NCT04304534

Brief Summary

The purpose of this study is to try to find the best dose of the new drug BAY 2433334 to give to participants and to look at how well BAY 2433334 works on top of a dual antiplatelet therapy (acetylsalicylic acid +/- clopidogrel) in patients following a recent heart attack (myocardial infarction) that happens when a blood vessel in the heart suddenly becomes blocked. BAY 2433334, works by blocking a step of the blood clotting process in our body and thins the blood and is a so called oral FXIa inhibitor.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,601

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Jun 2020

Geographic Reach
14 countries

160 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 8, 2020

Completed
3 days until next milestone

First Posted

Study publicly available on registry

March 11, 2020

Completed
3 months until next milestone

Study Start

First participant enrolled

June 17, 2020

Completed
1.7 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 21, 2022

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

February 21, 2022

Completed
1.1 years until next milestone

Results Posted

Study results publicly available

April 5, 2023

Completed
Last Updated

April 5, 2023

Status Verified

April 1, 2023

Enrollment Period

1.7 years

First QC Date

March 8, 2020

Results QC Date

February 19, 2023

Last Update Submit

April 3, 2023

Conditions

Outcome Measures

Primary Outcomes (2)

  • Efficacy - Number of Participants With Composite of CV Death, MI, Stroke and Stent Thrombosis (ST)

    CV death included death due to stroke, MI, heart failure or cardiogenic shock, sudden death or any other death due to other cardiovascular causes. Death due to non-traumatic hemorrhage was included. Acute MI was used when there was evidence of myocardial necrosis in a clinical setting consistent with acute myocardial ischemia. Stroke was defined as an acute episode of focal or global neurological dysfunction caused by an injury of the brain, spinal cord, or retina as a result of hemorrhage or infarction. ST was defined incorporating diagnostic certainty as well as timing: "Definite" ST: The highest level of certainty. Either angiographic or pathological confirmation of stent thrombosis. "Probable" ST: Regardless of the time after the index procedure, any MI that is related to documented acute ischemia in the territory of the implanted stent without angiographic confirmation of stent thrombosis and in the absence of any other obvious cause

    From baseline up to 52 weeks

  • Safety - Number of Participants With BARC Bleeding Definition Type 2, 3 and 5

    Type 2: any overt, actionable sign of hemorrhage that doesn't fit the criteria for type 3 or 5 but meets at least one of the following criteria: 1) requires nonsurgical, med intervention by a HCP, 2) leads to hospital or rise in level of care, or 3) prompt eval. Type 3a: 1) overt bleed + Hg drop of 3 to \<5 g/dl (provided Hg drop is related to bleed); 2 any transfusion with overt bleed. Type 3b: 1) overt bleed + Hg drop ≥5 g/dL (provided Hg drop is related to bleed); 2) cardiac tamponade; 3) bleed requiring surgical intervention for control (exclude dental/nasal /skin/hemorrhoid); 4) bleed requiring IV vasoactive agents. Type 3c: 1) ICH hemorrhage (doesn't include microbleeds or HT, does include intraspinal); subcategories confirmed by autopsy or imaging or LP; 2) intraocular bleed compromising vision. Type 5: fatal bleed. Type 5a: probable fatal bleed; no autopsy or image confirmation but clinical suspicion. Type 5b: definite fatal bleed; overt bleed or autopsy or image confirmation.

    From baseline up to 52 weeks

Secondary Outcomes (8)

  • Efficacy - Number of Participants With CV Death

    From baseline up to 52 weeks

  • Efficacy - Number of Participants With MI

    From baseline up to 52 weeks

  • Efficacy - Number of Participants With Stroke

    From baseline up to 52 weeks

  • Efficacy - Number of Participants With Stent Thrombosis

    From baseline up to 52 weeks

  • Efficacy - Number of Participants With All Cause Mortality

    From baseline up to 52 weeks

  • +3 more secondary outcomes

Study Arms (4)

BAY 2433334 high dose

EXPERIMENTAL
Drug: BAY2433334

BAY 2433334 medium dose

EXPERIMENTAL
Drug: BAY2433334

BAY 2433334 low dose

EXPERIMENTAL
Drug: BAY2433334

BAY2433334 matching placebo

PLACEBO COMPARATOR
Other: BAY2433334 matching placebo

Interventions

Tablet, taken orally once a day.

BAY 2433334 high doseBAY 2433334 low doseBAY 2433334 medium dose

Tablet, taken orally once a day.

BAY2433334 matching placebo

Eligibility Criteria

Age45 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Participants must be 45 years of age or older, at the time of signing the informed consent
  • Acute myocardial infarction (excluding MI associated with PCI or CABG revascularization procedures) with:
  • clinical symptoms of acute myocardial infarction AND
  • elevated biomarkers of myocardial necrosis (creatine kinase-muscle and brain isoenzyme \[CK-MB\] or cardiac troponins) AND
  • at least one of the following risk factors need to be fulfilled:
  • Age ≥ 65 years
  • Prior MI (before the index AMI event)
  • Prior peripheral arterial disease
  • Diabetes Mellitus
  • Prior coronary artery bypass grafting (CABG) AND
  • initial angiography and revascularization procedures, either PCI or CABG, as treatment for the index event performed before randomization. (Note: a planned, staged PCI procedure can be performed after randomization)
  • Plan for dual antiplatelet therapy (ASA + P2Y12 inhibitor) after hospital discharge for the index AMI
  • Randomization during hospitalization for the index AMI event and latest within 5 days of hospital admission
  • Capable of giving signed informed consent which includes compliance with the requirements and restrictions listed in the informed consent form (ICF) and in this protocol. Written informed consent has to be signed before any study-specific procedure.

You may not qualify if:

  • Hemodynamically significant ventricular arrhythmias or cardiogenic shock at time of randomization
  • Active bleeding; known bleeding disorder, history of major bleeding (intracranial, retroperitoneal, intraocular) or clinically significant gastrointestinal bleeding within last 6 months of randomization
  • Planned use or requirement of full dose and long term anticoagulation therapy during study conduct.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (160)

Valley Clinical Trials, Inc. - Covina

Covina, California, 91723, United States

Location

Florida Premier Cardiology

Boynton Beach, Florida, 33437, United States

Location

Clearwater Cardiovascular Associates | Clearwater, FL

Clearwater, Florida, 33756, United States

Location

Cardiology Associates Research Company

Daytona Beach, Florida, 32117, United States

Location

Southwest Florida Research

Naples, Florida, 34102, United States

Location

Cardiology Partners Clinical Research Institute

Palm Beach Gardens, Florida, 33410, United States

Location

Columbus Regional Research Institute

Columbus, Georgia, 31904, United States

Location

Reid Health

Richmond, Indiana, 47374, United States

Location

Midwest Heart & Vascular Specialists

Overland Park, Kansas, 66211, United States

Location

Cardiovascular Associates Research, LLC

Covington, Louisiana, 70433, United States

Location

Southern Clinical Research, LLC

Zachary, Louisiana, 70791, United States

Location

Maryland Cardiovascular Specialists

Baltimore, Maryland, 21229, United States

Location

White Oak Medical Center

Silver Spring, Maryland, 20904, United States

Location

St. Mary's/Duluth Clinic Health System

Duluth, Minnesota, 55805, United States

Location

Logan Health Research

Kalispell, Montana, 59901, United States

Location

Methodist Physicians Clinic

Omaha, Nebraska, 68114, United States

Location

The Valley Hospital, Inc.

Ridgewood, New Jersey, 07450, United States

Location

Trinity Medical WNY

Cheektowaga, New York, 14227, United States

Location

Jefferson Heart Institute

Philadelphia, Pennsylvania, 19107, United States

Location

Cardiovascular Research of Knoxville

Powell, Tennessee, 37849, United States

Location

PharmaTex Research, LLC

Amarillo, Texas, 79109, United States

Location

North Texas Research Associates

McKinney, Texas, 75071, United States

Location

Klinikum Klagenfurt am Wörthersee

Klagenfurt, Carinthia, 9020, Austria

Location

Universitätsklinikum St. Pölten

Sankt Pölten, Lower Austria, 3100, Austria

Location

Landesklinikum Wiener Neustadt

Wiener Neustadt, Lower Austria, 2700, Austria

Location

Medizinische Universität Graz

Graz, Styria, 8036, Austria

Location

Krankenhaus St. Josef Braunau

Braunau am Inn, Upper Austria, 5280, Austria

Location

Kepler Universitätsklinikum Campus III

Linz, Upper Austria, 4021, Austria

Location

Universitätsklinikum AKH Wien

Vienna, 1090, Austria

Location

Klinik Ottakring - Wilhelminenspital

Vienna, 1160, Austria

Location

Klinik Floridsdorf - Krankenhaus Nord

Vienna, 1210, Austria

Location

OL Vrouwziekenhuis - Campus Aalst

Aalst, 9300, Belgium

Location

Imeldaziekenhuis - St-Elisabethkliniek

Bonheiden, 2820, Belgium

Location

AZ Sint-Jan Brugge-Oostende | Sint-Jan - Cardiology

Bruges, 8000, Belgium

Location

CU Saint-Luc/UZ St-Luc

Bruxelles - Brussel, 1200, Belgium

Location

Ziekenhuis Oost-Limburg

Genk, 3600, Belgium

Location

Jessa Ziekenhuis

Hasselt, 3500, Belgium

Location

UZ Leuven Gasthuisberg

Leuven, 3000, Belgium

Location

CHR de la Citadelle - Cardiology

Liège, 4000, Belgium

Location

Fakultni nemocnice Brno

Brno, 625 00, Czechia

Location

Fakultni nemocnice u sv. Anny

Brno, 656 91, Czechia

Location

Nemocnice Ceske Budejovice, a.s. Department of kardiologie

České Budějovice, 370 01, Czechia

Location

Fakultni Nemocnice Hradec Kralove

Hradec Králové, 500 05, Czechia

Location

Fakultni nemocnice Plzen - Lochotin

Pilsen, 304 60, Czechia

Location

Fakultni nemocnice Kralovske Vinohrady

Prague, 10034, Czechia

Location

Vseobecna fakultni nemocnice v Praze

Prague, 12808, Czechia

Location

Institut Klinicke a Experimentalni Mediciny

Prague, 140 21, Czechia

Location

Fakultni nemocnice v Motole

Prague, 150 06, Czechia

Location

Ustredni vojenska nemocnice Praha

Prague, 169 02, Czechia

Location

Nemocnice Slany

Slaný, 274 01, Czechia

Location

Universitätsherzzentrum Freiburg - Bad Krozingen

Bad Krozingen, Baden-Wurttemberg, 79189, Germany

Location

St. Vinzenz-Hospital

Cologne, North Rhine-Westphalia, 50733, Germany

Location

Universitätsklinikum Essen

Essen, North Rhine-Westphalia, 45147, Germany

Location

Kliniken Maria Hilf GmbH

Mönchengladbach, North Rhine-Westphalia, 41063, Germany

Location

Sana-Klinikum Remscheid GmbH

Remscheid, North Rhine-Westphalia, 42859, Germany

Location

Forschungszentrum Ruhr - KliFoCenter GmbH

Witten, North Rhine-Westphalia, 58455, Germany

Location

Universitätsmedizin der Johannes Gutenberg Universität Mainz

Mainz, Rhineland-Palatinate, 55131, Germany

Location

Krankenhaus Dresden-Friedrichstadt

Dresden, Saxony, 01067, Germany

Location

Universitätsklinikum Hamburg Eppendorf (UKE)

Hamburg, 20246, Germany

Location

Universitätsklinikum Heidelberg

Heidelberg, 69120, Germany

Location

Allami Szivkorhaz

Balatonfüred, 8230, Hungary

Location

Budai Irgalmasrendi Korhaz

Budapest, 1023, Hungary

Location

University of Semmelweis/ Semmelweis Egyetem

Budapest, 1122, Hungary

Location

Eszak-Pesti Centrumkorhaz-Honvedkorhaz

Budapest, Hungary

Location

Debreceni Egyetem Klinikai Kozpont

Debrecen, 4032, Hungary

Location

Petz Aladar Megyei Oktato Korhaz

Győr, 9023, Hungary

Location

Pandy Kalman Korhaz

Gyula, 5700, Hungary

Location

Somogy Megyei Kaposi Mor Oktato Korhaz

Kaposvár, 7400, Hungary

Location

Josa Andras Hospital

Nyíregyháza, H-4400, Hungary

Location

Jasz-Nagykun-Szolnok Megyei Hetenyi Geza Korhaz

Szolnok, 5000, Hungary

Location

Zala Megyei Szent Rafael Korhaz

Zalaegerszeg, 8900, Hungary

Location

A.O. San Pio

Benevento, Campania, 82100, Italy

Location

ASL Caserta

Caserta, Campania, 81031, Italy

Location

A.O.U. di Ferrara

Ferrara, Emilia-Romagna, 44124, Italy

Location

Asl Roma 2

Rome, Lazio, 00157, Italy

Location

IRCCS Ospedale Policlinico San Martino

Genoa, Liguria, 16132, Italy

Location

Istituto Clinico Humanitas - Humanitas Mirasole S.p.A.

Milan, Lombardy, 20089, Italy

Location

IRCCS Centro Cardiologico Monzino S.p.A

Milan, Lombardy, 20138, Italy

Location

ASST Valle Olona

Varese, Lombardy, 21047, Italy

Location

A.O. S.Croce e Carle

Cuneo, Piedmont, 12100, Italy

Location

ASL TO3 di Collegno e Pinerolo

Turin, Piedmont, 10098, Italy

Location

A.O.U. di Sassari

Sassari, Sardinia, Italy

Location

A.O.U. Ospedali Riuniti "Umberto I - G.M.Lancisi - G.Salesi"

Ancona, The Marches, 60126, Italy

Location

AUSL Toscana Sud-Est

Grosseto, Tuscany, 58100, Italy

Location

ULSS3 Serenissima

Venezia, Veneto, 30035, Italy

Location

Daido Hospital, Social Medical Corporation Kojunkai

Nagoya, Aichi-ken, 457-8511, Japan

Location

Chiba-Nishi General Hospital

Matsudo, Chiba, 270-2251, Japan

Location

Fukuoka Tokushukai Hospital

Kasuga, Fukuoka, 816-0864, Japan

Location

Kokura Memorial Hospital

Kitakyushu, Fukuoka, 802-8555, Japan

Location

Ogaki Municipal Hospital

Ōgaki, Gifu, 503-8502, Japan

Location

Hokkaido Cardiovascular Hospital

Sapporo, Hokkaido, 064-8622, Japan

Location

Hyogo Prefectural Harima-Himeji General Medical Center

Himeji, Hyōgo, 670-8560, Japan

Location

Takahashi Hospital

Kobe, Hyōgo, 654-0026, Japan

Location

Nishinomiya Watanabe Cardiovascular Center

Nishinomiya, Hyōgo, 662-0911, Japan

Location

Tsukuba Medical Center Hospital

Tsukuba, Ibaraki, 305-8558, Japan

Location

Kanagawa Cardiovascular and Respiratory Center

Yokohama, Kanagawa, 236-0051, Japan

Location

Kishiwada Tokushukai Hospital

Kishiwada, Osaka, 596-0042, Japan

Location

Shin-Kuki General Hospital

Kukichūō, Saitama, 346-8530, Japan

Location

Saitama Sekishinkai Hospital

Sayama, Saitama, 350-1305, Japan

Location

Tokyo Medical and Dental University Hospital

Bunkyo-ku, Tokyo, 113-8519, Japan

Location

Fukui Prefectural Hospital

Fukui, 910-8526, Japan

Location

Japanese Red Cross Fukuoka Hospital

Fukuoka, 815-8555, Japan

Location

Saiseikai Kumamoto Hospital

Kumamoto, 861-4193, Japan

Location

Osaka General Medical Center

Osaka, 558-8558, Japan

Location

Oita Prefectural Hospital

Ōita, 870-8511, Japan

Location

Jeroen Bosch Ziekenhuis

's-Hertogenbosch, 5223 GZ, Netherlands

Location

Noord West Ziekenhuisgroep-Medisch Centrum Alkmaar

Alkmaar, 1815 JD, Netherlands

Location

Reinier de Graaf Gasthuis

Delft, 2625 AD, Netherlands

Location

Albert Schweitzer Ziekenhuis, Dordwijk

Dordrecht, 3318 AT, Netherlands

Location

Zuyderland Medisch Centrum

Heerlen, 6419 PC, Netherlands

Location

Elkerliek Ziekenhuis, Lokatie Helmond

Helmond, 5707 HA, Netherlands

Location

Leids Universitair Medisch Centrum

Leiden, 2333 ZA, Netherlands

Location

Universitair Medisch Centrum St. Radboud

Nijmegen, 6500 HB, Netherlands

Location

Canisius Wilhelmina Ziekenhuis

Nijmegen, 6532 SZ, Netherlands

Location

Bravis Ziekenhuis

Roosendaal, 4708 AE, Netherlands

Location

Ikazia Ziekenhuis

Rotterdam, 3083 AN, Netherlands

Location

VieCuri - Medisch Centrum voor Noord-Limburg locatie Venlo

Venlo, 5912 BL, Netherlands

Location

Gelre Ziekenhuizen Zutphen

Zutphen, 7207 AE, Netherlands

Location

Isala

Zwolle, 8025 AZ, Netherlands

Location

Uniwersytecki Szpital Kliniczny w Bialymstoku

Bialystok, 15-276, Poland

Location

Szpital sw. Wincentego a Paulo

Gdynia, 81-348, Poland

Location

Samodzielny Publiczny Specjalistyczny Szpital Zachodni

Grodzisk Mazowiecki, 05-825, Poland

Location

Uniwersytecki Szpital Kliniczny w Opolu

Opole, 45-401, Poland

Location

Kliniczny Szpital Wojewodzki Nr 2 im. Sw. Jadwigi Krolowej

Rzeszów, 35-301, Poland

Location

Uniwersyteckie Centrum Kliniczne Warszawskiego UM

Warsaw, 02-097, Poland

Location

Szpital Grochowski im. dr.med. Rafala Masztaka

Warsaw, 04-073, Poland

Location

Uniwersytecki Szpital Kliniczny UM we Wroclawiu

Wroclaw, 50-556, Poland

Location

Ciutat Sanitaria i Universitaria de la Vall d'Hebron

Barcelona, 08035, Spain

Location

Hospital de la Santa Creu i de Sant Pau | Cardiología

Barcelona, 08041, Spain

Location

Hospital Universitari de Bellvitge | Bellvitge Biomedical Research Institute - Cardiology - AF, Stroke Prevention

Barcelona, 08907, Spain

Location

Hospital Universitario Virgen de las Nieves|Cardiologia

Granada, 18014, Spain

Location

Hospital Ramon y Cajal | Cardiologia

Madrid, 28034, Spain

Location

Hospital Clinico Universitario San Carlos | Cardiologia

Madrid, 28040, Spain

Location

Hospital Universitario 12 de Octubre

Madrid, 28041, Spain

Location

Hospital Clinico Universitario Virgen de la Arrixaca | Neurology Department - Stroke

Murcia, 30120, Spain

Location

Hospital Universitario Virgen de la Macarena

Seville, 41071, Spain

Location

Inst Investigacio Sanitaria Pere Virgili | Hosp Univ Joan XXIII de Tarragona - Neurology - Stroke, No-Cardioembolic-Tia

Tarragona, 43005, Spain

Location

Hospital Gral. Univ. de Valencia | Cardiologia

Valencia, 46014, Spain

Location

Hospital Universitari i Politècnic La Fe | Cardiología

Valencia, 46026, Spain

Location

Falu Lasarett

Falun, 791 82, Sweden

Location

Sahlgrenska Universitetssjukhuset

Gothenburg, 413 45, Sweden

Location

Länssjukhuset Ryhov

Jönköping, 551 85, Sweden

Location

Skånes Universitetssjukhus

Lund, 222 42, Sweden

Location

Universitetssjukhuset Örebro

Örebro, 701 85, Sweden

Location

Danderyds sjukhus

Stockholm, 182 88, Sweden

Location

Länssjukhuset Sundsvall-Härnösand

Sundsvall, 851 86, Sweden

Location

Akademiska sjukhuset Hjärtforskningsmottagningen

Uppsala, 751 85, Sweden

Location

Västmanlands Sjukhus Västerås

Västerås, 721 89, Sweden

Location

Kantonsspital Baselland - Standort Liestal

Liestal, Basel-Landschaft, 4410, Switzerland

Location

Kantonsspital Aarau

Aarau, Canton of Aargau, 5001, Switzerland

Location

Centre Hospitalier Universitaire Vaudois (CHUV)

Lausanne, Canton of Vaud, 1011, Switzerland

Location

Kantonsspital Baden

Baden, 5404, Switzerland

Location

Hôpital Cantonal Universitaire de Genève

Geneva, 1205, Switzerland

Location

Luzerner Kantonsspital

Lucerne, 6000, Switzerland

Location

Ospedale regionale di Lugano

Lugano, 6900, Switzerland

Location

Lister Hospital

Stevenage, Hertfordshire, SG1 4AB, United Kingdom

Location

Freeman Hospital

Newcastle upon Tyne, Tyne and Wear, NE7 7DN, United Kingdom

Location

Worcestershire Acute Hospital Trust

Worcester, Worcestershire, WR5 1DD, United Kingdom

Location

Imperial College London

London, W12 0HS, United Kingdom

Location

Wythenshawe Hospital

Manchester, M23 9LT, United Kingdom

Location

Related Publications (2)

  • Whiteson HZ, Frishman WH. Factor XI/XIa Inhibitors: A New Approach to Anticoagulation. Cardiol Rev. 2025 Jul-Aug 01;33(4):306-311. doi: 10.1097/CRD.0000000000000624. Epub 2023 Dec 1.

  • Rao SV, Kirsch B, Bhatt DL, Budaj A, Coppolecchia R, Eikelboom J, James SK, Jones WS, Merkely B, Keller L, Hermanides RS, Campo G, Ferreiro JL, Shibasaki T, Mundl H, Alexander JH; PACIFIC AMI Investigators. A Multicenter, Phase 2, Randomized, Placebo-Controlled, Double-Blind, Parallel-Group, Dose-Finding Trial of the Oral Factor XIa Inhibitor Asundexian to Prevent Adverse Cardiovascular Outcomes After Acute Myocardial Infarction. Circulation. 2022 Oct 18;146(16):1196-1206. doi: 10.1161/CIRCULATIONAHA.122.061612. Epub 2022 Aug 27.

Related Links

Results Point of Contact

Title
Therapeutic Area Head
Organization
Bayer AG

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 8, 2020

First Posted

March 11, 2020

Study Start

June 17, 2020

Primary Completion

February 21, 2022

Study Completion

February 21, 2022

Last Updated

April 5, 2023

Results First Posted

April 5, 2023

Record last verified: 2023-04

Locations