NCT07011732

Brief Summary

The purpose of this study is to evaluate the efficacy and safety of KarXT + KarX-EC in adult participants with agitation related to Alzheimer's Disease.

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
352

participants targeted

Target at P25-P50 for phase_3 alzheimer-disease

Timeline
32mo left

Started Jul 2025

Typical duration for phase_3 alzheimer-disease

Geographic Reach
15 countries

157 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress24%
Jul 2025Dec 2028

First Submitted

Initial submission to the registry

June 2, 2025

Completed
8 days until next milestone

First Posted

Study publicly available on registry

June 10, 2025

Completed
1 month until next milestone

Study Start

First participant enrolled

July 10, 2025

Completed
3.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 24, 2028

Expected
14 days until next milestone

Study Completion

Last participant's last visit for all outcomes

December 8, 2028

Last Updated

April 30, 2026

Status Verified

April 1, 2026

Enrollment Period

3.4 years

First QC Date

June 2, 2025

Last Update Submit

April 29, 2026

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change from baseline on the Cohen-Mansfield Agitation Inventory-International Psychogeriatric Association (CMAI-IPA) total score at Week 14

    At Week 14

Secondary Outcomes (20)

  • Change from baseline on the Clinical Global Impressions-Severity (CGI-S) at Week 14

    At Week 14

  • Change from baseline on the CMAI-IPA Domains at Week 14

    At Week 14

  • Change from baseline on the CMAI Total Score at Week 14

    At Week 14

  • Number of participants with Occurrence of Response at Week 14

    At Week 14

  • Change from baseline on the Neuropsychiatric Inventory/Neuropsychiatric Inventory -Nursing Home (NPI/NPI-NH) Total Score at Week 14

    At Week 14

  • +15 more secondary outcomes

Study Arms (2)

KarXT + KarX-EC

EXPERIMENTAL
Drug: Xanomeline/Trospium Chloride CapsuleDrug: Xanomeline Enteric Capsule

Placebo

PLACEBO COMPARATOR
Drug: Placebo

Interventions

Specified dose on specified days

Also known as: KarXT, BMS-986510
KarXT + KarX-EC

Specified dose on specified days

Also known as: KarX-EC, BMS-986519
KarXT + KarX-EC

Specified dose on specified days

Placebo

Eligibility Criteria

Age55 Years - 90 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • \- A diagnosis of Alzheimer's disease (AD) in accordance with the 2024 Alzheimer's Association criteria with one of the following confirmations of AD pathology: i) Historical evidence of AD diagnosis with amyloid positron emission tomography (PET), Aβ42/40 ratio in CSF, pTau181/Aβ42 ratio in CSF or pTau217/Aβ42 ratio in plasma using an Health Authority (HA)-authorized diagnostic assay.
  • ii) If no historical evidence available: A. A plasma biomarker will be assessed for eligibility if allowed per regulatory requirements. The test cutoff(s) will be based on diagnostic use approval.
  • B. If a plasma biomarker assay cannot be used or if the assay result is inconclusive, conduct one the following:
  • Amyloid PET.
  • Aβ42/40 ratio or pTau181/Aβ42 ratio in CSF using an HA-authorized diagnostic assay.
  • Mini-Mental State Examination (MMSE) score of 5 to 22, inclusive, at Screening (Visit 1).
  • Have one identified caregiver who should have sufficient contact (approximately 10 hours a week or more) and is willing to:
  • i) Attend all visits and report on participant's status. ii) Oversee participant compliance with medication and study procedures. iii) Participate in the study assessments and provide informed consent to participate in the study.
  • History of agitation that meets the International Psychogeriatric Association (IPA) consensus definition for agitation in cognitive disorders with onset at least two weeks prior to Screening (Visit 1).
  • AD participants are required to have NPI/NPI-NH Agitation/Aggression score ≥ 4 at Screening (Visit 1) and Baseline (Visit 2).
  • CGI-S ≥ 4, as related to agitation, at Screening (Visit 1) and Baseline (Visit 2).
  • At least 1 of the following 3 criteria must be established from the CMAI-IPA at Screening (Visit 1) and Baseline (Visit 2; CMAI-IPA Physical/Verbal Aggression Positivity):
  • i) 1 or more aggressive behaviors occurring at least several times per week. ii) 2 or more aggressive behaviors occurring at least once or twice per week. iii) 3 or more aggressive behaviors occurring less than once per week.

You may not qualify if:

  • \- Medical Conditions: i) Agitation symptoms that are primarily attributable to a condition other than the AD causing the dementia.
  • ii) History of bipolar disorder, schizophrenia, or schizoaffective disorder. iii) History of (or at high risk for) urinary retention, gastric retention, or narrow-angle glaucoma as evaluated by the Investigator.
  • iv) Risk of suicidal behavior during the study as determined by the Investigator's clinical assessment and/or C-SSR.
  • \- Prior/Concomitant Therapy: i) Recent history of receiving monoamine oxidase inhibitors, anticonvulsants (eg, lamotrigine, divalproex), mood stabilizers (eg, lithium), tricyclic antidepressants (eg, imipramine, desipramine), or any other psychoactive medications except for as needed anxiolytics (eg, lorazepam).
  • A. Selective serotonin reuptake inhibitors and serotonin norepinephrine reuptake inhibitors taken at a stable dose for at least 8 weeks prior to Screening (Visit 1) may be permitted.
  • B. Mirtazapine or trazodone may be used as a hypnotic if started at least 8 weeks prior to Screening (Visit 1).

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (157)

Imaging Endpoints

Scottsdale, Arizona, 85258, United States

RECRUITING

Advanced Research Center (ARC) - Anaheim

Anaheim, California, 92805, United States

RECRUITING

Kaizen Brain Center

La Jolla, California, 92037, United States

RECRUITING

The Neurology Group

Pomona, California, 91767, United States

RECRUITING

Torrance Clinical Research

Torrance, California, 90505, United States

RECRUITING

Sunwise Clinical Research

Walnut Creek, California, 94596, United States

RECRUITING

Local Institution - 1630

Colorado Springs, Colorado, 80907, United States

WITHDRAWN

Local Institution - 1622

Maitland, Florida, 32751, United States

NOT YET RECRUITING

Local Institution - 1631

Maitland, Florida, 32751, United States

NOT YET RECRUITING

Local Institution - 1602

Miami, Florida, 33122, United States

NOT YET RECRUITING

Local Institution - 1618

Miami, Florida, 33135, United States

NOT YET RECRUITING

Hope Research Network - Miami

Miami, Florida, 33166, United States

RECRUITING

Local Institution - 1604

Miami, Florida, 33186, United States

ACTIVE NOT RECRUITING

Local Institution - 1608

Ocala, Florida, 34471, United States

NOT YET RECRUITING

Combined Research Orlando (CRO)

Orlando, Florida, 32807, United States

RECRUITING

Progressive Medical Research

Port Orange, Florida, 32127, United States

RECRUITING

Local Institution - 1661

Savannah, Georgia, 31406, United States

NOT YET RECRUITING

Local Institution - 1655

Marrero, Louisiana, 70072, United States

NOT YET RECRUITING

CBH Health

Gaithersburg, Maryland, 20877, United States

RECRUITING

Local Institution - 1663

Foxborough, Massachusetts, 02035-1309, United States

NOT YET RECRUITING

Boston Center for Memory

Newton, Massachusetts, 02459, United States

RECRUITING

Mayflower Clinical Research

South Dartmouth, Massachusetts, 02747, United States

RECRUITING

Elixia MA

Springfield, Massachusetts, 01103, United States

RECRUITING

Local Institution - 1665

Bloomfield Hills, Michigan, 48302, United States

NOT YET RECRUITING

Oakland Medical Research

Troy, Michigan, 48085, United States

RECRUITING

Redbird Research

Las Vegas, Nevada, 89119, United States

RECRUITING

Patient First MD

Middletown, New Jersey, 07748, United States

RECRUITING

Local Institution - 1664

Princeton, New Jersey, 08540, United States

NOT YET RECRUITING

Local Institution - 1610

Inwood, New York, 11096, United States

NOT YET RECRUITING

Mid Hudson Medical Research

New Windsor, New York, 12553, United States

RECRUITING

Five Towns Neurology PC -Woodmere - 923 Broadway

Woodmere, New York, 11598-1739, United States

RECRUITING

Local Institution - 1645

Woodmere, New York, 11598-1739, United States

WITHDRAWN

Local Institution - 1659

Centerville, Ohio, 45459, United States

NOT YET RECRUITING

Central States Research

Tulsa, Oklahoma, 74136, United States

RECRUITING

Local Institution - 1652

Columbia, South Carolina, 29205, United States

WITHDRAWN

Advanced Neurology Epilepsy and Sleep Center

El Paso, Texas, 79912, United States

RECRUITING

Wasatch Clinical Research, LLC

Salt Lake City, Utah, 84107, United States

RECRUITING

The Memory Clinic

Bennington, Vermont, 05201-9810, United States

RECRUITING

Local Institution - 1644

Seattle, Washington, 98122, United States

NOT YET RECRUITING

Kingfisher Cooperative

Spokane, Washington, 99201, United States

RECRUITING

Local Institution - 1001

La Plata, Buenos Aires, 1900, Argentina

NOT YET RECRUITING

Local Institution - 1002

Mar del Plata, Buenos Aires, B7602CBM, Argentina

NOT YET RECRUITING

Fundacion Estudios Clinicos

Rosario, Santa Fe Province, S2000DEJ, Argentina

RECRUITING

Local Institution - 1003

Buenos Aires, C1428AQK, Argentina

NOT YET RECRUITING

Local Institution - 1004

Córdoba, 5000, Argentina

NOT YET RECRUITING

Instituto Privado Kremer

Córdoba, 5004, Argentina

RECRUITING

Centro Medico Luquez

Córdoba, 5006, Argentina

RECRUITING

Local Institution - 1051

Brasília, Federal District, 70200730, Brazil

NOT YET RECRUITING

CECPAR - Centro de Estudos Clínicos do Paraná

Curitiba, Paraná, 80030-310, Brazil

RECRUITING

PUCTrials

Curitiba, Paraná, 80230-130, Brazil

RECRUITING

Local Institution - 1058

Porto Alegre, Rio Grande do Sul, 90430-001, Brazil

NOT YET RECRUITING

Hospital Moinhos de Vento

Porto Alegre, Rio Grande do Sul, 90560-032, Brazil

RECRUITING

Local Institution - 1057

Campinas, São Paulo, 13060-080, Brazil

NOT YET RECRUITING

Ruschel Medicina e Pesquisa Clínica

Rio de Janeiro, 22270-060, Brazil

RECRUITING

CPQuali Pesquisa Clínica

São Paulo, 01228-000, Brazil

RECRUITING

Clinica Viver - Centro de Desospitalizacao Humana

São Paulo, 04020-060, Brazil

RECRUITING

Medical Center Sveti Naum EOOD

Sofia, Sofia-Grad, 1113, Bulgaria

RECRUITING

Local Institution - 1104

Sofia, Sofia-Grad, 1202, Bulgaria

NOT YET RECRUITING

Medical Center Medconsult Pleven OOD

Pleven, 5800, Bulgaria

RECRUITING

Outpatient Clinic for Individual Practice for Specialized Medical Care in Psychiatry - Dr. Madlena Dimitrova Borisova

Razgrad, 7200, Bulgaria

RECRUITING

Medical Center Mladost

Varna, 9020, Bulgaria

RECRUITING

Local Institution - 1153

Hamilton, Ontario, ON L8M 1W9, Canada

NOT YET RECRUITING

Local Institution - 1755

London, Ontario, N6A 5W9, Canada

WITHDRAWN

London Health Sciences Centre-Victoria Campus

London, Ontario, N6A 5W9, Canada

RECRUITING

Sunnybrook Research Institute

Toronto, Ontario, M4N 3M5, Canada

RECRUITING

Centre for Addiction & Mental Health

Toronto, Ontario, M6J 1H4, Canada

RECRUITING

Ontario Shores Centre For Mental Health Sciences

Whitby, Ontario, L1N 5S9, Canada

RECRUITING

Local Institution - 1150

Montreal, Quebec, H4A 3T2, Canada

NOT YET RECRUITING

Xuanwu Hospital Capital Medical University

Beijing, Beijing Municipality, 100053, China

RECRUITING

Local Institution - 1810

Beijing, Beijing Municipality, 100088, China

NOT YET RECRUITING

Local Institution - 1815

Haidian District, Beijing Municipality, 100191, China

NOT YET RECRUITING

Local Institution - 1813

Chongqing, Chongqing Municipality, 630014, China

NOT YET RECRUITING

Local Institution - 1809

Guangzhou, Guangdong, 0, China

NOT YET RECRUITING

Shenzhen Kangning Hospital

Shenzhen, Guangdong, 518118, China

RECRUITING

Local Institution - 1802

Guangzhou, Guangzhou Province, 510260, China

NOT YET RECRUITING

Local Institution - 1803

Changsha, Hunan, 410008, China

NOT YET RECRUITING

Local Institution - 1801

Nanjing, Jiangsu, 210008, China

NOT YET RECRUITING

Local Institution - 1800

Shanghai, Shanghai Municipality, 200025, China

NOT YET RECRUITING

Local Institution - 1816

Xian, Shanxi, 710061, China

NOT YET RECRUITING

Local Institution - 1819

Chengdu, Sichuan, 610041, China

NOT YET RECRUITING

Tianjin Anding Hospital

Tianjin, Tianjin Municipality, 300074, China

RECRUITING

Local Institution - 1804

Hangzhou, Zhejiang, 310003, China

NOT YET RECRUITING

Local Institution - 1817

Hangzhou, 310016, China

NOT YET RECRUITING

Local Institution - 1812

Kunming, 650032, China

NOT YET RECRUITING

Local Institution - 1808

Tianjin, 300350, China

NOT YET RECRUITING

Local Institution - 1550

Zagreb, City of Zagreb, 10000, Croatia

NOT YET RECRUITING

Local Institution - 1553

Zagreb, City of Zagreb, 10000, Croatia

NOT YET RECRUITING

Local Institution - 1554

Rijeka, 51000, Croatia

NOT YET RECRUITING

Clinical Hospital Center Split

Split, HR-21000, Croatia

RECRUITING

General Hospital Varazdin

Varaždin, 42000, Croatia

RECRUITING

University Hospital of Patras

Pátrai, Achaḯa, 26504, Greece

RECRUITING

Henry Dunant Hospital Center

Athens, Attica, 115 26, Greece

RECRUITING

Aiginiteio University Hospital

Athens, Attikí, 115 28, Greece

RECRUITING

University General Hospital "ATTIKON" - General Hospital of West Attica "H AGIA VARVARA"

Chaïdári, Attikí, 124 62, Greece

RECRUITING

Eginition Hospital

Athens, 11528, Greece

RECRUITING

Local Institution - 1207

Athens, 15125, Greece

NOT YET RECRUITING

Local Institution - 1201

Ioannina, 45500, Greece

NOT YET RECRUITING

Euromedica General Clinic of Thessaloniki

Thessaloniki, 54645, Greece

RECRUITING

Local Institution - 1255

Ahmedabad, Gujarat, 380060, India

NOT YET RECRUITING

Local Institution - 1252

Hyderabad, Telangana, 500082, India

NOT YET RECRUITING

Local Institution - 1254

Varanasi, Uttar Pradesh, 221005, India

NOT YET RECRUITING

Local Institution - 1250

Kolkata, West Bengal, 700054, India

NOT YET RECRUITING

Local Institution - 1256

Delhi, 110 095, India

NOT YET RECRUITING

Local Institution - 1251

Hyderabad, 500034, India

NOT YET RECRUITING

Local Institution - 1253

New Delhi, 110029, India

NOT YET RECRUITING

Local Institution - 1301

Hadano, Kanagawa, 257-0003, Japan

NOT YET RECRUITING

Teikyo University Mizonokuchi Hospital

Kawasaki, Kanagawa, 213-8507, Japan

RECRUITING

Local Institution - 1304

Sakai, Osaka, 590-0018, Japan

NOT YET RECRUITING

National Hospital Organization Hizen Psychiatric Center

Kanzaki-Gun Yoshinogari-Cho, Saga-ken, 842-0192, Japan

RECRUITING

Rainbow and Sea Hospital

Karatsu-shi, Saga-ken, 847-0031, Japan

RECRUITING

Local Institution - 1305

Bunkyo-ku, Tokyo, 113-8603, Japan

NOT YET RECRUITING

Kuramitsu Hospital

Fukuoka, 819-0037, Japan

RECRUITING

Okayama City General Medical Center Okayama City Hospital

Okayama, 700-8557, Japan

RECRUITING

Local Institution - 1308

Shimotsuke-shi, Tochigi, 329-0498, Japan

NOT YET RECRUITING

Hospital Universitario de Saltillo

Saltillo, Coahuila, 25000, Mexico

RECRUITING

Boca Clinical Trials Mexico S.C.

Guadalajara, Jalisco, 44600, Mexico

RECRUITING

Innovacion y Desarrollo en Ciencias de la Salud

Mexico City, Mexico City, 14090, Mexico

RECRUITING

Local Institution - 1360

Mexico City, Mexico City, 14269, Mexico

NOT YET RECRUITING

AVIX Investigacion Clinica

Monterrey, Nuevo León, 64623, Mexico

RECRUITING

Local Institution - 1350

Monterrey, Nuevo León, 66460, Mexico

NOT YET RECRUITING

Local Institution - 1361

Mexico City, 10200, Mexico

NOT YET RECRUITING

Neurociencias PRISMA A.C.

San Luis Potosí City, 78216, Mexico

RECRUITING

Clinical Research Institute S.C.

Tlalnepantla, 54055, Mexico

RECRUITING

Local Institution - 1401

Coimbra, 3049, Portugal

NOT YET RECRUITING

Centro Hospitalar do Alto Ave

Guimarães, 4835-044, Portugal

RECRUITING

Local Institution - 1404

Lisbon, 1649-035, Portugal

NOT YET RECRUITING

Unidade Local de Saúde de Matosinhos SA

Senhora da Hora, 4464-513, Portugal

RECRUITING

Campus Neurologico Senior

Torres Vedras, 2560-280, Portugal

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Prof. Dr. Alexandru Obregia Psychiatry Hospital

Bucharest, Bucharest, 041919, Romania

RECRUITING

Local Institution - 1451

Bucharest, 010825, Romania

NOT YET RECRUITING

Local Institution - 1459

Bucharest, 060222, Romania

NOT YET RECRUITING

Prof Dr Alexandru Obregia Clinical Psychiatric Hospital- Centrul de Sanatate Mintala

Bucharest, 40874, Romania

RECRUITING

Local Institution - 1461

Constanța, 90123, Romania

NOT YET RECRUITING

Institutul de Psihiatrie Socola

Iași, 700282, Romania

RECRUITING

Local Institution - 1460

Sanpetru /Brasov, 507190, Romania

NOT YET RECRUITING

Local Institution - 1462

Sibiu, 550082, Romania

NOT YET RECRUITING

Oroitu CAE

Getxo, Bizkaia, 48993, Spain

RECRUITING

Hospital General Universitario de Elche

Elche (alicante), 03203, Spain

RECRUITING

Complejo Hospitalario Ruber Juan Bravo

Madrid, 28006, Spain

RECRUITING

Hospital Clinico San Carlos

Madrid, 28040, Spain

RECRUITING

Hospital Clinico Universitario Virgen de La Victoria

Málaga, 29010, Spain

RECRUITING

Clinica Universidad de Navarra

Pamplona, 31008, Spain

RECRUITING

Hospital Universitario de Salamanca - Complejo Asistencial Universitario de Salamanca

Salamanca, 37007, Spain

RECRUITING

Hospital Victoria Eugenia de Sevilla

Seville, 41009, Spain

RECRUITING

Hospital Mutua Terrassa

Terrassa, 8221, Spain

RECRUITING

Hospital Universitario De Rio Hortega

Valladolid, 47012, Spain

RECRUITING

Hospital Viamed Montecanal

Zaragoza, 50012, Spain

RECRUITING

Chang Gung Memorial Hospital at Kaohsiung

Kaohsiung Niao Sung Dist, Kaohsiung, 83301, Taiwan

RECRUITING

National Cheng Kung University Hospital

Tainan, Taiana, 704, Taiwan

RECRUITING

National Taiwan University Hospital

Taipei, 100229, Taiwan

RECRUITING

Taipei Veterans General Hospital

Taipei, 112, Taiwan

RECRUITING

Chang Gung Medical Foundation-Linkou Branch

Taoyuan, 333, Taiwan

RECRUITING

Related Links

MeSH Terms

Conditions

Alzheimer Disease

Interventions

xanomelinetrospium chloride

Condition Hierarchy (Ancestors)

DementiaBrain DiseasesCentral Nervous System DiseasesNervous System DiseasesTauopathiesNeurodegenerative DiseasesNeurocognitive DisordersMental Disorders

Study Officials

  • Bristol-Myers Squibb

    Bristol-Myers Squibb

    STUDY DIRECTOR

Central Study Contacts

BMS Clinical Trials Contact Center www.BMSClinicalTrials.com

CONTACT

First line of the email MUST contain NCT # and Site #.

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 2, 2025

First Posted

June 10, 2025

Study Start

July 10, 2025

Primary Completion (Estimated)

November 24, 2028

Study Completion (Estimated)

December 8, 2028

Last Updated

April 30, 2026

Record last verified: 2026-04

Data Sharing

IPD Sharing
Will share

BMS will provide access to individual anonymized participant data upon request from qualified researchers, and subject to certain criteria. Additional information regarding Bristol Myer Squibb's data sharing policy and process can be found at https://www.bms.com/researchers-and-partners/clinical-trials-and-research.html

Shared Documents
STUDY PROTOCOL, SAP, CSR
Time Frame
See Plan Description
Access Criteria
See Plan Description
More information

Locations