NCT03312907

Brief Summary

The purpose of this study is to assess whether co-administration of belimumab and a single cycle of rituximab will optimize treatment with belimumab, which will result in improvements of clinical status with a favorable safety profile, by comparing subjects randomized to belimumab plus rituximab versus belimumab plus rituximab-placebo. Approximately 292 subjects will be randomized in a 1:2:1 ratio to 1 of 3 treatment arms; belimumab plus rituximab-placebo (Arm A, control), belimumab plus rituximab (Arm B, combination), or belimumab plus standard therapy (Arm C, reference). Belimumab will be administered as subcutaneous (SC) and rituximab-placebo or rituximab will be administered by intravenous (IV) infusions. The total duration of the study is for 104 weeks.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
292

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Mar 2018

Typical duration for phase_3

Geographic Reach
11 countries

79 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 13, 2017

Completed
5 days until next milestone

First Posted

Study publicly available on registry

October 18, 2017

Completed
4 months until next milestone

Study Start

First participant enrolled

March 1, 2018

Completed
2.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 29, 2020

Completed
1.1 years until next milestone

Study Completion

Last participant's last visit for all outcomes

July 7, 2021

Completed
10 months until next milestone

Results Posted

Study results publicly available

April 25, 2022

Completed
Last Updated

February 18, 2025

Status Verified

January 1, 2025

Enrollment Period

2.2 years

First QC Date

October 13, 2017

Results QC Date

March 25, 2022

Last Update Submit

January 27, 2025

Conditions

Keywords

immunosuppressantsSystemic Lupus Erythematosus Disease Activity IndexBelimumabLupus Low Disease Activity StateSystemic Lupus Erythematosus

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants With a State of Disease Control at Week 52

    Percentage of participants with a state of disease control (Independent blinded assessor \[IBA\]) was defined as the percentage of participants with a Systemic Lupus Erythematosus Disease Activity Index 2000(SLEDAI-2K)score less than or equal to(\<=)2 achieved without immunosuppressants and with corticosteroids at a prednisone equivalent dose of \<=5 mg/day at Week 52. SLEDAI-2K was a weighted, cumulative index for measuring systemic lupus erythematosus (SLE) disease activity in previous 10 days,consisting 24 individual items in which signs and symptoms, laboratory tests and physician's assessment for each item within each of 9 organ systems were given a weighted score(1 to 8 with higher score indicating increased activity)and summed if present at the time of visit or in preceding 10 days. The SLEDAI-2K score was sum of all 24 individual items from the SLEDAI-2K, ranges from 0(no symptoms) to 105(presence of all defined symptoms) with higher scores representing increased disease activity.

    Week 52

Secondary Outcomes (27)

  • Percentage of Participants With a State of Clinical Remission at Week 64

    Week 64

  • Percentage of Participants With a State of Disease Control at Week 104

    Week 104

  • Percentage of Participants With a State of Disease Control by Visits

    Weeks 12, 26, 40, 52, 64, 80 and 104

  • Percentage of Participants With a State of Clinical Remission by Visits

    Weeks 64, 80 and 104

  • Percentage of Participants With a State of Complete Remission (CR) Sustained for at Least 24 Weeks During Week 52 to Week 104

    Week 52 to Week 104

  • +22 more secondary outcomes

Study Arms (3)

Belimumab + Placebo

PLACEBO COMPARATOR

Eligible subjects will receive Belimumab 200 milligrams (mg) to be administered subcutaneously (SC) on Day 1 and then weekly (i.e., every 7 days) through Week 52. Subjects will also receive rituximab-placebo to be administered by intravenous (IV) infusions at Weeks 4 and 6 in double blind manner. Subjects will receive standard therapy excluding Immunosuppressants and including anti-malarials, non-steroidal anti-inflammatory drugs (NSAIDs), and/or corticosteroids tapered down to prednisone equivalent of less than or equal to (\<=) 5 mg/day until Week 104. Subjects will not receive treatment after 52 weeks and will be in observation until Week 104.

Drug: BelimumabDrug: Rituximab-placeboDrug: Standard therapy (Excluding Immunosuppressants)Drug: Steroid Taper

Belimumab + Rituximab

EXPERIMENTAL

Eligible subjects will receive Belimumab 200 mg to be administered SC on Day 1 and then weekly (i.e., every 7 days) through Week 52. Subjects will also receive rituximab 1000 mg to be administered by IV infusions at Weeks 4 and 6 in double blind manner. Subjects will receive standard therapy excluding Immunosuppressants and including anti-malarials, NSAIDs, and/or corticosteroids tapered down to prednisone equivalent of \<= 5 mg/day until Week 104. Subjects will not receive treatment after 52 weeks and will be in observation until Week 104.

Drug: BelimumabDrug: RituximabDrug: Standard therapy (Excluding Immunosuppressants)Drug: Steroid Taper

Belimumab + Standard therapy

OTHER

Eligible subjects will receive open-label Belimumab 200 mg administered SC on Day 1 and then weekly (i.e., every 7 days) until Week 104. Subjects will also receive standard therapy including immunosuppressant, anti-malarials, NSAIDs, and/or corticosteroids tapered down to prednisone equivalent of \<= 5 mg/day until Week 104.

Drug: BelimumabDrug: Standard therapy (Including Immunosuppressants)Drug: Steroid Taper

Interventions

Belimumab will be administered as SC injection once weekly via autoinjector in thigh or abdomen

Belimumab + PlaceboBelimumab + RituximabBelimumab + Standard therapy

Rituximab will be administered as IV infusion of 1000mg at Week 4 and Week 6

Belimumab + Rituximab

Saline will be administered as IV infusions at Week 4 and Week 6

Belimumab + Placebo

Standard therapy will contain stable SLE medications including immunosuppressant to be administered from baseline through Week 104.

Belimumab + Standard therapy

Standard therapy excluding Immunosuppressant will contain anti-malarials, NSAIDs, and/or corticosteroids with prednisone dose equivalent to \<= 5 mg/day will administered through Week 104.

Belimumab + PlaceboBelimumab + Rituximab

Steroid taper will include prednisone doses equivalent to =\< 5 mg/day in all Arms through Week 104.

Belimumab + PlaceboBelimumab + RituximabBelimumab + Standard therapy

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Subjects must be \>=18 years of age at the time of signing the informed consent.
  • Subjects who have clinical diagnosis of SLE based on 4 or more of the 11 American College of Rheumatology (ACR) criteria.
  • Subjects who have a screening SLEDAI-2K score \>=6 (This refers to the total score. Serological activity, i.e., anti-double stranded deoxyribonucleic acid \[dsDNA\]) positivity and/or hypocomplementemia is not required to be present in SLEDAI-2K assessment, but are scored if present).
  • Subjects who have unequivocally positive autoantibody test results defined as an anti-nuclear (ANA) titer \>=1:80 and/or a positive anti-dsDNA (\>=30 International Units per milliliter \[IU/mL\]) serum antibody test from 2 independent time points as follows: Positive test results from 2 independent time points within the study screening period. Screening results must be based on the study's central laboratory results. Or, one positive historical test result and 1 positive test result during the screening period.
  • Subjects who are on a stable SLE treatment regimen consisting of any of these medications (alone or in combination) for a period of at least 30 days prior to Day 1 (i.e. day of first dose of study treatment) with the exception that switching one agent for another of the same class for tolerability or availability reasons, which will be allowed within 30 days of Day 1: Corticosteroids (prednisone or prednisone equivalent); For those subjects on alternating daily doses of steroids, use the average of 2 daily doses to calculate the average daily steroid dose; Any immunosuppressant or immunomodulatory agents including methotrexate, azathioprine, leflunomide, mycophenolate (including mycophenolate mofetil, mycophenolate mofetil hydrochloride, and mycophenolate sodium), calcineurin inhibitors (example \[e.g.\] tacrolimus, cyclosporine), sirolimus, oral cyclophosphamide, 6-mercaptopurine, mizoribine, or thalidomide; Anti-malarials (e.g., hydroxychloroquine, chloroquine, quinacrine); Non steroidal anti-inflammatory drugs (NSAIDs).
  • Male and/or female. A female subject is eligible to participate if she is not pregnant not breastfeeding, and at least one of the these conditions applies: Not a woman of childbearing potential (WOCBP) or A WOCBP who agrees to follow the contraceptive guidance during the treatment period and for at least 16 weeks after the last dose of belimumab, or at least 12 months after the last dose of rituximab or rituximab-placebo.
  • Capable of giving signed informed consent which includes compliance with the requirements and restrictions listed in the informed consent form (ICF) and in this protocol.

You may not qualify if:

  • Symptomatic herpes zoster within 3 months prior to screening.
  • Evidence of active or latent tuberculosis (TB). Documentation may include medical history and examination, chest X-rays (posterior, anterior, and lateral), and TB testing: either a positive tuberculin skin test (TST; defined as a skin induration ≥5 mm at 48 to 72 hours, regardless of Baccillus Calmette-Guerin (BCG) or other vaccination history) or a positive (not indeterminate) QuantiFERON-TB Gold Plus test.
  • Significant allergies to humanized monoclonal antibodies.
  • History of hypersensitivity to belimumab and/or rituximab or known to have titers of human anti-mouse antibody or history of hypersensitivity reactions when treated with other diagnostic or therapeutic monoclonal antibodies.
  • Lymphoma, leukemia, or any malignancy within the past 5 years (yrs) except for basal cell or squamous epithelial carcinomas of the skin that have been resected with no evidence of metastatic disease for 3 yrs.
  • Alanine transferase (ALT) greater than 2 times upper limit of normal (ULN).
  • Bilirubin greater than 1.5 times ULN (isolated bilirubin greater than 1.5 times ULN is acceptable if bilirubin is fractionated and direct bilirubin less than 35%).
  • Immunoglobulin A (IgA) deficiency (IgA level less than 10 milligram per deciliter \[mg/dL\]).
  • Immunoglobulin G (IgG) less than 250 mg/dL. For Germany only, IgG less than 400mg/dL.
  • Neutrophils less than 1.5 times 10\^9.
  • Current unstable liver or biliary disease per investigator assessment defined by the presence of ascites, encephalopathy, coagulopathy, hypoalbuminemia, esophageal or gastric varices, persistent jaundice, or cirrhosis.
  • Severe heart failure (New York Heart Association Class IV) or other severe, uncontrolled cardiac disease.
  • QT interval corrected (QTc) greater than 450 millisecond (msec) or QTc greater than 480 msec in subjects with bundle branch block.
  • Subjects who have a history of a major organ transplant (e.g., heart, lung, kidney, liver) or hematopoietic stem cell/marrow transplant.
  • Subjects who have clinical evidence of significant unstable or uncontrolled acute or chronic diseases not due to SLE (i.e., cardiovascular, pulmonary, hematologic, gastrointestinal, hepatic, renal, neurological, psychiatric, malignancy, or infectious diseases) which, in the opinion of the principal investigator, could confound the results of the study or put the subject at undue risk.
  • +17 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (79)

GSK Investigational Site

Birmingham, Alabama, 35294, United States

Location

GSK Investigational Site

La Mesa, California, 92020, United States

Location

GSK Investigational Site

San Leandro, California, 94578, United States

Location

GSK Investigational Site

Upland, California, 91786, United States

Location

GSK Investigational Site

Denver, Colorado, 80230, United States

Location

GSK Investigational Site

Aventura, Florida, 33180, United States

Location

GSK Investigational Site

Miami, Florida, 33136, United States

Location

GSK Investigational Site

Orlando, Florida, 32806-6264, United States

Location

GSK Investigational Site

Tamarac, Florida, 33321, United States

Location

GSK Investigational Site

Tampa, Florida, 33613, United States

Location

GSK Investigational Site

Tampa, Florida, 33614, United States

Location

GSK Investigational Site

Ann Arbor, Michigan, 48109-5542, United States

Location

GSK Investigational Site

Brighton, Michigan, 48116, United States

Location

GSK Investigational Site

Lansing, Michigan, 48910, United States

Location

GSK Investigational Site

Lansing, Michigan, 48917, United States

Location

GSK Investigational Site

Las Cruces, New Mexico, 88011, United States

Location

GSK Investigational Site

Manhasset, New York, 11030, United States

Location

GSK Investigational Site

New York, New York, 10016, United States

Location

GSK Investigational Site

New York, New York, 10032, United States

Location

GSK Investigational Site

Charlotte, North Carolina, 28204, United States

Location

GSK Investigational Site

Vandalia, Ohio, 45377, United States

Location

GSK Investigational Site

Oklahoma City, Oklahoma, 73102, United States

Location

GSK Investigational Site

Pittsburgh, Pennsylvania, 15224, United States

Location

GSK Investigational Site

Summerville, South Carolina, 29486, United States

Location

GSK Investigational Site

Austin, Texas, 78731, United States

Location

GSK Investigational Site

League City, Texas, 77573, United States

Location

GSK Investigational Site

Spokane, Washington, 99204, United States

Location

GSK Investigational Site

Glendale, Wisconsin, 53217, United States

Location

GSK Investigational Site

Ciudad Autonoma de Buenos Aires, Buenos Aires, C1046AAQ, Argentina

Location

GSK Investigational Site

La Plata, Buenos Aires, B1904CFH,, Argentina

Location

GSK Investigational Site

San Miguel de TucumĂ¡n, TucumĂ¡n Province, T4000AXL, Argentina

Location

GSK Investigational Site

Salvador, Estado de Bahia, 40.150-150, Brazil

Location

GSK Investigational Site

CuiabĂ¡, Mato Grosso, 78043-142, Brazil

Location

GSK Investigational Site

Juiz de Fora, Minas Gerais, 36010-570, Brazil

Location

GSK Investigational Site

SĂ£o JosĂ© do Rio Preto, SĂ£o Paulo, 15090-000, Brazil

Location

GSK Investigational Site

Hamilton, Ontario, L8S 4K1, Canada

Location

GSK Investigational Site

Toronto, Ontario, M5T 2S8, Canada

Location

GSK Investigational Site

Trois-Rivières, Quebec, G8Z 1Y2, Canada

Location

GSK Investigational Site

Saskatoon, Saskatchewan, S7K 0H6, Canada

Location

GSK Investigational Site

Brest, 29609, France

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GSK Investigational Site

Lille, 59037, France

Location

GSK Investigational Site

Paris, 75013, France

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GSK Investigational Site

Paris, 75571, France

Location

GSK Investigational Site

Pessac, 33604, France

Location

GSK Investigational Site

Strasbourg, 67091, France

Location

GSK Investigational Site

Hanover, Lower Saxony, 30625, Germany

Location

GSK Investigational Site

Kiel, Schleswig-Holstein, 24105, Germany

Location

GSK Investigational Site

Frankfurt, 60590, Germany

Location

GSK Investigational Site

Zapopan, Jalisco, 45070, Mexico

Location

GSK Investigational Site

MĂ©rida, YucatĂ¡n, 97070, Mexico

Location

GSK Investigational Site

Amersfoort, 3813 TZ, Netherlands

Location

GSK Investigational Site

Groningen, 9713 GZ, Netherlands

Location

GSK Investigational Site

Leiden, 2333 ZA, Netherlands

Location

GSK Investigational Site

The Hague, 2545 AA, Netherlands

Location

GSK Investigational Site

Utrecht, 3584 CX, Netherlands

Location

GSK Investigational Site

Chelyabinsk, 454076, Russia

Location

GSK Investigational Site

Kazan', 420097, Russia

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GSK Investigational Site

Kemerovo, 650066, Russia

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GSK Investigational Site

Moscow, 119435, Russia

Location

GSK Investigational Site

Novosibirsk, 630117, Russia

Location

GSK Investigational Site

Omsk, 644111, Russia

Location

GSK Investigational Site

Petrozavodsk, 185019, Russia

Location

GSK Investigational Site

Ryazan, 390026, Russia

Location

GSK Investigational Site

Saint Petersburg, 190068, Russia

Location

GSK Investigational Site

Ufa, 450005, Russia

Location

GSK Investigational Site

Ulyanovsk, 432063, Russia

Location

GSK Investigational Site

Yaroslavl, 150030, Russia

Location

GSK Investigational Site

Daegu, 700-721, South Korea

Location

GSK Investigational Site

Gwangju, 501-757, South Korea

Location

GSK Investigational Site

Incheon, 400-711, South Korea

Location

GSK Investigational Site

Seoul, 03080, South Korea

Location

GSK Investigational Site

Seoul, 133-792, South Korea

Location

GSK Investigational Site

Seoul, 137-701, South Korea

Location

GSK Investigational Site

Suwon, 443-380, South Korea

Location

GSK Investigational Site

Badalona, 08916, Spain

Location

GSK Investigational Site

Barcelona, 08035, Spain

Location

GSK Investigational Site

Valencia, 46017, Spain

Location

GSK Investigational Site

Valladolid, 47010, Spain

Location

GSK Investigational Site

Vigo (Pontevedra), 36214, Spain

Location

Related Publications (5)

  • Aranow C, Allaart CF, Amoura Z, Bruce IN, Cagnoli PC, Chatham WW, Clark KL, Furie R, Groark J, Urowitz MB, van Vollenhoven R, Daniels M, Fox NL, Gregan YI, Henderson RB, van Maurik A, Ocran-Appiah JC, Oldham M, Roth DA, Shanahan D, Tak PP, Teng YO. Efficacy and safety of sequential therapy with subcutaneous belimumab and one cycle of rituximab in patients with systemic lupus erythematosus: the phase 3, randomised, placebo-controlled BLISS-BELIEVE study. Ann Rheum Dis. 2024 Oct 21;83(11):1502-1512. doi: 10.1136/ard-2024-225686.

    PMID: 39159997BACKGROUND
  • Arends EJ, Zlei M, Tipton CM, Cotic J, Osmani Z, de Bie FJ, Kamerling SWA, van Maurik A, Dimelow R, Gregan YI, Fox NL, Rabelink TJ, Roth DA, Sanz I, van Dongen JJM, van Kooten C, Teng YKO. Disruption of memory B-cell trafficking by belimumab in patients with systemic lupus erythematosus. Rheumatology (Oxford). 2024 Sep 1;63(9):2387-2398. doi: 10.1093/rheumatology/keae286.

  • Hannon CW, McCourt C, Lima HC, Chen S, Bennett C. Interventions for cutaneous disease in systemic lupus erythematosus. Cochrane Database Syst Rev. 2021 Mar 9;3(3):CD007478. doi: 10.1002/14651858.CD007478.pub2.

  • Teng YKO, Bruce IN, Diamond B, Furie RA, van Vollenhoven RF, Gordon D, Groark J, Henderson RB, Oldham M, Tak PP. Phase III, multicentre, randomised, double-blind, placebo-controlled, 104-week study of subcutaneous belimumab administered in combination with rituximab in adults with systemic lupus erythematosus (SLE): BLISS-BELIEVE study protocol. BMJ Open. 2019 Mar 20;9(3):e025687. doi: 10.1136/bmjopen-2018-025687.

  • Parodis I, Lopez Benavides AH, Zickert A, Pettersson S, Moller S, Welin Henriksson E, Voss A, Gunnarsson I. The Impact of Belimumab and Rituximab on Health-Related Quality of Life in Patients With Systemic Lupus Erythematosus. Arthritis Care Res (Hoboken). 2019 Jun;71(6):811-821. doi: 10.1002/acr.23718.

MeSH Terms

Conditions

Lupus Erythematosus, Systemic

Interventions

belimumabRituximabStandard of Care

Condition Hierarchy (Ancestors)

Connective Tissue DiseasesSkin and Connective Tissue DiseasesAutoimmune DiseasesImmune System Diseases

Intervention Hierarchy (Ancestors)

Antibodies, Monoclonal, Murine-DerivedAntibodies, MonoclonalAntibodiesImmunoglobulinsImmunoproteinsBlood ProteinsProteinsAmino Acids, Peptides, and ProteinsSerum GlobulinsGlobulinsQuality Indicators, Health CareQuality of Health CareHealth Services AdministrationHealth Care Quality, Access, and Evaluation

Results Point of Contact

Title
GSK Response Center
Organization
GlaxoSmithKline

Study Officials

  • GSK Clinical Trials

    GlaxoSmithKline

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR
Expanded Access
Yes

Study Record Dates

First Submitted

October 13, 2017

First Posted

October 18, 2017

Study Start

March 1, 2018

Primary Completion

May 29, 2020

Study Completion

July 7, 2021

Last Updated

February 18, 2025

Results First Posted

April 25, 2022

Record last verified: 2025-01

Data Sharing

IPD Sharing
Will share

GSK will assess requests from qualified researchers for anonymized individual patient-level data (IPD) and related study documents. Data sharing is subject to certain criteria, conditions, and exceptions. For further information, refer to https://www.gsk-studyregister.com/About\_GSK\_Patient\_Level\_Data\_Sharing\_Final\_13July2023.pdf

Shared Documents
STUDY PROTOCOL, SAP, ICF, CSR
Time Frame
Anonymized IPD is made available within 6 months of publication of primary, key secondary and safety results for studies in product with approved indication(s) or terminated asset(s) across all indications.
Access Criteria
Anonymized IPD is shared with researchers whose proposals are approved by an Independent Review Panel and after a Data Sharing Agreement is in place. Access is provided for an initial period of 12 months but an extension may be granted, when justified, for up to 6 months.
More information

Locations