NCT05600309

Brief Summary

The purpose of this China extension study is to assess the safety and efficacy of coformulated favezelimab/pembrolizumab (MK-4280A) in adult Chinese participants with metastatic colorectal cancer. The study will also compare MK-4280A with the standard of care treatment of regorafenib and TAS-102 (trifluridine and tipiracil). The primary study hypothesis is that coformulated favezelimab/pembrolizumab (MK-4280A) is superior to standard of care with respect to overall survival.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
94

participants targeted

Target at below P25 for phase_3 colorectal-cancer

Timeline
Completed

Started Jun 2022

Shorter than P25 for phase_3 colorectal-cancer

Geographic Reach
1 country

24 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

June 14, 2022

Completed
4 months until next milestone

First Submitted

Initial submission to the registry

October 26, 2022

Completed
5 days until next milestone

First Posted

Study publicly available on registry

October 31, 2022

Completed
1.8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 15, 2024

Completed
6 months until next milestone

Study Completion

Last participant's last visit for all outcomes

February 21, 2025

Completed
7 months until next milestone

Results Posted

Study results publicly available

September 17, 2025

Completed
Last Updated

November 26, 2025

Status Verified

November 1, 2025

Enrollment Period

2.2 years

First QC Date

October 26, 2022

Results QC Date

July 31, 2025

Last Update Submit

November 17, 2025

Conditions

Keywords

Programmed Cell Death-1 (PD1, PD-1),Programmed Cell Death Receptor Ligand 1 (PDL1, PD-L1)Programmed Cell Death Receptor Ligand 2 (PDL2, PD-L2)

Outcome Measures

Primary Outcomes (1)

  • Overall Survival (OS)

    OS was defined as the time from randomization to death due to any cause.

    Up to approximately 26 months

Secondary Outcomes (5)

  • Progression-Free Survival (PFS) According Per Response Evaluation Criteria in Solid Tumors Version 1.1 (RECIST 1.1) as Assessed by Blinded Independent Central Review (BICR)

    Up to approximately 26 months

  • Objective Response Rate (ORR) Per RECIST 1.1 as Assessed by BICR

    Up to approximately 26 months

  • Duration of Response (DOR) Per RECIST 1.1 as Assessed by BICR

    Up to approximately 26 months

  • Number of Participants Who Experienced at Least One Adverse Event (AE)

    Up to approximately 20 months

  • Number of Participants Who Discontinued Study Treatment Due to an AE

    Up to approximately 17 months

Study Arms (2)

Favezelimab/Pembrolizumab

EXPERIMENTAL

Participants will receive coformulated favezelimab/pembrolizumab (800 mg/200 mg) intravenously (IV) on Day 1, then every 3 weeks (Q3W), for up to 35 infusions.

Biological: favezelimab/pembrolizumab

Standard of Care (Regorafenib or TAS-102)

ACTIVE COMPARATOR

At the Investigator's choice, participants will receive 160 mg regorafenib orally daily on Days 1-12 of each 28-day cycle or 35 mg/m\^2 TAS-102 orally twice daily on Days 1-5 and Days 8-12 of each 28-day cycle.

Drug: regorafenibDrug: TAS-102

Interventions

Coformulated favezelimab/pembrolizumab (800 mg/200 mg), IV infusion

Also known as: MK-4280A
Favezelimab/Pembrolizumab

Oral

Also known as: STIVARGA®, REGONIX®
Standard of Care (Regorafenib or TAS-102)

Oral

Also known as: LONSURF®
Standard of Care (Regorafenib or TAS-102)

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has a histologically confirmed colorectal adenocarcinoma that is metastatic and unresectable.
  • Has measurable disease per RECIST 1.1 as assessed by the local site investigator.
  • Has been previously treated for the disease and radiographically progressed on or after or could not tolerate standard treatment.
  • Submits an archival (≤ 5 years) or newly obtained tumor tissue sample or newly obtained tumor tissue sample that has not been previously irradiated.
  • Has an Eastern Cooperative Oncology Group Performance Score (ECOG PS) of 0 to 1 within 10 days prior to first dose of study intervention.
  • Has a life expectancy of at least 3 months, based on the investigator assessment.
  • Has the ability to swallow and retain oral medication and not have any clinically significant gastrointestinal abnormalities that might alter absorption.
  • Has adequate organ function.

You may not qualify if:

  • Has previously been found to have deficient mismatch repair/microsatellite instability-high (dMMR/MSI-H) tumor status.
  • Has known active central nervous system (CNS) metastases and/or carcinomatous meningitis or leptomeningeal disease.
  • Has a history of acute or chronic pancreatitis.
  • Has neuromuscular disorders associated with an elevated creatine kinase (eg, inflammatory myopathies, muscular dystrophy, amyotrophic lateral sclerosis, spinal muscular atrophy)
  • Has clinically significant cardiovascular disease within 12 months from first dose of study intervention, including New York Heart Association Class III or IV congestive heart failure, unstable angina, myocardial infarction, cerebral vascular accident, or cardiac arrhythmia associated with hemodynamic instability.
  • Has urine protein greater than or equal to 1g/24h.
  • A woman of childbearing potential who has a positive urine/serum pregnancy test within 24/72 hours prior to the first dose of study intervention.
  • Has received prior therapy with an anti-programmed cell death 1 (PD-1), anti-programmed death ligand 1 (PD-L1), or anti-programmed cell death ligand 2 (PD-L2), anti-lymphocyte activation gene 3 (LAG-3) antibody, with a tyrosine kinase inhibitor (TKI; eg, lenvatinib) other than rapidly accelerated fibrosarcoma (RAF) inhibitors (binimetinib is permitted if combined with a RAF inhibitor), or with an agent directed to another stimulatory or coinhibitory T-cell receptor (eg, cytotoxic T-lymphocyte-associated protein 4, OX-40, cluster of differentiation \[CD\] 137).
  • Has previously received regorafenib or TAS-102.
  • Has received prior systemic anticancer therapy including investigational agents within 28 days before randomization.
  • Has received prior radiotherapy within 2 weeks of start of study intervention. Participants must have recovered from all radiation-related toxicities, not require corticosteroids, and not have had radiation pneumonitis. A 1-week washout is permitted for palliative radiation (≤2 weeks of radiotherapy) to non-CNS disease.
  • Has received a live or live-attenuated vaccine within 30 days before the first dose of study intervention.
  • Has a known additional malignancy that is progressing or has required active treatment within the past 3 years.
  • Has severe hypersensitivity (≥Grade 3) to pembrolizumab and/or any of its excipients.
  • Has an active autoimmune disease that has required systemic treatment in past 2 years.
  • +6 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (24)

The Second Affiliated Hospital of Anhui Medical University ( Site 1179)

Hefei, Anhui, 230601, China

Location

Chongqing Cancer Hospital ( Site 1151)

Chongqing, Chongqing Municipality, 400030, China

Location

Fujian Province Cancer Hospital ( Site 1178)

Fuzhou, Fujian, 350014, China

Location

Sun Yat-Sen University Cancer Center ( Site 1150)

Guangzhou, Guangdong, 510060, China

Location

Southern Medical University Nanfang Hospital ( Site 1154)

Guangzhou, Guangdong, 510515, China

Location

The Sixth Affiliated Hospital of Sun Yat-sen University ( Site 1159)

Guangzhou, Guangdong, 510655, China

Location

Guangxi Medical University Affiliated Tumor Hospital ( Site 1158)

Nanning, Guangxi, 531021, China

Location

Hainan General Hospital ( Site 1177)

Haikou, Hainan, 570311, China

Location

Wuhan Union Hospital Cancer Center ( Site 1162)

Wuhan, Hubei, 430022, China

Location

Hubei Cancer Hospital ( Site 1152)

Wuhan, Hubei, 430079, China

Location

Xiangya Hospital Central South University ( Site 1171)

Changsha, Hunan, 410008, China

Location

Hunan Cancer Hospital ( Site 1174)

Changsha, Hunan, 410013, China

Location

The Third Xiangya Hospital of Central South University ( Site 1175)

Changsha, Hunan, 410013, China

Location

Changzhou Cancer Hospital-Department of Oncology ( Site 1183)

Changzhou, Jiangsu, 213000, China

Location

Affiliated Hospital of Jiangnan University(Wuxi Fourth People's Hospital ) ( Site 1185)

Wuxi, Jiangsu, 214122, China

Location

Jilin Cancer Hospital ( Site 1163)

Changchun, Jilin, 130012, China

Location

Jinan Central Hospital ( Site 1167)

Jinan, Shandong, 250000, China

Location

Shanghai Tenth People's Hospital ( Site 1170)

Shanghai, Shanghai Municipality, 200072, China

Location

Fudan University Shanghai Cancer Center ( Site 1176)

Shanghai, Shanghai Municipality, 201321, China

Location

West China Hospital Sichuan University ( Site 1172)

Chengdu, Sichuan, 332001, China

Location

Tianjin Medical University Cancer Institute and Hospital ( Site 1161)

Tianjin, Tianjin Municipality, 300060, China

Location

Yunnan Province Cancer Hospital-Colorectal surgery ( Site 1169)

Kunming, Yunnan, 650106, China

Location

Zhejiang Cancer Hospital ( Site 1180)

Hangzhou, Zhejiang, 310005, China

Location

Sir Run Run Shaw Hospital-Medical Oncology ( Site 1173)

Hangzhou, Zhejiang, 310018, China

Location

Related Links

MeSH Terms

Conditions

Colorectal NeoplasmsParkinson Disease 4, Autosomal Dominant Lewy Body

Interventions

pembrolizumabregorafenibtrifluridine tipiracil drug combination

Condition Hierarchy (Ancestors)

Intestinal NeoplasmsGastrointestinal NeoplasmsDigestive System NeoplasmsNeoplasms by SiteNeoplasmsDigestive System DiseasesGastrointestinal DiseasesColonic DiseasesIntestinal DiseasesRectal Diseases

Results Point of Contact

Title
Senior Vice President, Global Clinical Development
Organization
Merck Sharp & Dohme LLC

Study Officials

  • Medical Director

    Merck Sharp & Dohme LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Masking Details
None (Open-label)
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 26, 2022

First Posted

October 31, 2022

Study Start

June 14, 2022

Primary Completion

August 15, 2024

Study Completion

February 21, 2025

Last Updated

November 26, 2025

Results First Posted

September 17, 2025

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will share

https://trialstransparency.msdclinicaltrials.com/pdf/ProcedureAccessClinicalTrialData.pdf

More information

Locations