NCT05884671

Brief Summary

Rationale: To unravel the role of dopamine in gating of working memory, motivation and learning. Objective: The primary objective of this study is to isolate effects of blocking D2 receptor stimulation on gating of working memory, reinforcement learning and reward-based motivation, and their associated physiological changes (measured with fMRI and eye tracking). The secondary objective is to assess the degree to which the effects of D2 receptor action vary as a function of proxy measures of baseline dopamine levels. Study design: A double-blind placebo controlled within-subject design will be employed, in which young healthy participants are tested twice, once on placebo, and once on a low oral dose (400mg) of the D2 receptor antagonist sulpiride. This design and drug dose is commonly used in our lab without side effects (previously approved CMO protocols 2011/204, 2008/078 \& 2016/2646). Study population: Healthy human participants, 18 - 45 yr old. We will recruit 46 participants. Intervention: Participants will receive both 400 mg sulpiride and placebo, in separate sessions in a counterbalanced order. Main study parameters/endpoints: BOLD signal measured with fMRI, and behavioural performance on cognitive tasks. Nature and extent of the burden and risks associated with participation, benefit and group relatedness: Participants will attend 3 study sessions: A screening session and 2 pharmaco-fMRI sessions (sulpiride and placebo). Participants will complete a baseline battery of tasks and questionnaires, a structural MRI scan, as well as a battery of tasks both in and outside the scanner. On the day preceding each pharmaco-fMRI session, participants will have to adhere to some simple restrictions with respect to medication, alcohol and drug intake. On the day of testing participants will have to refrain from smoking and stimulant-containing drinks. Sulpiride can be administered safely without any relevant risk of serious adverse events and has been approved for clinical use in the Netherlands.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
47

participants targeted

Target at P25-P50 for not_applicable

Timeline
Completed

Started Sep 2021

Shorter than P25 for not_applicable

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 23, 2021

Completed
10 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 12, 2022

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

July 12, 2022

Completed
8 months until next milestone

First Submitted

Initial submission to the registry

March 21, 2023

Completed
2 months until next milestone

First Posted

Study publicly available on registry

June 1, 2023

Completed
Last Updated

September 21, 2023

Status Verified

September 1, 2023

Enrollment Period

10 months

First QC Date

March 21, 2023

Last Update Submit

September 19, 2023

Conditions

Outcome Measures

Primary Outcomes (14)

  • Working memory gating task: Reaction time

    Reaction time \[ms\] during selective vs. non-selective input- and output-gating to assess the ability (speed) to selectively input- and output-gate working memory representations at intervention (sulpiride) versus placebo.

    Measured at intervention day 1, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Working memory gating task: Reaction time

    Reaction time \[ms\] during selective vs. non-selective input- and output-gating to assess the ability (speed) to selectively input- and output-gate working memory representations at intervention (sulpiride) versus placebo.

    Measured at intervention day 2, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Working memory gating task: Accuracy

    Accuracy \[%\] during selective vs. non-selective input- and output-gating to assess the ability (correctness) to selectively input- and output-gate working memory representations at intervention (sulpiride) versus placebo.

    Measured at intervention day 1, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Working memory gating task: Accuracy

    Accuracy \[%\] during selective vs. non-selective input- and output-gating to assess the ability (correctness) to selectively input- and output-gate working memory representations at intervention (sulpiride) versus placebo.

    Measured at intervention day 2, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Working memory gating task: BOLD-response

    BOLD-response to selective vs. global cues, examined for both pre- and retro-cue conditions (i.e., input- and output-gating respectively) to assess the neural response to selective working memory gating at intervention (sulpiride) versus placebo.

    Measured at intervention day 1, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Working memory gating task: BOLD-response

    BOLD-response to selective vs. global cues, examined for both pre- and retro-cue conditions (i.e., input- and output-gating respectively) to assess the neural response to selective working memory gating at intervention (sulpiride) versus placebo.

    Measured at intervention day 2, 115 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Simon task: Accuracy

    Accuracy \[%\] during high and low average reward rate congruent and incongruent trials to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 1, 250 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Simon task: Accuracy

    Accuracy \[%\] during high and low average reward rate congruent and incongruent trials to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 2, 250 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Simon task: Reaction time

    Reaction time \[ms\] during high and low average reward rate congruent and incongruent trials to assess cognitive effort investment after intervention versus placebo

    Measured at intervention day 1, 250 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Simon task: Reaction time

    Reaction time \[ms\] during high and low average reward rate congruent and incongruent trials to assess cognitive effort investment after intervention versus placebo

    Measured at intervention day 2, 250 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Perceptual decision-making task: Accuracy

    Accuracy \[%\] as a function of average reward rate to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 1, 215 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Perceptual decision-making task: Accuracy

    Accuracy \[%\] as a function of average reward rate to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 2, 215 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Perceptual decision-making task: Reaction time

    Reaction time \[ms\] as a function of average reward rate to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 1, 215 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

  • Perceptual decision-making task: Reaction time

    Reaction time \[ms\] as a function of average reward rate to assess cognitive effort investment after intervention versus placebo.

    Measured at intervention day 2, 215 min after the pharmacological intervention took place. Measurements are compared regarding intervention type (drug versus placebo).

Secondary Outcomes (11)

  • Eye-blink rate

    Measured at baseline during intake session

  • Operation Span test

    Measured at baseline during intake session

  • Digit Span test

    Measured at baseline during intake session

  • Digit Span test

    Measured during intervention day 1 (sessions at least 14 days apart), 290 min after the pharmacological intervention took place

  • Digit Span test

    Measured during intervention day 2 (sessions at least 14 days apart), 290 min after the pharmacological intervention took place

  • +6 more secondary outcomes

Other Outcomes (40)

  • Diastolic blood pressure

    Measured at baseline on intervention day 1 (before pharmacological intervention took place)

  • Diastolic blood pressure

    Measured at baseline on intervention day 2 (before pharmacological intervention took place)

  • Diastolic blood pressure

    Measured 90 min post drug/placebo intake on intervention day 1

  • +37 more other outcomes

Study Arms (2)

Sulpiride

ACTIVE COMPARATOR

All study participants receive both placebo and the active medication (sulpiride 400mg), in a within-subjects , double-blind, randomized design.

Drug: Sulpiride 400 MG

Placebo

PLACEBO COMPARATOR

All study participants receive both placebo and the active medication (sulpiride 400mg), in a within-subjects , double-blind, randomized design.

Drug: Placebo

Interventions

All participants will receive one single dose of 400mg sulpiride. None of the participants will receive repeated doses. In order for the fMRI data acquisition to coincide with the time-window of maximal drug effects represented by a combination of plasma kinetics and physiological effects we will administer the drug 90 minutes prior to fMRI data acquisition.

Also known as: Dogmatil
Sulpiride

All participants will receive placebo during one of the sessions.

Placebo

Eligibility Criteria

Age18 Years - 45 Years
Sexall
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy volunteers between 18 and 45 years of age
  • Predominant right-handedness

You may not qualify if:

  • Presence of prolactin-dependent tumors (e.g., pituitary prolactinoma or breast cancer)
  • (History of) autonomic failure (e.g., vasovagal reflex syncope).
  • (History of) clinically significant hepatic, cardiac, obstructive respiratory, renal, cerebrovascular, cardiovascular, metabolic, ocular or pulmonary disease/disorders
  • (History of) epilepsy in adulthood (i.e. no insult after 18 years of age, no current medication for epilepsy and no insult in the last five years)
  • Diagnosis (or history of) endocrine treatment
  • Diagnosis (or history of) neuroendocrine treatment (e.g., phechromocytoma, hyperthyroidism, Cushing's syndrome)
  • (History of) melanoma
  • Hypersensitivity to sulpiride
  • One first degree or two or more second degree family members with a history of sudden death or ventricular arrhythmia
  • Abnormal QT interval (assessed via ECG)
  • Uncontrolled hypertension, defined as diastolic blood pressure at rest \> 95 mmHg or systolic blood pressure at rest \> 180 mmHg
  • Hypotension, defined as diastolic blood pressure \< 50 mm Hg or systolic \< 95 mm Hg
  • or resting pulse rate \< 45 beats/min
  • Diabetes
  • History of prescribed medication within the last month prior to the start of the study.
  • +26 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Donders Centre for Cognition, Radboud University

Nijmegen, Gelderland, Netherlands

Location

MeSH Terms

Interventions

Sulpiride

Intervention Hierarchy (Ancestors)

BenzamidesAmidesOrganic ChemicalsBenzoatesAcids, CarbocyclicCarboxylic AcidsBenzene DerivativesHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbons

Study Design

Study Type
interventional
Phase
not applicable
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
BASIC SCIENCE
Intervention Model
CROSSOVER
Model Details: This is a within-subjects (i.e., crossover), double-blind, randomized placebo-controlled study.
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Prof. Dr.

Study Record Dates

First Submitted

March 21, 2023

First Posted

June 1, 2023

Study Start

September 23, 2021

Primary Completion

July 12, 2022

Study Completion

July 12, 2022

Last Updated

September 21, 2023

Record last verified: 2023-09

Data Sharing

IPD Sharing
Will share

Following publication, raw and processed data will be archived for scientific integrity. The data use agreement gives access to the data, provided that certain conditions set by the local institutional guidelines as well as (inter)national (EU) law are met. Data sharing will be done using the Donders Institute research data repository (http://data.donders.ru.nl) in accordance to institutional and EU guidelines.

Shared Documents
ANALYTIC CODE
Time Frame
After publication
Access Criteria
As described on the website of the Donders Repository, shared data can be accessed via a persistent identifier. This identifier can be obtained directly from the authors or via a link in the publication. Also see: https://data.donders.ru.nl/doc/help/user-manual/access-shared-data/request-access.html?4
More information

Locations