII235

Arm 5

EXPERIMENTAL

DII235 dose 4

Drug: DII235

Interventions

DII235DRUG

Solution for injection

Arm 2Arm 3Arm 4Arm 5
SalineDRUG

solution for injection

Arm 1

Eligibility Criteria

Age18 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Signed informed consent must be obtained prior to participation in the study.
  • Male or female participants 18 to 80 years of age (inclusive) at the screening.
  • Lp(a) ≥ 150 nmol/L at screening, measured at the central laboratory.
  • Participants with evidence of atherosclerotic cardiovascular disease and/or type 2 diabetes mellitus.

You may not qualify if:

  • Severe renal dysfunction
  • Hepatic dysfunction
  • Malignancy within the last 5 years
  • Use of investigational medications as defined in the protocol
  • History or presence at screening of an underlying disease, or surgical, physical, medical, or psychiatric condition that, in the opinion of the Investigator, or sponsor if consulted, would potentially affect participant safety within the study or interfere with participating in or completing the study or with the interpretation of data

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (66)

Parkway Medical Center

Birmingham, Alabama, 35215, United States

RECRUITING

Heart Center Research Llc

Huntsville, Alabama, 35801, United States

RECRUITING

Cardiology and Medicine Clinic PA

Little Rock, Arkansas, 72204, United States

ACTIVE NOT RECRUITING

National Heart Institute

Beverly Hills, California, 90211, United States

RECRUITING

Alliance Clinical

Canoga Park, California, 91303, United States

RECRUITING

Excel Medical Clinical Trials LLC

Boca Raton, Florida, 33434, United States

ACTIVE NOT RECRUITING

Zenith Clinical Research

Hollywood, Florida, 33021, United States

ACTIVE NOT RECRUITING

Jacksonville Center for Clinical Research

Jacksonville, Florida, 32216, United States

RECRUITING

Flourish Res Acq LLC North Miami

Miami, Florida, 33138, United States

ACTIVE NOT RECRUITING

Inpatient Research Clinical LLC

Miami Lakes, Florida, 33014, United States

RECRUITING

Inpatient Research Clinical LLC

Miami Lakes, Florida, 33014, United States

ACTIVE NOT RECRUITING

Ocala Cardiovascular Research

Ocala, Florida, 34471, United States

ACTIVE NOT RECRUITING

SEC Clinical Research

Pensacola, Florida, 32503, United States

RECRUITING

Cardiology Partners Clinical Research Institute

Wellington, Florida, 33449, United States

ACTIVE NOT RECRUITING

Atlanta Heart Specialists LLC

Tucker, Georgia, 30084, United States

RECRUITING

AMR Chicago

Niles, Illinois, 60714, United States

RECRUITING

CV Ins of the South

Lafayette, Louisiana, 70503, United States

RECRUITING

Monroe Research Llc

West Monroe, Louisiana, 71291, United States

RECRUITING

Metropolitan Cardiovascular Consultants Llc

Beltsville, Maryland, 20705, United States

RECRUITING

Anderson Medical Research

Ft. Washington, Maryland, 20744, United States

RECRUITING

Capitol Cardiology Associates

Lanham, Maryland, 20706, United States

RECRUITING

AA Medical Research Center

Flint, Michigan, 48504, United States

RECRUITING

Trinity Health Michigan Heart

Ypsilanti, Michigan, 48197, United States

RECRUITING

Cardiology Associates of North MS

Tupelo, Mississippi, 38801, United States

RECRUITING

AB Clinical Trials

Las Vegas, Nevada, 89119, United States

RECRUITING

K and R Research LLC

Marion, Ohio, 43302, United States

RECRUITING

TCV Clinical Studies

Linwood, Pennsylvania, 19061, United States

ACTIVE NOT RECRUITING

Cardiology Consultants of Philadelphia

Yardley, Pennsylvania, 19067, United States

ACTIVE NOT RECRUITING

Apex Cardiology Research Associates of Jackson

Jackson, Tennessee, 38301, United States

RECRUITING

Alliance for Multispecialty Research

Knoxville, Tennessee, 37909, United States

RECRUITING

Angiocardiac Care of Texas PA

Houston, Texas, 77025, United States

ACTIVE NOT RECRUITING

Dallas Heart and Vascular Consultants PA

Houston, Texas, 77084, United States

ACTIVE NOT RECRUITING

Biopharma Informatic

Katy, Texas, 77479, United States

ACTIVE NOT RECRUITING

Clinical Trials of Texas

San Antonio, Texas, 78229, United States

ACTIVE NOT RECRUITING

Northwest Houston Clinical Research PLLC

Tomball, Texas, 77375, United States

ACTIVE NOT RECRUITING

Progressive Clinical Research

Bountiful, Utah, 84010, United States

ACTIVE NOT RECRUITING

Dominion Medical Associates

Richmond, Virginia, 23219, United States

ACTIVE NOT RECRUITING

MultiCare Ins Research Innovation

Puyallup, Washington, 98372, United States

RECRUITING

Novartis Investigative Site

Luoyang, Henan, 471002, China

ACTIVE NOT RECRUITING

Novartis Investigative Site

Shenyang, Liaoning, 110016, China

RECRUITING

Novartis Investigative Site

Wenzhou, Zhejiang, 325000, China

ACTIVE NOT RECRUITING

Novartis Investigative Site

Beijing, 100034, China

RECRUITING

Novartis Investigative Site

Munich, Bavaria, 81377, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Potsdam, Brandenburg, 14473, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Frankfurt am Main, Hesse, 60594, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Kaiserslautern, Rhineland-Palatinate, 67655, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Dresden, Saxony, 01307, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Bad Krozingen, 79189, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Bad Oeynhausen, 32545, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Berlin, 10787, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Dortmund, 44137, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Essen, 45147, Germany

WITHDRAWN

Novartis Investigative Site

Essen, 45359, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Gladbeck, 45968, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Magdeburg, 39120, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Münster, 48145, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Papenburg, 26871, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Rostock, 18057, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Rüdersdorf, 15562, Germany

WITHDRAWN

Novartis Investigative Site

Warendorf, 48231, Germany

ACTIVE NOT RECRUITING

Novartis Investigative Site

Matsudo, Chiba, 270-2251, Japan

ACTIVE NOT RECRUITING

Novartis Investigative Site

Takamatsu, Kagawa-ken, 7608557, Japan

ACTIVE NOT RECRUITING

Novartis Investigative Site

Miyhazaki, Miyazaki, 8802102, Japan

ACTIVE NOT RECRUITING

Novartis Investigative Site

Suita, Osaka, 5650853, Japan

RECRUITING

Novartis Investigative Site

Shinjuku Ku, Tokyo, 160-0008, Japan

RECRUITING

Novartis Investigative Site

Kyoto, 6078062, Japan

ACTIVE NOT RECRUITING

MeSH Terms

Conditions

Cardiovascular DiseasesAtherosclerosisHyperlipidemiasDyslipidemias

Interventions

Sodium Chloride

Condition Hierarchy (Ancestors)

ArteriosclerosisArterial Occlusive DiseasesVascular DiseasesLipid Metabolism DisordersMetabolic DiseasesNutritional and Metabolic Diseases

Intervention Hierarchy (Ancestors)

ChloridesHydrochloric AcidChlorine CompoundsInorganic ChemicalsSodium Compounds

Study Officials

  • Novartis Pharmaceuticals

    Novartis Pharmaceuticals

    STUDY DIRECTOR

Central Study Contacts

Novartis Pharmaceuticals

CONTACT

Novartis Pharmaceuticals

CONTACT

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Masking Details
In order to preserve the integrity of the study and to minimize bias, a randomized double-blind study design is being used.
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 14, 2025

First Posted

November 19, 2025

Study Start

December 2, 2025

Primary Completion (Estimated)

April 26, 2027

Study Completion (Estimated)

April 25, 2028

Last Updated

June 8, 2026

Record last verified: 2026-06

Data Sharing

IPD Sharing
Will share

Novartis is committed to sharing with qualified external researchers, access to patient-level data and supporting clinical documents from eligible studies. These requests are reviewed and approved by an independent review panel on the basis of scientific merit. All data provided is anonymized to respect the privacy of patients who have participated in the trial in line with applicable laws and regulations. This trial data availability is according to the criteria and process described on www.clinicalstudydatarequest.com

Locations