NCT02256553

Brief Summary

The purpose of this study is to assess the safety and tolerability of MK-3641 (short ragweed \[Ambrosia artemisiifolia\] extract, SCH 039641, RAGWITEK®) sublingual tablets and MK-7243 (Timothy grass \[Phleum pratense\] extract, SCH 697243, GRASTEK®) sublingual tablets co-administered in participants 18 through 65 years of age with both ragweed- and grass polled-induced allergic rhinitis, with or without conjunctivitis and with or without asthma. The primary endpoint is the percentage of participants who experience at least one event of local swelling after co-administration of MK-3641 and MK-7243 sublingual tablets.

Trial Health

100
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
102

participants targeted

Target at P50-P75 for phase_4

Timeline
Completed

Started Oct 2014

Shorter than P25 for phase_4

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

October 1, 2014

Completed
Same day until next milestone

Study Start

First participant enrolled

October 1, 2014

Completed
2 days until next milestone

First Posted

Study publicly available on registry

October 3, 2014

Completed
4 months until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2015

Completed
Same day until next milestone

Study Completion

Last participant's last visit for all outcomes

February 1, 2015

Completed
12 months until next milestone

Results Posted

Study results publicly available

January 18, 2016

Completed
Last Updated

March 3, 2017

Status Verified

January 1, 2017

Enrollment Period

4 months

First QC Date

October 1, 2014

Results QC Date

December 7, 2015

Last Update Submit

January 18, 2017

Conditions

Outcome Measures

Primary Outcomes (1)

  • Percentage of Participants Who Experienced at Least One Event of Local Swelling

    Events of local swelling included pharyngeal edema, laryngeal edema, mouth edema, oropharyngeal swelling, palatal edema, tongue swelling/edema, or throat tightness. Events that occurred during in-clinic dosing were to be monitored and recorded by clinic staff. A Side Effect Report Card was used in Periods I-III to collect information on adverse events identified by the World Allergy Organization (WAO) as local side effects of sublingual immunotherapy (SLIT) that occurred within the first 60 minutes after study drug intake. During Period I, participants were to complete the report card once a day after MK-7243 was administered. During Period II, participants were to complete the report card twice a day, once after each tablet was administered. During Period III, participants were to complete the report card once a day after both tablets were administered.

    During Period I, Period II and Period III (Up to 6 weeks)

Secondary Outcomes (3)

  • Percentage of Participants Who Experienced at Least One Event of Local Application Site Reaction

    During Period I, Period II and Period III (Up to 6 weeks)

  • Percentage of Participants Who Discontinued Study Drug Due to an Adverse Event (AE)

    During Period I, Period II and Period III (Up to 6 weeks)

  • Percentage of Participants Who Experienced at Least One Local Application Site Reaction That Required Symptomatic Treatment

    During Period I, Period II and Period III (Up to 6 weeks)

Study Arms (1)

MK-3641+ MK-7243

EXPERIMENTAL

Participants receive one MK-7243 tablet, SL QD in the evening for 14 days during Period I; one MK-3641 tablet, SL QD in the morning and one MK-7243 tablet, SL QD in the evening for 14 days during Period II; and one MK-3641 tablet, SL QD, and one MK-7243 tablet, SL QD, within 5 minutes of each other for 14 days during Period III.

Biological: MK-3641 12 Amb a 1-U (short ragweed extract)Biological: MK-7243 2800 BAU (Timothy grass extract)Drug: Rescue Medication

Interventions

12 units of Ambrosia artemisiifolia major allergen number 1 (Amb a 1-U) extract sublingual tablets

Also known as: SCH 039641, RAGWITEK®
MK-3641+ MK-7243

2800 bioequivalent allergen units (BAU) of Phleum pratense extract sublingual tablets

Also known as: SCH 697243, GRASTEK®
MK-3641+ MK-7243

Self-injectable epinephrine, to be administered for an anaphylactic reaction, including symptoms/signs of upper airway obstruction.

MK-3641+ MK-7243

Eligibility Criteria

Age18 Years - 65 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • Clinical history of physician-diagnosed ragweed- and grass pollen-induced rhinitis with or without conjunctivitis of \>1 year duration, with or without asthma
  • Female participants of childbearing potential must have a negative urine pregnancy test at Screening and Randomization Visits and must agree to remain abstinent or use (or have their partner use) any one of the acceptable methods of birth control within the projected duration of the study. Acceptable methods of birth control are: intrauterine device (IUD), diaphragm with spermicide, contraceptive sponge, condom, vasectomy, hormonal contraception.

You may not qualify if:

  • Unstable, uncontrolled or severe asthma treated with long-acting beta agonists (LABAs) at the time of Screening
  • Received immunosuppressive treatment within 3 months prior to Randomization (except steroids for allergic reactions other than asthma)
  • History of anaphylaxis with cardiorespiratory symptoms with prior immunotherapy, unknown cause, or inhalant allergen
  • Diagnosis of eosinophilic esophagitis
  • History of any severe systemic allergic reaction or any severe local reaction to sublingual allergen immunotherapy
  • Female and breastfeeding, pregnant or intending to become pregnant
  • Received another form of allergen immunotherapy with the past month
  • Previously exposed to MK-3641 (RAGWITEK®) or other sublingual ragweed immunotherapy
  • Previously exposed to MK-7243 (GRASTEK®) or other sublingual grass immunotherapy
  • Known history of allergy, hypersensitivity, or intolerance to the excipient ingredients of the study drug (except for Ambrosia artemisiifolia and/or Phleum pratense), or self-injectable epinephrine
  • Unable to or will not comply with the use of self-injectable epinephrine
  • Used an investigational drug within 30 days prior to Screening Visit, or plans to participate in another interventional clinical trial during the duration of this trial
  • Family member of the investigational or sponsor staff involved in this trial
  • Participating in this same trial at another investigational site.

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Related Publications (1)

  • Maloney J, Berman G, Gagnon R, Bernstein DI, Nelson HS, Kleine-Tebbe J, Kaur A, Li Q, Nolte H. Sequential Treatment Initiation with Timothy Grass and Ragweed Sublingual Immunotherapy Tablets Followed by Simultaneous Treatment Is Well Tolerated. J Allergy Clin Immunol Pract. 2016 Mar-Apr;4(2):301-9.e2. doi: 10.1016/j.jaip.2015.11.004. Epub 2016 Jan 2.

MeSH Terms

Conditions

Rhinitis, Allergic, Seasonal

Condition Hierarchy (Ancestors)

Rhinitis, AllergicRhinitisNose DiseasesRespiratory Tract DiseasesRespiratory HypersensitivityOtorhinolaryngologic DiseasesHypersensitivity, ImmediateHypersensitivityImmune System Diseases

Results Point of Contact

Title
Senior Vice President, Global Clinical Development
Organization
Merck Sharp & Dohme Corp.

Study Officials

  • Medical Director

    Merck Sharp & Dohme LLC

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restriction Type
OTHER
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 4
Allocation
NA
Masking
NONE
Purpose
TREATMENT
Intervention Model
SINGLE GROUP
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

October 1, 2014

First Posted

October 3, 2014

Study Start

October 1, 2014

Primary Completion

February 1, 2015

Study Completion

February 1, 2015

Last Updated

March 3, 2017

Results First Posted

January 18, 2016

Record last verified: 2017-01