NCT05291689

Brief Summary

This is an open-label, single arm, multicenter, Phase 2a study evaluating the efficacy, safety, and tolerability of MORF-057 in adult patients with Moderately to Severely Active Ulcerative Colitis (UC)

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
39

participants targeted

Target at P25-P50 for phase_2

Timeline
Completed

Started Apr 2022

Typical duration for phase_2

Geographic Reach
2 countries

17 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 10, 2022

Completed
13 days until next milestone

First Posted

Study publicly available on registry

March 23, 2022

Completed
21 days until next milestone

Study Start

First participant enrolled

April 13, 2022

Completed
1.5 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

October 18, 2023

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

November 26, 2024

Completed
3 months until next milestone

Study Completion

Last participant's last visit for all outcomes

February 19, 2025

Completed
Last Updated

March 11, 2026

Status Verified

February 1, 2026

Enrollment Period

1.5 years

First QC Date

March 10, 2022

Results QC Date

October 18, 2024

Last Update Submit

February 18, 2026

Conditions

Keywords

Ulcerative Colitis (UC)Inflammatory Bowel Disease (IBD)a4b7Moderately to severely active ulcerative colitisIntegrin

Outcome Measures

Primary Outcomes (1)

  • Main Cohort: Change From Baseline to Week 12 in the Robarts Histopathology Index (RHI) Score

    Robarts Histopathology Index (RHI) Score: the total RHI Score ranges from 0 (no disease activity) to 33 (severe disease activity)

    From baseline to 12 weeks

Secondary Outcomes (4)

  • Main Cohort: Change From Baseline to Week 12 in the Modified Mayo Clinic Score

    From baseline to 12 weeks

  • Main Cohort: Maximum Plasma Concentration (Cmax) During Multiple Doses of MORF-057

    12 weeks

  • Main Cohort: Time to Reach Cmax (Tmax) During Multiple Doses of MORF-057

    12 weeks

  • Main Cohort: Area Under the Curve (AUC) Following Multiple Doses of MORF-057

    12 weeks

Study Arms (1)

MORF-057

EXPERIMENTAL

Participants received MORF-057 100 milligrams (mg) orally twice daily for up to 78 weeks.

Drug: MORF-057

Interventions

MORF-057 is a small molecule that is designed to selectively inhibit integrin α4β7 and is administered orally.

Also known as: LY4268989
MORF-057

Eligibility Criteria

Age18 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has signs/symptoms of moderately to severely active UC for at least 3 months prior to Screening
  • Has evidence of UC extending at least 15 cm from the anal verge
  • Is bio-naïve or had an inadequate response, loss of response, or intolerance to other UC drugs
  • Agrees to abide by the study guidelines and requirements
  • Capable of giving signed informed consent

You may not qualify if:

  • Diagnosed with indeterminate colitis, microscopic colitis, ischemic colitis, radiation colitis, or Crohn's disease or has clinical findings suggestive of Crohn's disease
  • Has positive findings on a subjective neurological screening questionnaire
  • Has a concurrent, clinically significant, serious, unstable comorbidity
  • Primary non-responder to vedolizumab or other integrin inhibitors
  • Participation in any other interventional study or received any investigational therapy within 30 days
  • Previous exposure to MORF-057 and/or a known hypersensitivity to drugs with a similar mechanism to MORF-057
  • Unable to attend study visits or comply with study procedures

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (17)

Clinical Study Site

Tampa, Florida, 33609, United States

Location

Clinical Study Site

Lafayette, Louisiana, 70503, United States

Location

Clinical Study Site

Freehold, New Jersey, 07728, United States

Location

Clinical Study Site

Brooklyn, New York, 11235, United States

Location

Clinical Study Site

New York, New York, 10075, United States

Location

Clinical Study Site

Bydgoszcz, 85-794, Poland

Location

Clinical Study Site

Elblag, 82-300, Poland

Location

Clinical Study Site

Katowice, 40-748, Poland

Location

Clinical Study Site

Lodz, 90-349, Poland

Location

Clinical Study Site

Lodz, 90-752, Poland

Location

Clinical Study Site

Oświęcim, 32-600, Poland

Location

Clinical Study Site

Sopot, 81-756, Poland

Location

Clinical Study Site

Sosnowiec, 41-209, Poland

Location

Clinical Study Site

Staszów, 28-200, Poland

Location

Clinical Study Site

Tychy, 43-100, Poland

Location

Clinical Study Site

Warsaw, 00-728, Poland

Location

Clinical Study Site

Warsaw, 02-665, Poland

Location

Related Publications (1)

  • Sands BE, Schreiber S, Danese S, Kierkus J, Abhyankar B, Choi MY, Soo C, Wu Y, Sun F, Lee D, Cui D, Mangada M, Singhal P, Hussain A, Rogers BN, Peyrin-Biroulet L, Feagan BG. A Phase 2 Study of MORF-057, an Oral alpha4beta7 Integrin Inhibitor in Moderately to Severely Active Ulcerative Colitis. Clin Gastroenterol Hepatol. 2026 Feb;24(2):525-534. doi: 10.1016/j.cgh.2025.07.030. Epub 2025 Aug 6.

MeSH Terms

Conditions

Inflammatory Bowel DiseasesColitis, Ulcerative

Condition Hierarchy (Ancestors)

GastroenteritisGastrointestinal DiseasesDigestive System DiseasesIntestinal DiseasesColitisColonic Diseases

Results Point of Contact

Title
Chief Medical Officer
Organization
Eli Lilly and Company

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 10, 2022

First Posted

March 23, 2022

Study Start

April 13, 2022

Primary Completion

October 18, 2023

Study Completion

February 19, 2025

Last Updated

March 11, 2026

Results First Posted

November 26, 2024

Record last verified: 2026-02

Locations