NCT05422222

Brief Summary

The purpose of this study is to evaluate the pharmacokinetics, safety, tolerability and efficacy of VX-121/tezacaftor/deutivacaftor (VX-121/TEZ/D-IVA) in CF participants with at least 1 triple combination responsive (TCR) mutation in the cystic fibrosis transmembrane conductance regulator (CFTR) gene.

Trial Health

88
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
210

participants targeted

Target at P25-P50 for phase_3

Timeline
51mo left

Started Jun 2022

Longer than P75 for phase_3

Geographic Reach
10 countries

38 active sites

Status
recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress48%
Jun 2022Jun 2030

First Submitted

Initial submission to the registry

June 13, 2022

Completed
3 days until next milestone

First Posted

Study publicly available on registry

June 16, 2022

Completed
5 days until next milestone

Study Start

First participant enrolled

June 21, 2022

Completed
8 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 30, 2030

Expected
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

June 30, 2030

Last Updated

March 30, 2026

Status Verified

November 1, 2025

Enrollment Period

8 years

First QC Date

June 13, 2022

Last Update Submit

March 27, 2026

Conditions

Outcome Measures

Primary Outcomes (3)

  • Part A: Observed Pre-dose Plasma Concentration (Ctrough) of VX-121, TEZ, D-IVA, and Relevant Metabolites

    From Day 1 up to Day 22

  • Part A: Safety and Tolerability as Assessed by Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs)

    From Day 1 up to Day 50

  • Part B: Safety and Tolerability as Assessed by Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs)

    From Day 1 up to Week 28

Secondary Outcomes (19)

  • Part B: Absolute Change in Sweat Chloride (SwCl)

    From Baseline Through Week 24

  • Part B: Observed Pre-dose Plasma Concentration (Ctrough) of VX-121, TEZ, D-IVA, and Relevant Metabolites

    From Day 1 up to Week 16

  • Part B: Drug Acceptability Assessment Using Modified Facial Hedonic Scale

    At Day 1 and Week 24

  • Part B: Absolute Change in Percent Predicted Forced Expiratory Volume (ppFEV1)

    From Baseline Through Week 24

  • Part B: Number of Pulmonary Exacerbation (PEx)

    From Baseline Through Week 24

  • +14 more secondary outcomes

Study Arms (2)

Part A: VX-121/TEZ/D-IVA

EXPERIMENTAL

Participants will receive VX-121/TEZ/D-IVA in the morning.

Drug: VX-121/TEZ/D-IVA

Part B: VX-121/TEZ/D-IVA

EXPERIMENTAL

Participants will receive VX-121/TEZ/D-IVA in the morning with the dose(s) to be based on the outcome of Part A.

Drug: VX-121/TEZ/D-IVA

Interventions

Fixed-dose combination for oral administration.

Also known as: VX-121/VX-661/VX-561, VX-121/VX-661/CTP-656, VX-121/tezacaftor/deutivacaftor
Part A: VX-121/TEZ/D-IVAPart B: VX-121/TEZ/D-IVA

Eligibility Criteria

Age1 Year - 11 Years
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17)

You may qualify if:

  • Participants with stable CF and at least 1 TCR mutation (including F508del) in the CFTR gene

You may not qualify if:

  • History of solid organ, hematological transplantation, or cancer
  • Hepatic cirrhosis with portal hypertension, moderate hepatic impairment (Child Pugh Score 7 to 9), or severe hepatic impairment (Child Pugh Score 10 to 15)
  • Lung infection with organisms associated with a more rapid decline in pulmonary status

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (38)

Children's Hospital of Orange County

Orange, California, 92868, United States

COMPLETED

Stanford University Clinical and Translational Research Unit

Palo Alto, California, 94304, United States

COMPLETED

Children's Hospital of Colorado

Aurora, Colorado, 80045, United States

NOT YET RECRUITING

The Emory Clinic / Children's Healthcare of Atlanta at Egleston

Atlanta, Georgia, 30322, United States

COMPLETED

Ann & Robert H. Lurie Children's Hospital of Chicago

Chicago, Illinois, 60611, United States

COMPLETED

Riley Hospital for Children at Indiana University Health

Indianapolis, Indiana, 46202, United States

NOT YET RECRUITING

Boston Children's Hospital

Boston, Massachusetts, 02115, United States

NOT YET RECRUITING

Children's Respiratory and Critical Care Specialists, P.A., Children's Hospitals and Clinics of Minnesota

Minneapolis, Minnesota, 55404, United States

COMPLETED

The Children's Mercy Hospital

Kansas City, Missouri, 64108, United States

COMPLETED

Washington University School of Medicine / St. Louis Children's Hospital

St Louis, Missouri, 63110, United States

COMPLETED

Cohen Children's Medical Center

Lake Success, New York, 11042, United States

COMPLETED

Cincinnati Children's Hospital Medical Center

Cincinnati, Ohio, 45229, United States

COMPLETED

Rainbow Babies and Children's Hospital/University Hospitals Cleveland Medical Center

Cleveland, Ohio, 44106, United States

COMPLETED

Nationwide Children's Hospital

Columbus, Ohio, 43205, United States

COMPLETED

Oregon Health & Science University

Portland, Oregon, 97239, United States

COMPLETED

UPMC Children's Hospital of Pittsburgh

Pittsburgh, Pennsylvania, 15224, United States

COMPLETED

Texas Children's Hospital - Wallace Tower

Houston, Texas, 77030, United States

COMPLETED

Vermont Lung Center

Colchester, Vermont, 05446, United States

COMPLETED

American Family Childrens Hospital

Madison, Wisconsin, 53792, United States

COMPLETED

The Kids Research Institute Australia

Nedlands, Australia

NOT YET RECRUITING

Women's and Children's Hospital

North Adelaide, Australia

NOT YET RECRUITING

The Royal Children's Hospital

Parkville, Australia

NOT YET RECRUITING

Queensland Children's Hospital

South Brisbane, Australia

NOT YET RECRUITING

The Hospital for Sick Children

Toronto, Canada

NOT YET RECRUITING

British Columbia Children's Hospital

Vancouver, Canada

NOT YET RECRUITING

CHU Lyon - Hopital Femme Mere-Enfant

Bron, France

NOT YET RECRUITING

Hopital Necker, Enfants Malades

Paris, France

NOT YET RECRUITING

Charité - Paediatric Pulmonology Department

Berlin, Germany

NOT YET RECRUITING

Universitatsklinikum Essen

Essen, Germany

NOT YET RECRUITING

Medizinische Hochschule Hannover

Hanover, Germany

NOT YET RECRUITING

Erasmus Medical Center / Sophia Children's Hospital

Rotterdam, Netherlands

NOT YET RECRUITING

Starship Children's Hospital

Grafton, New Zealand

COMPLETED

Sahlgrenska Universitetssjukhuset

Gothenburg, Sweden

COMPLETED

Karolinska University Hospital - Pulmonology

Stockholm, Sweden

NOT YET RECRUITING

Inselspital - Universitaetsspital Bern

Bern, Switzerland

RECRUITING

Kinderspital Zurich

Zurich, Switzerland

NOT YET RECRUITING

Children and Young Adults Research Unit

Cardiff, United Kingdom

NOT YET RECRUITING

Great Ormond Street Hospital for Children

London, United Kingdom

NOT YET RECRUITING

Related Publications (1)

  • Hoppe JE, Kasi AS, Pittman JE, Jensen R, Thia LP, Robinson P, Tirakitsoontorn P, Ramsey B, Mall MA, Taylor-Cousar JL, McKone EF, Tullis E, Salinas DB, Zhu J, Chen YC, Rodriguez-Romero V, Sosnay PR, Davies G; VX21-121-105 Study Group. Vanzacaftor-tezacaftor-deutivacaftor for children aged 6-11 years with cystic fibrosis (RIDGELINE Trial VX21-121-105): an analysis from a single-arm, phase 3 trial. Lancet Respir Med. 2025 Mar;13(3):244-255. doi: 10.1016/S2213-2600(24)00407-7. Epub 2025 Jan 2.

MeSH Terms

Conditions

Cystic Fibrosis

Condition Hierarchy (Ancestors)

Pancreatic DiseasesDigestive System DiseasesLung DiseasesRespiratory Tract DiseasesGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and AbnormalitiesInfant, Newborn, Diseases

Central Study Contacts

Medical Information

CONTACT

Study Design

Study Type
interventional
Phase
phase 3
Allocation
NON RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
SEQUENTIAL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 13, 2022

First Posted

June 16, 2022

Study Start

June 21, 2022

Primary Completion (Estimated)

June 30, 2030

Study Completion (Estimated)

June 30, 2030

Last Updated

March 30, 2026

Record last verified: 2025-11

Data Sharing

IPD Sharing
Will not share

Details on Vertex data sharing criteria and process for requesting access can be found at: https://www.vrtx.com/our-science/clinical-trials-data-sharing/

Locations