NCT02345226

Brief Summary

The primary objective of this study is to evaluate the non-inferiority of switching to emtricitabine/rilpivirine/tenofovir alafenamide (FTC/RPV/TAF) fixed dose combination (FDC) as compared to continuing the non-nucleoside reverse transcriptase inhibitor (NNRTI) regimen of efavirenz /FTC/tenofovir disoproxil fumarate (EFV/FTC/TDF) FDC in virologically-suppressed HIV-1 infected participants.

Trial Health

93
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
881

participants targeted

Target at P75+ for phase_3

Timeline
Completed

Started Jan 2015

Typical duration for phase_3

Geographic Reach
9 countries

117 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

January 19, 2015

Completed
7 days until next milestone

First Posted

Study publicly available on registry

January 26, 2015

Completed
Same day until next milestone

Study Start

First participant enrolled

January 26, 2015

Completed
1.4 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

June 29, 2016

Completed
1.3 years until next milestone

Results Posted

Study results publicly available

October 19, 2017

Completed
1.2 years until next milestone

Study Completion

Last participant's last visit for all outcomes

January 2, 2019

Completed
Last Updated

January 2, 2020

Status Verified

December 1, 2019

Enrollment Period

1.4 years

First QC Date

January 19, 2015

Results QC Date

September 21, 2017

Last Update Submit

December 16, 2019

Conditions

Keywords

HIV

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Week 48 as Defined by the US FDA-defined Snapshot Algorithm

    The percentage of participants achieving HIV-1 RNA \< 50 copies/mL at Week 48 was analyzed using the snapshot algorithm, which defines a patient's virologic response status using only the viral load at the predefined time point within an allowed window of time, along with study drug discontinuation status.

    Week 48

Secondary Outcomes (11)

  • Percentage of Participants With HIV-1 RNA ≥ 50 Copies/mL at Week 48 as Defined by the US FDA-defined Snapshot Algorithm

    Week 48

  • Percentage of Participants With HIV-1 RNA ≥ 50 Copies/mL at Week 96 as Defined by the US FDA-defined Snapshot Algorithm

    Week 96

  • Percentage of Participants With HIV-1 RNA < 50 Copies/mL at Week 96 as Defined by the US FDA-defined Snapshot

    Week 96

  • Change From Baseline in CD4+ Cell Count at Week 48

    Baseline; Week 48

  • Change From Baseline in CD4+ Cell Count at Week 96

    Baseline; Week 96

  • +6 more secondary outcomes

Study Arms (3)

FTC/RPV/TAF

EXPERIMENTAL

FTC/RPV/TAF plus EFV/FTC/TDF placebo for at least 96 weeks.

Drug: FTC/RPV/TAFDrug: EFV/FTC/TDF Placebo

EFV/FTC/TDF

ACTIVE COMPARATOR

EFV/FTC/TDF plus FTC/RPV/TAF placebo for at least 96 weeks.

Drug: EFV/FTC/TDFDrug: FTC/RPV/TAF Placebo

Open Label Extension Phase

EXPERIMENTAL

After the Week 96 visit, participants will be given the option to receive open label FTC/RPV/TAF for up to an additional 48 weeks. In countries where FTC/RPV/TAF is not yet commercially available, participants will be given the option to receive open-label FTC/RPV/TAF and attend visits every 12 weeks until FTC/RPV/TAF becomes commercially available, or until Gilead elects to discontinue the study, whichever occurs first.

Drug: FTC/RPV/TAF

Interventions

200/25/25 mg FDC tablets administered orally once daily

Also known as: Odefsey®
FTC/RPV/TAFOpen Label Extension Phase

Tablets administered orally once daily

FTC/RPV/TAF

600/200/300 mg FDC tablets administered orally once daily

Also known as: Atripla®
EFV/FTC/TDF

Tablets administered orally once daily

EFV/FTC/TDF

Eligibility Criteria

Age18 Years+
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • The ability to understand and sign a written informed consent form, which must be obtained prior to initiation of study procedures
  • Currently receiving EFV/FTC/TDF FDC for ≥ 6 consecutive months preceding the screening visit
  • Documented plasma HIV-1 RNA levels \< 50 copies/mL (or undetectable HIV-1 RNA level according to the local assay being used if the limit of detection is \> 50 copies/mL) for ≥ 6 months preceding the screening visit. Unconfirmed virologic elevation of ≥ 50 copies/mL after previously reaching viral suppression (transient detectable viremia, or "blip") and prior to screening is acceptable
  • Have no documented resistance to any of the study agents at any time in the past
  • HIV-1 RNA \< 50 copies/mL at the screening visit
  • Hepatic transaminases (AST and ALT) ≤ 5 × upper limit of normal (ULN)
  • Total bilirubin ≤ 1.5 mg/dL, or normal direct bilirubin
  • Adequate hematologic function (absolute neutrophil count ≥ 1,000/mm\^3; platelets ≥ 50,000/mm\^3; hemoglobin ≥ 8.5 g/dL)
  • Serum amylase ≤ 5 × ULN (individuals with serum amylase \> 5 × ULN will remain eligible if serum lipase is ≤ 5 × ULN)
  • Normal ECG (or if abnormal, determined by the Investigator to be not clinically significant)
  • Adequate renal function: Estimated glomerular filtration rate ≥ 50 mL/min according to the Cockcroft-Gault formula

You may not qualify if:

  • Hepatitis B surface antigen (HBsAg) positive
  • Hepatitis C antibody positive with detectable hepatitis C virus (HCV) RNA (individuals who have HCV antibody but no detectable HCV RNA are eligible to enroll)
  • Individuals experiencing or with a medical history of decompensated cirrhosis (e.g., ascites, encephalopathy, etc.)
  • Females who are breastfeeding
  • Positive serum pregnancy test
  • Current alcohol or substance use judged by the Investigator to potentially interfere with the individual's study compliance
  • A history of malignancy within the past 5 years (prior to screening) or ongoing malignancy other than cutaneous Kaposi's sarcoma (KS), basal cell carcinoma, or resected, non-invasive cutaneous squamous carcinoma. Individuals with cutaneous KS are eligible, but must not have received any systemic therapy for KS within 30 days of Baseline/Day 1 and must not be anticipated to require systemic therapy during the study
  • Active, serious infections (other than HIV-1 infection) requiring parenteral antibiotic or antifungal therapy within 30 days prior to Baseline/Day 1
  • Any other clinical condition or prior therapy that, in the opinion of the Investigator, would make the individual unsuitable for the study or unable to comply with dosing requirements
  • Participation in any other clinical trial (including observational trials) without prior approval from the sponsor is prohibited while participating in this trial
  • Individuals receiving ongoing therapy with any of the disallowed medications listed in the protocol, including drugs not to be used with FTC, RPV and/or TAF; or individuals with any known allergies to the excipients of FTC/RPV/TAF

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (117)

Maricopa Integrated Health System

Phoenix, Arizona, 85004, United States

Location

Spectrum Medical Group

Phoenix, Arizona, United States

Location

AHF Research Center

Beverly Hills, California, United States

Location

Pacific Oaks Medical Group

Beverly Hills, California, United States

Location

Long Beach Education and Research Consultants

Long Beach, California, United States

Location

Kaiser Permanente

Los Angeles, California, United States

Location

Southern California Men's Medical Group

Los Angeles, California, United States

Location

Tarrant County ID Associates

Los Angeles, California, United States

Location

Kaiser Permanente

Sacramento, California, United States

Location

University of California-UC Davis

Sacramento, California, United States

Location

La Playa Medical Group and Clinical Research

San Diego, California, United States

Location

Kaiser Permanente

San Francisco, California, United States

Location

Optimus Medical

San Francisco, California, United States

Location

Kaiser Permanente

San Leandro, California, United States

Location

Los Angeles BioMedical Institute at Harbor-UCLA Medical Center

Torrance, California, United States

Location

University of Colorado

Aurora, Colorado, United States

Location

Apex Research Institute

Denver, Colorado, United States

Location

Yale University School of Medicine

New Haven, Connecticut, United States

Location

World Health Clinicians' CIRCLE CARE Center

Norwalk, Connecticut, United States

Location

Capital Medical Associates, P.C.

Washington D.C., District of Columbia, United States

Location

Medical Faculty Associates, Inc.

Washington D.C., District of Columbia, United States

Location

Whitman Walker Clinic

Washington D.C., District of Columbia, United States

Location

Gary Richmond, MD, PA, Inc.

Fort Lauderdale, Florida, United States

Location

Therafirst Medical Centers

Fort Lauderdale, Florida, United States

Location

Midway Immunology & Research Center, LLC

Ft. Pierce, Florida, United States

Location

AIDS Healthcare Foundation

Miami, Florida, United States

Location

University of Miami

Miami, Florida, United States

Location

AIDS Healthcare Foundation

Miami Beach, Florida, United States

Location

Orlando Immunology Center

Orlando, Florida, United States

Location

Infectious Diseases Associates of NW Florida, P.A.

Pensacola, Florida, United States

Location

Hillsborough County Health Dept.

Tampa, Florida, United States

Location

Infectious Disease Research Institute Inc.

Tampa, Florida, United States

Location

St. Joseph's Comprehensive Research Institute

Tampa, Florida, United States

Location

AIDS Research & Treatment Center of the Treasure Coast

Vero Beach, Florida, United States

Location

Triple O Research Institute, P.A.

West Palm Beach, Florida, United States

Location

Rowan Tree Medical PA

Wilton Manors, Florida, United States

Location

AIDS Research Consortium of Atlanta

Atlanta, Georgia, United States

Location

Atlanta ID Group

Atlanta, Georgia, United States

Location

Infectious Disease Specialists of Atlanta

Decatur, Georgia, United States

Location

Mercer University School of Medicine

Macon, Georgia, United States

Location

Chatham County Health Department

Savannah, Georgia, United States

Location

The CORE Foundation

Chicago, Illinois, United States

Location

Indiana University Medical Center

Indianapolis, Indiana, United States

Location

Boston University Medical Center

Boston, Massachusetts, United States

Location

Brigham and Women's

Boston, Massachusetts, United States

Location

MetroWest Medical Center

Framingham, Massachusetts, United States

Location

Baystate Infectious Diseases Clinical Research

Springfield, Massachusetts, United States

Location

The Research Institute

Springfield, Massachusetts, United States

Location

Be Well Medical Center

Berkley, Michigan, United States

Location

Henry Ford Health System

Detroit, Michigan, United States

Location

Hennepin County Medical Center

Minneapolis, Minnesota, United States

Location

Southampton Healthcare, Inc.

St Louis, Missouri, United States

Location

Saint Michael's Medical Center

Newark, New Jersey, United States

Location

South Jersey Infectious Disease

Somers Point, New Jersey, United States

Location

Southwest CARE Center

Santa Fe, New Mexico, United States

Location

Upstate Infectious Diseases Associates

Albany, New York, United States

Location

North Shore University Hospital

Manhasset, New York, United States

Location

Columbia University Medical Center/ New York Presbyterian

New York, New York, United States

Location

Jacobi Medical Center

The Bronx, New York, United States

Location

Montefiore Medical Center

The Bronx, New York, United States

Location

University of North Carolina at Chapel Hill

Chapel Hill, North Carolina, United States

Location

Infectious Disease Consultants, PA

Charlotte, North Carolina, United States

Location

The Brody School of Medicine

Greenville, North Carolina, United States

Location

Rosedale Infectious Diseases

Huntersville, North Carolina, United States

Location

The Ohio State University

Columbus, Ohio, United States

Location

University of Pennsylvania

Philadelphia, Pennsylvania, United States

Location

The Miriam Hospital

Providence, Rhode Island, United States

Location

Medical University of South Carolina

Charleston, South Carolina, United States

Location

Central Texas Clinical Research

Austin, Texas, United States

Location

North Texas Infectious Diseases Consultants

Dallas, Texas, United States

Location

Southwest Infectious Disease Clinical Research, Inc.

Dallas, Texas, United States

Location

Trinity Health and Wellness Center/AIDS Arms, Inc.

Dallas, Texas, United States

Location

AIDS Arms, Inc./Trinity Health & Wellness Center

Fort Worth, Texas, United States

Location

Gordon E. Crofoot, MD, PA

Houston, Texas, United States

Location

Research Access Network

Houston, Texas, United States

Location

DCOL Center for Clinical Research

Longview, Texas, United States

Location

Clinical Alliance for Research & Education - Infectious Diseases, LLC (CARE-ID)

Annandale, Virginia, United States

Location

Peter Shalit, MD

Seattle, Washington, United States

Location

Premier Clinical Research

Spokane, Washington, United States

Location

CHU Saint-Pierre University Hospital

Brussels, Belgium

Location

Cliniques Universitaires UCL Saint-Luc

Brussels, Belgium

Location

University of Alberta

Edmonton, Alberta, Canada

Location

Spectrum Health

Vancouver, British Columbia, Canada

Location

Health Sciences Centre

Winnipeg, Manitoba, Canada

Location

Maple Leaf Research

Toronto, Ontario, Canada

Location

University Health Network

Toronto, Ontario, Canada

Location

Clinique medicale l'Actuel

Montreal, Quebec, Canada

Location

Clinique OPUS

Montreal, Quebec, Canada

Location

McGill University Health Centre

Montreal, Quebec, Canada

Location

Hopital Bichat Claude Bernard

Paris, France

Location

Hopital Saint Louis

Paris, France

Location

Chu Tours

Tours, France

Location

Zentrum für Infektiologie Berlin Prenzlauer Berg GmbH (zibp)

Berlin, Germany

Location

University of Bonn

Bonn, Germany

Location

Universitat zu Koln

Cologne, Germany

Location

Center for HIV and Hepatogastroenterology

Düsseldorf, Germany

Location

Universitätsklinikum Essen

Essen, Germany

Location

Infektiologikum

Frankfurt, Germany

Location

ICH Study Center Hamburg

Hamburg, Germany

Location

Universitaetsklinikum Hamburg-Eppendorf

Hamburg, Germany

Location

MUC Research GmbH

München, Germany

Location

Clinical Research Puerto Rico Inc

San Juan, Puerto Rico

Location

Hope Clinical Research

San Juan, Puerto Rico

Location

University of Puerto Rico School of Medicine

San Juan, Puerto Rico

Location

Hospital General Universitario de Alicante

Alicante, Spain

Location

Hospital Clinic i Provincial

Barcelona, Spain

Location

Hospital del Mar

Barcelona, Spain

Location

Hospital Universitary de Bellvitge

Barcelona, Spain

Location

Hospital Universitario 12 de Octubre

Madrid, Spain

Location

Hospital Universitario La Paz

Madrid, Spain

Location

University Hospital Basel

Basel, Switzerland

Location

Geneva University Hospital

Geneva, Switzerland

Location

Centre Hospitalier Universitaire Vaudois

Lausanne, Switzerland

Location

Barts & The London NHS Trust

London, United Kingdom

Location

King's College Hospital

London, United Kingdom

Location

Mortimer Market Centre

London, United Kingdom

Location

The Royal Free Hampstead NHS Trust

London, United Kingdom

Location

Related Publications (11)

  • Hagins D, Orkin C, Daar ES, Mills A, Brinson C, DeJesus E, Post FA, Morales-Ramirez J, Thompson M, Osiyemi O, Rashbaum B, Stellbrink HJ, Martorell C, Liu H, Liu YP, Porter D, Collins SE, SenGupta D, Das M. Switching to coformulated rilpivirine (RPV), emtricitabine (FTC) and tenofovir alafenamide from either RPV, FTC and tenofovir disoproxil fumarate (TDF) or efavirenz, FTC and TDF: 96-week results from two randomized clinical trials. HIV Med. 2018 Nov;19(10):724-733. doi: 10.1111/hiv.12664. Epub 2018 Aug 12.

  • Mills A, Brinson C, Martorell C, Crofoot G, Daar E, Osiyemi O, et al. Switching to RPV/FTC/TAF from RPV/FTC/TDF or EFV/FTC/TDF: Week 96 Results. Conference on Retroviruses and Opportunistic Infections, Boston. March 4-7, 2018, Abstract 504.

    RESULT
  • Arribas JR, Rockstroh J, Post, Yazdanpanah Y, Cavassini, DeJesus E, et al. Bone and renal safety of switching to rilpivirine/emtricitabine/tenofovir alafenamide (RPV/FTC/TAF) from single-tablet regimens (STRs) containing efavirenz/emtricitabine/tenofovir disoproxil fumarate (EFV/FTC/TDF) or rilpivirine/emtricitabine/tenofovir disoproxil fumarate (RPV/FTC/TDF): Week 48 subgroup analysis in patients at risk of or with comorbidities. Abstract accepted for presentation at the 16th European AIDS Conference, 2017 25-27 October Milan, Italy.

    RESULT
  • Porter DP, KulkarniR, Cao H, SenGupta D, and White KL. No Emergent Resistance in HIV-1 Virologically-Suppressed Subjects Who Switched to RPV/FTC/TAF [Poster 1381]. ID Week 2017 4-8 October; San Diego, California.

    RESULT
  • E DeJesus, M Ramgopal, G Crofoot, P Ruane, A LaMarca. J-M Molina et al. Efficacy and Safety of Switching to RPV/FTC/TAF in Older Adults. 8th International Workshop on HIV and Aging 2017 2-3 October, New York, New York.

    RESULT
  • Molina JM, DeJesus E, Rijnders B, Post FAV, B., Stoeckle M, ThalmeA, et al. Efficacy and Safety of Switching From RPV/FTC/TDF or EFV/FTC/TDF to RPV/FTC/TAF in Black Adults [Presentation MOPEB0291]. 9th IAS Conference on HIV Science 2017 23-26 July Paris, France.

    RESULT
  • Rockstroh J, Orkin C, Yazdanpanah Y, Di Perri GDS, P. E., Arribas JR, Brinkman K, et al. Switching From TDF to TAF Improves Bone and Renal Safety Independent of Age, Sex, Race, or 3rd Agent: Results From Pooled Analysis (N=3816) of Virologically Suppressed HIV-1 Infected Adults [Presentation MOPEB0289]. 9th IAS Conference on HIV Science; 2017 23 26 July Paris, France.

    RESULT
  • DeJesus E, Ramgopal M, Crofoot G, Ruane P, LaMarca A, Mills A, Martorell CT, de Wet J, Stellbrink HJ, Molina JM, Post FA, Valero IP, Porter D, Liu Y, Cheng A, Quirk E, SenGupta D, Cao H. Switching from efavirenz, emtricitabine, and tenofovir disoproxil fumarate to tenofovir alafenamide coformulated with rilpivirine and emtricitabine in virally suppressed adults with HIV-1 infection: a randomised, double-blind, multicentre, phase 3b, non-inferiority study. Lancet HIV. 2017 May;4(5):e205-e213. doi: 10.1016/S2352-3018(17)30032-2. Epub 2017 Mar 2.

  • Majeed SR, Shao Y, Garner W, Scott J, Pérez-Ruixo C, SenGupta D, et al. Evaluation of RPV/FTC/TAF Exposure-Efficacy and Exposure-Safety Relationships [Poster 427]. Conference on Retroviruses and Opportunistic Infections (CROI) 2017 13-16 February; Seattle, Washington.

    RESULT
  • Hagins D, Mills A, Martorell C, Walmsley S, Gallant J, Tebas P, et al. Efficacy and Safety of Switching to RPV/FTC/TAF in Women [Abstract 12]. 7th International Workshop on HIV & Women; 2017 11-12 February; Seattle, Washington.

    RESULT
  • Orkin C, DeJesus E, Ramgopal M, Crofoot G, Ruane P, LaMarca A, et al. 48 Week Results from two studies: Switching to RPV/FTC/TAF from EFV/FTC/TDF (Study 1160) or RPV/FTC/TDF (Study 1216) [Presentation]. HIV Glasgow; 2016 23-26 October; Glasgow, United Kingdom.

    RESULT

MeSH Terms

Interventions

Efavirenz, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination

Intervention Hierarchy (Ancestors)

TenofovirOrganophosphonatesOrganophosphorus CompoundsOrganic ChemicalsOxazinesHeterocyclic Compounds, 1-RingHeterocyclic CompoundsEmtricitabineDeoxycytidineCytidinePyrimidine NucleosidesPyrimidinesAdeninePurinesHeterocyclic Compounds, 2-RingHeterocyclic Compounds, Fused-RingDrug CombinationsPharmaceutical Preparations

Results Point of Contact

Title
Gilead Clinical Study Information Center
Organization
Gilead Sciences

Study Officials

  • Gilead Study Director

    Gilead Sciences

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

January 19, 2015

First Posted

January 26, 2015

Study Start

January 26, 2015

Primary Completion

June 29, 2016

Study Completion

January 2, 2019

Last Updated

January 2, 2020

Results First Posted

October 19, 2017

Record last verified: 2019-12

Data Sharing

IPD Sharing
Will share

Qualified external researchers may request IPD for this study after study completion. For more information, please visit our website at http://www.gilead.com/research/disclosure-and transparency

Shared Documents
STUDY PROTOCOL, SAP
Time Frame
18 months after study completion
Access Criteria
A secured external environment with username, password, and RSA code
More information

Locations