NCT07218926

Brief Summary

The purpose of this study is to find out if a new drug, called IDRX-42 (also known as GSK6042981), is effective in treating adults with a type of cancer called Gastrointestinal Stromal Tumors (GIST) when compared to another drug named sunitinib. The study will see if IDRX-42 works well and is safe for participants whose GIST has spread or cannot be surgically removed, and who have already taken the drug imatinib.

Trial Health

83
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
450

participants targeted

Target at P50-P75 for phase_3

Timeline
56mo left

Started Dec 2025

Longer than P75 for phase_3

Geographic Reach
5 countries

20 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress9%
Dec 2025Nov 2030

First Submitted

Initial submission to the registry

October 17, 2025

Completed
4 days until next milestone

First Posted

Study publicly available on registry

October 21, 2025

Completed
1 month until next milestone

Study Start

First participant enrolled

December 3, 2025

Completed
2.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 30, 2028

Expected
2.5 years until next milestone

Study Completion

Last participant's last visit for all outcomes

November 29, 2030

Last Updated

January 30, 2026

Status Verified

January 1, 2026

Enrollment Period

2.5 years

First QC Date

October 17, 2025

Last Update Submit

January 29, 2026

Conditions

Keywords

GSK6042981IDRX-42SunitinibImatinibGastrointestinal Stromal Tumors

Outcome Measures

Primary Outcomes (1)

  • Progression-Free Survival (PFS)

    PFS is defined as time from the date of randomization to the date of disease progression or death due to any cause, whichever occurs first.

    Up to approximately 130 weeks

Secondary Outcomes (13)

  • Overall Survival (OS)

    Up to approximately 261 weeks

  • Progression-Free Survival (PFS)

    Up to approximately 261 weeks

  • Confirmed Overall Objective Response Rate (ORR)

    Up to approximately 261 weeks

  • Time to Response (TTR)

    Up to approximately 261 weeks

  • Time from initial study randomization to second disease progression or death after starting the next line of treatment (PFS2)

    Up to approximately 261 weeks

  • +8 more secondary outcomes

Study Arms (2)

IDRX-42 (GSK6042981)

EXPERIMENTAL
Drug: IDRX-42

Sunitinib

ACTIVE COMPARATOR
Drug: Sunitinib

Interventions

Sunitinib will be administered.

Sunitinib

IDRX-42 will be administered.

Also known as: GSK6042981
IDRX-42 (GSK6042981)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants with histologically or cytologically confirmed GIST that is metastatic and/or surgically unresectable.
  • Documented disease progression on or intolerance to imatinib administered for first-line treatment of unresectable/metastatic disease.
  • Tumor tissue must be available to be submitted to the central laboratory for retrospective biomarker analysis. The sample may be from archival tissue or a new biopsy. Tissue samples are not required to be submitted centrally prior to randomization.

You may not qualify if:

  • Known untreated or active central nervous system metastases.
  • Participants with a known allergy or hypersensitivity to any component of IDRX-42 (GSK6042981) or sunitinib. Participants with a history of Stevens-Johnson syndrome on a prior Tyrosine kinase inhibitor (TKI) are excluded.
  • Has a malignancy (except disease under study) that has progressed or required active treatment within the past 24 months except for basal cell or squamous cell carcinomas of the skin or in-situ carcinomas \[e.g., breast, cervix, bladder\] that have been resected with no evidence of metastatic disease.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (20)

GSK Investigational Site

Boston, Massachusetts, 02215, United States

RECRUITING

GSK Investigational Site

Omaha, Nebraska, 68130, United States

RECRUITING

GSK Investigational Site

New York, New York, 10032, United States

RECRUITING

GSK Investigational Site

Philadelphia, Pennsylvania, 19111, United States

RECRUITING

GSK Investigational Site

Knoxville, Tennessee, 37920, United States

RECRUITING

GSK Investigational Site

Houston, Texas, 77030, United States

RECRUITING

GSK Investigational Site

Tacoma, Washington, 98405, United States

RECRUITING

GSK Investigational Site

Toronto, Ontario, M5G 2M9, Canada

RECRUITING

GSK Investigational Site

Chiba, 277-8577, Japan

RECRUITING

GSK Investigational Site

Ehime, 791-0280, Japan

RECRUITING

GSK Investigational Site

Fukuoka, 812-8582, Japan

RECRUITING

GSK Investigational Site

Hokkaido, 060-8648, Japan

RECRUITING

GSK Investigational Site

Kanagawa, 247-8533, Japan

RECRUITING

GSK Investigational Site

Osaka, 565-0871, Japan

RECRUITING

GSK Investigational Site

Tokyo, 104-0045, Japan

RECRUITING

GSK Investigational Site

Changhua, 500, Taiwan

RECRUITING

GSK Investigational Site

Kaohsiung City, 807, Taiwan

RECRUITING

GSK Investigational Site

Taipei, 100, Taiwan

RECRUITING

GSK Investigational Site

London, SW3 6JJ, United Kingdom

RECRUITING

GSK Investigational Site

Manchester, M20 4BX, United Kingdom

RECRUITING

MeSH Terms

Conditions

Gastrointestinal NeoplasmsGastrointestinal Stromal Tumors

Interventions

IDRX-42Sunitinib

Condition Hierarchy (Ancestors)

Digestive System NeoplasmsNeoplasms by SiteNeoplasmsDigestive System DiseasesGastrointestinal DiseasesNeoplasms, Connective TissueNeoplasms, Connective and Soft TissueNeoplasms by Histologic Type

Intervention Hierarchy (Ancestors)

PyrrolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsIndolesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-Ring

Central Study Contacts

US GSK Clinical Trials Call Center

CONTACT

EU GSK Clinical Trials Call Center

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 17, 2025

First Posted

October 21, 2025

Study Start

December 3, 2025

Primary Completion (Estimated)

May 30, 2028

Study Completion (Estimated)

November 29, 2030

Last Updated

January 30, 2026

Record last verified: 2026-01

Data Sharing

IPD Sharing
Will not share

GSK will assess requests from qualified researchers for anonymized individual patient-level data and related study documents. Data sharing is subject to certain criteria, conditions, and exceptions. For further information, refer to https://www.gsk-studyregister.com/About\_GSK\_Patient\_Level\_Data\_Sharing\_Final\_13July2023.pdf.

Locations