NCT02586155

Brief Summary

The purpose of this study is to determine whether bromodomain extraterminal domain (BET) inhibition treatment with RVX000222 in high-risk type 2 diabetes mellitus patients with coronary artery disease increases the time to major adverse cardiovascular events.

Trial Health

98
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Strong global presence with extensive site network
Enrollment
2,425

participants targeted

Target at P75+ for phase_3 diabetes-mellitus-type-2

Timeline
Completed

Started Nov 2015

Longer than P75 for phase_3 diabetes-mellitus-type-2

Geographic Reach
15 countries

214 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 21, 2015

Completed
5 days until next milestone

First Posted

Study publicly available on registry

October 26, 2015

Completed
6 days until next milestone

Study Start

First participant enrolled

November 1, 2015

Completed
5.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 30, 2020

Completed
7 months until next milestone

Study Completion

Last participant's last visit for all outcomes

June 21, 2021

Completed
2 months until next milestone

Results Posted

Study results publicly available

August 20, 2021

Completed
Last Updated

August 20, 2021

Status Verified

July 1, 2021

Enrollment Period

5.1 years

First QC Date

October 21, 2015

Results QC Date

June 21, 2021

Last Update Submit

July 23, 2021

Conditions

Outcome Measures

Primary Outcomes (1)

  • Incidence of First Occurrence of Adjudication-confirmed Narrowly Defined MACE

    Incidence of first occurrence of MACE narrowly defined as a single composite endpoint of Cardiovascular (CV) Death (including undetermined cause of death) or Non-fatal Myocardial Infarction (MI) or Stroke. If a subject has multiple events, only the first event contributing to the composite endpoint is counted.

    120 weeks

Secondary Outcomes (13)

  • Incidence of First Occurrence of Adjudication-confirmed Broadly Defined MACE

    120 weeks

  • Incidence of Hospitalization for Congestive Heart Failure (CHF)

    120 weeks

  • Incidence of All-cause Mortality

    120 weeks

  • Change in Apolipoprotein A1 (ApoA-I) Concentration From Baseline Over Time Within and Between Treatment Groups

    120 weeks

  • Change in Apolipoprotein B (apoB) Concentration From Baseline Over Time Within and Between Treatment Groups

    120 weeks

  • +8 more secondary outcomes

Study Arms (2)

High-Intensity statin therapy+RVX000222

EXPERIMENTAL

Daily dose 100 mg capsule b.i.d. with high-intensity statin therapy (atorvastatin or rosuvastatin)

Drug: ApabetaloneDrug: AtorvastatinDrug: Rosuvastatin

High-Intensity statin therapy+Placebo

ACTIVE COMPARATOR

Placebo (for RVX000222 100 mg capsule) b.i.d. with high-intensity statin therapy (atorvastatin or rosuvastatin)

Drug: PlaceboDrug: AtorvastatinDrug: Rosuvastatin

Interventions

100 mg capsule

Also known as: RVX000222
High-Intensity statin therapy+RVX000222

Capsule manufactured to mimic RVX000222 100 mg capsule

Also known as: Placebo (for RVX000222)
High-Intensity statin therapy+Placebo

High-Intensity Statin

Also known as: Lipitor
High-Intensity statin therapy+PlaceboHigh-Intensity statin therapy+RVX000222

High-Intensity Statin

Also known as: Crestor
High-Intensity statin therapy+PlaceboHigh-Intensity statin therapy+RVX000222

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • ACS event of either unstable angina or myocardial infarction 7-90 days prior Visit 1:
  • Unstable angina: for a qualifying unstable angina event, each of components (a), (b), and (c) must be satisfied: a.) Characteristic ischemic pain or discomfort in chest/associated referral areas, occurring at rest/with minimal exertion b.) ECG changes consistent with acute myocardial ischemia based on new/presumed ST elevation/depression or T-wave inversion c.) Objective evidence of obstructive CAD based on 1+ of the following: i. New/presumed new evidence of myocardial ischemia/infarction by perfusion imaging ii. New/presumed new regional wall motion abnormality iii. Current evidence of at least 1 epicardial coronary artery stenosis ≥70% by coronary angiography iv. Need for coronary revascularization for the index ACS event, including a percutaneous coronary intervention (PCI) with or without coronary stenting.
  • Prior MI 7-90 days prior screening treated with or without a percutaneous coronary intervention (PCI). For a qualifying event of MI 2 of the following 3 criteria must be satisfied: a.) Characteristic ischemic chest pain/pain in associated referral areas b.) Dynamic elevation of troponin T/I or CKMB if troponinT/I is unavailable at local lab (at least \>ULN for lab) c.) Development of new Q-waves in ≥2 adjacent ECG leads or development of new dominant R wave in V1
  • Documented diagnosis of T2DM (1+ of the following criteria): Documented history of T2DM, History of taking diabetes medication, and/or HbA1c ≥6.5% at Visit 1
  • For males HDL-C\<40 mg/dL(1.04 mmol/L), for females HDL-C\<45 mg/dL(1.17 mmol/L) at Visit 1
  • Subjects currently not on high intensity statin therapy could start rosuvastatin at Visit 1 and those currently on therapy besides atorvastatin/rosuvastatin can be switched to rosuvastatin at Visit 1
  • Female subjects of non-childbearing potential (post-surgical sterilization/post-menopausal) or if childbearing potential have neg urine pregnancy test and be willing and able to use non-hormonal birth control (non-hormonal IUD, condom or diaphragm) or remain abstinent from Screening to Follow-up Visit
  • Give signed informed consent

You may not qualify if:

  • Heart disease which will w/in 90 days of Visit 1 likely need coronary bypass, PCI, cardiac transplantation, surgical repair and/or replacement
  • Previous/current diagnosis of severe heart failure or documented LVEF\<25% determined by contrast left ventriculography, radionuclide ventriculography or echocardiography. Absence of LVEF measurement in subject w/out a previous/current diagnosis of heart failure does not exclude entry into study
  • Evidence of cardiac EP instability incl. history of uncontrolled ventricular arrhythmias, atrial fibrillation/flutter or supraventricular tachycardias w/ a ventricular response HR\>100bpm at rest w/in 4 wks prior Visit 1
  • CABG w/in 90 days prior Visit 1
  • Evidence of severe renal impairment as determined by either eGFR\<30 mL/min/1.7m2 at Visit 1 or current need for dialysis
  • Uncontrolled hypertension defined as 2 consecutive measurements of sitting BP of systolic\>180 mmHg or diastolic\>100 mmHg at Visit 1
  • Treatment w/ immunosuppressants w/in 12 mos prior Visit 1
  • Use of fibrates at any dose or niacin/nicotinic acid 250+ mg w/in 30 days prior Visit 1
  • Known allergy/sensitivity to any ingredient in IMP
  • History of intolerance to atorvastatin/rosuvastatin
  • Triglycerides\>400 mg/dL (4.52 mmol/L) at Visit 1
  • Any medical/surgical condition which might significantly alter absorption, distribution, metabolism or excretion of medication
  • Evidence of cirrhosis from liver imaging/biopsy, history of hepatic encephalopathy, esophageal/gastric varices, active hepatitis or prior porta-caval shunt procedure or a Child-Pugh score of ≥5 points
  • ALT/AST\>1.5xULN by central lab at Visit 1
  • Tot. bilirubin\>ULN by central lab at Visit 1
  • +8 more criteria

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (214)

Instituto de Investigaciones Clinicas Bahia Blanca

Bahía Blanca, Argentina

Location

Bioclinica Buenos Aires

Buenos Aires, Argentina

Location

Centro Privado de Enfermedades Cardiovasculares

Buenos Aires, Argentina

Location

Consultorios Asociados Endocronología E Investigación Clínica Aplicada

Buenos Aires, Argentina

Location

Instituto Cardiovascular de Buenos Aires

Buenos Aires, Argentina

Location

Sanatorio Guemes

Buenos Aires, Argentina

Location

Clinica Coronel Suarez

Coronel Suárez, Argentina

Location

Instituto de Cardiologia de Corrientes Juana Francisca Cabral

Corrientes, Argentina

Location

CEMAIC

Córdoba, Argentina

Location

Centro Médico Colón

Córdoba, Argentina

Location

Centro Médico Luquez

Córdoba, Argentina

Location

Clínica Privada Del Prado Sociedad de Responsabilidad Limitada

Córdoba, Argentina

Location

Fundación Clínica Colombo

Córdoba, Argentina

Location

Hospital Cordoba

Córdoba, Argentina

Location

Hospital San Roque

Córdoba, Argentina

Location

Instituto Del Corazón

Córdoba, Argentina

Location

Instituto Modelo de Cardiologia

Córdoba, Argentina

Location

Instituto Médico DAMIC

Córdoba, Argentina

Location

Ipac Caraffa

Córdoba, Argentina

Location

Sanatorio Allende

Córdoba, Argentina

Location

Centro Médico Libertad

Haedo, Argentina

Location

CIMEL

Lanús, Argentina

Location

Instituto de Investigaciones Clínicas Mar Del Plata

Mar del Plata, Argentina

Location

Hospital Central

Mendoza, Argentina

Location

DIM Clinica Privada

Ramos Mejía, Argentina

Location

Instituto de Hematologia Y Medicina Clinica

Rosario, Argentina

Location

Sanatorio Britanico de Rosario

Rosario, Argentina

Location

Prevencion Cardio Vascular

Salta, Argentina

Location

Grupo Medico Alem

San Isidro, Argentina

Location

Bioclinica Tucumán

San Miguel de Tucumán, Argentina

Location

Centro Modelo de Cardiologia

San Miguel de Tucumán, Argentina

Location

Investigaciones Clinicas Tucuman

San Miguel de Tucumán, Argentina

Location

Centro de Investigaciones Clínicas Del Litoral SRL

Santa Fe, Argentina

Location

Sanatorio San Francisco

Santiago del Estero, Argentina

Location

Clínica FUSAVIM Privada

Villa María, Argentina

Location

Instituto de Investigaciones Clínicas Zárate

Zárate, Argentina

Location

Flinders Medical Centre

Bedford Park, Australia

Location

ZNA Middelheim

Antwerp, Belgium

Location

Imelda VZW

Bonheiden, Belgium

Location

AZ Turnhout

Turnhout, Belgium

Location

Multiprofile Hospital For Active Treatment Dr Tota Venkova

Gabrovo, Bulgaria

Location

Multiprofile Hospital for Active Treatment - Prof. Dr. Paraskev Stoyanov AD

Lovech, Bulgaria

Location

Multiprofile Hospital For Active Treatment - Pazardzhik AD

Pazardzhik, Bulgaria

Location

University Multiprofile Hospital for Active Treatment - Dr. Georgi Stranski EAD

Pleven, Bulgaria

Location

Multiprofile Hospital For Active Treatment - Dr. Bratan Shukerov AD

Smolyan, Bulgaria

Location

Acibadem City Clinic Multiprofile Hospital for Active Treatment Tokuda

Sofia, Bulgaria

Location

City Clinic University Multiprofile Hospital for Active Treatment EOOD

Sofia, Bulgaria

Location

Medical Center Kardiohelp EOOD

Sofia, Bulgaria

Location

Second Multiprofile Hospital for Active Treatment Sofia

Sofia, Bulgaria

Location

Synexus Affiliate - Diagnostic and Consulting Center Ascendent

Sofia, Bulgaria

Location

University Multiprofile Hospital for Active Treatment Aleksandrovska EAD

Sofia, Bulgaria

Location

University Multiprofile Hospital for Active Treatment and Emergency Medicine N. I. Pirogov EAD

Sofia, Bulgaria

Location

Medical Center Orfey OOD

Stara Zagora, Bulgaria

Location

Multiprofile Hospital for Active Treatment Sveta Marina EAD

Varna, Bulgaria

Location

General Hospital Karlovac

Karlovac, Croatia

Location

Special Hospital for medicinal rehabilitation Krapinske Toplice

Krapinske Toplice, Croatia

Location

Clinical Hospital Osijek

Osijek, Croatia

Location

General Hospital Dr Josip Bencevic

Slavonski Brod, Croatia

Location

General Hospital Virovitica

Virovitica, Croatia

Location

Clinical Hospital Sveti duh

Zagreb, Croatia

Location

DRK Kliniken Berlin Westend

Berlin, Germany

Location

Medizinisches Versorgungszentrum am Küchwald GmbH

Chemnitz, Germany

Location

Zentrum für Klinische Prüfung in der Facharztzentrum Dresden Neustadt Gbr

Dresden, Germany

Location

Katholisches Krankenhaus St. Johann Nepomuk

Erfurt, Germany

Location

Heidelberger Praxisklinik für Kardiologie

Heidelberg, Germany

Location

Klinikum Hoyerswerda

Hoyerswerda, Germany

Location

Studienzentrum Dr.Appel

Kassel, Germany

Location

Asklepios Klinik Langen

Langen, Germany

Location

Klinikum Leverkusen GmbH

Leverkusen, Germany

Location

Bajai Szent Rókus Kórház

Baja, Hungary

Location

Grof Tisza Istvan Korhaz Berettyoujfalu

Berettyóújfalu, Hungary

Location

Bajcsy-Zsilinszky Korhaz es Rendelointezet

Budapest, Hungary

Location

Del-pesti Centrumkorhaz- Orszagos Hematologiai és Infektologiai Intezet

Budapest, Hungary

Location

Gottsegen Gyorgy Orszagos Kardiologiai Intezet

Budapest, Hungary

Location

Magyar Honvédség Egészségügyi Központ

Budapest, Hungary

Location

Semmelweis Egyetem

Budapest, Hungary

Location

Synexus (DRS) - Synexus Magyarország Kft. Budapest

Budapest, Hungary

Location

Szent Margit Korhaz

Budapest, Hungary

Location

Szent Rókus Kórház és Intézményei

Budapest, Hungary

Location

Selye János Kórház

Komárom, Hungary

Location

TaNaMed Kft.

Mosonmagyaróvár, Hungary

Location

Kanizsai Dorottya Kórház

Nagykanizsa, Hungary

Location

Coromed-SMO Kft.

Pécs, Hungary

Location

Szegedi Tudomanyegyetem Szent-Gyorgyi Albert Klinikai Kozpont

Szeged, Hungary

Location

Tolna Megyei Balassa János Kórház

Szekszárd, Hungary

Location

Fejer Megyei Szent Gyorgy Egyetemi Oktato Korhaz

Székesfehérvár, Hungary

Location

Barzilai Medical Center

Ashkelon, Israel

Location

Soroka University Medical Centre

Beersheba, Israel

Location

Hillel Yaffe Medical Center

Hadera, Israel

Location

Bnei Zion Medical Center

Haifa, Israel

Location

Lady Davis Carmel Medical Center

Haifa, Israel

Location

Linn Medical Center Clalit Health Services

Haifa, Israel

Location

Rambam Medical Center

Haifa, Israel

Location

Edith Wolfson Medical Center

Holon, Israel

Location

Hadassah University Hospital Ein Kerem

Jerusalem, Israel

Location

Hadassah University Hospital Mount Scopus

Jerusalem, Israel

Location

Shaare Zedek Medical Center

Jerusalem, Israel

Location

Meir Medical Center

Kefar Sava, Israel

Location

Galilee Medical Center

Nahariya, Israel

Location

Nazareth EMMS Hospital

Nazareth, Israel

Location

Chaim Sheba Medical Center

Ramat Gan, Israel

Location

Kaplan Medical Center

Rehovot, Israel

Location

ZIV Medical Center

Safed, Israel

Location

Clalit Health Medical Center

Tel Aviv, Israel

Location

Tel Aviv Sourasky Medical Center

Tel Aviv, Israel

Location

Baruch Padeh Poriya Medical Center

Tiberias, Israel

Location

Fundacion Cardiovascular de Aguascalientes AC

Aguascalientes, Mexico

Location

Hospital Cardiológica Aguascalientes

Aguascalientes, Mexico

Location

Investigacion en Salud y Metabolismo S.C.

Chihuahua City, Mexico

Location

Centro Para el Desarrollo de la Medicina y de Asistencia Especializada SC

Culiacán, Mexico

Location

Centro de Investigacion y Atencion de Diabetes, Endocrinologia y Nutricion

Durango, Mexico

Location

Arechavaleta Granell Maria del Rosario

Guadalajara, Mexico

Location

Centro de Investigacion Medica Biologica Y de Terapia Avanzada SC

Guadalajara, Mexico

Location

Unidad de Investigacion Clinica Cardiometabolica de Occidente SC

Guadalajara, Mexico

Location

Hospital Angeles Leon

León, Mexico

Location

Centro de Investigación Biomedica y Farmaceutica

Mexico City, Mexico

Location

Clinica Integral del Paciente Diabetico y Obeso

Mexico City, Mexico

Location

Fundación de Atención e Investigación Médica Lindavista S.C.

Mexico City, Mexico

Location

Sanatorio y Servicios Médicos Obregón S.A. de C.V.

Mexico City, Mexico

Location

Centro de Desarrollo Biomédico

Mérida, Mexico

Location

Instituto Cardiovascular de Monclova

Monclova, Mexico

Location

Hospital Universitario Dr. Jose Eleuterio González

Monterrey, Mexico

Location

IMED Internal Medicine Clin Trials

Monterrey, Mexico

Location

Unidad de Investigación Clínica En Medicina SC

Monterrey, Mexico

Location

Diabetes Total, S.A de C.V.

Pachuca, Mexico

Location

Investigacion Biomedica Aplicada de Hidalgo S.A. de C.V.

Pachuca, Mexico

Location

Cardioarritmias e Investigación S.C.

San Luis Potosí City, Mexico

Location

Hospital Central Dr Ignacio Morones Prieto

San Luis Potosí City, Mexico

Location

INBIOMEDYC Toluca

Toluca, Mexico

Location

Centro de Alta Especialidad Dr. Rafael Lucio

Veracruz, Mexico

Location

Dr. Humberto Alvarez Lopez

Zapopan, Mexico

Location

Meander Medisch Centrum

Amersfoort, Netherlands

Location

OLVG locatie Oost

Amsterdam, Netherlands

Location

VU Medisch Centrum

Amsterdam, Netherlands

Location

Podlaski Osrodek Kardiologii Poradnia Prywatna

Bialystok, Poland

Location

Malopolskie Centrum Sercowo-Naczyniowe

Chrzanów, Poland

Location

Polsko-Amerykanskie Kliniki Serca

Dąbrowa Górnicza, Poland

Location

Gabinet Kardiologiczno-Internistyczny

Gdynia, Poland

Location

Niepubliczny Zaklad Opieki Zdrowotnej Centrum Uslug Medycznych Promont-Med.

Kielce, Poland

Location

Diamond Clinic

Krakow, Poland

Location

Szpital Specjalistyczny im. Jozefa Dietla w Krakowie

Krakow, Poland

Location

Zespol Przychodni Specjalistycznych DIAB-END-COR Sp. z o.o.

Krakow, Poland

Location

Prywatna Praktyka Lekarska MAZ-MEDICA Maciej R.Mazurkiewicz

Lodz, Poland

Location

Uniwersytecki Szpital Kliniczny im. Wojskowej Akademii Medycznej Centralny Szpital Weteranow

Lódz, Poland

Location

Polsko-Amerykanskie Kliniki Serca

Nysa, Poland

Location

Pro Corde, Dom Medyczny

Opole, Poland

Location

Medicome Sp. z o.o.

Oświęcim, Poland

Location

Rodzinne Centrum Zdrowia

Otwock, Poland

Location

Niepubliczny Zaklad Opieki Zdrowotnej Specjalistyczna Przychodnia Lekarska "MEDIKARD"

Płock, Poland

Location

Niepubliczny Zaklad Opieki Zdrowotnej Centrum Medyczne SBB

Tarnobrzeg, Poland

Location

Centrum Medyczne doktorA

Warsaw, Poland

Location

Instytut Kardiologii im Prymasa Tysiaclecia Kardynala Stefana Wyszynskiego

Warsaw, Poland

Location

Niepubliczny Zaklad Opieki Zdrowotnej AURUM

Warsaw, Poland

Location

Centrum Kardiologiczne Pro Corde Sp. z o.o. Niepubliczny Zaklad Opieki Zdrowotnej

Wroclaw, Poland

Location

Wro Medica

Wroclaw, Poland

Location

City Clinical Hospital #6

Chelyabinsk, Russia

Location

Federal Budget Healthcare Institution Medici - sanitary unit of Ministry of internal affairs of Russ

Kemerovo, Russia

Location

Research Institute of Complex Cardiovascular Pathology

Kemerovo, Russia

Location

Krasnodar Regional Clinical Hospital #2

Krasnodar, Russia

Location

Moscow City State Budgetary Healthcare Institution City Clinical Hospital named after V.V. Veresayev

Moscow, Russia

Location

Russian Cardiology Research and Production Center

Moscow, Russia

Location

City Hospital 13

Nizhny Novgorod, Russia

Location

State Budgetary Healthcare Institution of Novosibirsk Region City Clinical Hospital No. 19

Novosibirsk, Russia

Location

Republican Hospital n.a. V.A. Baranov

Petrozavodsk, Russia

Location

Municipal Budgetary Healthcare Institution City Emergency Hospital

Rostov-on-Don, Russia

Location

International Medical Center SOGAZ

Saint Petersburg, Russia

Location

North-West State Medical University n.a. I.I. Mechnikov

Saint Petersburg, Russia

Location

St Petersburg City Outpatient Clinic #109

Saint Petersburg, Russia

Location

Saratov State Medical University

Saratov, Russia

Location

State Healthcare Institution Regional Clinical Cardiologic Dispensary

Saratov, Russia

Location

City Hospital #4

Sochi, Russia

Location

Research Cardiology Institute of Tomsk Scientific Center of RAMS Siberian Branch

Tomsk, Russia

Location

State Budgetary Healthcare Institution of Vladimir Region City Hospital No. 4

Vladimir, Russia

Location

Ural State Medical University

Yekaterinburg, Russia

Location

Clinical Center of Serbia

Belgrade, Serbia

Location

Clinical Hospital Centar Zvezdara

Belgrade, Serbia

Location

Clinical Hospital Center Bezanijska Kosa

Belgrade, Serbia

Location

Clinical Hospital Centre Zemun

Belgrade, Serbia

Location

Euromedik

Belgrade, Serbia

Location

Institute of Cardiovascular Diseases Dedinje

Belgrade, Serbia

Location

KBC Dr Dragisa Misovic Dedinje

Belgrade, Serbia

Location

Military Medical Academy

Belgrade, Serbia

Location

Institute of Cardiovascular Diseases of Vojvodina

Kamenitz, Serbia

Location

Clinical Center Kragujevac

Kragujevac, Serbia

Location

Clinical Center Nis

Niš, Serbia

Location

Institute Niska Banja

Niška Banja, Serbia

Location

Clinical Centre of Vojvodina

Novi Sad, Serbia

Location

General Hospital Uzice

Užice, Serbia

Location

Health Center Zajecar

Zaječar, Serbia

Location

ALIAN, s.r.o

Bardejov, Slovakia

Location

CARDIOCONSULT, s.r.o.

Bratislava, Slovakia

Location

Univerzitna nemocnica Bratislava

Bratislava, Slovakia

Location

Kardio-Onkologia, s.r.o.

Dolný Kubín, Slovakia

Location

CARDIO D&R, s.r.o. Kosice

Košice, Slovakia

Location

Zeleznicne zdravotnictvo Kosice, s.r.o.

Košice, Slovakia

Location

KARDIOMED s.r.o.

Lučenec, Slovakia

Location

MEDI M&M s.r.o.

Moldava nad Bodvou, Slovakia

Location

Nemocnica s poliklinikou Nove Mesto nad Vahom n.o.

Nové Mesto nad Váhom, Slovakia

Location

Cardioinvest s. r. o.

Nové Zámky, Slovakia

Location

DIAB s.r.o.

Rožňava, Slovakia

Location

MEDIVASA, s.r.o.

Žilina, Slovakia

Location

Changhua Christian Hospital

Changhua, Taiwan

Location

Kaohsiung Chang Gung Memorial Hospital

Kaohsiung City, Taiwan

Location

Kaohsiung Veterans General Hospital

Kaohsiung City, Taiwan

Location

Mackay Memorial Hospital-Taipei branch

New Taipei City, Taiwan

Location

China Medical University Hospital

Taichung, Taiwan

Location

National Cheng Kung University Hospital

Tainan, Taiwan

Location

Cathay General Hospital

Taipei, Taiwan

Location

Chi Mei Medical Center

Taipei, Taiwan

Location

Far Eastern Memorial Hospital

Taipei, Taiwan

Location

National Taiwan University Hospital

Taipei, Taiwan

Location

Taipei Veterans General Hospital

Taipei, Taiwan

Location

Tri-Service General Hospital

Taipei, Taiwan

Location

Chang Gung Medical Foundation Linkou Branch (Clinical Research Center)

Taoyuan, Taiwan

Location

Related Publications (5)

  • Ray KK, Nicholls SJ, Buhr KA, Ginsberg HN, Johansson JO, Kalantar-Zadeh K, Kulikowski E, Toth PP, Wong N, Sweeney M, Schwartz GG; BETonMACE Investigators and Committees. Effect of Apabetalone Added to Standard Therapy on Major Adverse Cardiovascular Events in Patients With Recent Acute Coronary Syndrome and Type 2 Diabetes: A Randomized Clinical Trial. JAMA. 2020 Apr 28;323(16):1565-1573. doi: 10.1001/jama.2020.3308.

  • Schwartz GG, Nicholls SJ, Toth PP, Sweeney M, Halliday C, Johansson JO, Wong NCW, Kulikowski E, Kalantar-Zadeh K, Ginsberg HN, Ray KK. Relation of insulin treatment for type 2 diabetes to the risk of major adverse cardiovascular events after acute coronary syndrome: an analysis of the BETonMACE randomized clinical trial. Cardiovasc Diabetol. 2021 Jun 22;20(1):125. doi: 10.1186/s12933-021-01311-9.

  • Haarhaus M, Gilham D, Kulikowski E, Magnusson P, Kalantar-Zadeh K. Pharmacologic epigenetic modulators of alkaline phosphatase in chronic kidney disease. Curr Opin Nephrol Hypertens. 2020 Jan;29(1):4-15. doi: 10.1097/MNH.0000000000000570.

  • Ray KK, Nicholls SJ, Ginsberg HD, Johansson JO, Kalantar-Zadeh K, Kulikowski E, Toth PP, Wong N, Cummings JL, Sweeney M, Schwartz GG. Effect of selective BET protein inhibitor apabetalone on cardiovascular outcomes in patients with acute coronary syndrome and diabetes: Rationale, design, and baseline characteristics of the BETonMACE trial. Am Heart J. 2019 Nov;217:72-83. doi: 10.1016/j.ahj.2019.08.001. Epub 2019 Aug 9.

  • Gilham D, Tsujikawa LM, Sarsons CD, Halliday C, Wasiak S, Stotz SC, Jahagirdar R, Sweeney M, Johansson JO, Wong NCW, Kalantar-Zadeh K, Kulikowski E. Apabetalone downregulates factors and pathways associated with vascular calcification. Atherosclerosis. 2019 Jan;280:75-84. doi: 10.1016/j.atherosclerosis.2018.11.002. Epub 2018 Nov 14.

Related Links

MeSH Terms

Conditions

Diabetes Mellitus, Type 2Coronary Artery Disease

Interventions

apabetaloneAtorvastatinRosuvastatin Calcium

Condition Hierarchy (Ancestors)

Diabetes MellitusGlucose Metabolism DisordersMetabolic DiseasesNutritional and Metabolic DiseasesEndocrine System DiseasesCoronary DiseaseMyocardial IschemiaHeart DiseasesCardiovascular DiseasesArteriosclerosisArterial Occlusive DiseasesVascular Diseases

Intervention Hierarchy (Ancestors)

PyrrolesAzolesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsHeptanoic AcidsFatty AcidsLipidsSulfonamidesAmidesOrganic ChemicalsFluorobenzenesHydrocarbons, FluorinatedHydrocarbons, HalogenatedHydrocarbonsSulfonesSulfur CompoundsPyrimidines

Results Point of Contact

Title
Sr. Director of Clinical Operations
Organization
Resverlogix Corp.

Study Officials

  • Kausik Ray, MD

    Imperial College London

    STUDY CHAIR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
No

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
TRIPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR
Purpose
PREVENTION
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 21, 2015

First Posted

October 26, 2015

Study Start

November 1, 2015

Primary Completion

November 30, 2020

Study Completion

June 21, 2021

Last Updated

August 20, 2021

Results First Posted

August 20, 2021

Record last verified: 2021-07

Data Sharing

IPD Sharing
Will not share

Locations