NCT06353347

Brief Summary

The goal of this clinical study is to evaluate the efficacy and safety of berberine ursodeoxycholate (HTD1801) compared to placebo in patients with type 2 diabetes inadequately controlled with metformin.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
551

participants targeted

Target at P75+ for phase_3 type-2-diabetes-mellitus

Timeline
Completed

Started Nov 2023

Geographic Reach
1 country

64 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

November 13, 2023

Completed
5 months until next milestone

First Submitted

Initial submission to the registry

April 3, 2024

Completed
6 days until next milestone

First Posted

Study publicly available on registry

April 9, 2024

Completed
8 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

December 12, 2024

Completed
8 months until next milestone

Study Completion

Last participant's last visit for all outcomes

July 30, 2025

Completed
Last Updated

November 26, 2025

Status Verified

November 1, 2025

Enrollment Period

1.1 years

First QC Date

April 3, 2024

Last Update Submit

November 19, 2025

Conditions

Outcome Measures

Primary Outcomes (1)

  • Primary Endpoint: mean change in HbA1c

    Mean change in HbA1c from baseline to Week 24

    24 Weeks

Secondary Outcomes (6)

  • Double-blind (DB) Phase: mean change in fasting plasma glucose

    24 Weeks

  • DB Phase: mean change in 2-hour postprandial glucose

    24 Weeks

  • DB Phase: proportion of patients achieving HbA1c <7.0%

    24 Weeks

  • DB Phase: proportion of patients achieving HbA1c <6.5%

    24 Weeks

  • DB Phase: mean change in insulin sensitivity (HOMA-IR)

    24 Weeks

  • +1 more secondary outcomes

Other Outcomes (6)

  • Open-Label Extension (OLE) Phase: mean change in HbA1c

    52 Weeks

  • OLE Phase: mean change in 2-Hour postprandial glucose

    52 Weeks

  • OLE Phase: proportion of patients achieving HbA1c <7.0%

    52 Weeks

  • +3 more other outcomes

Study Arms (2)

HTD1801

EXPERIMENTAL

Administered orally twice daily (BID)

Drug: HTD1801

Placebo

PLACEBO COMPARATOR

Administered orally BID

Drug: Placebo

Interventions

HTD1801 1000 mg administered orally BID as four capsules

Also known as: berberine ursodeoxycholate
HTD1801

Matching placebo administered orally BID as four capsules

Placebo

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Have been diagnosed with type 2 diabetes
  • Received a stable dose of metformin monotherapy for at least 8 weeks prior to screening
  • If used any glucose-lowering drugs other than metformin within the 8 weeks prior to screening such use was ≤7 days and was discontinued at least 4 weeks prior to screening
  • Have HbA1c ≥7.5% to ≤11.0% (screening) and HbA1c ≥7.0% to ≤10.5% (pre-randomization)
  • Have fasting plasma glucose ≤13.9 mmol/L (screening and pre-randomization)
  • Have a body mass index ≥19.0 kg/m\^2 to ≤35.0 kg/m\^2

You may not qualify if:

  • Have type 1 diabetes
  • Have had any acute diabetic complications within 12 months prior to screening
  • Have had any Grade 3 hypoglycemic event within 12 months prior to screening
  • Have had proliferative retinopathy or macular degeneration, severe diabetic neuropathy, or diabetic foot
  • Have been taking any weight loss medication or dietary supplement, have participated in a weight loss program, or have adhered to a special diet within 12 weeks prior to screening
  • Have used insulin or an insulin analogue for more than 14 days within 12 months prior to screening
  • Have used any hypoglycemic drug other than metformin during the 4-week run-in period prior to randomization
  • Have had weight gain or loss ≥5% during the 4-week run-in period prior to randomization

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (64)

Baogang Hospital of Inner Mongolia

Baotou, China

Location

Beijing Friendship Hospital, Capital Medical University

Beijing, China

Location

Beijing Luhe Hospital Capital Medical University

Beijing, China

Location

Beijing Pinggu Hospital

Beijing, China

Location

Peking Union Medical College Hospital

Beijing, China

Location

Peking University People's Hospital

Beijing, China

Location

The Second Norman Bethune Hospital of Jilin University

Changchun, China

Location

The First People's Hospital of Changde City

Changde, China

Location

Hunan Provincial People's Hospital

Changsha, China

Location

The Third Xiangya Hospital of Central South University

Changsha, China

Location

Chongqing University Three Gorges Hospital

Chongqing, China

Location

The Third People's Hospital of Datong

Datong, China

Location

Nanfang Hospital, Southern Medical University

Guangzhou, China

Location

Handan First Hospital

Handan, China

Location

The Fourth Affiliated Hospital of Harbin Medical University

Harbin, China

Location

Anhui Provincial Hospital

Hefei, China

Location

The Second Hospital of Anhui Medical University

Hefei, China

Location

Hengshui People's Hospital (Harrison International Peace Hospital)

Hengshui, China

Location

Heze Municipal Hospital

Heze, China

Location

Huai'an First People's Hospital

Huai'an, China

Location

Huangshi Central Hospital

Huangshi, China

Location

Huizhou Municipal Central Hospital

Huizhou, China

Location

Huzhou Central Hospital

Huzhou, China

Location

Jinan Central Hospital

Jinan, China

Location

Jingzhou Central Hospital

Jingzhou, China

Location

Jinzhou Central Hospital

Jinzhou, China

Location

The First People's Hospital of Kashgar

Kashgar, China

Location

Hebei Petro China Center Hospital

Langfang, China

Location

Liaocheng People's Hospital

Liaocheng, China

Location

The First Affiliated Hospital of Henan University of Science and Technology (Jinghua)

Luoyang, China

Location

The First Affiliated Hospital of Henan University of Science and Technology (Kaiyuan)

Luoyang, China

Location

Nanjing Drum Tower Hospital - The Affiliated Hospital of Nanjing University Medical School

Nanjing, China

Location

Nanjing First Hospital

Nanjing, China

Location

Nanjing Jiangning Hospital

Nanjing, China

Location

Sir Run Run Hospital Nanjing Medical University

Nanjing, China

Location

The Second Affiliated Hospital of Nanjing Medical University

Nanjing, China

Location

The First People's Hospital of Nanning

Nanning, China

Location

The First Affiliated Hospital of Nanyang Medical College

Nanyang, China

Location

Panjin Liaohe Oilfield Gem Flower Hospital

Panjin, China

Location

The First Hospital of Qiqihar

Qiqihar, China

Location

Shanghai East Hospital of Tongji University

Shanghai, China

Location

Shanghai Pudong New Area People's Hospital

Shanghai, China

Location

Shengjing Hospital of China Medical University

Shenyang, China

Location

The Sixth People's Hospital of Shenyang

Shenyang, China

Location

Shenzhen People's Hospital

Shenzhen, China

Location

The University of Hong Kong - Shenzhen Hospital

Shenzhen, China

Location

Taihe Hospital

Shiyan, China

Location

Siping City Central People's Hospital

Siping, China

Location

The First Affiliated Hospital of Suzhou University

Suzhou, China

Location

People's Hospital of Tianjin

Tianjin, China

Location

Tonghua Central Hospital

Tonghua, China

Location

The Central Hospital of Wuhan

Wuhan, China

Location

Yijishan Hospital of Wannan Medical College

Wuhu, China

Location

The First People's Hospital of Xiangtan City

Xiangtan, China

Location

The Affiliated Hospital of Xuzhou Medical University

Xuzhou, China

Location

Yanan University Affiliated Hospital

Yanan, China

Location

Yueyang People's Hospital

Yueyang, China

Location

Yuncheng Central Hospital

Yuncheng, China

Location

The Second Affiliated Hospital of Zhengzhou University

Zhengzhou, China

Location

Affiliated Hospital of Jiangsu University

Zhenjiang, China

Location

Zhumadian Central Hospital

Zhumadian, China

Location

Zhuzhou Central Hospital

Zhuzhou, China

Location

Zibo Central Hospital

Zibo, China

Location

The First People's Hospital of Zunyi

Zunyi, China

Location

MeSH Terms

Conditions

Diabetes Mellitus, Type 2

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System Diseases

Study Officials

  • Kui Liu, MD

    Shenzhen HighTide Biopharmaceutical Ltd.

    STUDY DIRECTOR

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

April 3, 2024

First Posted

April 9, 2024

Study Start

November 13, 2023

Primary Completion

December 12, 2024

Study Completion

July 30, 2025

Last Updated

November 26, 2025

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will not share

Locations