NCT04136171

Brief Summary

To evaluate the efficacy of eplontersen compared to placebo in participants with ATTR-CM receiving available standard of care (SoC).

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
1,438

participants targeted

Target at P75+ for phase_3

Timeline
2mo left

Started Mar 2020

Longer than P75 for phase_3

Geographic Reach
20 countries

139 active sites

Status
active not recruiting

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Progress98%
Mar 2020Aug 2026

First Submitted

Initial submission to the registry

October 21, 2019

Completed
2 days until next milestone

First Posted

Study publicly available on registry

October 23, 2019

Completed
5 months until next milestone

Study Start

First participant enrolled

March 13, 2020

Completed
6.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 1, 2026

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

August 1, 2026

Expected
Last Updated

August 8, 2025

Status Verified

August 1, 2025

Enrollment Period

6.1 years

First QC Date

October 21, 2019

Last Update Submit

August 6, 2025

Conditions

Keywords

TTRAmyloidosisCardiomyopathy

Outcome Measures

Primary Outcomes (1)

  • Composite Outcome of Cardiovascular (CV) Mortality and Recurrent CV Clinical Events up to Week 140

    Baseline up to Week 140

Secondary Outcomes (8)

  • Change From Baseline in the 6-minute Walk Test (6MWT) Distance at Week 140

    Baseline to Week 140

  • Change From Baseline in the Kansas City Cardiomyopathy Questionnaire (KCCQ) Scores at Week 140

    Baseline to Week 140

  • Recurrent CV Clinical Events up to Week 140

    Baseline up to Week 140

  • All-Cause Mortality up to Week 160

    Baseline up to Week 160

  • All-Cause Mortality up to Week 140

    Baseline up to Week 140

  • +3 more secondary outcomes

Study Arms (2)

Eplontersen

EXPERIMENTAL

Eplontersen by subcutaneous injection once every 4 weeks

Drug: Eplontersen

Placebo

PLACEBO COMPARATOR

Eplontersen-matching placebo by subcutaneous injection once every 4 weeks

Drug: Placebo

Interventions

Eplontersen by subcutaneous injection

Also known as: ION-682884, IONIS-TTR-LRx
Eplontersen

Eplontersen-matching placebo by subcutaneous injection

Placebo

Eligibility Criteria

Age18 Years - 90 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Females must be non-pregnant and non-lactating, and either surgically sterile or post-menopausal or abstinent. If engaged in sexual relations of child-bearing potential, agree to use 1 highly effective contraceptive method
  • Males must be surgically sterile or, abstinent or, if engaged in sexual relations with a woman of child-bearing potential, the participant or the participant's non-pregnant female partner must be using a highly effective contraceptive method
  • Amyloid deposits in cardiac or non-cardiac tissue confirmed by Congo Red (or equivalent) staining OR technetium scintigraphy (99mTc -3,3-diphosphono-1,2- propanodicarboxylic acid \[DPD-Tc\], 99m Tc-pyrophosphate \[PYP-Tc\], or 99m Tc-hydroxymethylene-diphosphonate \[HMDP-Tc\]) with Grade 2 or 3 cardiac uptake in the absence of abnormal light chains ratio, centrally confirmed
  • End-diastolic interventricular septum thickness of \> 12 millimeters (mm) on Screening echocardiogram
  • New York Heart Association (NYHA) class I-III

You may not qualify if:

  • Acute coronary syndrome, unstable angina, stroke, transient ischemic attack (TIA), coronary revascularization, cardiac device implantation, cardiac valve repair, or major surgery within 3 months of Screening
  • Cardiomyopathy not primarily caused by ATTR-CM, for example, cardiomyopathy due to hypertension, valvular heart disease, or ischemic heart disease
  • Monoclonal gammopathy of undetermined significance (MGUS) and/or alterations in immunoglobulin free light chain (FLC) ratio unless fat, bone marrow, or heart biopsy confirming the absence of light chain and the presence of TTR protein by mass spectrometry or immunoelectron microscopy. For participants with chronic kidney disease (CKD) and without presence of monoclonal protein in blood and urine, the acceptable FLC ratio is 0.26-2.25. Results different from that may be discussed with local hematologist, Investigator and Medical Monitor if the risks associated with the biopsy outweigh the benefits
  • Prior liver or heart transplant, and/or Left Ventricular Assist Device (LVAD) or anticipated liver transplant or LVAD within 1 year after randomization
  • Current or previous treatment with Tegsedi™ (inotersen) or Onpattro™ (patisiran) or other oligonucleotide or ribonucleic acid (RNA) therapeutic (including small interfering ribonucleic acid \[siRNA\]; does not apply to COVID-19 mitochondrial \[mRNA\] vaccinations)
  • Current treatment with diflunisal, doxycycline, with or without ursodeoxycholic acid, and/or non-dihydropyridine calcium-channel blocker (e.g., verapamil, diltiazem). Participants receiving any of these agents must respect a wash-out period of 14 days before randomization.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (142)

Mayo Clinic - Arizona

Phoenix, Arizona, 85054, United States

Location

Altman Clinical and Translational Research Institute Center for Clinical Research

La Jolla, California, 92037, United States

Location

Cedars-Sinai Medical Center

Los Angeles, California, 90048, United States

Location

University of California, San Francisco (UCSF) - Medical Center

San Francisco, California, 94143, United States

Location

Stanford Hospital

Stanford, California, 94305, United States

Location

University of Colorado Hospital - Anschutz Medical Campus

Aurora, Colorado, 80045, United States

Location

MedStar Washington Hospital Center

Washington D.C., District of Columbia, 20010, United States

Location

The George Washington Medical Faculty Associates - Foggy Bottom North Pavilion

Washington D.C., District of Columbia, 20037, United States

Location

Cleveland Clinic Florida

Weston, Florida, 33331, United States

Location

Emory Heart and Vascular Center - Emory Clifton Campus

Atlanta, Georgia, 30322, United States

Location

Piedmont Heart of Fayetteville

Fayetteville, Georgia, 30214, United States

Location

Northwestern University

Chicago, Illinois, 60611, United States

Location

The University of Chicago Medical Center

Chicago, Illinois, 60637, United States

Location

Loyola University Medical Center

Maywood, Illinois, 60153, United States

Location

Indiana University Health

Indianapolis, Indiana, 46202, United States

Location

University of Kansas Medical Center

Kansas City, Kansas, 66160, United States

Location

Louisiana State University Health Sciences Center

New Orleans, Louisiana, 70112, United States

Location

Tulane University Heart and Vascular Institute

New Orleans, Louisiana, 70112, United States

Location

Ochsner Health System

New Orleans, Louisiana, 70121, United States

Location

University of Maryland Medical Center

Baltimore, Maryland, 21201, United States

Location

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

Location

Brigham and Women's Hospital

Boston, Massachusetts, 02115, United States

Location

Boston University School of Medicine

Boston, Massachusetts, 02118, United States

Location

Henry Ford Health System

Detroit, Michigan, 48202, United States

Location

Minneapolis Heart Institute

Minneapolis, Minnesota, 55407, United States

Location

Mayo Clinic - Rochester

Rochester, Minnesota, 55905, United States

Location

Saint Luke's Hospital of Kansas City

Kansas City, Missouri, 64111, United States

Location

Barnes-Jewish Hospital

St Louis, Missouri, 63110, United States

Location

New York University Langone Cardiology Associates

New York, New York, 10016, United States

Location

Columbia University Irving Medical Center

New York, New York, 10034, United States

Location

Weill Cornell Medicine Cardiology

New York, New York, 10065, United States

Location

Laurelton Heart Specialists

Rosedale, New York, 11422, United States

Location

The University of North Carolina at Chapel Hill

Chapel Hill, North Carolina, 27599, United States

Location

Duke University Medical Center

Durham, North Carolina, 27710, United States

Location

Carl and Edyth Lindner Research Center at The Christ Hospital

Cincinnati, Ohio, 45219, United States

Location

University Hospitals Cleveland Medical Center

Cleveland, Ohio, 44106, United States

Location

Cleveland Clinic Main Campus

Cleveland, Ohio, 44195, United States

Location

The Ohio State University College of Medicine

Columbus, Ohio, 43210, United States

Location

Oregon Health and Science University

Portland, Oregon, 97239, United States

Location

Lancaster General Hospital

Lancaster, Pennsylvania, 17602, United States

Location

Penn Presbyterian Medical Center

Philadelphia, Pennsylvania, 19104, United States

Location

University of Pittsburgh Medical School

Pittsburgh, Pennsylvania, 15261, United States

Location

Medical University of South Carolina

Charleston, South Carolina, 29425, United States

Location

Vanderbilt University Medical Center

Nashville, Tennessee, 37232, United States

Location

University of Texas Southwestern Medical Center

Dallas, Texas, 75390, United States

Location

Houston Methodist Hospital

Houston, Texas, 77030, United States

Location

University of Utah

Salt Lake City, Utah, 84112, United States

Location

Virginia Commonwealth University (VCU)

Richmond, Virginia, 23298, United States

Location

University of Washington

Seattle, Washington, 98195, United States

Location

University of Wisconsin - Madison

Madison, Wisconsin, 53792, United States

Location

Froedtert & Medical College of Wisconsin

Milwaukee, Wisconsin, 53226, United States

Location

Instituto Cardiovascular de Buenos Aires

Ciudad Autonoma de Buenos Aires, Buenos Aires, C1428ART, Argentina

Location

Hospital Italiano de Buenos Aires

Ciudad Autónoma de Buenos Aires, Buenos Aires, C1199ABB, Argentina

Location

Liverpool Hospital

Liverpool, New South Wales, 2170, Australia

Location

The Westmead Institute for Medical Research

Westmead, New South Wales, NSW 2145, Australia

Location

Princess Alexandra Hospital

Woolloongabba, Queensland, 4102, Australia

Location

Advara Heartcare

Leabrook, South Australia, 5068, Australia

Location

Royal Hobart Hospital

Hobart, Tasmania, 7000, Australia

Location

Box Hill Hospital

Box Hill, Victoria, 3128, Australia

Location

Advara HeartCare

Joondalup, Western Australia, 6027, Australia

Location

Advara HeartCare Murdoch

Murdoch, Western Australia, 6150, Australia

Location

Medizinische Universität Graz

Graz, Styria, 8036, Austria

Location

Medizinische Universität Innsbruck

Innsbruck, Tyrol, 6020, Austria

Location

Medizinische Universität Wien

Vienna, 1090, Austria

Location

Ziekenhuis Oost-Limburg - Campus Sint-Jan

Genk, Limburg, 3600, Belgium

Location

Algemeen Ziekenhuis Sint-Jan Brugge-Oostende - Campus Sint-Jan

Bruges, West-Vlaanderen, 8000, Belgium

Location

Universidade Estadual de Campinas

Campinas, 13083881, Brazil

Location

Hospital Moinhos de Vento

Porto Alegre, 90560-030, Brazil

Location

Centro Avançado de Pesquisa e Estudos para o Diagnóstico CAPED

Ribeirão Preto, 14026-900, Brazil

Location

Hospital das Clínicas da Faculdade de Medicina de Ribeirão Preto

Ribeirão Preto, 14040-030, Brazil

Location

A Beneficência Portuguesa de São Paulo - Unidade Mirante

São Paulo, 01323-030, Brazil

Location

Instituto Dante Pazzanese de Cardiologia

São Paulo, 04012-909, Brazil

Location

Instituto do Coração de São Paulo

São Paulo, 05403-000, Brazil

Location

University of Calgary

Calgary, Alberta, T2N 4Z6, Canada

Location

Gordon and Leslie Diamond Health Care Centre

Vancouver, British Columbia, V5Z 1M9, Canada

Location

University Hospital - London Health Sciences Centre

London, Ontario, N6A 5A5, Canada

Location

Toronto General Hospital

Toronto, Ontario, M5G 2M9, Canada

Location

Centre Hospitalier de l'Université de Montréal (CHUM)

Montreal, Quebec, H2X 0C1, Canada

Location

Hôpital Regional de Rimouski

Rimouski, Quebec, G5L 5T1, Canada

Location

Fakultní Nemocnice u sv. Anny v Brn

Brno, South Moravian, 656 91, Czechia

Location

Vseobecna Fakultni Nemocnice v Praze

Prague, 128 08, Czechia

Location

Institut Klinické a Experimentální Medicíny

Prague, 140 21, Czechia

Location

Rigshospitalet

Copenhagen, Capital Region, 2100, Denmark

Location

Odense Universitetshospital

Odense, Region Syddanmark, 5000, Denmark

Location

Hôpital Rangueil

Toulouse, Occitanie, 31059, France

Location

Hôpitaux Universitaires Henri Mondor

Créteil, 94010, France

Location

Centre Hospitalier Départemental Vendée

La Roche-sur-Yon, 85925, France

Location

Hôpital de la Timone

Marseille, 13005, France

Location

Hôpital Haut-Lévêque

Pessac, 33604, France

Location

Centre Hospitalier Universitaire De Nantes - Hôpital Nord Laennec

Saint-Herblain, 44805, France

Location

Universitätsklinikum des Saarlandes

Homburg, Saarland, 66421, Germany

Location

Charité Campus Mitte

Berlin, 10117, Germany

Location

Charité Universitätsmedizin Berlin

Berlin, 13353, Germany

Location

Uniklinik Koln

Cologne, 50937, Germany

Location

Universitaetsklinikum Heidelberg - Zentrum fur Innere Medizin

Heidelberg, 69120, Germany

Location

Universitätsklinikum Münster

Münster, 48149, Germany

Location

Universitätsklinikum Würzburg

Würzburg, 97078, Germany

Location

Alexandra General Hospital

Athens, 11528, Greece

Location

Rambam Health Care Campus

Haifa, 3109601, Israel

Location

Hadassah University Hospital Ein Kerem

Jerusalem, 9112001, Israel

Location

Kaplan Medical Center

Rehovot, Israel

Location

Azienda Ospedaliero Universitaria Delle Marche

Ancona, 60126, Italy

Location

Azienda Ospedaliero-Universitaria di Bologna Policlinico Sant Orsola-Malpighi

Bologna, 40138, Italy

Location

Azienda Ospedaliero - Universitaria Careggi

Florence, 50139, Italy

Location

Azienda Ospedale - Università di Padova

Padua, 35128, Italy

Location

Fondazione IRCCS Policlinico San Matteo

Pavia, 27100, Italy

Location

Fondazione Toscana Gabriele Monasterio per la Ricerca Medica e di Sanita Pubblica

Pisa, 56126, Italy

Location

Azienda Ospedaliera - Universitaria Sant' Andrea

Roma, 00189, Italy

Location

Uwajima City Hospital

Uwajima-shi, Ehime, 798-8510, Japan

Location

Hospital of the University of Occupational and Environmental Health

Kitakyushu-shi, Fukuoka, 807-8555, Japan

Location

Kurume University Hospital

Kurume-shi, Fukuoka, 830-0011, Japan

Location

Sapporo Medical University Hospital

Sapporo, Hokkaido, 060-8543, Japan

Location

Saiseikai Fukuoka General Hospital

Fukuoka, Hukuoka, 810-0001, Japan

Location

Kokura Memorial Hospital

Kitakyushu, Hukuoka, 802-8555, Japan

Location

University Hospital Kyoto Prefectural University of Medicine

Kyoto, Kyoto, 602-8566, Japan

Location

Shinshu University Hospital

Matsumoto, Nagano, 390-8621, Japan

Location

Okayama University Hospital

Okayama, Okayama-ken, 700-8558, Japan

Location

Osaka Metropolitan University Hospital

Osaka, Osaka, 545-8586, Japan

Location

Hamamatsu University Hospital

Hamamatsu, Shizuoka, 431-3192, Japan

Location

Keio University Hospital

Shinjuku-Ku, Tokyo, 160-8582, Japan

Location

Kumamoto University Hospital

Kumamoto, 860-8556, Japan

Location

Krakowski Szpital Specjalistyczny im. Jana Pawa II

Krakow, 31-202, Poland

Location

Narodowy Instytut Kardiologii Stefana kardyna Wyszyskiego - Pastwowy Instytut Badawczy

Warsaw, 04-628, Poland

Location

Hospital da Senhora da Oliveira - Guimarães

Guimarães, 4835-044, Portugal

Location

Centro Hospitalar Universitário de Lisboa Central - Hospital de Santa Marta

Lisbon, 1169-024, Portugal

Location

Centro Hospitalar Universitário do Porto - Hospital Geral de Santo Antonio

Porto, 4099-001, Portugal

Location

Centro Hospitalar Universitário de São João

Porto, 4200-319, Portugal

Location

Veterans Affairs Caribbean Healthcare System

San Juan, 00921, Puerto Rico

Location

Hospital Universitari Vall d'Hebrón

Barcelona, 08035, Spain

Location

Hospital Universitario Puerta de Hierro - Majadahonda

Majadahonda, 28222, Spain

Location

Hospital Clínico Universitario Virgen de la Arrixaca

Murcia, 30120, Spain

Location

Complejo Hospitalario Universitario de Santiago

Santiago de Compostela, 15706, Spain

Location

Sahlgrenska Universitetssjukhuset

Gothenburg, 413 45, Sweden

Location

Skellefteå lasarett

Skellefteå, 931 86, Sweden

Location

Synexus - Scotland Clinical Research Centre

Glasgow, Scotland, G20 0SP, United Kingdom

Location

Synexus - Wales

Cardiff, Wales, CF15 9SS, United Kingdom

Location

Synexus Midlands Clinical Research Centre

Edgbaston, B15 2SQ, United Kingdom

Location

Synexus - North Tees Clinical Research Centre

Hexham, TS19 8PE, United Kingdom

Location

Synexus - Manchester Clinical Research Centre

Liverpool, L22 0LG, United Kingdom

Location

Synexus - Merseyside Clinical Research Centre

Liverpool, L22 0LG, United Kingdom

Location

Royal Free London NHS Foundation Trust

London, HR3M+6R, United Kingdom

Location

Richmond Pharmacology

London, SE1 1YR, United Kingdom

Location

MeSH Terms

Conditions

AmyloidosisCardiomyopathies

Interventions

eplontersen

Condition Hierarchy (Ancestors)

Proteostasis DeficienciesMetabolic DiseasesNutritional and Metabolic DiseasesHeart DiseasesCardiovascular Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, INVESTIGATOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 21, 2019

First Posted

October 23, 2019

Study Start

March 13, 2020

Primary Completion

April 1, 2026

Study Completion (Estimated)

August 1, 2026

Last Updated

August 8, 2025

Record last verified: 2025-08

Data Sharing

IPD Sharing
Will share

Ionis may share anonymized individual participant data, aggregated clinical data, and other types of data that support the results in this study. Data requests from qualified researchers will be considered once all three of the following criteria are met: (1) 12 months from marketing approval of the study drug in both the United States and European Union; (2) 18 months from conclusion of the study; and (3) 6 months from publication of study article. Access would be via a secure environment and is contingent upon approval of a research proposal and entry into an appropriate data use agreement. Requests to access data can be submitted via the website https://vivli.org/ourmember/ionis/.

Locations