NCT02600507

Brief Summary

The study will evaluate the efficacy and safety of ITI-007 adjunctive to lithium or valproate in a randomized, double-blind, parallel-group, placebo-controlled, multi-center study in patients diagnosed with Bipolar I or Bipolar II disorder having a major depressive episode.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
529

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Mar 2016

Typical duration for phase_3

Geographic Reach
5 countries

71 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

November 5, 2015

Completed
4 days until next milestone

First Posted

Study publicly available on registry

November 9, 2015

Completed
4 months until next milestone

Study Start

First participant enrolled

March 7, 2016

Completed
4.3 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 2, 2020

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

July 2, 2020

Completed
2.9 years until next milestone

Results Posted

Study results publicly available

May 17, 2023

Completed
Last Updated

May 17, 2023

Status Verified

April 1, 2021

Enrollment Period

4.3 years

First QC Date

November 5, 2015

Results QC Date

April 24, 2023

Last Update Submit

April 24, 2023

Conditions

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline in Montgomery-Åsberg Depression Rating Scale (MADRS) Total Score

    The Montgomery-Åsberg Depression Rating Scale (MADRS) is a clinician-rated 10 item scale to assess depressive symptoms. Each item is rated on a 7-point scale from 0-6. The total score ranges from 0 to 60 with a higher score indicating increased severity of depressive symptoms.

    Baseline to Day 43

Secondary Outcomes (1)

  • Change From Baseline in Clinical Global Impression Scale-Bipolar Version-Severity (CGI-BP-S) Depression Score

    Baseline to Day 43

Study Arms (3)

Lumateperone 28 mg (ITI-007 40 mg tosylate)

EXPERIMENTAL

Lumateperone 28 mg (ITI-007 40 mg tosylate) administered orally as capsules once daily for 6 weeks

Drug: Lumateperone (ITI-007)

Lumateperone 42 mg (ITI-007 60 mg tosylate)

EXPERIMENTAL

Lumateperone 42 mg (ITI-007 60 mg tosylate) administered orally as capsules once daily for 6 weeks

Drug: Lumateperone (ITI-007)

Placebo

PLACEBO COMPARATOR

Placebo administered orally as visually-matched capsules once daily for 6 weeks

Drug: Placebo

Interventions

Lumateperone 28 mg (ITI-007 40 mg tosylate)Lumateperone 42 mg (ITI-007 60 mg tosylate)
Placebo

Eligibility Criteria

Age18 Years - 75 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • male or female subjects of any race, ages 18-75 inclusive, with a clinical diagnosis of Bipolar I or Bipolar II disorder
  • experiencing a current major depressive episode
  • treatment with either lithium or valproate and inadequate therapeutic response of depressive symptoms

You may not qualify if:

  • any subject unable to provide informed consent
  • any female subject who is pregnant or breastfeeding
  • any subject judged to be medically inappropriate for study participation

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (71)

Clinical Site

Rogers, Arkansas, United States

Location

Clinical Site

Cerritos, California, United States

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Costa Mesa, California, United States

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Culver City, California, United States

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Garden Grove, California, United States

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Glendale, California, United States

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Lemon Grove, California, United States

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Oceanside, California, United States

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Pico Rivera, California, United States

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Riverside, California, United States

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San Diego, California, United States

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Santa Rosa, California, United States

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Sherman Oaks, California, United States

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Temecula, California, United States

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Jacksonville, Florida, United States

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Lauderhill, Florida, United States

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Miami, Florida, United States

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Orange City, Florida, United States

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Orlando, Florida, United States

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Atlanta, Georgia, United States

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Savannah, Georgia, United States

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Chicago, Illinois, United States

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Lake Charles, Louisiana, United States

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Baltimore, Maryland, United States

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O'Fallon, Missouri, United States

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St Louis, Missouri, United States

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Las Vegas, Nevada, United States

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Berlin, New Jersey, United States

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Cherry Hill, New Jersey, United States

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Toms River, New Jersey, United States

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Cedarhurst, New York, United States

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New York, New York, United States

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Rochester, New York, United States

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Staten Island, New York, United States

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Charlotte, North Carolina, United States

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Cincinnati, Ohio, United States

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Dayton, Ohio, United States

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Garfield Heights, Ohio, United States

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Allentown, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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The Woodlands, Texas, United States

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Everett, Washington, United States

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Burgas, Bulgaria

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Kardzhali, Bulgaria

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Lovech, Bulgaria

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Pleven, Bulgaria

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Plovdiv, Bulgaria

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Rousse, Bulgaria

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Sofia, Bulgaria

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Varna, Bulgaria

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Veliko Tarnovo, Bulgaria

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Vratsa, Bulgaria

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Moscow, Russia

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Nizhny Novgorod, Russia

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Omsk, Russia

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Saint Petersburg, Russia

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Samara, Russia

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Saratov, Russia

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Tomsk, Russia

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Belgrade, Serbia

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Kovin, Serbia

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Novi Sad, Serbia

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Šumadija, Serbia

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Ivano-Frankivsk, Ukraine

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Kharkiv, Ukraine

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Kropyvnytskyi, Ukraine

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Odesa, Ukraine

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Poltava, Ukraine

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Smila, Ukraine

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Vasylkiv, Ukraine

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Clinical Site

Vinnytsia, Ukraine

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Related Publications (1)

  • Suppes T, Durgam S, Kozauer SG, Chen R, Lakkis HD, Davis RE, Satlin A, Vanover KE, Mates S, McIntyre RS, Tohen M. Adjunctive lumateperone (ITI-007) in the treatment of bipolar depression: Results from a randomized placebo-controlled clinical trial. Bipolar Disord. 2023 Sep;25(6):478-488. doi: 10.1111/bdi.13310. Epub 2023 Feb 26.

MeSH Terms

Conditions

Bipolar Disorder

Interventions

lumateperone

Condition Hierarchy (Ancestors)

Bipolar and Related DisordersMood DisordersMental Disorders

Results Point of Contact

Title
ITI Clinical Trials
Organization
Intra-Cellular Therapies, Inc.

Study Officials

  • Susan Kozauer, MD

    Intra-Cellular Therapies, Inc.

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

November 5, 2015

First Posted

November 9, 2015

Study Start

March 7, 2016

Primary Completion

July 2, 2020

Study Completion

July 2, 2020

Last Updated

May 17, 2023

Results First Posted

May 17, 2023

Record last verified: 2021-04

Locations