NCT03158506

Brief Summary

This is an open-label, single center, 1-period study in healthy adult male subjects to assess absorption, metabolism, and excretion of HMS5552 after a single oral administration of 50 mg (90 μCi) of \[14C\]-HMS5552.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
6

participants targeted

Target at below P25 for phase_1

Timeline
Completed

Started Mar 2017

Geographic Reach
1 country

1 active site

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

March 29, 2017

Completed
8 days until next milestone

Primary Completion

Last participant's last visit for primary outcome

April 6, 2017

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

April 6, 2017

Completed
1 month until next milestone

First Submitted

Initial submission to the registry

May 10, 2017

Completed
8 days until next milestone

First Posted

Study publicly available on registry

May 18, 2017

Completed
Last Updated

December 31, 2018

Status Verified

April 1, 2017

Enrollment Period

8 days

First QC Date

May 10, 2017

Last Update Submit

December 27, 2018

Conditions

Outcome Measures

Primary Outcomes (4)

  • Total radioactivity in blood, plasma urine and feces

    Peak plasma concentration (Cmax)

    Up to 168 hours

  • Total radioactivity in blood, plasma urine and feces

    Area under the plasma concentration versus time curve (AUC)

    Up to 168 hours

  • Total radioactivity in blood, plasma urine and feces

    Time to reach Cmax (Tmax)

    Up to 168 hours

  • Total radioactivity in blood, plasma urine and feces

    Total radioactivity in urine and faeces at each time interval and cumulative radioactivity (mass balance)

    Up to 168 hours

Secondary Outcomes (4)

  • Concentrations of HMS5552 and its metabolites in plasma, urine and feces

    Up to 168 hours

  • Number of participants with adverse events as a measure of safety and tolerability

    Up to 168 hours

  • Concentrations of HMS5552 and its metabolites in plasma, urine and feces

    Up to 168 hours

  • Concentrations of HMS5552 and its metabolites in plasma, urine and feces

    Up to 168 hours

Study Arms (1)

[C14]-labelled HMS5552

EXPERIMENTAL
Drug: HMS5552

Interventions

\[14C\]-labelled HMS5552

[C14]-labelled HMS5552

Eligibility Criteria

Age19 Years - 55 Years
Sexmale
Healthy VolunteersYes
Age GroupsAdult (18-64)

You may qualify if:

  • Healthy, adult, male 19-55 years of age
  • Weight at least 50 kg, and BMI within the range of 18-30 kg/m2
  • Written informed consent must be obtained before any assessment is performed

You may not qualify if:

  • History or presence of clinically significant medical, surgical or psychiatric condition or disease in the opinion of the Investigator or designee which might significantly alter the absorption, distribution, metabolism and excretion of drugs.
  • History or presence of alcoholism or drug abuse.
  • Smoker.
  • Abnormal bowel habits.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Celerion

Lincoln, Nebraska, 68502, United States

Location

MeSH Terms

Interventions

Dorzagliatin

Study Officials

  • Charles Tomek, MD

    Celerion

    PRINCIPAL INVESTIGATOR

Study Design

Study Type
interventional
Phase
phase 1
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

May 10, 2017

First Posted

May 18, 2017

Study Start

March 29, 2017

Primary Completion

April 6, 2017

Study Completion

April 6, 2017

Last Updated

December 31, 2018

Record last verified: 2017-04

Data Sharing

IPD Sharing
Will not share

Locations