NCT02580305

Brief Summary

This is a phase 2a, proof-of-concept, 26-week, double-blind, multicenter, randomized, parallel group, placebo-controlled study to compare the efficacy and safety of treatment with SUVN-502 to placebo treatment in subjects with moderate Alzheimer's disease receiving stable doses of donepezil HCl and memantine HCl.

Trial Health

87
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
564

participants targeted

Target at P75+ for phase_2

Timeline
Completed

Started Sep 2015

Typical duration for phase_2

Geographic Reach
1 country

71 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

Study Start

First participant enrolled

September 1, 2015

Completed
2 months until next milestone

First Submitted

Initial submission to the registry

October 17, 2015

Completed
3 days until next milestone

First Posted

Study publicly available on registry

October 20, 2015

Completed
4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

November 5, 2019

Completed
2 days until next milestone

Study Completion

Last participant's last visit for all outcomes

November 7, 2019

Completed
3.6 years until next milestone

Results Posted

Study results publicly available

June 9, 2023

Completed
Last Updated

June 9, 2023

Status Verified

May 1, 2023

Enrollment Period

4.2 years

First QC Date

October 17, 2015

Results QC Date

April 17, 2023

Last Update Submit

May 16, 2023

Conditions

Keywords

SUVN-5025-HT6Phase 2CognitionDonepezilMemantineAlzheimer's DiseaseTriple CombinationProof of Concept (POC)

Outcome Measures

Primary Outcomes (1)

  • Change From Baseline to Week-26 in Alzheimer's Disease Assessment Scale-Cognitive Subscale 11 (ADAS-Cog 11)

    Mean change from baseline at week 26 is assessed for ADAS-Cog11 score. The ADAS-Cog11 is a structured scale that evaluates memory, orientation, attention, reasoning, language, and constructional praxis. ADAS-Cog11 measures cognition by assessing 11 metrics impaired in AD: word recall; commands; constructional praxis; naming objects and fingers; ideational praxis; orientation; word recognition; remembering test instructions; spoken language ability; word-finding difficulty; and comprehension of spoken language. The scale ranges from 0 to 70, with higher scores indicate greater impairment.

    Baseline to Week 26

Secondary Outcomes (4)

  • Change From Baseline to Week-26 in Clinical Dementia Rating Scale - Sum of Boxes (CDR-SB)

    Baseline to Week 26

  • Change From Baseline to Week-26 in Alzheimer's Disease Cooperative Study Group-Activities of Daily Living (ADCS-ADL)

    Baseline to Week 26

  • Change From Baseline to Week-26 in Neuropsychiatric Inventory (NPI)

    Baseline to Week 26

  • Change From Baseline to Week-26 in Change in Mini Mental State Examination (MMSE)

    Baseline to Week 26

Study Arms (3)

Experimental: SUVN-502 Low dose (50 mg)

ACTIVE COMPARATOR

SUVN-502 Low dose adjunct to base treatment with Donepezil and Memantine

Drug: SUVN-502Drug: DonepezilDrug: Memantine

Experimental: SUVN-502 High dose (100 mg)

ACTIVE COMPARATOR

SUVN-502 High dose adjunct to base treatment with Donepezil and Memantine

Drug: SUVN-502Drug: DonepezilDrug: Memantine

Placebo

PLACEBO COMPARATOR

Placebo adjunct to base treatment with Donepezil and Memantine

Drug: PlaceboDrug: DonepezilDrug: Memantine

Interventions

Once-daily, tablets, orally

Also known as: Masupirdine
Experimental: SUVN-502 High dose (100 mg)Experimental: SUVN-502 Low dose (50 mg)

Once-daily, tablets, orally

Placebo

Donepezil HCl (10 mg, once a day)

Also known as: Namzaric
Experimental: SUVN-502 High dose (100 mg)Experimental: SUVN-502 Low dose (50 mg)Placebo

Memantine HCl (10 mg, twice a day or 28 mg extended-release, once a day).

Also known as: Namenda XR®
Experimental: SUVN-502 High dose (100 mg)Experimental: SUVN-502 Low dose (50 mg)Placebo

Eligibility Criteria

Age50 Years - 85 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Has a diagnosis of probable Alzheimer's disease based on the National Institute of Neurological and Communicative Disorders and Stroke and the Alzheimer's Disease and Related Disorders Association (NINCDS-ADRDA) criteria at least 1 year prior to the screening visit.
  • Has a score between 12 and 20 inclusive on the MMSE at the screening and baseline visits.
  • Has a MRI or CT scan performed within 12 months prior to screening with findings consistent with the diagnosis of dementia due to Alzheimer's disease without any other clinically significant comorbid pathologies.
  • Must be receiving treatment with stable doses of donepezil HCl and memantine HCl for at least 3 months prior to the screening visit
  • Availability of an eligible and reliable caregiver
  • Must be living in the community or an assisted living facility.
  • Must be ambulatory or ambulatory aided (use of cane or walker).
  • Is not pregnant or planning to become pregnant during the study.
  • Subject (or subject's legally acceptable representative) and caregiver must sign an Informed Consent to participate in the study.

You may not qualify if:

  • Has a diagnosis of dementia due to other than Alzheimer's Disease
  • Is taking cholinesterase inhibitors other than donepezil HCl or taking doses of donepezil HCl other than 10 mg
  • Is taking doses of memantine HCl other than 10 mg bid or Namenda XR® 28 mg qd.
  • Has uncontrolled cardiac disease or hypertension.
  • Has clinically significant renal or hepatic impairment.
  • Has cancer or a malignant tumor, untreated thyroid disorder or has a history of seizure disorder
  • Is treated or likely to require treatment during the study, with any medications prohibited by the study protocol.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (71)

Banner Alzheimer's Institute

Phoenix, Arizona, 85006, United States

Location

Barrow Neurological Institute

Phoenix, Arizona, 85013, United States

Location

Territory Neurology & Research Institute

Tucson, Arizona, 85704, United States

Location

ATP Clinical Research, Inc.

Costa Mesa, California, 92626, United States

Location

Neuro-Pain Medical Center Inc

Fresno, California, 93710, United States

Location

Neurology Center of North Orange County

Fullerton, California, 72835, United States

Location

Senior Clinical Trials, Inc.

Laguna Hills, California, 92653, United States

Location

Collaborative Neuroscience Network, LLC

Long Beach, California, 90806, United States

Location

Easton Center for Alzheimer's Disease Research at UCLA

Los Angeles, California, 90095, United States

Location

Paradigm Research

San Diego, California, 92117, United States

Location

Associated Neurologists of South Connecticut

Fairfield, Connecticut, 06824, United States

Location

JEM Research Institute

Atlantis, Florida, 33462, United States

Location

Bradenton Research Center, Inc

Bradenton, Florida, 34205, United States

Location

Brain Matters Research

Delray Beach, Florida, 33445, United States

Location

Jacksonville Center for Clinical Research

Jacksonville, Florida, 32216, United States

Location

CCM Clinical Research Group

Miami, Florida, 33186, United States

Location

Collier Neurologic Specialists

Naples, Florida, 34102, United States

Location

Palm Beach Neurological Center

Palm Beach Gardens, Florida, 33410, United States

Location

Anchor Neuroscience

Pensacola, Florida, 32502, United States

Location

Emerald Coast Center for Neurological Disorders

Pensacola, Florida, 32514, United States

Location

Neurostudies Inc

Port Charlotte, Florida, 33952, United States

Location

The Roskamp Institute, Inc.

Sarasota, Florida, 34243, United States

Location

Brain Matters Research

Stuart, Florida, 34997, United States

Location

Neurology Clinical Research, Inc.

Sunrise, Florida, 33351, United States

Location

Axiom Clinical Research of Florida

Tampa, Florida, 33609, United States

Location

Olympian Clinical Research

Tampa, Florida, 33609, United States

Location

Stedman Clinical Trials

Tampa, Florida, 33613, United States

Location

University of South Florida - Byrd Alzheimer's Institute

Tampa, Florida, 33613, United States

Location

iResearch Atlanta, LLC

Decatur, Georgia, 30030, United States

Location

Advocate Lutheran General Hospital

Park Ridge, Illinois, 60068, United States

Location

Southern Illinois School of Medicine

Springfield, Illinois, 62702, United States

Location

Indiana University Health - University Hospital

Indianapolis, Indiana, 46202, United States

Location

Cotton-O'Neil Clinical Research Center

Topeka, Kansas, 66606, United States

Location

KU Medical Center Wichita Clinical Trial Unit

Wichita, Kansas, 67214, United States

Location

University Of Kentucky

Lexington, Kentucky, 40536, United States

Location

Pennington Biomedical Research Center

Baton Rouge, Louisiana, 70808, United States

Location

Acadia Hospital

Bangor, Maine, 04402, United States

Location

Sheppard Pratt Health System

Baltimore, Maryland, 21204, United States

Location

Clinical Research Professionals

St Louis, Missouri, 63141, United States

Location

Princeton Medical Institute

Princeton, New Jersey, 08540, United States

Location

Advanced Memory Research Institute of NJ, PC - Internal Medicine

Rahway, New Jersey, 07065, United States

Location

Advanced Memory Research Institute

Toms River, New Jersey, 08755, United States

Location

Biobehavioral Health

Toms River, New Jersey, 08755, United States

Location

Neurology Specialists of Monmouth County

West Long Branch, New Jersey, 07764, United States

Location

Neurological Associates of Albany, PC

Albany, New York, 12208, United States

Location

Integrative Clinical Trials, LLC

Brooklyn, New York, 11229, United States

Location

SPRI Clinical Trials, LLC

Brooklyn, New York, 11235, United States

Location

Mid Hudson Medical Research

New Windsor, New York, 12553, United States

Location

New York University

New York, New York, 10016, United States

Location

Eastside Comprehensive Medical Center, LLC

New York, New York, 10021, United States

Location

Manhattan Behavioral Medicine

New York, New York, 10022, United States

Location

Upstate University Hospital (SUNY Health Science Center)

Syracuse, New York, 13210, United States

Location

Five Towns Neuroscience Research

Woodmere, New York, 11598, United States

Location

New Hope Clinical Research

Charlotte, North Carolina, 28211, United States

Location

Alzheimer Memory Center

Charlotte, North Carolina, 28270, United States

Location

Richard Weisler, MD, PA

Raleigh, North Carolina, 27609, United States

Location

Ohio Clinical Research Partners, LLC

Canton, Ohio, 44718, United States

Location

Valley Medical Research

Centerville, Ohio, 45459, United States

Location

Cleveland Clinic Main Campus

Cleveland, Ohio, 44195, United States

Location

IPS Research Company

Oklahoma City, Oklahoma, 73103, United States

Location

Lynn Health Science Institute

Oklahoma City, Oklahoma, 73112, United States

Location

Tulsa Clinical Research, LLC

Tulsa, Oklahoma, 74104, United States

Location

Lehigh Valley Health Network

Allentown, Pennsylvania, 18103, United States

Location

Northeastern Pennsylvania Memory and Alzheimers Center

Plains, Pennsylvania, 18705, United States

Location

Roper St. Francis Healthcare

Charleston, South Carolina, 29401, United States

Location

University of North Texas Health Science Center

Fort Worth, Texas, 76107, United States

Location

Shepherd Healthcare

Lewisville, Texas, 75067, United States

Location

Radiant Research, Inc.

San Antonio, Texas, 78229, United States

Location

Wasatch Clinical Research

Salt Lake City, Utah, 84107, United States

Location

Center for Alzheimer's Care, Imaging and Research

Salt Lake City, Utah, 84108, United States

Location

Independent Psychiatric Consultants, SC, dba

Waukesha, Wisconsin, 53188, United States

Location

Related Publications (3)

  • Nirogi R, Jayarajan P, Benade V, Shinde A, Goyal VK, Jetta S, Ravula J, Abraham R, Grandhi VR, Subramanian R, Pandey SK, Badange RK, Mohammed AR, Jasti V, Ballard C, Cummings J. Potential beneficial effects of masupirdine (SUVN-502) on agitation/aggression and psychosis in patients with moderate Alzheimer's disease: Exploratory post hoc analyses. Int J Geriatr Psychiatry. 2022 Oct;37(10):10.1002/gps.5813. doi: 10.1002/gps.5813.

  • Nirogi R, Ieni J, Goyal VK, Ravula J, Jetta S, Shinde A, Jayarajan P, Benade V, Palacharla VRC, Dogiparti DK, Jasti V, Atri A, Cummings J. Effect of masupirdine (SUVN-502) on cognition in patients with moderate Alzheimer's disease: A randomized, double-blind, phase 2, proof-of-concept study. Alzheimers Dement (N Y). 2022 Jun 1;8(1):e12307. doi: 10.1002/trc2.12307. eCollection 2022.

  • Nirogi R, Goyal VK, Benade V, Subramanian R, Ravula J, Jetta S, Shinde A, Pandey SK, Jayarajan P, Jasti V, Cummings J. Effect of Concurrent Use of Memantine on the Efficacy of Masupirdine (SUVN-502): A Post Hoc Analysis of a Phase 2 Randomized Placebo-Controlled Study. Neurol Ther. 2022 Dec;11(4):1583-1594. doi: 10.1007/s40120-022-00390-4. Epub 2022 Jul 31.

Related Links

MeSH Terms

Conditions

Alzheimer Disease

Interventions

1-((2-bromophenyl)sulfonyl)-5-methoxy-3-((4-methyl-1-piperazinyl)methyl)-1H-indole dimesylate monohydrateDonepezilNamzaricMemantine

Condition Hierarchy (Ancestors)

DementiaBrain DiseasesCentral Nervous System DiseasesNervous System DiseasesTauopathiesNeurodegenerative DiseasesNeurocognitive DisordersMental Disorders

Intervention Hierarchy (Ancestors)

IndansIndenesPolycyclic Aromatic HydrocarbonsHydrocarbons, AromaticHydrocarbons, CyclicHydrocarbonsOrganic ChemicalsPiperidinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsPolycyclic CompoundsAmantadineAdamantaneBridged-Ring Compounds

Results Point of Contact

Title
Ramakrishna Nirogi, PhD
Organization
Suven Life Sciences

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
GT60
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 17, 2015

First Posted

October 20, 2015

Study Start

September 1, 2015

Primary Completion

November 5, 2019

Study Completion

November 7, 2019

Last Updated

June 9, 2023

Results First Posted

June 9, 2023

Record last verified: 2023-05

Locations