NCT02187003

Brief Summary

This is a clinical study evaluating the efficacy and safety of rivipansel (GMI-1070) in treating subjects with sickle cell disease (SCD) who are 6 years of age or older experiencing a pain crisis necessitating hospitalization.

Trial Health

90
On Track

Trial Health Score

Automated assessment based on enrollment pace, timeline, and geographic reach

Enrollment
345

participants targeted

Target at P50-P75 for phase_3

Timeline
Completed

Started Jun 2015

Typical duration for phase_3

Geographic Reach
2 countries

142 active sites

Status
completed

Health score is calculated from publicly available data and should be used for screening purposes only.

Trial Relationships

Click on a node to explore related trials.

Study Timeline

Key milestones and dates

First Submitted

Initial submission to the registry

June 12, 2014

Completed
28 days until next milestone

First Posted

Study publicly available on registry

July 10, 2014

Completed
11 months until next milestone

Study Start

First participant enrolled

June 17, 2015

Completed
3.9 years until next milestone

Primary Completion

Last participant's last visit for primary outcome

May 3, 2019

Completed
2 months until next milestone

Study Completion

Last participant's last visit for all outcomes

June 27, 2019

Completed
5.7 years until next milestone

Results Posted

Study results publicly available

March 11, 2025

Completed
Last Updated

March 11, 2025

Status Verified

February 1, 2025

Enrollment Period

3.9 years

First QC Date

June 12, 2014

Results QC Date

February 26, 2024

Last Update Submit

February 18, 2025

Conditions

Keywords

Sickle Cell AnemiaSickle Cell DiseaseSickle Cell Disorderspain crisisvaso-occlusive crisisrivipanselGMI-1070selectin inhibitorSCDVOC

Outcome Measures

Primary Outcomes (1)

  • Time to Readiness for Discharge From Hospital

    Time to readiness-for-discharge from hospital was defined as the difference (in hours) between the time and date when all criteria for readiness-for-discharge were met and the start time and date of the first infusion (loading dose) of study drug. Criteria for readiness-for-discharge were met when all of the applicable 6 criteria (in relation to treatment of VOC and complications related to the VOC) were documented to have occurred. The six criteria were: 1) only oral pain medication was required, 2) acute complications related to the VOC (such as acute chest syndrome, stroke, priapism) had resolved to the extent that management could be in an outpatient setting, 3) IV opioids had been discontinued, 4) IV hydration had been discontinued, 5) IV antibiotics had been discontinued and 6) red blood cell (RBC) transfusion was no longer required for treatment of this VOC.

    Day 1 up to the latest day when all 6 criteria of readiness-for-discharge were met (up to an average of Day 8)

Secondary Outcomes (5)

  • Time to Discharge From Hospital

    Day 1 up to the latest day when the order of hospital discharge was issued by a qualified healthcare provider (up to an average of Day 8)

  • Cumulative Intravenous (IV) Opioids Consumption From Time of Loading Dose of Study Drug to Discharge From Hospital

    Day 1 up to the latest day when IV opioid was discontinued (up to an average of Day 8)

  • Time to Discontinuation of Intravenous (IV) Opioids

    Day 1 up to the latest day when IV opioid was discontinued (up to an average of Day 8)

  • Cumulative Intravenous (IV) Opioids Consumption Within First 24 Hours Post-Loading Dose of Study Drug

    24 hours post first IV infusion of loading dose of study drug on Day 1

  • Percentage of Participants Re-hospitalized for Vaso-Occlusive Crisis (VOC) Within 3 Days of Discharge From Hospital

    Within 3 days of discharge from hospital, where discharge from hospital was any day from Day 1 to an average of Day 8

Other Outcomes (9)

  • Number of Participants With Treatment Emergent Adverse Events (AEs) and Serious Adverse Events (SAEs) as Per Genotype

    Day 1 up to the 35-day post discharge visit (up to an average of Day 43)

  • Number of Participants With Treatment Emergent Adverse Event (AEs) as Per Severity

    Day 1 up to the 35-day post discharge visit (up to an average of Day 43)

  • Number of Participants With Clinical Laboratory Abnormalities

    Day 1 up to the 35-day post discharge visit (up to an average of Day 43)

  • +6 more other outcomes

Study Arms (2)

Rivipansel Treatment Arm

EXPERIMENTAL
Drug: Rivipansel

Placebo Treatment Arm

PLACEBO COMPARATOR
Other: Placebo

Interventions

Rivipansel (GMI-1070) will be infused intravenously every 12 hours up to 15 doses maximum. Subjects aged 12 and over who weigh more than 40 kilograms will receive a dose of 1680 mg of rivipansel, followed by a dose of 840 mg of rivipansel every 12 hours. All subjects aged 6 to 11 years and any subject who weighs 40 kilograms or less, will receive weight-based dosing (mg/kg) of 40 mg/kg of rivipansel (maximum of 1680 mg) followed by a dose of 20 mg/kg of rivipansel (maximum of 840 mg) every 12 hours.

Also known as: GMI-1070
Rivipansel Treatment Arm
PlaceboOTHER

Placebo (phosphate buffered saline) will be infused intravenously every 12 hours up to 15 doses maximum.

Also known as: phosphate buffered saline (PBS)
Placebo Treatment Arm

Eligibility Criteria

Age6 Years+
Sexall
Healthy VolunteersNo
Age GroupsChild (0-17), Adult (18-64), Older Adult (65+)

You may qualify if:

  • At least 6 years of age.
  • Documented diagnosis of sickle cell disease.
  • Diagnosis of vaso-occlusive crisis necessitating admission to the hospital with treatment including IV opioids.
  • Able to receive the first dose of study drug within 24 hours from the administration of IV opioids.

You may not qualify if:

  • Serious systemic infection
  • Acute Chest Syndrome
  • Serious concomitant medical problems (for example, stroke)
  • SCD pain atypical of VOC
  • Severe renal or hepatic impairment
  • Chronic pain rather than a presentation of acute VOC

Contact the study team to confirm eligibility.

Sponsors & Collaborators

Study Sites (142)

University of South Alabama Children's and Women's Hospital

Mobile, Alabama, 36604, United States

Location

Arkansas Children's Hospital Research Pharmacy

Little Rock, Arkansas, 72202, United States

Location

Arkansas Children's Hospital

Little Rock, Arkansas, 72202, United States

Location

UCSF Benioff Children's Hospital Oakland

Oakland, California, 94609, United States

Location

UC Davis Medical Center Main Hospital

Sacramento, California, 95817, United States

Location

UC Davis Medical Center

Sacramento, California, 95817, United States

Location

University of California Davis Medical Center

Sacramento, California, 95817, United States

Location

University of Colorado CTRC

Aurora, Colorado, 80045, United States

Location

University of Colorado Hospital

Aurora, Colorado, 80045, United States

Location

Howard University Center for Sickle Cell Disease

Washington D.C., District of Columbia, 20001, United States

Location

Medstar Health Research Institute

Washington D.C., District of Columbia, 20010, United States

Location

Howard University Hospital

Washington D.C., District of Columbia, 20060, United States

Location

Golisano Children's Hospital of Southwest Florida

Fort Myers, Florida, 33908, United States

Location

UF Health Davis Cancer Pavillion and Shands Med Plaza

Gainesville, Florida, 32608, United States

Location

UF Health Shands Cancer Hospital

Gainesville, Florida, 32608, United States

Location

UF Health Shands Hospital

Gainesville, Florida, 32610, United States

Location

Jackson Memorial Hospital

Miami, Florida, 33136, United States

Location

University Of Miami

Miami, Florida, 33136, United States

Location

Investigational Drug Service Tampa General Hospital

Tampa, Florida, 33606, United States

Location

Tampa General Hospital Center of Research Excellence

Tampa, Florida, 33606, United States

Location

Tampa General Hospital

Tampa, Florida, 33606, United States

Location

University of South Florida

Tampa, Florida, 33606, United States

Location

St. Joseph's Children's Hospital

Tampa, Florida, 33607, United States

Location

Children's Hematology and Oncology Associates

West Palm Beach, Florida, 33407, United States

Location

St. Mary's Medical Center

West Palm Beach, Florida, 33407, United States

Location

Children's Healthcare of Atlanta Aflac Cancer and Blood Disorders Center

Atlanta, Georgia, 30303, United States

Location

Grady Health System

Atlanta, Georgia, 30303, United States

Location

Children's Healthcare of Atlanta Aflac Cancer and Blood Disorders Center

Atlanta, Georgia, 30322, United States

Location

Emory Children's Center

Atlanta, Georgia, 30322, United States

Location

Children's Healthcare of Atlanta Aflac Cancer and Blood Disorders Center

Atlanta, Georgia, 30342, United States

Location

Children's Healthcare of Atlanta: Scottish Rite Campus

Atlanta, Georgia, 30342, United States

Location

Augusta University Clinical Research Pharmacy

Augusta, Georgia, 30912, United States

Location

Augusta University Medical Center

Augusta, Georgia, 30912, United States

Location

Augusta University

Augusta, Georgia, 30912, United States

Location

Memorial Family Medicine Ctr. @Memorial Health Univ Med Ct

Savannah, Georgia, 31404, United States

Location

Memorial Health University Medical Center

Savannah, Georgia, 31404, United States

Location

University of Illinois at Chicago Clinical Research Center

Chicago, Illinois, 60612, United States

Location

University of Illinois Hospital and Health Sciences System

Chicago, Illinois, 60612, United States

Location

The University of Chicago/Comer Children's Hospital

Chicago, Illinois, 60637, United States

Location

University of Chicago, Investigational Drug Service Pharmacy

Chicago, Illinois, 60637, United States

Location

University of Iowa Hospitals and Clinics

Iowa City, Iowa, 52242, United States

Location

Kosair Charities Pediatric Clinical Research Unit

Louisville, Kentucky, 40202, United States

Location

Norton Children´s Hospital

Louisville, Kentucky, 40202, United States

Location

The Novak Center for Children's Health

Louisville, Kentucky, 40202, United States

Location

University of Louisville Health Sciences Center

Louisville, Kentucky, 40202, United States

Location

University of Louisville Physicians Pediatric Hematology Oncology

Louisville, Kentucky, 40202, United States

Location

Our Lady of the Lake Regional Medical Center

Baton Rouge, Louisiana, 70808, United States

Location

St. Jude Affiliate Clinic

Baton Rouge, Louisiana, 70808, United States

Location

Our Lady of the Lake Physician Group-Medical Oncology

Baton Rouge, Louisiana, 70809, United States

Location

University of Maryland Medical System Investigational Pharmacy

Baltimore, Maryland, 21201, United States

Location

University of Maryland Medical System

Baltimore, Maryland, 21201, United States

Location

Johns Hopkins Medicine

Baltimore, Maryland, 21205, United States

Location

The Johns Hopkins University School of Medicine

Baltimore, Maryland, 21205, United States

Location

The Johns Hopkins Hospital

Baltimore, Maryland, 21287-6180, United States

Location

Johns Hopkins Medicine

Baltimore, Maryland, 21287, United States

Location

Boston Children's Hospital

Boston, Massachusetts, 02115, United States

Location

Brigham and Womens Hospital

Boston, Massachusetts, 02115, United States

Location

Center for Clinical Investigation, Brigham & Women's Hospital

Boston, Massachusetts, 02115, United States

Location

Investigational Drug Services

Boston, Massachusetts, 02115, United States

Location

Boston Medical Center E7E

Boston, Massachusetts, 02118, United States

Location

Boston Medical Center

Boston, Massachusetts, 02118, United States

Location

Boston University Medical Center

Boston, Massachusetts, 02118, United States

Location

Children's Hospital of Michigan

Detroit, Michigan, 48201, United States

Location

Detroit Medical Center Pharmacy

Detroit, Michigan, 48201, United States

Location

Wayne State University / Detroit Receiving Hospital

Detroit, Michigan, 48201, United States

Location

University of Mississippi Medical Center-Outpatient Clinical Research Unit

Jackson, Mississippi, 39216, United States

Location

University Of Mississippi Medical Center

Jackson, Mississippi, 39216, United States

Location

Children's Mercy Hospital

Kansas City, Missouri, 64108, United States

Location

Center for Outpatient Health

St Louis, Missouri, 63108, United States

Location

Barnes-Jewish Hospital Department of Pharmacy

St Louis, Missouri, 63110, United States

Location

Barnes-Jewish Hospital

St Louis, Missouri, 63110, United States

Location

Center for Advanced Medicine

St Louis, Missouri, 63110, United States

Location

Washington University School of Medicine

St Louis, Missouri, 63110, United States

Location

Bristol Myers Squibb Children's Hospital at Robert Wood Johnson University Hospital

New Brunswick, New Jersey, 08901, United States

Location

Rutgers-Robert Wood Johnson Medical School

New Brunswick, New Jersey, 08901, United States

Location

Rutgers Cancer Institute Of New Jersey

New Brunswick, New Jersey, 08903, United States

Location

Kings County Hospital Center - Pharmacy Department

Brooklyn, New York, 11203, United States

Location

Kings County Hospital Center

Brooklyn, New York, 11203, United States

Location

State University of New York (SUNY) - Downstate Medical Center

Brooklyn, New York, 11203, United States

Location

SUNY Downstate Medical Center University Hospital of Brooklyn

Brooklyn, New York, 11203, United States

Location

Icahn School of Medicine at Mount Sinai

New York, New York, 10029, United States

Location

Columbia University Medical Center Research Pharmacy

New York, New York, 10032, United States

Location

MS CHONY Pediatric Emergency Department

New York, New York, 10032, United States

Location

MS CHONY Pediatric Hematology/Oncology Unit

New York, New York, 10032, United States

Location

Staten Island University Hospital

Staten Island, New York, 10305, United States

Location

Jacobi Medical Center

The Bronx, New York, 10461, United States

Location

Duke University Hospital

Durham, North Carolina, 27710, United States

Location

Duke University Medical Center

Durham, North Carolina, 27710, United States

Location

East Carolina University Brody School of Medicine

Greenville, North Carolina, 27834, United States

Location

Leo W. Jenkins Cancer Center

Greenville, North Carolina, 27834, United States

Location

Vidant Medical Center

Greenville, North Carolina, 27834, United States

Location

University of Cincinnati Medical Center/ Investigational Pharmacy

Cincinnati, Ohio, 45219, United States

Location

University of Cincinnati Medical Center/Research Office

Cincinnati, Ohio, 45219, United States

Location

University of Cincinnati Medical Center

Cincinnati, Ohio, 45219, United States

Location

University of Cincinnati Physicians Company LLC

Cincinnati, Ohio, 45219, United States

Location

University of Cincinnati- Hoxworth Building

Cincinnati, Ohio, 45219, United States

Location

UC Health Ridgeway Hospital

Cincinnati, Ohio, 45229, United States

Location

The Ohio State University Wexner Medical Center East

Columbus, Ohio, 43203, United States

Location

Nationwide Childrens Hospital

Columbus, Ohio, 43205, United States

Location

The Ohio State University Investigational Drug Services

Columbus, Ohio, 43210, United States

Location

The Ohio State University James Comprehensive Cancer Hospital & Solove Research Institute

Columbus, Ohio, 43210, United States

Location

The Ohio State University Wexner Medical Center

Columbus, Ohio, 43210, United States

Location

Five Rivers Medical Surgical Health Center

Dayton, Ohio, 45402, United States

Location

Miami Valley Hospital

Dayton, Ohio, 45409, United States

Location

Einstein Medical Center Philadelphia

Philadelphia, Pennsylvania, 19141, United States

Location

UPMC Presbyterian

Pittsburgh, Pennsylvania, 15213, United States

Location

Children's Hospital of Pittsburgh of UPMC

Pittsburgh, Pennsylvania, 15224, United States

Location

UPMC Hillman Cancer Center

Pittsburgh, Pennsylvania, 15232, United States

Location

Hasbro Children's Hospital

Providence, Rhode Island, 02903, United States

Location

Rhode Island Hospital-Pharmacy Service

Providence, Rhode Island, 02903, United States

Location

Rhode Island Hospital

Providence, Rhode Island, 02903, United States

Location

The Miriam Hospital

Providence, Rhode Island, 02906, United States

Location

Medical University of South Carolina - Hospital

Charleston, South Carolina, 29425, United States

Location

Medical University of South Carolina Lifespan Comprehensive Sickle Cell Center

Charleston, South Carolina, 29425, United States

Location

Medical University of South Carolina

Charleston, South Carolina, 29425, United States

Location

MUSC Investigational Drug Services

Charleston, South Carolina, 29425, United States

Location

Cook Children's Hematology and Oncology Center

Fort Worth, Texas, 76104, United States

Location

Cook Children's Medical Center

Fort Worth, Texas, 76104, United States

Location

Cook Children's Hematology and Oncology Center-Grapevine

Grapevine, Texas, 76051, United States

Location

Texas Children's Hospital - Clinical Research Center

Houston, Texas, 77030, United States

Location

Texas Children´s Hospital

Houston, Texas, 77030, United States

Location

University of Texas Medical School

Houston, Texas, 77030, United States

Location

Primary Children's Hospital

Salt Lake City, Utah, 84113, United States

Location

Main Hospital - Virginia Commonwealth University

Richmond, Virginia, 23298, United States

Location

Virginia Commonwealth University-Investigational Drug Services

Richmond, Virginia, 23298, United States

Location

Virginia Commonwealth University

Richmond, Virginia, 23298, United States

Location

Royal Alexandra Hospital

Edmonton, Alberta, T5H 3V9, Canada

Location

Miseracordia Community Hospital

Edmonton, Alberta, T5R 4H5, Canada

Location

Kaye Edmonton Clinic 3 C

Edmonton, Alberta, T6G 1Z1, Canada

Location

University of Alberta Hospital, Pharmacy Services

Edmonton, Alberta, T6G 1Z1, Canada

Location

Stollery Children's Hospital

Edmonton, Alberta, T6G 2B7, Canada

Location

University of Alberta Hospital

Edmonton, Alberta, T6G 2B7, Canada

Location

Research transition Facility

Edmonton, Alberta, T6G 2V2, Canada

Location

Grey Nuns Community Hospital

Edmonton, Alberta, T6L 5X8, Canada

Location

St. Paul's Hospital

Vancouver, British Columbia, V6E 1M7, Canada

Location

St. Paul's Hospital

Vancouver, British Columbia, V6Z 1Y6, Canada

Location

Children's Hospital Of Eastern Ontario

Ottawa, Ontario, K1H 8L1, Canada

Location

University Health Network, Toronto General Hospital

Toronto, Ontario, M5G 2C4, Canada

Location

The Hospital for Sick Children

Toronto, Ontario, M5G1X8, Canada

Location

Centre Hospitalier Universitaire Sainte-Justine

Montreal, Quebec, H3T 1C5, Canada

Location

McGill University Health Centre, Royal Victoria Hospital

Montreal, Quebec, H4A 3J1, Canada

Location

The Montreal Children's Hospital/ McGill University Health Centre

Montreal, Quebec, H4A 3J1, Canada

Location

Related Publications (2)

  • Dampier CD, Telen MJ, Wun T, Brown RC, Desai P, El Rassi F, Fuh B, Kanter J, Pastore Y, Rothman J, Taylor JG, Readett D, Sivamurthy KM, Tammara B, Tseng LJ, Lozier JN, Thackray H, Magnani JL, Hassell KL; RESET Investigators. A randomized clinical trial of the efficacy and safety of rivipansel for sickle cell vaso-occlusive crisis. Blood. 2023 Jan 12;141(2):168-179. doi: 10.1182/blood.2022015797.

  • Rebelo AL, Chevalier MT, Russo L, Pandit A. Role and therapeutic implications of protein glycosylation in neuroinflammation. Trends Mol Med. 2022 Apr;28(4):270-289. doi: 10.1016/j.molmed.2022.01.004. Epub 2022 Feb 1.

MeSH Terms

Conditions

Anemia, Sickle CellVaso-Occlusive Crises

Interventions

rivipansel

Condition Hierarchy (Ancestors)

Anemia, Hemolytic, CongenitalAnemia, HemolyticAnemiaHematologic DiseasesHemic and Lymphatic DiseasesHemoglobinopathiesGenetic Diseases, InbornCongenital, Hereditary, and Neonatal Diseases and Abnormalities

Results Point of Contact

Title
Head of Regulatory
Organization
Biossil Inc.

Study Officials

  • Pfizer CT.gov Call Center

    Pfizer

    STUDY DIRECTOR

Publication Agreements

PI is Sponsor Employee
No
Restrictive Agreement
Yes

Study Design

Study Type
interventional
Phase
phase 3
Allocation
RANDOMIZED
Masking
QUADRUPLE
Who Masked
PARTICIPANT, CARE PROVIDER, INVESTIGATOR, OUTCOMES ASSESSOR
Purpose
TREATMENT
Intervention Model
PARALLEL
Sponsor Type
INDUSTRY
Responsible Party
SPONSOR

Study Record Dates

First Submitted

June 12, 2014

First Posted

July 10, 2014

Study Start

June 17, 2015

Primary Completion

May 3, 2019

Study Completion

June 27, 2019

Last Updated

March 11, 2025

Results First Posted

March 11, 2025

Record last verified: 2025-02

Data Sharing

IPD Sharing
Will not share

Locations