NCT04643093

Brief Summary

The study is to evaluate whether the efficacy of 1PC111 is superior to pitavastatin and ezetimibe in patients with primary hypercholesterolemia or mixed dyslipidemia in the 12 week treatment period.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
390

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Aug 2020

Shorter than P25 for phase_3

Geographic Reach
3 countries

34 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

August 1, 2020

Completed
4 months until next milestone

First Submitted

Initial submission to the registry

November 22, 2020

Completed
2 days until next milestone

First Posted

Study publicly available on registry

November 24, 2020

Completed
9 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

August 19, 2021

Completed
2 months until next milestone

Study Completion

Last participant's last visit for all outcomes

October 5, 2021

Completed
Last Updated

May 18, 2022

Status Verified

May 1, 2022

Enrollment Period

1 year

First QC Date

November 22, 2020

Last Update Submit

May 17, 2022

Conditions

Keywords

Primary HypercholesterolemiaMixed Dyslipidemias

Outcome Measures

Primary Outcomes (1)

  • The efficacy of 1PC111 is superior to pitavastatin and ezetimibe in patients

    12 week treatment period

Secondary Outcomes (1)

  • The efficacy and safety profile of 1PC111 , pitavastatin and ezetimibe during the treatment period and 2 week follow up period.

    12 week treatment period

Study Arms (3)

Pitavastatin

ACTIVE COMPARATOR

Pitavastatin

Drug: Pitavastatin

Ezetimibe

ACTIVE COMPARATOR

Ezetimibe

Drug: Ezetimibe

1PC111

EXPERIMENTAL

1PC111

Drug: 1PC111

Interventions

Pitavastatin, QD

Pitavastatin

Ezetimibe, QD

Ezetimibe
1PC111DRUG

1PC111, QD

1PC111

Eligibility Criteria

Age20 Years - 80 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Primary hypercholesterolemia or mixed dyslipidemia
  • Subject meeting All of the following diagnoses at Baseline visit:
  • TG≦350 mg/dL
  • ALT and AST≦ 2.5 times of upper limit of normal (ULN) with no acute liver disease
  • Creatine kinase (CK) concentration≦2 times of UL N
  • Creatinine≦1.5 mg/dL
  • Subject who is willing and able to provide inform ed consent

You may not qualify if:

  • Female who is or intends to be pregnant or breast feeding, or has childbearing potential but without effective contraception.
  • Subject with documented HIV
  • Subject with uncontrolled hypothyroidism according to the investigator's judgment
  • Subject with unstable cardiovascular disease (CVD), including but not limited to congestive heart failure (CHF) defined as New York Heart Association class III or IV, unstable angina, unstable arrhythmia according to the investigator's judgment
  • Subject with unstable hepatic or biliary disorders, including but not limited to acute hepatitis, acute exacerbation of chronic hepatitis, liver cirrhosis, liver cancer, jaundice , and chronic hepatitis B or C under antiviral therapy
  • Subject with the following medical histories:
  • History of malignancy, exceptions made for the following malignancies: a)those determined to be cured or in remission for ≥ 5 years, b) curatively resected basal cell or squamous cell skin cancers, c) cervical cancer in situ, or resected colonic polyps
  • Acute coronary syndrome with or without cardiac catheterization within the past 9 months
  • Therapeutic cardiac catheterization (due to reasons other than acute coronary syndrome) within the past 6 months
  • Any unstable comorbidities or clinical conditions , including laboratory abnormalities which could lead to unacceptable risk to subject or confound data interpretation , per investigatiors judgment
  • Use any lipid lowering agent within 6 weeks prior to initiating the study treatment ( recheck this criterion at Day 1)
  • Use cyclosporine within 6 weeks prior to initiating the study treatment (recheck this criterion at Day 1)
  • Use any investigational product within 6 weeks prior to initiating the study treatment ( recheck this criterion at Day 1)

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (34)

Paratus Clinical Research Western Sydney

Blacktown, Australia

Location

Northern Beaches Clinical Research

Brookvale, Australia

Location

Emeritus Research

Camberwell, Australia

Location

Paratus Clinical Research Central Coast

Kanwal, Australia

Location

Southern Clinical Trials - Waitemata Ltd.

Auckland, New Zealand

Location

Southern Clinical Trials Totara

Auckland, New Zealand

Location

Southern Clinical Trials Group Ltd

Christchurch, New Zealand

Location

Lakeland Clinical Trials Waikato

Hamilton, New Zealand

Location

Southern Clinical Trials Tasman

Nelson, New Zealand

Location

Lakeland Clinical Trials Rotorua

Rotorua, New Zealand

Location

Culloden Research Ltd.

Tauranga, New Zealand

Location

Changhua Christian Hospital

Changhua, Taiwan

Location

Chiayi Christian Hospital

Chiayi City, Taiwan

Location

E-Da Hospital

Kaohsiung City, Taiwan

Location

Kaohsiung Chang Gung Memorial Hospital of the C.G.M.F.

Kaohsiung City, Taiwan

Location

Kaohsiung Medical University Hospital

Kaohsiung City, Taiwan

Location

Kaohsiung Veterans General Hospital

Kaohsiung City, Taiwan

Location

China Medical University Hospital

Taichung, Taiwan

Location

Chung Shan Medical University Hospital

Taichung, Taiwan

Location

Kuang Tien General Hospital

Taichung, Taiwan

Location

Taichung Veterans General Hospital

Taichung, Taiwan

Location

Chi Mei Medical Center

Tainan, Taiwan

Location

National Cheng Kung University Hospital

Tainan, Taiwan

Location

Tainan Municipal Hospital (Managed By Show Chwan Medical Care Corporation)

Tainan, Taiwan

Location

Cathay General Hospital

Taipei, Taiwan

Location

Cheng Hsin General Hospital

Taipei, Taiwan

Location

Far Eastern Memorial Hospital

Taipei, Taiwan

Location

National Taiwan University Hospital

Taipei, Taiwan

Location

Shin Kong Wu Ho-Su Memorial Hospital

Taipei, Taiwan

Location

Taipei Medical University Hospital

Taipei, Taiwan

Location

Taipei Veterans General Hospital

Taipei, Taiwan

Location

Tamsui Mackay Memorial Hospital

Taipei, Taiwan

Location

Tri-Service General Hospital

Taipei, Taiwan

Location

Chang Gung Medical Foundation- LinKuo Branch

Taoyuan District, Taiwan

Location

Related Publications (1)

  • Chou MT, McGirr A, Jong GP, Chao TH, Lee IT, Huang CY, Chen CP, Hsieh CH, Lu CH, Sheu WH. Effect of 1PC111, a Fixed-dose Combination of Pitavastatin and Ezetimibe, Versus Pitavastatin or Ezetimibe Monotherapy on Lipid Profiles in Patients With Hypercholesterolemia or Mixed Dyslipidemia: A Randomized, Double-blind, Multicenter, Phase III Study. Clin Ther. 2022 Oct;44(10):1272-1281. doi: 10.1016/j.clinthera.2022.08.006. Epub 2022 Aug 25.

MeSH Terms

Interventions

pitavastatinEzetimibe

Intervention Hierarchy (Ancestors)

AzetidinesAzetinesHeterocyclic Compounds, 1-RingHeterocyclic Compounds

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Masking Details
Double-Blind
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 22, 2020

First Posted

November 24, 2020

Study Start

August 1, 2020

Primary Completion

August 19, 2021

Study Completion

October 5, 2021

Last Updated

May 18, 2022

Record last verified: 2022-05

Locations