NCT02250872

Brief Summary

Cisplatin is a potent chemotherapeutic agent, however, its nephrotoxicity manifested by acute kidney injury (AKI) often limits applicability. Dipeptidylpeptidase-4 (DPP4) inhibitors are well known to improve glucose intolerance by augmentation of endogenous glucagon like peptide (GLP-1) and glucose-dependent insulinotropic peptide (GIP). DPP4 inhibitor also has the potential anti-apoptotic and renoprotective effect in a mouse model of cisplatin-induced AKI. This is a single-center, randomized, double-blind, parallel-group, placebo-controlled, prospective study to investigate the renoprotective effect of DPP4 inhibitor on cisplatin-induced AKI. A total 182 patients, who are scheduled to treat with cisplatin, will be recruited and randomly assigned to either Gemigliptin or placebo groups. Subjects will take study drugs for 8 days starting from one day before cisplatin treatment. Serum creatinine (Cr) and estimated glomerular filtration rate (eGFR) will be measured at 7 days after cisplatin treatment.

Trial Health

43
At Risk

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Trial has exceeded expected completion date
Enrollment
182

participants targeted

Target at P75+ for phase_2 cancer

Timeline
Completed

Started Dec 2014

Typical duration for phase_2 cancer

Geographic Reach
1 country

1 active site

Status
unknown

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

September 24, 2014

Completed
2 days until next milestone

First Posted

Study publicly available on registry

September 26, 2014

Completed
2 months until next milestone

Study Start

First participant enrolled

December 1, 2014

Completed
3.2 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

February 1, 2018

Completed
4 months until next milestone

Study Completion

Last participant's last visit for all outcomes

June 1, 2018

Completed
Last Updated

April 20, 2016

Status Verified

April 1, 2016

Enrollment Period

3.2 years

First QC Date

September 24, 2014

Last Update Submit

April 18, 2016

Conditions

Keywords

CisplatinNephrotoxicityGemigliptinDPP4 inhibitor

Outcome Measures

Primary Outcomes (1)

  • Incidence of acute kidney injury defined as any of the followings

    * Increase in sCr by ≥ 0.3 mg/dl * Increase in sCr to ≥ 1.5 times baseline * Decrease in eGFR to ≥ 25% All subjects receive Gemigliptin or placebo at a total dose of 100mg (50mg twice a day) for 8 consecutive days, serum creatinine will be measured.

    up to 7 days

Secondary Outcomes (2)

  • delta Cr

    Time Frame: up to 7 days

  • delta eGFR

    up to 7 days

Study Arms (2)

Experimental: Gemigliptin and Cisplatin

ACTIVE COMPARATOR

Gemigliptin 100mg daily in two divided doses for 8 days starting from one day before cisplatin-treatment

Drug: GemigliptinDrug: Cisplatin

Control arm

PLACEBO COMPARATOR

Placebo 100mg daily in two divided doses for 8 days starting from one day before cisplatin-treatment

Drug: PlaceboDrug: Cisplatin

Interventions

Gemigliptin 100mg in 2 divided doses plus cisplatin

Also known as: Zemiglo
Experimental: Gemigliptin and Cisplatin

100mg in 2 divided doses plus cisplatin

Also known as: Identical inert tablet to mimic gemigliptin (50mg)
Control arm

All patients will receive intravenous cisplatin

Control armExperimental: Gemigliptin and Cisplatin

Eligibility Criteria

Age18 Years - 70 Years
Sexall
Healthy VolunteersNo
Age GroupsAdult (18-64), Older Adult (65+)

You may qualify if:

  • age \> 18 years
  • cancer patients treated with intravenous cisplatin
  • written consent

You may not qualify if:

  • Diabetes mellitus
  • Chronic kidney disease stage IV-V (eGFR \< 30ml/min/1.73m2)
  • History of transplantation
  • History of acute kidney injury before randomization
  • Use of other nephrotoxic agents such as non steroidal anti-inflammatory drugs, aminoglycosides, colistin, vancomycin
  • Receiving contrast media during last 72 hours
  • Liver disease (bilirubin \> 2 mg/dl, transaminase levels \>2.5 times the upper limit normal)
  • Active infection
  • Patients with high risks of dehydration owing to poor oral intake
  • High blood pressure (\> 180/110 mmHg despite antihypertensive medications)
  • Hypersensitivity to Gemigliptin or its excipients
  • Low compliance to Gemigliptin treatment

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (1)

Seoul National University Bundang Hospital

Seongnam-si, Gyeonggi-do, 463-707, South Korea

RECRUITING

Related Publications (2)

  • Katagiri D, Hamasaki Y, Doi K, Okamoto K, Negishi K, Nangaku M, Noiri E. Protection of glucagon-like peptide-1 in cisplatin-induced renal injury elucidates gut-kidney connection. J Am Soc Nephrol. 2013 Dec;24(12):2034-43. doi: 10.1681/ASN.2013020134. Epub 2013 Oct 3.

  • Baek SH, Kim SH, Kim JW, Kim YJ, Lee KW, Na KY. Effects of a DPP4 inhibitor on cisplatin-induced acute kidney injury: study protocol for a randomized controlled trial. Trials. 2015 May 29;16:239. doi: 10.1186/s13063-015-0772-4.

Related Links

MeSH Terms

Conditions

Neoplasms

Interventions

LC15-0444Cisplatin

Intervention Hierarchy (Ancestors)

Chlorine CompoundsInorganic ChemicalsNitrogen CompoundsPlatinum Compounds

Study Officials

  • Ki Young Na

    Seoul National University Bundang Hospital

    PRINCIPAL INVESTIGATOR

Central Study Contacts

Ki Young Na

CONTACT

Study Design

Study Type
interventional
Phase
phase 2
Allocation
RANDOMIZED
Masking
DOUBLE
Who Masked
PARTICIPANT, CARE PROVIDER
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
OTHER
Responsible Party
PRINCIPAL INVESTIGATOR
PI Title
Professor

Study Record Dates

First Submitted

September 24, 2014

First Posted

September 26, 2014

Study Start

December 1, 2014

Primary Completion

February 1, 2018

Study Completion

June 1, 2018

Last Updated

April 20, 2016

Record last verified: 2016-04

Locations