NCT04986202

Brief Summary

This is a randomised, double-blind, placebo-controlled, multi-center sequential phase 2b and Phase 3 study to evaluate the efficacy and safety of AZD4831 administered for up to 48 Weeks in participants with heart failure with left ventricular ejection fraction \> 40%. The study will consist of 2 separate parts, Part A and Part B, approximately 660 participants will be randomised in Part A, 820 in Part B.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
711

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Jun 2021

Geographic Reach
18 countries

171 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 18, 2021

Completed
12 days until next milestone

Study Start

First participant enrolled

June 30, 2021

Completed
1 month until next milestone

First Posted

Study publicly available on registry

August 2, 2021

Completed
2.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

March 27, 2024

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

March 27, 2024

Completed
1.4 years until next milestone

Results Posted

Study results publicly available

August 27, 2025

Completed
Last Updated

August 27, 2025

Status Verified

July 1, 2025

Enrollment Period

2.7 years

First QC Date

June 18, 2021

Results QC Date

March 26, 2025

Last Update Submit

August 8, 2025

Conditions

Keywords

Heart failureHeart failure with preserved ejection fractionHFpEF

Outcome Measures

Primary Outcomes (2)

  • Kansas City Cardiomyopathy Questionnaire -Total Symptom Score

    Kansas City Cardiomyopathy Questionnaire -Total Symptom Score change from baseline at 16 weeks compared with placebo Part A. The score ranges from 0 to 100, where a higher score represents a better patient outcome

    Baseline - 16 weeks

  • Six Minute Walk Distance

    Six Minute Walk Distance change from baseline at 16 weeks compared with placebo Part A

    Baseline - 16 weeks

Secondary Outcomes (9)

  • Kansas City Cardiomyopathy Questionnaire-Total Symptom Score

    Baseline - 24 and 48 weeks

  • Six Minute Walk Distance

    Baseline - 24 and 48 weeks

  • N-terminal Pro-brain Natriuretic Peptide (NT-proBNP)

    Baseline - 16, 24 and 48 weeks

  • Left Ventricular Global Longitudinal Strain (LV-GLS)

    Baseline - 16 and 24 weeks

  • Left Atrial Volume Index (LAVI)

    Baseline - 16 and 24 weeks

  • +4 more secondary outcomes

Other Outcomes (5)

  • Adverse Events

    Baseline - 52 weeks

  • Vital Signs

    Baseline - 52 weeks

  • Clinical Laboratory (Haematology)

    Baseline - 52 weeks

  • +2 more other outcomes

Study Arms (5)

Part A 2.5 mg

EXPERIMENTAL

AZD4831 2.5 mg

Drug: AZD4831

Part A 5 mg

EXPERIMENTAL

AZD4831 5 mg

Drug: AZD4831

Part A Placebo

PLACEBO COMPARATOR

Placebo

Other: Placebo

Part B Dose based on Part A

EXPERIMENTAL

AZD4831 Dose based on Part A

Drug: AZD4831

Part B Placebo

PLACEBO COMPARATOR

Placebo

Other: Placebo

Interventions

AZD4831

Part A 2.5 mgPart A 5 mgPart B Dose based on Part A
PlaceboOTHER

Placebo

Part A PlaceboPart B Placebo

Eligibility Criteria

Age40 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Part A
  • ≥ 40 to ≤ 85 years of age, at the time of signing the informed consent.
  • Documented stable symptomatic HF (New York Heart Association Class II-IV) for at least 1 month at Screening (Visit 1) (transient HF in the setting of an MI does not qualify), with a medical history of typical symptoms of HF and receiving optimal therapy for HF as determined by the health-care physician.
  • LVEF \> 40% at Screening (Visit 1). All participants will undergo a local echocardiogram at the Screening (Visit 1) with central reading to confirm the LVEF \> 40% eligibility criteria before randomisation.
  • MWD ≥ 30 meters and ≤ 400 meters at Screening (Visit 1) and Randomisation (Visit 3). Difference in 6MWD between Screening and Randomisation must be \< 50 meters.
  • KCCQ-TSS ≤ 90 points at Screening (Visit 1) and Randomisation (Visit 3)
  • NT-proBNP ≥ 250 pg/mL (sinus rhythm) or ≥ 500 pg/mL (atrial fibrillation/flutter) at Screening (Visit 1) for patients with BMI ≤30 kg/m2.
  • NT-proBNP ≥ 200 pg/mL (sinus rhythm) or ≥ 400 pg/mL (atrial fibrillation/flutter) at Screening (Visit 1) for patients with BMI \> 30 kg/m2.
  • The ECG performed at Screening should be used for heart rhythm evaluation.
  • At least one of the following:
  • Structural heart disease, ie, LA enlargement and/or left ventricular hypertrophy at the echocardiogram performed at Screening (Visit 1). Left atrial enlargement is defined by at least 1 of the following: LA width (diameter) ≥ 3.8 cm or LA length ≥ 5.0 cm, or LA area ≥ 20 cm2 or LA volume ≥ 55 mL or LAVI \> 34 mL/m2. Left ventricular hypertrophy is defined by septal thickness or posterior wall thickness ≥ 1.1 cm or LVMI \> 95 g/m2 in women and \> 115 g/m2 in men.
  • Spectral tissue Doppler echocardiography - E/e' ratio (average of septal and lateral) ≥ 13 at rest at the echocardiogram performed at Screening (Visit 1).
  • Indirectly estimated elevation of PASP by TRmax velocity \> 2.8 m/s (280 cm/s) (PASP \> 35 mmHg) at the echocardiogram performed at Screening (Visit 1) OR directly measured pulmonary capillary wedge pressure \> 15 mmHg at rest within the past 12 months or \> 25 mmHg at exercise documented by right heart catheterisation within 12 months prior to Screening (Visit 1).
  • HF decompensation within 6 months before Randomisation (Visit 3), defined as hospitalisation for HF or IV diuretic treatment for HF during an urgent, unscheduled visit without hospitalisation.
  • Body mass index ≥ 18.0 kg/m2 and ≤ 45.0 kg/m2
  • +17 more criteria

You may not qualify if:

  • Part A
  • eGFR \< 30 mL/min/1.73m2 (Chronic Kidney Disease-Epidemiology Collaboration formula) at Screening (Visit 1).
  • \. Systolic blood pressure \< 90 mmHg or ≥ 160 mmHg if not on treatment with ≥ 3 blood pressure lowering medications or ≥ 180 mmHg irrespective of treatments at Randomisation
  • \. Heart rate \> 110 bpm or \< 50 bpm at Randomisation
  • \. Life expectancy \< 3 years due to other reasons than cardiovascular disease.
  • \. History or ongoing allergy/hypersensitivity reactions to drugs (including but not limited to rash, angioedema, acute urticaria).
  • \. Presence of any disease or condition rather than HF constituting the main reason for limiting the ability to exercise/reduced exercise capacity.
  • \. Current decompensated HF and/or NT-proBNP \> 5000 pg/mL at Screening (Visit 1)
  • \. Documented history of ejection fraction ≤ 40%.i.e. HF with recovered ejection fraction. Transient ejection fraction decrease e.g. in the setting of an MI does not apply
  • \. Any planned cardiovascular procedure (eg, coronary revascularisation, ablation of atrial fibrillation/flutter, valve repair/replacement, aortic aneurysm surgery, etc).
  • \. Any cardiac event (eg, myocardial infarction, unstable angina), coronary revascularisation (percutaneous coronary intervention or coronary artery bypass grafting), ablation of atrial fibrillation/flutter, valve repair/replacement, implantation of a cardiac resynchronisation therapy device within 12 weeks prior to Screening (Visit 1) or between Screening and Randomisation. Patients who underwent a successful atrial fibrillation/flutter cardioversion, can be enrolled in the study after 4 weeks.
  • \. Hb \< 110 g/L (male) and \< 100 g/L (female) or iron-deficiency with/without anaemia requiring ongoing or planned IV iron treatment.
  • \. Participants with hyperthyroidism, uncontrolled hypothyroidism (including but not limited to TSH ≥10 mIU/mL), or any clinically significant thyroid disease as judged by the investigator.
  • \. ALT or AST ≥ 2 × ULN at Screening (Visit 1).
  • \. Pulmonary arterial hypertension, chronic pulmonary embolism, severe pulmonary disease including COPD (ie, requiring home oxygen, chronic nebulizer therapy or chronic oral steroid therapy, or hospitalization for exacerbation of COPD requiring ventilatory support within 12 months prior to Screening (Visit 1).
  • +9 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (171)

Research Site

Alexander City, Alabama, 35010, United States

Location

Research Site

Little Rock, Arkansas, 72205, United States

Location

Research Site

Sacramento, California, 95821, United States

Location

Research Site

Miami, Florida, 33144, United States

Location

Research Site

Miami Beach, Florida, 33140, United States

Location

Research Site

Ocala, Florida, 34471, United States

Location

Research Site

Evanston, Illinois, 60208, United States

Location

Research Site

Hazel Crest, Illinois, 60429, United States

Location

Research Site

Shreveport, Louisiana, 71105, United States

Location

Research Site

Baltimore, Maryland, 21229, United States

Location

Research Site

St Louis, Missouri, 63136, United States

Location

Research Site

Buffalo, New York, 14215, United States

Location

Research Site

New York, New York, 10019, United States

Location

Research Site

Rosedale, New York, 11422, United States

Location

Research Site

Chapel Hill, North Carolina, 27599, United States

Location

Research Site

Pinehurst, North Carolina, 28374, United States

Location

Research Site

Cleveland, Ohio, 44195, United States

Location

Research Site

Philadelphia, Pennsylvania, 19107, United States

Location

Research Site

Knoxville, Tennessee, 37916, United States

Location

Research Site

Tullahoma, Tennessee, 37388, United States

Location

Research Site

Norfolk, Virginia, 23510, United States

Location

Research Site

Bedford Park, 5042, Australia

Location

Research Site

Chermside, 4032, Australia

Location

Research Site

Concord, 2139, Australia

Location

Research Site

Frankston, 3199, Australia

Location

Research Site

Aalst, 9300, Belgium

Location

Research Site

Dendermonde, 9200, Belgium

Location

Research Site

Hasselt, 3500, Belgium

Location

Research Site

Huy, 4500, Belgium

Location

Research Site

Kortrijk, 8500, Belgium

Location

Research Site

Leuven, 3000, Belgium

Location

Research Site

Roeselare, 8800, Belgium

Location

Research Site

Brasília, 72145-450, Brazil

Location

Research Site

Campina Grande do Sul, 83430000, Brazil

Location

Research Site

Campinas, 13060-080, Brazil

Location

Research Site

Campinas, 13092133, Brazil

Location

Research Site

Canoas, 92425-020, Brazil

Location

Research Site

Curitiba, 80730-150, Brazil

Location

Research Site

Porto Alegre, 90035-903, Brazil

Location

Research Site

Ribeirão Preto, 14026-020, Brazil

Location

Research Site

Ribeirão Preto, 14051-140, Brazil

Location

Research Site

Rio de Janeiro, 22061-080, Brazil

Location

Research Site

São Paulo, 01228-200, Brazil

Location

Research Site

Blagoevgrad, 2700, Bulgaria

Location

Research Site

Pleven, 5804, Bulgaria

Location

Research Site

Plovdiv, 4003, Bulgaria

Location

Research Site

Sofia, 1202, Bulgaria

Location

Research Site

Sofia, 1309, Bulgaria

Location

Research Site

Sofia, 1407, Bulgaria

Location

Research Site

Sofia, 1431, Bulgaria

Location

Research Site

Sofia, 1527, Bulgaria

Location

Research Site

Sofia, 1606, Bulgaria

Location

Research Site

Sofia, 1784, Bulgaria

Location

Research Site

Varna, 9000, Bulgaria

Location

Research Site

Guelph, Ontario, N1H 1B1, Canada

Location

Research Site

Newmarket, Ontario, L3Y 2P6, Canada

Location

Research Site

North York, Ontario, M9N 1W4, Canada

Location

Research Site

Ottawa, Ontario, K1Y 4W7, Canada

Location

Research Site

Toronto, Ontario, M6G 1M2, Canada

Location

Research Site

Waterloo, Ontario, N2T 0C1, Canada

Location

Research Site

Chicoutimi, Quebec, G7H 7K9, Canada

Location

Research Site

Trois-Rivières, Quebec, G9A 4P3, Canada

Location

Research Site

Brno, 625 00, Czechia

Location

Research Site

Broumov, 55001, Czechia

Location

Research Site

Jaroměř, 551 01, Czechia

Location

Research Site

Kolín, 280 02, Czechia

Location

Research Site

Louny, 440 01, Czechia

Location

Research Site

Pilsen, 320 00, Czechia

Location

Research Site

Prague, 110 00, Czechia

Location

Research Site

Prague, 121 11, Czechia

Location

Research Site

Příbram, 261 01, Czechia

Location

Research Site

Zlín, 760 01, Czechia

Location

Research Site

Århus N, 8200, Denmark

Location

Research Site

Copenhagen, 2300, Denmark

Location

Research Site

Copenhagen O, 2100, Denmark

Location

Research Site

Hvidovre, 2650, Denmark

Location

Research Site

København NV, 2400, Denmark

Location

Research Site

Roskilde, 4000, Denmark

Location

Research Site

Viborg, 8800, Denmark

Location

Research Site

Bayonne, 64100, France

Location

Research Site

Dijon, 21079, France

Location

Research Site

La Tronche, 38043, France

Location

Research Site

Le Coudray, 28630, France

Location

Research Site

Montauban, 82017, France

Location

Research Site

Montpellier, 34295, France

Location

Research Site

Paris, 75010, France

Location

Research Site

Paris, 75015, France

Location

Research Site

Pierre-Bénite, 69495, France

Location

Research Site

Rennes, 35033, France

Location

Research Site

Saint-Brieuc, 22027, France

Location

Research Site

Toulon, 83100, France

Location

Research Site

Toulouse, 31059, France

Location

Research Site

Tourcoing, 59208, France

Location

Research Site

Balatonfüred, 8230, Hungary

Location

Research Site

Budapest, 1096, Hungary

Location

Research Site

Budapest, 1122, Hungary

Location

Research Site

Nyíregyháza, 4400, Hungary

Location

Research Site

Fukui-shi, 910-8526, Japan

Location

Research Site

Higashiohmi-shi, 527-8505, Japan

Location

Research Site

Iwakuni-shi, 740-8510, Japan

Location

Research Site

Kanazawa, 920-8650, Japan

Location

Research Site

Kasugai-shi, 487-0016, Japan

Location

Research Site

Kishiwada-shi, 596-0042, Japan

Location

Research Site

Kure-shi, 737-0023, Japan

Location

Research Site

Kyoto, 612-8555, Japan

Location

Research Site

Matsumoto-shi, 390-8621, Japan

Location

Research Site

Minamiku, 861-4193, Japan

Location

Research Site

Nagano, 399-8695, Japan

Location

Research Site

Naha, 902-8511, Japan

Location

Research Site

Otaru-shi, 047-8510, Japan

Location

Research Site

Ōita, 870-8511, Japan

Location

Research Site

Ōmihachiman, 523-0082, Japan

Location

Research Site

Sagamihara-shi, 252-5188, Japan

Location

Research Site

Toshima-ku, 171-0014, Japan

Location

Research Site

Ueda-shi, 386-8610, Japan

Location

Research Site

Uwajima-shi, 798-8510, Japan

Location

Research Site

Yokohama, 245-8575, Japan

Location

Research Site

's-Hertogenbosch, 5223 GZ, Netherlands

Location

Research Site

Amsterdam, 1081 HV, Netherlands

Location

Research Site

Deventer, 7416 SE, Netherlands

Location

Research Site

Heerlen, 6419 PC, Netherlands

Location

Research Site

The Hague, 2545 AA, Netherlands

Location

Research Site

Bydgoszcz, 85-079, Poland

Location

Research Site

Lublin, 20-044, Poland

Location

Research Site

Rzeszów, 35-055, Poland

Location

Research Site

Skierniewice, 96-100, Poland

Location

Research Site

Tarnów, 33-100, Poland

Location

Research Site

Tczew, 83-110, Poland

Location

Research Site

Tychy, 43-100, Poland

Location

Research Site

Warsaw, 02-677, Poland

Location

Research Site

Warsaw, 02-758, Poland

Location

Research Site

Warsaw, 04-749, Poland

Location

Research Site

Wołomin, 05-200, Poland

Location

Research Site

Aramil, 624002, Russia

Location

Research Site

Kemerovo, 650002, Russia

Location

Research Site

Moscow, 119991, Russia

Location

Research Site

Moscow, 121205, Russia

Location

Research Site

Moscow, 121552, Russia

Location

Research Site

Novosibirsk, 630055, Russia

Location

Research Site

Perm, 614007, Russia

Location

Research Site

Saint Petersburg, 195067, Russia

Location

Research Site

Tver', 170036, Russia

Location

Research Site

Banská Bystrica, 974 01, Slovakia

Location

Research Site

Bratislava, 821 07, Slovakia

Location

Research Site

Brezno, 977 01, Slovakia

Location

Research Site

Košice, 04022, Slovakia

Location

Research Site

Košice, 044 24, Slovakia

Location

Research Site

Nitra, 949 01, Slovakia

Location

Research Site

Prešov, 080 01, Slovakia

Location

Research Site

Gothenburg, 413 45, Sweden

Location

Research Site

Jönköping, 551 85, Sweden

Location

Research Site

Lund, 222 21, Sweden

Location

Research Site

Norrköping, 603 79, Sweden

Location

Research Site

Örebro, 701 85, Sweden

Location

Research Site

Stockholm, 118 83, Sweden

Location

Research Site

Stockholm, 171 76, Sweden

Location

Research Site

Stockholm, 18288, Sweden

Location

Research Site

Kaohsiung City, 807, Taiwan

Location

Research Site

Kaohsiung City, 81362, Taiwan

Location

Research Site

Kaohsiung City, 833, Taiwan

Location

Research Site

Taichung, 40201, Taiwan

Location

Research Site

Taichung, 40447, Taiwan

Location

Research Site

Taichung, 40705, Taiwan

Location

Research Site

Tainan, 70403, Taiwan

Location

Research Site

Tainan, 710, Taiwan

Location

Research Site

Taipei, 100, Taiwan

Location

Research Site

Taipei, 110, Taiwan

Location

Research Site

Taipei, Taiwan

Location

Research Site

Taoyuan District, 333, Taiwan

Location

Research Site

Eskişehir, 26480, Turkey (Türkiye)

Location

Research Site

Izmir, 35340, Turkey (Türkiye)

Location

Related Publications (1)

  • Lund LH, Lam CSP, Pizzato PE, Gabrielsen A, Michaelsson E, Nelander K, Ericsson H, Holden J, Folkvaljon F, Mattsson A, Collen A, Aurell M, Whatling C, Baldus S, Drelich G, Goudev A, Merkely B, Bergh N, Shah SJ. Rationale and design of ENDEAVOR: A sequential phase 2b-3 randomized clinical trial to evaluate the effect of myeloperoxidase inhibition on symptoms and exercise capacity in heart failure with preserved or mildly reduced ejection fraction. Eur J Heart Fail. 2023 Sep;25(9):1696-1707. doi: 10.1002/ejhf.2977. Epub 2023 Aug 22.

Related Links

MeSH Terms

Conditions

Heart Failure

Interventions

AZD4831

Condition Hierarchy (Ancestors)

Heart DiseasesCardiovascular Diseases

Results Point of Contact

Title
Global Clinical Lead
Organization
AstraZeneca

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
No

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 18, 2021

First Posted

August 2, 2021

Study Start

June 30, 2021

Primary Completion

March 27, 2024

Study Completion

March 27, 2024

Last Updated

August 27, 2025

Results First Posted

August 27, 2025

Record last verified: 2025-07

Data Sharing

IPD Sharing
Will share

Qualified researchers can request access to anonymized individual patient-level data from AstraZeneca group of companies sponsored clinical trials via the request portal. All request will be evaluated as per the AZ disclosure commitment: https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure. Yes, indicates that AZ are accepting requests for IPD, but this does not mean all requests will be shared.

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
AstraZeneca will meet or exceed data availability as per the commitments made to the EFPIA Pharma Data Sharing Principles. For details of our timelines, please rerefer to our disclosure commitment at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
Access Criteria
When a request has been approved AstraZeneca will provide access to the de-identified individual patient-level data in an approved sponsored tool . Signed Data Sharing Agreement (non-negotiable contract for data accessors) must be in place before accessing requested information. Additionally, all users will need to accept the terms and conditions of the SAS MSE to gain access. For additional details, please review the Disclosure Statements at https://astrazenecagrouptrials.pharmacm.com/ST/Submission/Disclosure.
More information

Locations