NCT02438007

Brief Summary

The purpose of this study is to compare galeterone to enzalutamide in men expressing androgen receptor spice variant-7 mRNA (AR-V7) in metastatic (M1) castrate resistant prostate cancer (CRPC).

Trial Health

63
Monitor

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
953

participants targeted

Target at P75+ for phase_3 prostate-cancer

Timeline
Completed

Started Jun 2015

Shorter than P25 for phase_3 prostate-cancer

Geographic Reach
8 countries

117 active sites

Status
terminated

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

March 19, 2015

Completed
2 months until next milestone

First Posted

Study publicly available on registry

May 8, 2015

Completed
24 days until next milestone

Study Start

First participant enrolled

June 1, 2015

Completed
1.1 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

July 1, 2016

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

November 1, 2016

Completed
Last Updated

March 15, 2023

Status Verified

September 1, 2017

Enrollment Period

1.1 years

First QC Date

March 19, 2015

Last Update Submit

March 13, 2023

Conditions

Outcome Measures

Primary Outcomes (1)

  • Radiographic Progression-free survival

    ≥ 8 months

Secondary Outcomes (2)

  • Overall Survival

    ≥ 8 months

  • Time to Initiation of Cytotoxic Chemotherapy

    ≥ 8 months

Other Outcomes (6)

  • Skeletal-related Events

    ≥ 8 months

  • Safety measured by clinical safety laboratories and adverse events

    ≥ 8 months

  • Prostate Specific Antigen (PSA) Response ≥ 50%

    ≥ 8 months

  • +3 more other outcomes

Study Arms (2)

Galeterone

EXPERIMENTAL
Drug: Galeterone

Enzalutamide

ACTIVE COMPARATOR
Drug: Enzalutamide

Interventions

2550 mg galeterone tablets once daily PO

Also known as: TOK-001
Galeterone

160 mg enzalutamide capsules once daily PO

Also known as: Xtandi®
Enzalutamide

Eligibility Criteria

Age18 Years+
Sexmale
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Progressive metastatic (M1) disease on androgen deprivation therapy
  • Detectable AR-V7 from circulating tumors (CTCs)
  • ECOG performance status 0 or 1

You may not qualify if:

  • Prior treatment with second generation anti-androgens (e.g. abiraterone, enzalutamide)
  • Prior treatment with chemotherapy for CRPC

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (117)

Pinnacle Oncology Hematology

Scottsdale, Arizona, 85258, United States

Location

University Of Arizona Cancer Center

Tucson, Arizona, 85724, United States

Location

City of Hope

Duarte, California, 91010, United States

Location

USC Norris Comprehensive Cancer Center

Los Angeles, California, 90033, United States

Location

UCLA Jonsson Comprehensive Cancer Center

Los Angeles, California, 90095, United States

Location

Prostate Oncology Specialists, Inc.

Marina del Rey, California, 90292, United States

Location

UC Davis Cancer Center

Sacramento, California, 95817, United States

Location

San Bernardino Urological Associates

San Bernardino, California, 92404, United States

Location

Urology Speciality Group

Torrance, California, 90505, United States

Location

University of Colorado Cancer Center Anschultz Cancer Pavilion

Aurora, Colorado, 80045, United States

Location

The Urology Center of Colorado

Denver, Colorado, 80211, United States

Location

Yale University School of Medicine

New Haven, Connecticut, 06510, United States

Location

Georgetown University Medical Center

Washington D.C., District of Columbia, 20007, United States

Location

Sibley Memorial Hospital

Washington D.C., District of Columbia, 20016, United States

Location

Boca Raton Community Hospital, Inc.

Boca Raton, Florida, 33486, United States

Location

University of Florida Health Cancer Center

Orlando, Florida, 32806, United States

Location

Moffitt Cancer Center

Tampa, Florida, 33612, United States

Location

First Urology

Jeffersonville, Indiana, 47130, United States

Location

Tulane Medical Center

New Orleans, Louisiana, 70115, United States

Location

Regional Urology, LLC

Shreveport, Louisiana, 71106, United States

Location

University of Maryland Greenenbaum Cancer Center

Baltimore, Maryland, 21201, United States

Location

Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins

Baltimore, Maryland, 21205, United States

Location

Walter Reed National Military Medical Center

Bethesda, Maryland, 20307, United States

Location

Massachusetts General Hospital

Boston, Massachusetts, 02114, United States

Location

Dana-Farber Cancer Institute

Boston, Massachusetts, 02115, United States

Location

Beth Israel Deaconess Medical Center

Boston, Massachusetts, 02215, United States

Location

University of Michigan Health System

Ann Arbor, Michigan, 48109, United States

Location

Karmanos Cancer Center

Detroit, Michigan, 48201, United States

Location

Urology Cancer Center and GU Research Network

Omaha, Nebraska, 68130, United States

Location

Coastal Urology Associates

Brick, New Jersey, 08724, United States

Location

Brooklyn Urology Research Group

Brooklyn, New York, 11215, United States

Location

Advanced Urology Centers of New York

Plainview, New York, 11803, United States

Location

Premier Medical Group of the Hudson Valley

Poughkeepsie, New York, 12601, United States

Location

Associated Medical Professionals of NY

Syracuse, New York, 13210, United States

Location

University of North Carolina Lineberger Cancer Center

Chapel Hill, North Carolina, 27599, United States

Location

Carolina Urology Partners, PLLC

Charlotte, North Carolina, 28277, United States

Location

Carolina Urology Partners

Concord, North Carolina, 28025, United States

Location

The Urology Group

Cincinnati, Ohio, 45212, United States

Location

Clinical Research Solutions

Middleburg Heights, Ohio, 44130, United States

Location

Oregon Urology Institute

Springfield, Oregon, 97477, United States

Location

Lancaster Urology

Lancaster, Pennsylvania, 17604, United States

Location

Fox Chase Cancer Center

Philadelphia, Pennsylvania, 19111, United States

Location

UPMC Cancer Centers

Pittsburgh, Pennsylvania, 15232, United States

Location

Carolina Urologic Research Center

Myrtle Beach, South Carolina, 29572, United States

Location

Urology Associates Clinical Research

Nashville, Tennessee, 37209, United States

Location

Urology Clinics of North Texas

Dallas, Texas, 75231, United States

Location

Texas Oncology/Baylor University Medical Center

Dallas, Texas, 75246, United States

Location

Urology San Antonio

San Antonio, Texas, 78229, United States

Location

Virginia Urology

Richmond, Virginia, 23235, United States

Location

Urology of Virginia

Virginia Beach, Virginia, 23462, United States

Location

The University of Wisconsin Paul P. Carbone Comprehensive Cancer Center

Madison, Wisconsin, 53792, United States

Location

St. George Private Hospital, Oncology Day Care Centre

Kogarah, New South Wales, 2217, Australia

Location

Ashford Cancer Centre/Adelaide Cancer Centre Research

Kurralta Park, New South Wales, 5037, Australia

Location

North Coast Cancer Institute

Port Macquarie, New South Wales, 2444, Australia

Location

Prince of Wales Hospital

Randwick, New South Wales, 2031, Australia

Location

Macquarie University

Sydney, New South Wales, 2109, Australia

Location

Peninsula Specialist Centre

Kippa-Ring, Queensland, 4102, Australia

Location

ICON Cancer Care

Southport, Queensland, 4215, Australia

Location

Princess Alexandra Hospital

Woolloongabba, Queensland, 4102, Australia

Location

Ashford Cancer Centre/Adelaide Cancer Centre Research

Kurralta Park, South Australia, 5037, Australia

Location

Box Hill Hospital

Box Hill, Victoria, 3128, Australia

Location

Monash Medical Centre

East Bentleigh, Victoria, 3165, Australia

Location

Peter MacCallum Cancer Centre

East Melbourne, Victoria, 3002, Australia

Location

Cabrini Hospital

Malvern, Victoria, 3144, Australia

Location

Jules Bordet Institute Clinique d'Oncologie Medicale

Brussels, B-1000, Belgium

Location

Universitair Ziekenhuis Gent

Ghent, B-9000, Belgium

Location

Jessa Ziekenhuis

Hasselt, B-3500, Belgium

Location

CHU Sart Tilman

Liège, 4000, Belgium

Location

British Columbia Cancer

Kelowna, British Columbia, V1Y 5L3, Canada

Location

British Columbia Cancer

Vancouver, British Columbia, V5Z 4E6, Canada

Location

London Health Sciences Centre

London, Ontario, N6A 4L6, Canada

Location

Sunnybrook Research Institute

Toronto, Ontario, M4N 3M5, Canada

Location

Princess Margaret Hospital

Toronto, Ontario, M5G 2M9, Canada

Location

Centre Hospitalier De I'Universite de Montreal

Montreal, Quebec, H2L 4M1, Canada

Location

Centre Hospitalier Universitaire de Quebec

Québec, Quebec, G1R 3S1, Canada

Location

Centre Paul Papin

Angers, 49055, France

Location

Institut Sainte Catherine

Avignon, 84918, France

Location

Institut Bergonié

Bordeaux, 33076, France

Location

Centre François Baclesse

Caen, 14076, France

Location

Service de Médecine Interne Onco-Hématologie

La Roche-sur-Yon, 85925, France

Location

Clinique Victor Hugo Centre Jean Bernard

Le Mans, 72000, France

Location

Centre Léon Bérard

Lyon, 69008, France

Location

Hôpital Edouard Herriot

Lyon, Cedex 03, France

Location

Centre Antoine Lacassagne

Nice, 06189, France

Location

Centre René Gauducheau

Saint-Herblain, 44805, France

Location

Institut de Cancérologie de l'Ouest

Saint-Herblain, 44805, France

Location

Institut de Cancerlogie de la Loire

Saint-Priest-en-Jarez, 42271, France

Location

Institut Gustave-Roussy

Villejuif, 94805, France

Location

Centro Oncologico c/o Presidio Ospedaliero San Donato - Arezzo

Arezzo, 52100, Italy

Location

Unità Operativa di Oncologia Ospedale Civile degli Infe

Faenza (RA), 48018, Italy

Location

Romagnolo per lo Studio e la Cura dei Tumori IRST-IRCCS - Oncologia medica

Meldola (FC), 47014, Italy

Location

AOU "S. Luigi", SCDU Oncologia Medica

Orbassano (Torino), 10043, Italy

Location

Az. Ospedaliera San Camillo-Forlanini

Roma, 00152, Italy

Location

University of Turin

Torino, 10126, Italy

Location

Santa Chiara Hospital

Trento, 38122, Italy

Location

Hospital Clínic i Provincial de Barcelona-Oncology

Barcelona, 08036, Spain

Location

Instituto Catalan de Oncologia (Hospital Durans i Reynals)

Barcelona, 08908, Spain

Location

Hospital General Universitario de Elche

Elche, 3203, Spain

Location

Hospital General Universitario Gregorio Marañón

Madrid, 28009, Spain

Location

Spanish National Cancer Research Centre

Madrid, 28050, Spain

Location

Fundación Althaia Manresa

Manresa, 08243, Spain

Location

Unidad Cnio Ibima de Investigacion en Prostata

Málaga, Spain

Location

Hospital Son Espases - Oncología

Palma de Mallorca, 07010, Spain

Location

Hospital Clinico Universitario de Navarra

Pamplona, 31008, Spain

Location

Consorci Hospitalari de Parc Taulí

Sabadell, 08208, Spain

Location

Hospital Universitario Virgen del Rocio

Seville, 41013, Spain

Location

IVO-Oncología Médica

Valencia, 46009, Spain

Location

CR-UK Institute for Cancer Studies

Birmingham, England, B15 2PR, United Kingdom

Location

Sussex Cancer Centre

Brighton, England, BN2 5BE, United Kingdom

Location

University College of London Hospitals

London, England, NWI 2PG, United Kingdom

Location

Guy's and St. Thomas' NHS Foundation Trust

London, England, SE1 9RT, United Kingdom

Location

Southampton General Hospital

Southampton, England, SO16 6YD, United Kingdom

Location

University of Surrey Post Graduate Medical Hospital

Surrey, England, GU2 7WG, United Kingdom

Location

Royal Marsden Hospital

Surrey, England, SM2 5PT, United Kingdom

Location

The Royal Cornwall Hospital

Truro, England, TR1 3LJ, United Kingdom

Location

The Beatson West of Scotland Cancer Centre

Glasgow, Scotland, G12 0YN, United Kingdom

Location

Velindre Hospital

Cardiff, Wales, CF14 2TL, United Kingdom

Location

Related Publications (1)

  • Aragon-Ching JB. The promising role of poly(ADP-ribose) polymerase inhibitors in prostate cancer. Asian J Androl. 2016 Jul-Aug;18(4):592-3. doi: 10.4103/1008-682X.172821.

MeSH Terms

Conditions

Prostatic Neoplasms

Interventions

3-hydroxy-17-(1H-benzimidazole-1-yl)androsta-5,16-dieneenzalutamide

Condition Hierarchy (Ancestors)

Genital Neoplasms, MaleUrogenital NeoplasmsNeoplasms by SiteNeoplasmsGenital Diseases, MaleGenital DiseasesUrogenital DiseasesProstatic DiseasesMale Urogenital Diseases

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
NONE
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

March 19, 2015

First Posted

May 8, 2015

Study Start

June 1, 2015

Primary Completion

July 1, 2016

Study Completion

November 1, 2016

Last Updated

March 15, 2023

Record last verified: 2017-09

Locations